| 4-[(2S,5S,11S,14R)-14-Benzyl-11-(carboxymethyl)-5-[3-(diaminomethylideneamino)propyl]-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]butanoic acid | IC50 | 38800.0 [1] |
| 3-[1-Oxo-6-(1,2,3,4-tetrahydropyrimido[1,2-a]benzimidazol-9-yloxy)-3,4-dihydroisoquinolin-2-yl]-3-pyridin-3-ylpropanoic acid | IC50 | 5.0 [1] |
| 3-(1,3-Benzodioxol-5-yl)-3-[1-oxo-6-(1,2,3,4-tetrahydropyrimido[1,2-a]benzimidazol-9-yloxy)-3,4-dihydroisoquinolin-2-yl]propanoic acid | IC50 | 14.0 [1] |
| 3-[1-Oxo-6-(1,2,3,4-tetrahydropyrimido[1,2-a]benzimidazol-9-yloxy)-3,4-dihydroisoquinolin-2-yl]propanoic acid | IC50 | 310.0 [1] |
| 3-(4-(2-Amino-1-methyl-1H-benzo[d]imidazol-4-yloxy)benzamido)propanoic acid | IC50 | 2050.0 [1] |
| 3-(5-(2-Amino-1-methyl-1H-benzo[d]imidazol-4-yloxy)-1-oxoisoindolin-2-yl)propanoic acid | IC50 | 4800.0 [1] |
| 3-[6-(2-Amino-1-methylbenzimidazol-4-yl)oxy-1-oxo-3,4-dihydroisoquinolin-2-yl]propanoic acid | IC50 | 600.0 [1] |
| 3-[7-(2-Amino-1-methylbenzimidazol-4-yl)oxy-1-oxo-4,5-dihydro-3H-2-benzazepin-2-yl]propanoic acid | IC50 | 4300.0 [1] |
| (2R)-3-(Thiophene-3-carbonylamino)-2-[(2,4,6-trichlorophenyl)sulfonylamino]propanoic acid | IC50 | 24.0 [1] |
| (2R)-3-(Furan-3-carbonylamino)-2-[(3-methoxyphenyl)sulfonylamino]propanoic acid | IC50 | 208.0 [1] |
| (R)-3-(Furan-3-carboxamido)-2-(pyridine-3-sulfonamido)propanoic acid | IC50 | 793.0 [1] |
| (2R)-3-[[2-(Furan-3-yl)-2-oxoethyl]amino]-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 8000.0 [1] |
| (2R)-3-(Methanesulfonamido)-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 50000.0 [1] |
| (2R)-3-[(2-Phenylacetyl)amino]-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 50000.0 [1] |
| (2R)-3-(Thiophene-3-carbonylamino)-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 44.0 [1] |
| (2R)-3-(Furan-3-carbonylamino)-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 32.0 [1] |
| (2R)-3-Benzamido-2-[(2-chlorophenyl)sulfonylamino]propanoic acid | IC50 | 260.0 [1] |
| (2R)-3-Benzamido-2-[(2-methoxyphenyl)sulfonylamino]propanoic acid | IC50 | 729.0 [1] |
| (2R)-3-(3-Oxo-1H-isoindol-2-yl)-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 975.0 [1] |
| (2R)-3-[(2-Methoxybenzoyl)amino]-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 78.0 [1] |
| (2R)-3-(Furan-3-carbonylamino)-2-[(2-methylphenyl)sulfonylamino]propanoic acid | IC50 | 260.0 [1] |
| (2R)-3-Benzamido-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 120.0 [1] |
| (2R)-3-Acetamido-2-(benzenesulfonamido)propanoic acid | IC50 | 9100.0 [1] |
| (2R)-3-(Pyridine-3-carbonylamino)-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 81.0 [1] |
| (2R)-3-Benzamido-2-[(2-iodophenyl)sulfonylamino]propanoic acid | IC50 | 25.0 [1] |
| (2R)-3-Benzamido-2-[(2,6-dichlorophenyl)sulfonylamino]propanoic acid | IC50 | 118.0 [1] |
| (2R)-2-[(3-Cyanophenyl)sulfonylamino]-3-(furan-3-carbonylamino)propanoic acid | IC50 | 98.0 [1] |
| (2R)-3-(Methoxycarbonylamino)-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 50000.0 [1] |
| (2S)-3-Acetamido-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 8000.0 [1] |
| (2R)-3-Benzamido-2-[(2-methylsulfonylphenyl)sulfonylamino]propanoic acid | IC50 | 4600.0 [1] |
| (2R)-3-(Furan-3-carbonylamino)-2-[(2-methoxyphenyl)sulfonylamino]propanoic acid | IC50 | 700.0 [1] |
| (R)-3-Acetamido-2-(tert-butoxycarbonylamino)propanoic acid | IC50 | 50000.0 [1] |
| (2R)-3-Acetamido-2-[methyl-(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 50000.0 [1] |
| (2R)-2-[(2,4-Dichlorophenyl)sulfonylamino]-3-(thiophene-3-carbonylamino)propanoic acid | IC50 | 8.0 [1] |
| (2R)-3-Amino-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 50000.0 [1] |
| (2R)-3-(Butanoylamino)-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 30000.0 [1] |
| (2R)-3-[(2-Methylpropan-2-yl)oxycarbonylamino]-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 50000.0 [1] |
| (2R)-3-(Benzylamino)-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 50000.0 [1] |
| (2R)-3-Acetamido-2-(benzylsulfonylamino)propanoic acid | IC50 | 50000.0 [1] |
| (2R)-3-[(2-Methyl-1,3-oxazole-4-carbonyl)amino]-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 41.0 [1] |
| (2R)-3-Benzamido-2-[(2-methylphenyl)sulfonylamino]propanoic acid | IC50 | 320.0 [1] |
| (2R)-3-Benzamido-2-[(2,3-dichlorophenyl)sulfonylamino]propanoic acid | IC50 | 62.0 [1] |
| (2R)-3-Acetamido-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 800.0 [1] |
| (R)-3-Acetamido-2-(2,6-dichlorobenzamido)propanoic acid | IC50 | 50000.0 [1] |
| (R)-3-Acetamido-2-benzamidopropanoic acid | IC50 | 50000.0 [1] |
| (R)-3-Acetamido-2-(phenoxycarbonylamino)propanoic acid | IC50 | 50000.0 [1] |
| (2R)-3-[(2-Methylpyrazole-3-carbonyl)amino]-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 11.0 [1] |
| (2R)-3-(Pyrimidine-5-carbonylamino)-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 63.0 [1] |
| (2R)-3-(Pyridine-4-carbonylamino)-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 301.0 [1] |
| (2R)-2-[(2,3-Dichlorophenyl)sulfonylamino]-3-(thiophene-3-carbonylamino)propanoic acid | IC50 | 19.0 [1] |
| 2-[(2S,5R,8S,11S)-5-Benzyl-11-[3-(diaminomethylideneamino)propyl]-8-[[4-[[[2-[2-[2-[2-[(2E)-2-[3-[(19S)-19-ethyl-19-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4,6,8,10,15(20)-heptaen-10-yl]propylidene]hydrazinyl]-2-oxoethoxy]ethoxy]ethoxy]acetyl]amino]methyl]phenyl]methyl]-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]acetic acid | IC50 | 11000.0 [1] |
| 2-[(2S,5R,8S,11S)-5-Benzyl-11-[3-(diaminomethylideneamino)propyl]-8-[4-[2-[(Z)-[(19S)-19-ethyl-19-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4,6,8,10,15(20)-heptaen-10-yl]methylideneamino]oxyethylamino]-4-oxobutyl]-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]acetic acid | IC50 | 5800.0 [1] |
| 4-[[4-[(2S,5S,11S,14R)-14-Benzyl-11-(carboxymethyl)-5-[3-(diaminomethylideneamino)propyl]-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]phenyl]methylamino]-4-oxobutanoic acid | IC50 | 33700.0 [1] |
| 2-[(2S,5R,8S,11S)-5-Benzyl-11-[3-(diaminomethylideneamino)propyl]-8-[[4-[[[4-[2-[(E)-[(19S)-19-ethyl-19-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4,6,8,10,15(20)-heptaen-10-yl]methylideneamino]oxyethylamino]-4-oxobutanoyl]amino]methyl]phenyl]methyl]-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]acetic acid | IC50 | 100000.0 [1] |
| 2-[(2S,5R,8S,11S)-5-Benzyl-11-[3-(diaminomethylideneamino)propyl]-8-[[4-[[[2-[2-[2-[2-[2-[(E)-[(19S)-19-ethyl-19-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4,6,8,10,15(20)-heptaen-10-yl]methylideneamino]oxyethylamino]-2-oxoethoxy]ethoxy]ethoxy]acetyl]amino]methyl]phenyl]methyl]-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]acetic acid | IC50 | 8300.0 [1] |
| 2-[(2S,5R,8S,11S)-5-Benzyl-11-[3-(diaminomethylideneamino)propyl]-8-[[4-[[[2-[2-[2-[2-[(2E)-2-[[(19S)-19-ethyl-19-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4,6,8,10,15(20)-heptaen-10-yl]methylidene]hydrazinyl]-2-oxoethoxy]ethoxy]ethoxy]acetyl]amino]methyl]phenyl]methyl]-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]acetic acid | IC50 | 4800.0 [1] |
| 2-[(2S,5R,8S,11S)-5-Benzyl-11-[3-(diaminomethylideneamino)propyl]-8-[4-[[[2-[2-[2-(2-hydrazinyl-2-oxoethoxy)ethoxy]ethoxy]acetyl]amino]methyl]phenyl]-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]acetic acid | IC50 | 15600.0 [1] |
| 2-[(2S,5R,8S,11S)-5-Benzyl-8-[4-[[[2-[2-[2-(carboxymethoxy)ethoxy]ethoxy]acetyl]amino]methyl]phenyl]-11-[3-(diaminomethylideneamino)propyl]-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]acetic acid | IC50 | 18800.0 [1] |