![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_f0193f5276395ac51bc314c2ce4fc0c3.svg) | Mibefradil | IC50 | 130.0 [1], 181.0 [2], 1000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_54fa1df58338066d74c0171644a913bb.svg) | N,3-Bis(4-fluorophenyl)-5-pyridin-4-yl-3,4-dihydropyrazole-2-carboxamide | IC50 | 33.0 [1], 220.0 [2], 1700.0 [3] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_930013c9bfe5e54bf92595f70af47ec4.svg) | N-((1-(2-(Tert-Butylamino)-2-oxoethyl)piperidin-4-yl)methyl)-3-chloro-5-fluorobenzamide | IC50 | 73.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_77a621d46f70126639b55033f633b6aa.svg) | CID 24765479 | IC50 | 8.2 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_e49fd68b8d0e620242090f7ae222ad7b.svg) | N-[[5-(2-Methylpropyl)-1-phenylpyrazol-3-yl]methyl]benzenesulfonamide | IC50 | 5800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_011692593cb9bed117be0130bcb96326.svg) | 3-Chloro-2,5,5-trimethyl-N-[[2-(propan-2-yloxymethyl)phenyl]methyl]-6,7-dihydro-4H-isoindole-1-carboxamide | IC50 | 6.6 [1], 130.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_d8882629bd9b8f1148cac7733e73c0de.svg) | 3-(4-Chlorophenyl)-N-(3,4-difluorophenyl)-2-propan-2-yl-2,7-diazaspiro[3.5]nonane-7-carboxamide | IC50 | 174.0 [1], 340.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_94ee17801bc4b7f45644ebd29e01d83d.svg) | 3-(4-Chlorophenyl)-N-(3,5-difluorophenyl)-2-propan-2-yl-2,7-diazaspiro[3.5]nonane-7-carboxamide | IC50 | 138.0 [1], 328.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_f71fddf3a0d3ecc7904f94184ae6c288.svg) | 7-(6-Chloro-1H-benzimidazol-2-yl)-2-(3-chloro-4-fluorophenyl)-1-pyridin-2-yl-2,7-diazaspiro[3.5]nonan-3-one | IC50 | 71.0 [1], 78.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_a8145457033a8f0b4bd6fea73643e30e.svg) | 2-(3-Chlorophenyl)-7-[5-fluoro-6-(trifluoromethyl)-1H-benzimidazol-2-yl]-1-pyridin-2-yl-2,7-diazaspiro[3.5]nonan-3-one | IC50 | 44.0 [1], 63.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_292798b96d6ddb47b31332583dd8ae71.svg) | 2-(3-Chloro-4-fluorophenyl)-7-[5-fluoro-6-(trifluoromethyl)-1H-benzimidazol-2-yl]-1-pyridin-2-yl-2,7-diazaspiro[3.5]nonan-3-one | IC50 | 29.0 [1], 106.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_e669cb4be55857574ee0fbeb893884bd.svg) | 2-(3-Cyanophenyl)-N-(3,5-difluorophenyl)-3-oxo-1-pyridin-2-yl-2,7-diazaspiro[3.5]nonane-7-carboxamide | IC50 | 2377.0 [1], 19300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_5b9d3d93930ba1064fb374fc064f3fdf.svg) | Methyl (2S,3S)-2-[[3-(4-chlorophenyl)-2-propan-2-yl-2,7-diazaspiro[3.5]nonane-7-carbonyl]amino]-3-methylpentanoate | IC50 | 733.0 [1], 3197.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_f0b6b1b6d0b9c309974a5f51df00c407.svg) | N-(3,5-Difluorophenyl)-3-(4-fluorophenyl)-2-propan-2-yl-2,7-diazaspiro[3.5]nonane-7-carboxamide | IC50 | 172.0 [1], 995.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_fa689dad2cd978763cbf2e0f4c3e8c9d.svg) | Methyl (2S,3S)-2-[[1-(4-chlorophenyl)-2-(3-fluorophenyl)-3-oxo-2,7-diazaspiro[3.5]nonane-7-carbonyl]amino]-3-methylpentanoate | IC50 | 109.0 [1], 872.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_c29b6633bc116eff58716398e7b56b82.svg) | 2-(3-Chloro-4-fluorophenyl)-N-(3,5-difluorophenyl)-3-pyridin-2-yl-2,7-diazaspiro[3.5]nonane-7-carboxamide | IC50 | 41.0 [1], 291.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_e0de0a502e47d0e15a6600fdcefe4397.svg) | 2-(3-Chloro-4-fluorophenyl)-N-(3,5-difluorophenyl)-3-oxo-1-pyridin-2-yl-2,7-diazaspiro[3.5]nonane-7-carboxamide | IC50 | 42.0 [1], 176.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_fc2b0ef9af534447df62799d39703917.svg) | 2-(3-Chloro-4-fluorophenyl)-N-(3,4-difluorophenyl)-3-oxo-1-pyridin-2-yl-2,7-diazaspiro[3.5]nonane-7-carboxamide | IC50 | 402.0 [1], 17700.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_e8d0c1584f11887448b34f2a8d31aa43.svg) | 2-(3,4-Difluorophenyl)-3-oxo-1-pyridin-2-yl-N-[3-(trifluoromethyl)phenyl]-2,7-diazaspiro[3.5]nonane-7-carboxamide | IC50 | 176.0 [1], 283.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_d025da7bd71e8b2cbe37a099a34a69fc.svg) | 2-(3-Chlorophenyl)-N-(3,4-difluorophenyl)-3-oxo-1-pyridin-2-yl-2,7-diazaspiro[3.5]nonane-7-carboxamide | IC50 | 118.0 [1], 652.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_83c5069efcdc890cfd4330e2d862fa2a.svg) | 2-(3-Chlorophenyl)-N-(3,5-difluorophenyl)-3-oxo-1-pyridin-2-yl-2,7-diazaspiro[3.5]nonane-7-carboxamide | IC50 | 200.0 [1], 3490.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_75ea3a15159bf347101a955732fce64a.svg) | 7-(5-Chloro-6-fluoro-1H-benzimidazol-2-yl)-2-(3-chloro-4-fluorophenyl)-1-pyridin-2-yl-2,7-diazaspiro[3.5]nonan-3-one | IC50 | 60.0 [1], 84.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_0ddfc0382db93feadcc1143e01aafb3a.svg) | Cyano (2S,3S)-2-[[1-(4-chlorophenyl)-2-(3-fluorophenyl)-3-oxo-2,7-diazaspiro[3.5]nonane-7-carbonyl]amino]-3-methylpentanoate | IC50 | 35.0 [1], 17000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_9ffa733b44dbf9418b40a570f9de40c3.svg) | Methyl (2S,3S)-2-[[3-(4-chlorophenyl)-2-cyclopropyl-2,7-diazaspiro[3.5]nonane-7-carbonyl]amino]-3-methylpentanoate | IC50 | 325.0 [1], 713.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_af21967b53bfd2b826ca060f1d6b9c87.svg) | N-[[1-[2-(Tert-butylcarbamoylamino)ethyl]-4-(hydroxymethyl)piperidin-4-yl]methyl]-3,5-dichlorobenzamide | IC50 | 600.0 [1], 1200.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_2f396015dd3e84f1397988e4b6cdaffb.svg) | 8-Prenylnaringenin | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_6d769aa9526664c40191c0bd93326b38.svg) | NNC 55-0396 dihydrochloride | IC50 | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_51491790f6dc0e1f82f40025f5821d46.svg) | Sophoraflavanone G | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_0059e281ee1c8332255ffd38925c22eb.svg) | (R)-2-(4-Cyclopropylphenyl)-N-(1-(5-(2,2,2-trifluoroethoxy)pyridin-2-yl)ethyl)acetamide | IC50 | 92.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_2477d5ffbb98229152a04684816828b6.svg) | 1-[4-(Diphenylmethyl)-1-piperazinyl]-3,3-diphenyl-1-propanone | IC50 | 45000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_9b45fa7c41d4f6e3e6fa07d5e0489a47.svg) | (S)-4',5,7-Trihydroxy-6-prenylflavanone | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_a462c0bfa1d0e2a99d0468fe87ed726c.svg) | Auglurant | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_ba83dc79262458d01764950d1b6af431.svg) | 1-[3-(3,5-Dimethylpiperidine-1-carbonyl)benzenesulfonyl]-2-methyl-2,3-dihydro-1H-indole | IC50 | 3000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_865e442b08866850e5be87403820558c.svg) | N-Benzyl-2-[2-[5-(dimethylamino)pentyl-methylamino]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]acetamide;dihydrochloride | IC50 | 3600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_32593ab9e8f26835ff9e5fa89ce98aed.svg) | N-(1-Benzyl-1H-pyrazol-3-yl)benzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_4f5a1ee200fbb94ced49cd871f25ebcc.svg) | N-(1-Benzylpyrazol-3-yl)-2-phenylacetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_25a671d01c5314045b84690115b71784.svg) | 3-Fluoro-N-[[5-(2-methylpropyl)-1-phenylpyrazol-3-yl]methyl]benzenesulfonamide | IC50 | 2080.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_bdaebf3e2c11faf34d57af15dea12c0b.svg) | N-[1-[(5-Cyanopyridin-2-yl)methyl]pyrazol-3-yl]-2-[4-[1-(trifluoromethyl)cyclopropyl]phenyl]acetamide | IC50 | 18.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_d838f5f6c5209d24629c9402bb67a545.svg) | N-Benzyl-2-[2-[5-(dimethylamino)pentyl-methylamino]-6,8-difluoro-3-(4-phenylphenyl)-4H-quinazolin-4-yl]acetamide | IC50 | 5600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_1b95b25c2550bc68521b60171bcdde32.svg) | N-[(4-Fluorophenyl)methyl]-2-[3-(4-phenylphenyl)-2-[4-(2-pyrrolidin-1-ylethyl)piperazin-1-yl]-4H-quinazolin-4-yl]acetamide | IC50 | 5100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_878a482729b833a0834e68c7bbb1d6cd.svg) | 6-[[[1-[2-(7-Methoxy-2-oxoquinoxalin-1-yl)ethyl]piperidin-4-yl]amino]methyl]-4H-pyrido[3,2-b][1,4]oxazin-3-one | IC50 | 333000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_d689892c42c70ddff66c315b09e72743.svg) | [(1S,2S)-2-[2-[3-(1H-Benzimidazol-2-yl)propyl-methylamino]ethyl]-6-fluoro-1-propan-2-yl-3,4-dihydro-1H-naphthalen-2-yl] 2-methylpropanoate | IC50 | 149.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_19a54a26b2488d227f82c36d47245b22.svg) | Propan-2-yl 4-(3-chlorophenyl)-6-methyl-3-[3-[methyl-(4-phenoxybenzoyl)amino]propyl]-2-oxo-1,4-dihydropyrimidine-5-carboxylate | IC50 | 180.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_bb1d622c709b3a01ff279448f778ea61.svg) | Benzyl N-[2-[3-[benzyl-(3-chlorophenyl)sulfamoyl]anilino]-2-oxoethyl]-N-methylcarbamate | IC50 | 110.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_299d0b03fea867f9073621ca7bfc2e6c.svg) | Benzyl N-[2-[3-[(3-chlorophenyl)-[2-oxo-2-(propan-2-ylamino)ethyl]sulfamoyl]anilino]-2-oxoethyl]-N-methylcarbamate | IC50 | 1700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_7f6ec9a0fb29208bf55c5e2a0247ede2.svg) | Propan-2-yl 2-(3-chloro-N-[3-[3-(phenylmethoxycarbonylamino)propanoylamino]phenyl]sulfonylanilino)acetate | IC50 | 420.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_327bbcf54521b6862d7d521dd0184f84.svg) | Propan-2-yl 2-(3-chloro-N-[3-(3-phenylpropanoylamino)phenyl]sulfonylanilino)acetate | IC50 | 540.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_b0d9878cb766b26a9c655e9f2722ca36.svg) | Propan-2-yl 2-(3-chloro-N-[3-[[2-[methyl(phenylmethoxycarbonyl)amino]acetyl]amino]phenyl]sulfonylanilino)acetate | IC50 | 240.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_67e513f455b360d465aade2685b707be.svg) | N-[[4-Methyl-5-(2-methylpropyl)-1-phenylpyrazol-3-yl]methyl]benzenesulfonamide | IC50 | 4300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_bbfe737f7f05f9ba2dc25624a5b1d2ee.svg) | 2-[4-(Dimethylamino)phenyl]-N-[1-[(4-fluorophenyl)methyl]pyrazol-3-yl]acetamide | IC50 | 12.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_7d8330e63a7ab090476c65c01cec8d56.svg) | N-[1-[(4-Cyano-3-fluorophenyl)methyl]pyrazol-3-yl]-2-[4-(dimethylamino)phenyl]acetamide | IC50 | 14.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_27acca67234a8b83659df2d2b234c2a8.svg) | N-[1-[(3,5-Difluoro-4-methoxyphenyl)methyl]pyrazol-3-yl]-2-[4-(dimethylamino)phenyl]acetamide | IC50 | 7.8 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_ccbf5bd8f6256a79dafc8d74e74610a3.svg) | 2-[4-(Dimethylamino)phenyl]-N-[1-[(4-methylphenyl)methyl]pyrazol-3-yl]acetamide | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_b368a548d0447e71dc730586577ff478.svg) | N-[1-[(4-Cyanophenyl)methyl]pyrazol-3-yl]-2-[4-(dimethylamino)phenyl]acetamide | IC50 | 20.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_8d85cac1a61bcd1ae3a984e7201f4e65.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-[6-(dimethylamino)pyridin-3-yl]acetamide | IC50 | 46.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_6e31401d1fc2a51ccaa21a9a9fa5ffb4.svg) | N-[1-[[4-(Difluoromethoxy)phenyl]methyl]pyrazol-3-yl]-2-[4-(dimethylamino)phenyl]acetamide | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_ba9759f81982117d7269eed1947d3be9.svg) | 2-[4-(Dimethylamino)phenyl]-N-[1-[[4-(trifluoromethoxy)phenyl]methyl]pyrazol-3-yl]acetamide | IC50 | 5.1 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_c600fb4f3d11e81691ac5814f19a6b7f.svg) | N-[1-[(4-Chlorophenyl)methyl]pyrazol-3-yl]-2-[4-(dimethylamino)phenyl]acetamide | IC50 | 4.1 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_05f0450c8870f0c328609839e9d94a56.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-[4-(dimethylamino)phenyl]acetamide | IC50 | 3.4 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_8b0666fec5cce5cc5c0888655f5ec24e.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-[6-[(3S)-3-fluoropyrrolidin-1-yl]pyridin-3-yl]acetamide | IC50 | 21.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_afc965692104603b543742c94c22d8d5.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-[4-(3-fluorooxetan-3-yl)phenyl]acetamide | IC50 | 13.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_ed2fbafcc2ccf561c9a32410c450c7a2.svg) | 2-(6-Cyclopropylpyridin-3-yl)-N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]acetamide | IC50 | 220.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_ca06acabaad5b5426140dc1285e4e5b3.svg) | 2-[4-(Dimethylamino)phenyl]-N-[1-[(4-methoxyphenyl)methyl]pyrazol-3-yl]acetamide | IC50 | 47.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_a58c89dec3276d6f7aadb447315bcafe.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-(1H-indol-6-yl)acetamide | IC50 | 5.3 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_e830fd54289b9eea3d710bd4fed353bf.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-[4-(oxetan-3-yloxy)phenyl]acetamide | IC50 | 32.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_227d26b76f0172b6428458f06bf13609.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-(1-methylpyrrolo[2,3-b]pyridin-5-yl)acetamide | IC50 | 35.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_5330ce2e4570c55020a74555943931fb.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-(1H-indol-5-yl)acetamide | IC50 | 14.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_8ca26ef53f30d42d441fce7179208d29.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-(4-propan-2-ylphenyl)acetamide | IC50 | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_2038c48d438d42c36bc596518a7cc97b.svg) | 2-[4-(3,3-Difluorocyclobutyl)oxyphenyl]-N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]acetamide | IC50 | 11.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_da0091434e3739261e361b345822eeb0.svg) | 2-(4-Tert-butylphenyl)-N-[1-[(5-cyanopyridin-2-yl)methyl]pyrazol-3-yl]acetamide | IC50 | 7.5 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_cf226c259c9edc869a5cbbb91a10e0f4.svg) | 2-[4-(3,3-Difluorocyclobutyl)phenyl]-N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]acetamide | IC50 | 6.1 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_a031997dbba0f0e387338ca22767b08a.svg) | N-[2-[(3,4-Difluorophenyl)methyl]triazol-4-yl]-2-(1-methylindazol-5-yl)acetamide | IC50 | 8.6 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_dece8a540b188d817e14400ee34cf6f3.svg) | ABT-639 hydrochloride | IC50 | 2300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_8e764b68bb342ee732c629084d4aeba3.svg) | [(1S,2R,4S)-2-[2-[3-(1H-Benzimidazol-2-yl)propyl-methylamino]ethyl]-6-fluoro-4-methoxy-1-propan-2-yl-3,4-dihydro-1H-naphthalen-2-yl] 2-methylpropanoate | IC50 | 318.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_bbd692fd295a4917108f28a827101f15.svg) | [(1S,2R,4R)-2-[2-[3-(1H-Benzimidazol-2-yl)propyl-methylamino]ethyl]-6-fluoro-4-phenylmethoxy-1-propan-2-yl-3,4-dihydro-1H-naphthalen-2-yl] 2-methylpropanoate | IC50 | 132.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_1d0816badf3f36d340ac6f25d55d1b40.svg) | [(1S,2R,4S)-2-[2-[3-(1H-Benzimidazol-2-yl)propyl-methylamino]ethyl]-6-fluoro-4-phenylmethoxy-1-propan-2-yl-3,4-dihydro-1H-naphthalen-2-yl] 2-methylpropanoate | IC50 | 113.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_a5b696fabff177cf7ce29d26af6f1e74.svg) | [(1S,2R,4R)-2-[2-[3-(1H-Benzimidazol-2-yl)propyl-methylamino]ethyl]-6-fluoro-4-hydroxy-1-propan-2-yl-3,4-dihydro-1H-naphthalen-2-yl] 2-methylpropanoate | IC50 | 107.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_0e030a1636e29960a54cc73c3825017d.svg) | [(1S,2R,4S)-2-[2-[3-(1H-Benzimidazol-2-yl)propyl-methylamino]ethyl]-6-fluoro-4-hydroxy-1-propan-2-yl-3,4-dihydro-1H-naphthalen-2-yl] 2-methylpropanoate | IC50 | 76.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_de696624bbe33eb459b24c1b7ef677e1.svg) | [(1S,8S,9S)-9-[2-[3-(1H-Benzimidazol-2-yl)propyl-methylamino]ethyl]-9-tricyclo[6.2.2.02,7]dodeca-2,4,6-trienyl] 2-methoxyacetate | IC50 | 361.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_4560f99ece7cbf8878ad3de3ad3cd18a.svg) | [(1S,8S,9S)-9-[2-[3-(1H-Benzimidazol-2-yl)propyl-methylamino]ethyl]-9-tricyclo[6.2.2.02,7]dodeca-2,4,6-trienyl] cyclopropanecarboxylate | IC50 | 210.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_6a2d194eb50ec40a2b40d28897051680.svg) | [(1S,8S,9S)-9-[2-[3-(1H-Benzimidazol-2-yl)propyl-methylamino]ethyl]-3,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-trien-9-yl] 2-methylpropanoate | IC50 | 2065.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_89231bb0439fd5767f4c3f82e5933031.svg) | [(1S,2S)-2-[2-[3-(1H-Benzimidazol-2-yl)propyl-methylamino]ethyl]-6-fluoro-4,4-dimethyl-1-propan-2-yl-1,3-dihydronaphthalen-2-yl] 2-methoxyacetate | IC50 | 207.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_634845a20f1db8bea2c7fb7825d8e48b.svg) | [(1S,2S,4R)-2-[2-[3-(1H-Benzimidazol-2-yl)propyl-methylamino]ethyl]-4-butyl-6-fluoro-1-propan-2-yl-3,4-dihydro-1H-naphthalen-2-yl] 2-methoxyacetate | IC50 | 193.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_021518e26968b8a5fd1adcfb74291934.svg) | [(1S,2R,4R)-2-[2-[3-(1H-Benzimidazol-2-yl)propyl-methylamino]ethyl]-6-fluoro-4-methoxy-1-propan-2-yl-3,4-dihydro-1H-naphthalen-2-yl] 2-methylpropanoate | IC50 | 557.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_ac8c4d3fabe18ca81fedbe86a825e711.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-[6-(3,3-difluoropyrrolidin-1-yl)pyridin-3-yl]acetamide | IC50 | 6.7 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_0b3310d6ce08dd3afd47816f22ea5f10.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-[6-(2,2,2-trifluoroethoxy)pyridin-3-yl]acetamide | IC50 | 140.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_bc7dbb045135c69299207bfe0ad25682.svg) | N-[1-[(5-Cyanopyridin-2-yl)methyl]pyrazol-3-yl]-2-[3-ethyl-4-(2,2,2-trifluoroethoxy)phenyl]acetamide | IC50 | 7.8 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_0cf9e9ccd421656e56762f9eaac8f97d.svg) | N-[1-[(5-Cyanopyridin-2-yl)methyl]pyrazol-3-yl]-2-[3-methyl-4-(trifluoromethoxy)phenyl]acetamide | IC50 | 25.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_31dfeb00dd4088c3db5b02e709e8f022.svg) | N-[1-[(5-Cyanopyridin-2-yl)methyl]pyrazol-3-yl]-2-[3-methyl-4-(3,3,3-trifluoropropoxy)phenyl]acetamide | IC50 | 18.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_7329fc71a0b4aea8482e9aa0e8c9b064.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-(1-methylindazol-5-yl)acetamide | IC50 | 8.4 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_65ab047f9a83871df533bef503221178.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-(1,3,3-trimethyl-2-oxoindol-5-yl)acetamide | IC50 | 3.8 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_1c4146bebef03dea63bf42c6b7a42c4f.svg) | N-[1-[(5-Cyanopyridin-2-yl)methyl]pyrazol-3-yl]-2-[3-methyl-4-(2,2,2-trifluoroethoxy)phenyl]acetamide | IC50 | 7.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_3a455dea3633f832da16b30918de1baa.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-(3-methyl-2-oxo-1,3-benzoxazol-6-yl)acetamide | IC50 | 15.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_92bce33f608ab742f1bc1dfbbc085935.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-[4-(3-methyloxetan-3-yl)phenyl]acetamide | IC50 | 4.3 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_2cb13dec8818c32befd3b770d280f554.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-[4-[(3-methyloxetan-3-yl)methoxy]phenyl]acetamide | IC50 | 34.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_16fbbdb2f79224989553048e5b091be0.svg) | 2-[(1-Phenyl-5-propan-2-ylpyrazol-3-yl)methyl]-3H-1,2-benzothiazole 1,1-dioxide | IC50 | 2520.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_7d19de73f3bde0c23d5ec68d4b859929.svg) | 2-[[1-(4-Fluorophenyl)-5-propan-2-ylpyrazol-3-yl]methyl]-3H-1,2-benzothiazole 1,1-dioxide | IC50 | 2320.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_b8e141f2bd5b87fa73353cedf66854c3.svg) | Ethyl 3-[3-[2-(benzhydrylcarbamothioyl)hydrazinyl]-3-oxopropyl]-6-methyl-4-(3-nitrophenyl)-2-oxo-1,4-dihydropyrimidine-5-carboxylate | IC50 | 340.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_8aca67fa827e3c8ef3cf3156c55ab2fc.svg) | (3R,5S)-N,1-Dibenzyl-3,5-dimethyl-3,5-dihydro-2H-pyrido[3,4-e][1,4]diazepine-4-carboxamide | IC50 | 102.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1h-subunit_c7bb7e667d7eeb64cde2ce9ef26c506d.svg) | (5S)-N,1-Dibenzyl-5-methyl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide | IC50 | 241.0 [1] |