![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_01814a6086009d7440d5f435a324c600.svg) | Verapamil | IC50 | 150.0 [1], 23500.0 [2], 24000.0 [3], 47000.0 [4], 50000.0 [5] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_1232c84d43d4865ebdc5de8d7663a19f.svg) | Nifedipine | IC50 | 22.0 [1], 50.0 [2], 55.0 [3] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_1232c84d43d4865ebdc5de8d7663a19f.svg) | Nifedipine | Ki | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_f0193f5276395ac51bc314c2ce4fc0c3.svg) | Mibefradil | IC50 | 202.0 [1], 250.0 [2], 108000.0 [3], 288000.0 [4] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_f2beac4f632265172541ae8f16f89706.svg) | Nicardipine | IC50 | 250.0 [1], 9600.0 [2], 24100.0 [3] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_5c516e5fa259eb4dabbdf74f9982ff4f.svg) | Testosterone | IC50 | 34.0 [1], 38.4 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_d7f779d5cfb5b4dbb918458849a386b9.svg) | Halothane | IC50 | 1800000.0 [1], 14500000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_d807cd36eea3bdcc2c2c3e9b5d13b932.svg) | Lamotrigine | IC50 | 1258925.41 [1], 1584893.19 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_95b92c7a51ad4bb33df4aec269cfa5fa.svg) | Moxifloxacin | IC50 | 168900.0 [1], 398107.17 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_9677690a14053e2d953ed858e7325389.svg) | Amlodipine | IC50 | 1200.0 [1], 4200.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_7de5848be93196a6906eba944a298431.svg) | Sunitinib | IC50 | 79432.82 [1], 199526.23 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_986db0437f20070dfb14143a9f1b018d.svg) | Dasatinib | IC50 | 251188.64 [1], 398107.17 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_b429be022623e6dba89dbd55075672bf.svg) | Duloxetine | IC50 | 25118.86 [1], 100000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_755000a88f2651809d912de0f446bcfe.svg) | Lapatinib | IC50 | 1995262.31 [1], 15848931.92 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_f59214b920b0faf58103b7de887f46c7.svg) | Nilotinib | IC50 | 199526.23 [1], 3162277.66 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_611aee8360ba5f29cd9711190dfe1482.svg) | Vardenafil | IC50 | 15848.93 [1], 251188.64 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_01451c73b9c1f68aac3778db2f20814c.svg) | Dofetilide | IC50 | 158489.32 [1], 1023000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_e8bd31cd17a67cd8d7da95b1194a4650.svg) | Paliperidone | IC50 | 398107.17 [1], 1000000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_1c1cf29c7c7877942e85aa24d7e4f4fa.svg) | Cilnidipine | IC50 | 5300.0 [1], 12700.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_0c688849f6944f0c7d94d2ee0e5b5379.svg) | Barnidipine | IC50 | 1200.0 [1], 3100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_7a64ef32c888ae868ad08218ba91330e.svg) | Omarigliptin | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_99f04051f3a3c2e2d86079a90b1965c9.svg) | 2-(2-Amino-1,3-thiazol-4-yl)-N-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]acetamide | IC50 | 8200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_1db85a3a54706807cc7926de1f7164a1.svg) | 5-O-[(3R)-1-Benzylpiperidin-3-yl] 3-O-methyl 2,6-dimethyl-4-(3-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxylate | IC50 | 4900.0 [1], 13800.0 [2] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_5d76064ddc2dff8b46597ab1ba156fa1.svg) | (6S)-N-[4-[[(2S,5R)-5-[(R)-Hydroxy(pyridin-3-yl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole-6-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_722c621ffb02e379ed12b3dedfac01e8.svg) | (4R)-N-[4-[[(2S,5R)-5-[(R)-Hydroxy(pyridin-3-yl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5,6-dihydro-4H-cyclopenta[d][1,3]thiazole-4-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_28dba8f145b0b6293925c8c01ab57119.svg) | Estradiol | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_c70f5b79af37726016ec15cea0b55e94.svg) | Propranolol | IC50 | 21000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_444fa0db37706d6efa6c25fb3dd7c1de.svg) | Phenytoin | IC50 | 125000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_693b10fcf0f1bf3ce26f73cb27aee812.svg) | Fluoxetine | IC50 | 5400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_a047ba0a887d642df2938965c5266c0d.svg) | Ketamine | IC50 | 1800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_be4565ca8c20c1d9804fa640fd1584d5.svg) | Risperidone | IC50 | 125000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_ce2451a6dd9c86e3ec85025ead605266.svg) | Sildenafil | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_1651d7921a8facf41c6a5623ae7707ce.svg) | Diltiazem | IC50 | 44000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_d9d88c2a7bdabc45b702c06047b28bae.svg) | Quinidine | IC50 | 19820.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_fac222a9fee62d9cda063e5aabf1d4d4.svg) | 3-Isobutyl-1-methylxanthine | IC50 | 466000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_cfe3816ade941c998d8ece3061f8eb29.svg) | Remifentanil | IC50 | 38900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_9c9b6aadd4f8caa0bf86f9d7bbd70a7c.svg) | Sotalol | IC50 | 1023000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_6c5a78e8ca55529a3f6c3b506ecb26d6.svg) | Clotrimazole | IC50 | 590.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_8276105e0fe6a29070aaaab8ba4ded14.svg) | Nimodipine | IC50 | 110.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_6833af5a00e4820a7dec88d7ed0f4ead.svg) | Thioridazine | IC50 | 1320.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_4a2f7aa95b8e5fa8d1122874409c701a.svg) | Tadalafil | IC50 | 398107.17 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_79b99809a4327da541aa2304e553f873.svg) | Terfenadine | IC50 | 1320.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_b22ee7becceb5ad9c31ec4529677de35.svg) | Sitagliptin | IC50 | 100000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_a51b30f2494a45cccba6c8c3f14d39bb.svg) | Nitrendipine | Ki | 0.25 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_47f0bc6989009707a0e42006229bb2b9.svg) | Darunavir | IC50 | 1584893.19 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_ed79e2ddfcc7ee74d79415fe78de029e.svg) | Isradipine | IC50 | 2.2 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_e062b395a3ae7be9147860ab78c92beb.svg) | Tolterodine | IC50 | 25118.86 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_8ae9092a1acc8d5031d0a55ff520619e.svg) | Nebivolol | IC50 | 15848.93 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_0e03e9bd3ca5182dc5be5efc63b439c2.svg) | Deferasirox | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_e4d51706ccafae108b5baa824e5faa47.svg) | Gallopamil | IC50 | 17.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_4e787c15d05c81e9c577c24aa928fd0f.svg) | Bepridil | IC50 | 1400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_85bfeb5c1c0028708a30ec66fc1bbd21.svg) | Seliciclib | IC50 | 23400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_89204000491e48a54045d07bf3547c1f.svg) | Nisoldipine | IC50 | 3.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_be653f89bf9757f77ea6b06dba105b92.svg) | Alfuzosin | IC50 | 199526.23 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_5f96c8f50bc42c594915fbb1bfe0241d.svg) | Solifenacin | IC50 | 6309.57 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_ae4efaf952050c7b6a68b7e059211d8a.svg) | Doripenem | IC50 | 1995.26 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_6abe2f67827e0a50fdfd56dd09f893a8.svg) | Ambrisentan | IC50 | 2511886.43 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_d59e5533784cda90bc61ea3a0051826f.svg) | Palonosetron | IC50 | 398107.17 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_2caadd3ec7b2c08ae34435ae889a6a0b.svg) | Darifenacin | IC50 | 1584893.19 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_2f8b1a65fcaa2c2002b0eddc770532aa.svg) | Silodosin | IC50 | 794328.23 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_03f8951aef77ea138df5d258fb4ba4fa.svg) | Alvimopan | IC50 | 5011.87 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_0bf6f40a4e7b3a84ba22250897caab6e.svg) | Lacosamide | IC50 | 50118.72 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_8aac1ffdcc9b7b03b14d7a1abbfd2880.svg) | Norfluoxetine | IC50 | 1130.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_71388e561bf42bba3f364eabe9f69aa4.svg) | Propiverine | IC50 | 41700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_8bc21e734d2a7dc7d08f16b4864d59fd.svg) | Carbamimidothioic acid 2-[4-[(4-nitrophenyl)methoxy]phenyl]ethyl ester | IC50 | 3200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_5a8a609f90bde5e664777901c493d6de.svg) | 2-(4-((2,5-Difluorobenzyl)oxy)phenoxy)-5-ethoxyaniline | IC50 | 3600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_85d9e705a4afe045c96132caae2d94be.svg) | Pinaverium | IC50 | 1750.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_a7a3e6c074f97d267148d315bdd54aa0.svg) | Oliceridine | IC50 | 36000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_0059e281ee1c8332255ffd38925c22eb.svg) | (R)-2-(4-Cyclopropylphenyl)-N-(1-(5-(2,2,2-trifluoroethoxy)pyridin-2-yl)ethyl)acetamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_e58637f0d4a87ff8f46c8ad80ca08fcf.svg) | Vibegron | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_9182e75261c4c9a90083bb44381e7fec.svg) | L-796568 Free base | IC50 | 1700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_24597878df01113a50b5f94b00373ccd.svg) | 2-[(8R)-8-(3,5-Difluorophenyl)-8-methyl-10-oxo-6,9-diazaspiro[4.5]decan-9-yl]-N-[(3S)-2-oxospiro[1H-pyrrolo[2,3-b]pyridine-3,6'-5,7-dihydrocyclopenta[b]pyridine]-3'-yl]acetamide | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_961fef6d9b37084f97f3b08338435ffd.svg) | Tert-butyl N-[(2R)-1-oxo-1-[[(3R)-2-oxo-1-propan-2-yl-4,5-dihydro-3H-1-benzazepin-3-yl]amino]-3-[2-(trifluoromethoxy)phenyl]propan-2-yl]carbamate | IC50 | 3500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_d9df6cb5b3ce07978c9872c6cce8fd49.svg) | 5-[2-[4-[2-[4-(Tetrazol-1-yl)phenyl]acetyl]piperazin-1-yl]ethyl]-3H-2-benzofuran-1-one | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_9e0411d99b7e1fca741170518542c99e.svg) | 4-Methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide | IC50 | 15848.93 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_b920ffcf05fc069fcbaacc5435cdfce4.svg) | Zuranolone | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_298a6e14548d62f654e1b7817f68cb6e.svg) | Diethyl 2,6-dimethyl-4-[3-methyl-5-(2-naphthalen-1-ylethyl)-1,2-oxazol-4-yl]-1,4-dihydropyridine-3,5-dicarboxylate | Ki | 4.11 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_a894f01cd57434cd61158e9f7cb543a7.svg) | 3-Methyl-4-[4-[8-[(3-methylpyridin-2-yl)methyl]-2,4-dioxo-1-pyrimidin-4-yl-1,3,8-triazaspiro[4.5]decan-3-yl]phenyl]benzoic acid | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_31f5cdd5538ed447671f883fd2327e26.svg) | [2-(4-Chloro-2-fluoroanilino)-5-methyl-1,3-thiazol-4-yl]-[(2S,3S)-2,3-dimethylpiperidin-1-yl]methanone | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_8a2f8f3e300806cab9b0c0dd34da2841.svg) | Diethyl 2,6-dimethyl-4-[3-methyl-5-(2-phenylethyl)-1,2-oxazol-4-yl]-1,4-dihydropyridine-3,5-dicarboxylate | Ki | 22.9 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_89ef53acc5f4febd13075c144db1d790.svg) | Diethyl 2,6-dimethyl-4-[3-methyl-5-(2-naphthalen-2-ylethyl)-1,2-oxazol-4-yl]-1,4-dihydropyridine-3,5-dicarboxylate | Ki | 20.2 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_199aeeda3e6afca13020526be33230a1.svg) | Diethyl 2,6-dimethyl-4-[3-phenyl-5-(2-phenylethyl)-1,2-oxazol-4-yl]-1,4-dihydropyridine-3,5-dicarboxylate | Ki | 72.9 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_eab1794bdd96b417c47c9e4c8a44e5b6.svg) | Diethyl 2,6-dimethyl-4-[3-methyl-5-[2-(4-phenylphenyl)ethyl]-1,2-oxazol-4-yl]-1,4-dihydropyridine-3,5-dicarboxylate | Ki | 18.2 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_bdaebf3e2c11faf34d57af15dea12c0b.svg) | N-[1-[(5-Cyanopyridin-2-yl)methyl]pyrazol-3-yl]-2-[4-[1-(trifluoromethyl)cyclopropyl]phenyl]acetamide | IC50 | 2410.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_9f7a7b5c3accd993ffeca78fdc7e9d2f.svg) | 4-[4-[2-Chloro-5-(trifluoromethoxy)phenyl]-2,6-dimethylphenoxy]butanoic acid | IC50 | 12840.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_41c16009b349922ed73ddcbe1ad421d1.svg) | 3-[5-[2-Fluoro-5-(trifluoromethoxy)phenyl]-1-benzofuran-2-yl]propanoic acid | IC50 | 15090.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_ed48d688ada8524574dfb20d32cdde9c.svg) | Diethyl 2,6-dimethyl-4-(3-phenyl-5-propan-2-yl-1,2-oxazol-4-yl)-1,4-dihydropyridine-3,5-dicarboxylate | Ki | 417.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_878a482729b833a0834e68c7bbb1d6cd.svg) | 6-[[[1-[2-(7-Methoxy-2-oxoquinoxalin-1-yl)ethyl]piperidin-4-yl]amino]methyl]-4H-pyrido[3,2-b][1,4]oxazin-3-one | IC50 | 92000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_8cc56188b1d303404e0f06888f78ea89.svg) | (2R,3S,5R)-2-(2,5-Difluorophenyl)-5-(4,6-dihydro-1H-pyrrolo[3,4-c]pyrazol-5-yl)oxan-3-amine | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_5994d6c14cea7177c91a90f6234f9f76.svg) | N-[(4R)-4-(4-Methoxyphenyl)-3-[2-(4-methoxyphenyl)ethyl]-2-oxoimidazolidin-1-yl]methanesulfonamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_b0d9ac4fe33242893feb005ff0ba84de.svg) | Diethyl 4-(3,5-dimethyl-1,2-oxazol-4-yl)-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylate | Ki | 27.1 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_bc356f7fffd5550a7ff966da033391cd.svg) | Diethyl 2,6-dimethyl-4-(5-methyl-3-phenyl-1,2-oxazol-4-yl)-1,4-dihydropyridine-3,5-dicarboxylate | Ki | 13.9 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_d689892c42c70ddff66c315b09e72743.svg) | [(1S,2S)-2-[2-[3-(1H-Benzimidazol-2-yl)propyl-methylamino]ethyl]-6-fluoro-1-propan-2-yl-3,4-dihydro-1H-naphthalen-2-yl] 2-methylpropanoate | IC50 | 347.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_bcc6ec9c025fb81db6d6c70d187bc904.svg) | 2-(3,4-Dimethoxyphenyl)-2-[3-(N-methyl-3,4-dimethoxyphenethylamino)cyclohexyl]-3-methylbutyronitrile | IC50 | 270.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_f23f9c20d2eaafea7d76e059ab52ac5f.svg) | Diethyl 2,6-dimethyl-4-[3-methyl-5-[2-(2-phenylphenyl)ethyl]-1,2-oxazol-4-yl]-1,4-dihydropyridine-3,5-dicarboxylate | Ki | 91.1 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_05f0450c8870f0c328609839e9d94a56.svg) | N-[1-[(3,4-Difluorophenyl)methyl]pyrazol-3-yl]-2-[4-(dimethylamino)phenyl]acetamide | IC50 | 7100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_da0091434e3739261e361b345822eeb0.svg) | 2-(4-Tert-butylphenyl)-N-[1-[(5-cyanopyridin-2-yl)methyl]pyrazol-3-yl]acetamide | IC50 | 2420.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_fd2ac0800fae4f219e9d1ae243ad27e1.svg) | 10-[4-(2,1,3-Benzoxadiazol-4-yl)-2,6-dimethyl-5-propan-2-yloxycarbonyl-1,4-dihydropyridine-3-carbonyl]oxydecyl-trimethylazanium | IC50 | 70.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_1d939e2239673e5db0f300e9057d3c35.svg) | 8-[(2R)-2-Hydroxy-2-(4-methyl-1-oxo-3H-2-benzofuran-5-yl)ethyl]-2-(1-methyl-6-oxopyridazin-3-yl)-2,8-diazaspiro[4.5]decan-1-one | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/voltage-gated-l-type-calcium-channel-alpha-1c-subunit_14a32e2186170085b8462d9da6902620.svg) | (1S,3R)-3-[8-Amino-1-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]imidazo[1,5-a]pyrazin-3-yl]cyclohexane-1-carboxylic acid | IC50 | 30000.0 [1] |