Voltage-gated potassium channel subunit Kv4.3 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Sildenafil	IC50	501187.23 [1]
	Everolimus	IC50	10000000.0 [1]
	Sunitinib	IC50	50118.72 [1]
	Dasatinib	IC50	316227.77 [1]
	Duloxetine	IC50	100000.0 [1]
	Nelfinavir	IC50	5011872.34 [1]
	Sitagliptin	IC50	100000000.0 [1]
	Nilotinib	IC50	3162277.66 [1]
	Raltegravir	IC50	5011872.34 [1]
	Darunavir	IC50	100000.0 [1]
	Vardenafil	IC50	79432.82 [1]
	Tolterodine	IC50	12589.25 [1]
	Nebivolol	IC50	50118.72 [1]
	Deferasirox	IC50	50118.72 [1]
	Paliperidone	IC50	63095.73 [1]
	Etravirine	IC50	3162277.66 [1]
	Alfuzosin	IC50	1000000.0 [1]
	Solifenacin	IC50	50118.72 [1]
	Eltrombopag	IC50	1584893.19 [1]
	Ambrisentan	IC50	251188.64 [1]
	Darifenacin	IC50	12589.25 [1]
	Silodosin	IC50	316227.77 [1]
	Acacetin	IC50	9300.0 [1]
	Desvenlafaxine	IC50	5011872.34 [1]
	N-[(3S,4R)-6-Cyano-3-hydroxy-2,2-dimethyl-3,4-dihydrochromen-4-yl]-N-methylethanesulfonamide	IC50	1400.0 [1]
	6-[[[1-[2-(7-Methoxy-2-oxoquinoxalin-1-yl)ethyl]piperidin-4-yl]amino]methyl]-4H-pyrido[3,2-b][1,4]oxazin-3-one	IC50	100000.0 [1]
	N-[(4R)-4-(4-Methoxyphenyl)-3-[2-(4-methoxyphenyl)ethyl]-2-oxoimidazolidin-1-yl]methanesulfonamide	IC50	3870.0 [1]
	N-[6-[(1S)-1-(4-Fluorophenyl)-2,2-dipyridin-3-ylethyl]pyridin-2-yl]methanesulfonamide	IC50	2300.0 [1]
	N-(4-Morpholin-4-ylcyclohexyl)-5-(oxan-4-yl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine	IC50	30000.0 [1]
	[(7S)-5-(Methoxymethyl)-7-(1-methylindol-2-yl)-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl]-[(2S)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methanone	IC50	5800.0 [1]
	3-[6-[2-Carbamoyl-6-(trifluoromethoxy)indol-1-yl]pyridin-2-yl]butanoic acid	IC50	33000.0 [1]
	(1R)-1-[2-(3,5-Dichlorophenyl)pyridin-3-yl]-2,2-dipyridin-3-ylethanol	IC50	8300.0 [1]
	2-[[[4-[(1R)-1-Amino-2-(7-fluoro-2-oxoquinoxalin-1-yl)ethyl]cyclohexyl]amino]methyl]-8H-pyrimido[5,4-b][1,4]oxazin-7-one	IC50	100000.0 [1]
	N-[[1-[2-(Tert-butylcarbamoylamino)ethyl]-4-(hydroxymethyl)piperidin-4-yl]methyl]-3,5-dichlorobenzamide	IC50	33000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 34 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Voltage-gated potassium channel subunit Kv4.3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/voltage-gated-potassium-channel-subunit-kv4-3-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, December 21). Quest Database™ Voltage-gated potassium channel subunit Kv4.3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/voltage-gated-potassium-channel-subunit-kv4-3-inhibitors-ic50-ki.
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