| Apstatin | IC50 | 2900.0 [1], 6100.0 [2] |
| CID 10336627 | IC50 | 230.0 [1], 430.0 [2] |
| (2S)-1-[(3R,4S)-4-Amino-3-hydroxy-6-methylheptanoyl]-N-[(2S)-1-amino-1-oxopropan-2-yl]pyrrolidine-2-carboxamide | IC50 | 1000000.0 [1], 2000000.0 [2] |
| (2S)-1-[(2S,3S)-3-Amino-2-hydroxy-5-methylhexanoyl]-N-[(2S)-1-amino-1-oxopropan-2-yl]pyrrolidine-2-carboxamide | IC50 | 58000.0 [1], 88000.0 [2] |
| (2S)-1-[(2S,4R)-1-[(2S,3R)-3-Amino-2-hydroxy-4-phenylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]-N-[(2S)-1-amino-1-oxopropan-2-yl]pyrrolidine-2-carboxamide | IC50 | 470000.0 [1], 600000.0 [2] |
| 2-[(2S)-2-[[(2S)-1-Amino-1-oxopropan-2-yl]carbamoyl]pyrrolidin-1-yl]-4-phenylbutanoic acid | IC50 | 2600.0 [1], 8400.0 [2] |
| (2S)-1-[(4R)-3-[(2S,3R)-3-Amino-2-hydroxy-4-phenylbutanoyl]-1,3-thiazolidine-4-carbonyl]-N-[(2S)-1-amino-1-oxopropan-2-yl]pyrrolidine-2-carboxamide | IC50 | 11000.0 [1], 18000.0 [2] |
| (2S)-1-[(2R,3R)-3-Amino-2-hydroxy-5-methylhexanoyl]-N-[(2S)-1-amino-1-oxopropan-2-yl]pyrrolidine-2-carboxamide | IC50 | 30000.0 [1], 31000.0 [2] |
| (2S)-1-[(2S,3R)-3-Amino-2-hydroxy-5-methylhexanoyl]-N-[(2S)-1-amino-1-oxopropan-2-yl]pyrrolidine-2-carboxamide | IC50 | 130.0 [1], 230.0 [2] |
| (2S)-1-[(2S)-1-[(2S,3R)-3-Amino-2-hydroxy-4-phenylbutanoyl]pyrrolidine-2-carbonyl]pyrrolidine-2-carboxamide | IC50 | 79000.0 [1], 89000.0 [2] |
| (2S)-N-[(2S)-1-Amino-1-oxopropan-2-yl]-1-[2-(hydroxycarbamoyl)cyclohexanecarbonyl]pyrrolidine-2-carboxamide | IC50 | 1300000.0 [1], 9000000.0 [2] |
| (2S)-N-[(2S)-1-Amino-1-oxopropan-2-yl]-1-(2-sulfanylcyclopentanecarbonyl)pyrrolidine-2-carboxamide | IC50 | 300000.0 [1], 390000.0 [2] |
| (2S)-1-[(2S)-1-[(2S,3R)-3-Amino-2-hydroxy-4-phenylbutanoyl]pyrrolidine-2-carbonyl]-N-[(2S)-1-[[(2S)-1-[[(2R)-1-amino-1-oxo-3-sulfanylpropan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]pyrrolidine-2-carboxamide | IC50 | 2800.0 [1], 3400.0 [2] |
| 2-[[6-[(3R)-3-Amino-3-methylpiperidin-1-yl]-1,3-dimethyl-2,4-dioxopyrrolo[3,2-d]pyrimidin-5-yl]methyl]-4-fluorobenzonitrile | IC50 | 50000.0 [1] |
| (3R)-1-[(2S)-1-[(2S,4S)-4-Fluoro-1-[(2S)-4-methyl-2-sulfanylpentanoyl]pyrrolidine-2-carbonyl]pyrrolidine-2-carbonyl]pyrrolidine-3-carboxylic acid | IC50 | 3.7 [1] |
| (3S)-1-[(2S)-1-[(2S)-1-[(2S)-4-Methyl-2-sulfanylpentanoyl]pyrrolidine-2-carbonyl]pyrrolidine-2-carbonyl]pyrrolidine-3-carboxylic acid | IC50 | 26.0 [1] |
| (2S)-2-[Methyl-[(2S)-1-[(2S)-1-[(2S)-4-methyl-2-sulfanylpentanoyl]pyrrolidine-2-carbonyl]pyrrolidine-2-carbonyl]amino]propanoic acid | IC50 | 3.9 [1] |
| (2R)-1-[(2S)-1-[(2S)-1-[(2S)-4-Methyl-2-sulfanylpentanoyl]pyrrolidine-2-carbonyl]pyrrolidine-2-carbonyl]pyrrolidine-2-carboxylic acid | IC50 | 9.7 [1] |