![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_f0193f5276395ac51bc314c2ce4fc0c3.svg) | Mibefradil | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_5fe8c3e316406ba1c7b9e03e98f9c275.svg) | N-Benzyl-2-[2-[5-(dimethylamino)pentyl-methylamino]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]acetamide | IC50 | 41.0 [1], 41.3 [2], 260.0 [3] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_67294eecd01c7dd489f6b3b484f8cd8c.svg) | N-[[4-[(4-Methylphenyl)sulfonylamino]phenyl]methyl]-2-(3-phenyl-2-piperidin-1-yl-4H-quinazolin-4-yl)acetamide | IC50 | 169.82 [1], 170.0 [2], 250.0 [3] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_2bb689ddc1c3e508cb92682d831f7ea2.svg) | Methyl 2-(2-(5-aminopentylamino)-3-(biphenyl-4-yl)-3,4-dihydroquinazolin-4-yl)acetate | IC50 | 559.76 [1], 560.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_5c9afb920f1f246824c74e33c665f955.svg) | N-[[4-[(4-Fluorophenyl)sulfonylamino]phenyl]methyl]-2-(3-phenyl-2-piperidin-1-yl-4H-quinazolin-4-yl)acetamide | IC50 | 110.0 [1], 200.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_d59dac732f9315714f21dd72f791be11.svg) | N-Benzyl-2-(3-phenyl-2-piperidin-1-yl-4H-quinazolin-4-yl)acetamide | IC50 | 900.0 [1], 1160.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_7df7a64fe584dcebf0b4d63342fa6643.svg) | N-Benzyl-2-[2-[methyl(5-pyrrolidin-1-ylpentyl)amino]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]acetamide | IC50 | 260.0 [1], 260.02 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_1b7e495e646d3983091593ffdebcb62f.svg) | Tert-butyl N-[5-[4-[2-(benzylamino)-2-oxoethyl]-2-(4-phenylanilino)-4H-quinazolin-3-yl]pentyl]carbamate | IC50 | 169.82 [1], 170.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_71bd90b88a34a71d71df6f3385a6abd3.svg) | 2-[2-(5-Aminopentylimino)-3-(4-phenylphenyl)-1,4-dihydroquinazolin-4-yl]-N-benzylacetamide | IC50 | 130.0 [1], 130.02 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_2ba105520f0d3af298ba54fc99d4e03f.svg) | Methyl 2-[2-[5-[(2-methylpropan-2-yl)oxycarbonylamino]pentylimino]-3-(4-phenylphenyl)-1,4-dihydroquinazolin-4-yl]acetate | IC50 | 679.2 [1], 680.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_34045fa732833c6c7e3d5a71a6ea291e.svg) | Tert-butyl N-[5-[[4-[2-(benzylamino)-2-oxoethyl]-3-(4-phenylphenyl)-1,4-dihydroquinazolin-2-ylidene]amino]pentyl]carbamate | IC50 | 159.96 [1], 160.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_837276853661820f5722e8566c3c2802.svg) | Methyl 2-[2-[5-(dimethylamino)pentyl-methylamino]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]acetate | IC50 | 230.0 [1], 230.14 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_feca8145ffd7aeea69e4c3c54f897f15.svg) | Methyl 2-(3-(5-aminopentyl)-2-(biphenyl-4-ylamino)-3,4-dihydroquinazolin-4-yl)acetate | IC50 | 299.92 [1], 300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_9bc2bbd55bbe20f393d7f3df8729e564.svg) | Methyl 5-((3-(1H-benzo[d]imidazol-2-yl)propyl)(methyl)amino)-2-(4-bromophenyl)-2-isopropylpentanoate | IC50 | 8.17 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_54fa1df58338066d74c0171644a913bb.svg) | N,3-Bis(4-fluorophenyl)-5-pyridin-4-yl-3,4-dihydropyrazole-2-carboxamide | IC50 | 29.0 [1], 450.0 [2], 1800.0 [3] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_930013c9bfe5e54bf92595f70af47ec4.svg) | N-((1-(2-(Tert-Butylamino)-2-oxoethyl)piperidin-4-yl)methyl)-3-chloro-5-fluorobenzamide | IC50 | 37.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_865e442b08866850e5be87403820558c.svg) | N-Benzyl-2-[2-[5-(dimethylamino)pentyl-methylamino]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]acetamide;dihydrochloride | IC50 | 41.0 [1], 260.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_1df4ee68c91fd740bc4f1330f65b9fe7.svg) | N-Benzyl-2-[2-(4-methyl-piperazin-1-yl)-3-phenyl-3,4-dihydro-quinazolin-4-yl]-acetamide | IC50 | 35800.0 [1], 35809.64 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_a87e10faafd7a09aac192be612517270.svg) | 2-(3-Ethyl-2-piperidin-1-yl-4H-quinazolin-4-yl)-N-[[4-[(4-methylphenyl)sulfonylamino]phenyl]methyl]acetamide | IC50 | 959.4 [1], 960.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_77a621d46f70126639b55033f633b6aa.svg) | CID 24765479 | IC50 | 1.2 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_01198966efdcf6510510e24816f814f3.svg) | N-[(4-Aminophenyl)methyl]-2-(3-phenyl-2-piperidin-1-yl-4H-quinazolin-4-yl)acetamide | IC50 | 13031.67 [1], 14400.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_3e12d3576b8e0f069fcce2c8ad8ce1ac.svg) | N-Benzyl-2-[3-(4-nitro-phenyl)-2-piperidin-1-yl-3,4-dihydro-quinazolin-4-yl]-acetamide | IC50 | 2338.84 [1], 2500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_bf1b35e9ab59d885b7c2ff9aa4fce35d.svg) | 2,3-Diphenyl-3,4-dihydroquinazoline-4-acetic acid methyl ester | IC50 | 10690.55 [1], 10700.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_0c21bf9a1b187e73ff99c4f74a26096b.svg) | N-Benzyl-2-(2-morpholin-4-yl-3-phenyl-3,4-dihydro-quinazolin-4-yl)-acetamide | IC50 | 21577.44 [1], 21600.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_9d390a3a241a4b061527090981df05f8.svg) | Tert-butyl N-[5-[[4-[2-(benzylamino)-2-oxoethyl]-3-phenyl-1,4-dihydroquinazolin-2-ylidene]amino]pentyl]carbamate | IC50 | 570.0 [1], 570.16 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_a479cef9b53fdfe6887b23ea1c39519f.svg) | 2-Piperidino-3-phenyl-3,4-dihydroquinazoline-4-acetic acid methyl ester | IC50 | 27669.42 [1], 27700.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_914af8aaa05a4ff57508832fc9cbb7d8.svg) | 3-[(4-Chlorophenyl)methyl]-N-[3-(2-ethylpiperidin-1-yl)propyl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide | IC50 | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_6d864651dca60be3428a67b9ebab31a6.svg) | Methyl 2-[3-[5-[(2-methylpropan-2-yl)oxycarbonylamino]pentyl]-2-(4-phenylanilino)-4H-quinazolin-4-yl]acetate | IC50 | 369.83 [1], 370.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_07eb266d5d18da3909e507105b330ce6.svg) | Methyl 2-[2-[methyl(5-pyrrolidin-1-ylpentyl)amino]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]acetate | IC50 | 339.63 [1], 340.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_568e93061809483c852d88c9a0c933ad.svg) | 2-[3-(5-Amino-pentyl)-2-(biphenyl-4-ylamino)-3,4-dihydro-quinazolin-4-yl]-N-benzyl-acetamide | IC50 | 139.96 [1], 140.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_89b7832a3c34a32a810c469abff8ee64.svg) | Methyl 2-[2-[methyl(5-pyrrolidin-1-ylpentyl)amino]-3-phenyl-4H-quinazolin-4-yl]acetate | IC50 | 5834.45 [1], 5840.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_1a5b1358f69f5a00083c2c9a80a377d5.svg) | N-Benzyl-2-[2-[methyl(5-pyrrolidin-1-ylpentyl)amino]-3-phenyl-4H-quinazolin-4-yl]acetamide | IC50 | 4197.59 [1], 4200.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_b71d45d9d9a4c68d53b73fc66df739c5.svg) | 3-[(3-Fluorophenyl)methyl]-2,4-dioxo-N-(2-piperidin-1-ylethyl)-1H-quinazoline-7-carboxamide | IC50 | 16870.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_911b4f606d3876bd51ef10477e066c62.svg) | 3-[(4-Fluorophenyl)methyl]-2,4-dioxo-N-(2-piperidin-1-ylethyl)-1H-quinazoline-7-carboxamide | IC50 | 9230.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_db141d8190ff7c0ae98414a9584c7cce.svg) | 3-[(4-Chlorophenyl)methyl]-2,4-dioxo-N-(2-piperidin-1-ylethyl)-1H-quinazoline-7-carboxamide | IC50 | 2080.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_5593a129039a59c81c8c4cf26bc51b9c.svg) | 3-[(4-Chlorophenyl)methyl]-2,4-dioxo-N-(3-piperidin-1-ylpropyl)-1H-quinazoline-7-carboxamide | IC50 | 1950.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_c55e79dfbc4bd56dbf55a84ed0a9a501.svg) | 3-[(4-Chlorophenyl)methyl]-N-[2-(2-ethylpiperidin-1-yl)ethyl]-2,4-dioxo-1H-quinazoline-7-carboxamide | IC50 | 3380.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_f169863be82804b8c543ef83162a64fc.svg) | 3-[(4-Chlorophenyl)methyl]-2,4-dioxo-N-(2-pyrrolidin-1-ylethyl)-1H-quinazoline-7-carboxamide | IC50 | 2460.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_554be7e56f0bc44b28df96b42ac64d08.svg) | 2-[2-(Dimethylamino)-3-phenyl-4H-quinazolin-4-yl]-N-[(4-nitrophenyl)methyl]acetamide | IC50 | 349.95 [1], 350.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_0207ddca66f09c1a43c903c303f0c3ee.svg) | 2-(3-Ethyl-2-piperidin-1-yl-4H-quinazolin-4-yl)-N-[[4-[(4-fluorophenyl)sulfonylamino]phenyl]methyl]acetamide | IC50 | 1039.92 [1], 1040.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_75dbfa63ee8df00194e8dabc637dcdda.svg) | 2-[2-(Dimethylamino)-3-phenyl-4H-quinazolin-4-yl]-N-[[4-[(4-methylphenyl)sulfonylamino]phenyl]methyl]acetamide | IC50 | 629.51 [1], 630.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_49674384ac0c1fd333d9c3bb492c7b86.svg) | Methyl 2-(4-bromophenyl)-2-isopropyl-5-(4-(2-methoxyphenyl)piperazin-1-yl)pentanoate | IC50 | 95.0 [1], 95040.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_deea40505005edbf988353f9688dd344.svg) | 1-[4-[(2,4-Dichlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one | IC50 | 4.0 [1], 33.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_011692593cb9bed117be0130bcb96326.svg) | 3-Chloro-2,5,5-trimethyl-N-[[2-(propan-2-yloxymethyl)phenyl]methyl]-6,7-dihydro-4H-isoindole-1-carboxamide | IC50 | 200.0 [1], 810.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_a3e1833ad3a101d8b2731163c455dae4.svg) | 3,5-Dichloro-N-{[(3S,4R)-1-(3,3-dimethylbutyl)-3-fluoropiperidin-4-yl]methyl}benzamide | IC50 | 25.0 [1], 43.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_2f396015dd3e84f1397988e4b6cdaffb.svg) | 8-Prenylnaringenin | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_51491790f6dc0e1f82f40025f5821d46.svg) | Sophoraflavanone G | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_0059e281ee1c8332255ffd38925c22eb.svg) | (R)-2-(4-Cyclopropylphenyl)-N-(1-(5-(2,2,2-trifluoroethoxy)pyridin-2-yl)ethyl)acetamide | IC50 | 89.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_9b45fa7c41d4f6e3e6fa07d5e0489a47.svg) | (S)-4',5,7-Trihydroxy-6-prenylflavanone | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_e63ec13a2e7ac4885f405bfd8d962714.svg) | 3-(4-Methoxybenzyl)-2,4-dioxo-N-(3-piperidin-1-ylpropyl)-1,2,3,4-tetrahydroquinazoline-7-carboxamide | IC50 | 3110.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_0dc43da0ca767bdb6ade04bfbdc36b25.svg) | 3-(4-Chlorobenzyl)-7-(1-methylpiperazine-4-carbonyl)-2-thioxo-2,3-dihydroquinazolin-4(1H)-one | IC50 | 11390.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_1169e852f4da804d40ba196bb6f0c94a.svg) | 3-[(4-Chlorophenyl)methyl]-N-[2-(dimethylamino)ethyl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide | IC50 | 53500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_cdf2ee2047e2a4cf980c5a72a6a2515c.svg) | 3-[(4-Chlorophenyl)methyl]-N-[3-(4-methylpiperidin-1-yl)propyl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide | IC50 | 1100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_32593ab9e8f26835ff9e5fa89ce98aed.svg) | N-(1-Benzyl-1H-pyrazol-3-yl)benzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_4f5a1ee200fbb94ced49cd871f25ebcc.svg) | N-(1-Benzylpyrazol-3-yl)-2-phenylacetamide | IC50 | 1140.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_e49fd68b8d0e620242090f7ae222ad7b.svg) | N-[[5-(2-Methylpropyl)-1-phenylpyrazol-3-yl]methyl]benzenesulfonamide | IC50 | 5650.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_25a671d01c5314045b84690115b71784.svg) | 3-Fluoro-N-[[5-(2-methylpropyl)-1-phenylpyrazol-3-yl]methyl]benzenesulfonamide | IC50 | 3200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_bdaebf3e2c11faf34d57af15dea12c0b.svg) | N-[1-[(5-Cyanopyridin-2-yl)methyl]pyrazol-3-yl]-2-[4-[1-(trifluoromethyl)cyclopropyl]phenyl]acetamide | IC50 | 6.4 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_97cd6f15ed8767cc8fa04dec34fcbc3f.svg) | 3-[(4-Chlorophenyl)methyl]-N-[3-(2-ethylpiperidin-1-yl)propyl]-2,4-dioxo-1H-quinazoline-7-carboxamide | IC50 | 1520.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_75a06adc70a77179482377ed4356d9ad.svg) | 3-[(4-Chlorophenyl)methyl]-N-[3-(2-methylpiperidin-1-yl)propyl]-2,4-dioxo-1H-quinazoline-7-carboxamide | IC50 | 3720.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_abef69811c7bfb7ca930de50936f8a0c.svg) | 4-Amino-1-(4-((4-chlorophenyl)(phenyl)methyl)piperazin-1-yl)butan-1-one | IC50 | 3710.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_22fc3673f35c6008a88f7d4fdcb2de8a.svg) | 2-[2-(Dimethylamino)-3-ethyl-4H-quinazolin-4-yl]-N-[[4-[(4-fluorophenyl)sulfonylamino]phenyl]methyl]acetamide | IC50 | 4102.04 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_dcf74d2e23a94fb40ab8c0bf2ea99680.svg) | 2-[2-(Dimethylamino)-3-ethyl-4H-quinazolin-4-yl]-N-[[4-[(4-methylphenyl)sulfonylamino]phenyl]methyl]acetamide | IC50 | 1119.44 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_4466bc117cbe65bb64383b7df95e7106.svg) | N-Benzyl-2-[2-(dimethylamino)-3-ethyl-4H-quinazolin-4-yl]acetamide | IC50 | 24154.61 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_50e2ba887ab921136464b81b7dbaa218.svg) | N-Benzyl-2-(3-ethyl-2-piperidin-1-yl-4H-quinazolin-4-yl)acetamide | IC50 | 4581.42 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_954cc018239254fd1d83f19716936292.svg) | N-[2-Ethyl-2-(4-fluorophenyl)butyl]-1-(2-phenylethyl)piperidine-4-carboxamide | IC50 | 89.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_2e95e342f1400958817b83882919c314.svg) | 2-[2-[4-[2-(Dimethylamino)ethyl]piperazin-1-yl]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]-N-[(4-fluorophenyl)methyl]acetamide | IC50 | 320.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_23ab1a1a82f787548231911346c8bb6d.svg) | 2-[2-[4-[2-(Dimethylamino)ethyl]piperazin-1-yl]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]-N-[(4-methoxyphenyl)methyl]acetamide | IC50 | 310.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_1e99513e6232b3d6f30775ffe9dfb8a2.svg) | 1-[4-[(2-Chlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one | IC50 | 141.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_846bd99a8b65614c0b717974a0a5a115.svg) | 1-[4-[(2,6-Dichlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_d75c0b21e3a48609f223f257be31b576.svg) | 1-[4-[(2,4-Dimethylphenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one | IC50 | 35.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_783b60eaacaa2c56dcbbb572ef0460f2.svg) | 1-[4-[(3-Chlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one | IC50 | 55.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_0e807f9c38942328015e719811ed5cc7.svg) | 1-[4-[(3,4-Dichlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_ba1c5cef925381578fb6a173179adce1.svg) | N-[[3-[2-(Trifluoromethyl)phenyl]-1,2-oxazol-5-yl]methyl]-2-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]ethanamine | IC50 | 1020.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_c6223b173e37f7a96727d559f4d10ba0.svg) | (2S)-1-[4-[(4-Chlorophenyl)methyl]piperazin-1-yl]-3-(4-fluorophenoxy)propan-2-ol | IC50 | 1560.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_f665a7659706e671e61179114de272e8.svg) | 1-{4-[(4-Chloro-phenyl)-phenyl-methyl]-piperazin-1-yl}-3,3-diphenyl-propan-1-one | IC50 | 81.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_f6ec092ecb742bb8d12cb93fa4ee53fc.svg) | 1-[4-[Bis(4-methoxyphenyl)methyl]piperazin-1-yl]-3,3-diphenylpropan-1-one | IC50 | 745.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_81dedf1de803be5e281ae0e797c51579.svg) | 1-[4-[(2,3-Dichlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one | IC50 | 63.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_c2f40ebe0ab0fddae46cf299782a0447.svg) | 2-[4-(2,4-Dimethylphenyl)piperazin-1-yl]-N-[[3-[2-(trifluoromethyl)phenyl]-1,2-oxazol-5-yl]methyl]ethanamine | IC50 | 1530.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_ea78e858a68f7212121417db368c14fe.svg) | 1-[4-[(3,5-Dichlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_bbfe737f7f05f9ba2dc25624a5b1d2ee.svg) | 2-[4-(Dimethylamino)phenyl]-N-[1-[(4-fluorophenyl)methyl]pyrazol-3-yl]acetamide | IC50 | 4.2 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_7d8330e63a7ab090476c65c01cec8d56.svg) | N-[1-[(4-Cyano-3-fluorophenyl)methyl]pyrazol-3-yl]-2-[4-(dimethylamino)phenyl]acetamide | IC50 | 3.1 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_27acca67234a8b83659df2d2b234c2a8.svg) | N-[1-[(3,5-Difluoro-4-methoxyphenyl)methyl]pyrazol-3-yl]-2-[4-(dimethylamino)phenyl]acetamide | IC50 | 3.2 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_ccbf5bd8f6256a79dafc8d74e74610a3.svg) | 2-[4-(Dimethylamino)phenyl]-N-[1-[(4-methylphenyl)methyl]pyrazol-3-yl]acetamide | IC50 | 7.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_b368a548d0447e71dc730586577ff478.svg) | N-[1-[(4-Cyanophenyl)methyl]pyrazol-3-yl]-2-[4-(dimethylamino)phenyl]acetamide | IC50 | 11.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_8d85cac1a61bcd1ae3a984e7201f4e65.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-[6-(dimethylamino)pyridin-3-yl]acetamide | IC50 | 12.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_6e31401d1fc2a51ccaa21a9a9fa5ffb4.svg) | N-[1-[[4-(Difluoromethoxy)phenyl]methyl]pyrazol-3-yl]-2-[4-(dimethylamino)phenyl]acetamide | IC50 | 6.8 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_ba9759f81982117d7269eed1947d3be9.svg) | 2-[4-(Dimethylamino)phenyl]-N-[1-[[4-(trifluoromethoxy)phenyl]methyl]pyrazol-3-yl]acetamide | IC50 | 2.2 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_c600fb4f3d11e81691ac5814f19a6b7f.svg) | N-[1-[(4-Chlorophenyl)methyl]pyrazol-3-yl]-2-[4-(dimethylamino)phenyl]acetamide | IC50 | 1.1 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_05f0450c8870f0c328609839e9d94a56.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-[4-(dimethylamino)phenyl]acetamide | IC50 | 1.5 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_8b0666fec5cce5cc5c0888655f5ec24e.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-[6-[(3S)-3-fluoropyrrolidin-1-yl]pyridin-3-yl]acetamide | IC50 | 2.5 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_afc965692104603b543742c94c22d8d5.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-[4-(3-fluorooxetan-3-yl)phenyl]acetamide | IC50 | 4.3 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_ed2fbafcc2ccf561c9a32410c450c7a2.svg) | 2-(6-Cyclopropylpyridin-3-yl)-N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]acetamide | IC50 | 15.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_ca06acabaad5b5426140dc1285e4e5b3.svg) | 2-[4-(Dimethylamino)phenyl]-N-[1-[(4-methoxyphenyl)methyl]pyrazol-3-yl]acetamide | IC50 | 23.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_a58c89dec3276d6f7aadb447315bcafe.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-(1H-indol-6-yl)acetamide | IC50 | 1.9 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_e830fd54289b9eea3d710bd4fed353bf.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-[4-(oxetan-3-yloxy)phenyl]acetamide | IC50 | 4.6 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_227d26b76f0172b6428458f06bf13609.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-(1-methylpyrrolo[2,3-b]pyridin-5-yl)acetamide | IC50 | 7.1 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_5330ce2e4570c55020a74555943931fb.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-(1H-indol-5-yl)acetamide | IC50 | 2.3 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_8ca26ef53f30d42d441fce7179208d29.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-(4-propan-2-ylphenyl)acetamide | IC50 | 1.4 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-t-type-calcium-channel-alpha-1g-subunit_2038c48d438d42c36bc596518a7cc97b.svg) | 2-[4-(3,3-Difluorocyclobutyl)oxyphenyl]-N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]acetamide | IC50 | 1.4 [1] |