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Vascular endothelial growth factor receptor Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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VandetanibIC5025.0 [1], 400.0 [2]
N-(4-Bromo-2-fluorophenyl)-6-methoxy-7-[2-(triazol-1-yl)ethoxy]quinazolin-4-amineIC5050.0 [1]
6-(4-Methoxyphenyl)-3-(3-thienyl)-pyrazolo(1,5-a)pyrimidineIC50387.0 [1]
Pyrazolo[1,5-a]pyrimidine 1aIC50622.0 [1]
Pyrazolo[1,5-a]pyrimidine 2cIC50150.0 [1]
ErlotinibIC50250.0 [1]
VatalanibIC50100.0 [1]
PD173074IC50190.0 [1]
Raf265(chir-265)IC5020.0 [1]
PDGF Receptor Tyrosine Kinase Inhibitor IVIC503100.0 [1]
N-(4-Chloro-2-fluorophenyl)-6,7-dimethoxyquinazolin-4-amineIC501000.0 [1]
N-(4-Chlorophenylsulfonyl)benzamideIC5022000.0 [1]
4-[2-[4-(3-Phenylpyrazolo[1,5-a]pyrimidin-6-yl)phenoxy]ethyl]morpholineIC5032.0 [1]
2-Oxazolamine, N,5-diphenyl-IC503000.0 [1]
N-[2,4-Dichlorobenzoyl]phenylsulfonamideIC50530.0 [1]
2,4-Dichloro-N-(4-chlorophenyl)sulfonylbenzamideIC50170.0 [1]
4-[2-(3-Tert-butylanilino)-1-methylbenzimidazol-5-yl]oxy-N-methylpyridine-2-carboxamideIC505.0 [1]
N-[5-(Ethylsulfonyl)-2-methoxyphenyl]-5-[3-(2-pyridinyl)phenyl]-1,3-oxazol-2-amineIC50370.0 [1]
N-(3-Methylphenyl)-5-phenyl-1,3-oxazol-2-amineIC501700.0 [1]
4-[(5-Phenyl-1,3-oxazol-2-yl)amino]benzenesulfonamideIC504660.0 [1]
N-(3,5-Dimethoxyphenyl)-5-phenyl-1,3-oxazol-2-amineIC501690.0 [1]
5-Phenyl-N-(3,4,5-trimethoxyphenyl)-1,3-oxazol-2-amineIC50420.0 [1]
2-Anilino-5-aryloxazole 20IC501310.0 [1]
2-Anilino-5-aryloxazole 24IC507600.0 [1]
2-Anilino-5-aryloxazole 27IC501650.0 [1]
2-Anilino-5-aryloxazole 28IC50350.0 [1]
1-[3-(2-{[5-(Ethylsulfonyl)-2-methoxyphenyl]amino}-1,3-oxazol-5-yl)phenyl]ethanoneIC5013900.0 [1]
2-Anilino-5-aryloxazole 44IC5040.0 [1]
Unii-8FX9DP2Y1WIC501000.0 [1]
2,4-Difluoro-N-methoxy-5-[[6-(5-methyl-1,3,4-oxadiazol-2-yl)-5-propan-2-ylpyrrolo[2,1-f][1,2,4]triazin-4-yl]amino]benzamideIC507.6 [1]
N-(4-Chloro-2-fluorophenyl)-6-methoxy-7-(2-methoxyethoxy)quinazolin-4-amineIC5040.0 [1]
Pyrazolo[1,5-a]pyrimidine 4eIC5018.0 [1]
4-[2-[4-(3-Pyridin-4-ylpyrazolo[1,5-a]pyrimidin-6-yl)phenoxy]ethyl]morpholineIC5031.0 [1]
3-[[5-[6-[(3-Chlorophenyl)amino]pyrazinyl]-3-pyridinyl]amino]-1-propanolIC505.0 [1]
5-[[6-[5-(Difluoromethyl)-1,3,4-oxadiazol-2-yl]-5-propan-2-ylpyrrolo[2,1-f][1,2,4]triazin-4-yl]amino]-2,4-difluoro-N-methoxybenzamideIC5017.0 [1]
2,4-Difluoro-N-methoxy-5-[[6-(5-methyl-1,3-oxazol-2-yl)-5-propan-2-ylpyrrolo[2,1-f][1,2,4]triazin-4-yl]amino]benzamideIC501.1 [1]
2,4-Difluoro-N-methoxy-5-[[6-[5-(methylsulfonylmethyl)-1,3,4-oxadiazol-2-yl]-5-propan-2-ylpyrrolo[2,1-f][1,2,4]triazin-4-yl]amino]benzamideIC502.1 [1]
2,4-Dichloro-N-(3,4-dichlorophenyl)sulfonylbenzamideIC50460.0 [1]
(3-Chloro-4-fluoro-phenyl)-(5-methyl-pyrrolo[2,1-f][1,2,4]triazin-4-yl)-amineIC502500000.0 [1]
5-[[6-[5-[Difluoro(methylsulfonyl)methyl]-1,3,4-oxadiazol-2-yl]-5-propan-2-ylpyrrolo[2,1-f][1,2,4]triazin-4-yl]amino]-2,4-difluoro-N-methoxybenzamideIC5027.0 [1]
1-(3-Cyanophenyl)-3-(4,6,8,9-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,7,10,12-hexaen-3-yl)ureaIC50200.0 [1]
1-(4-Fluorophenyl)-3-(4,6,8,9-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,7,10,12-hexaen-3-yl)ureaIC50631.0 [1]
1-(4,6,8,9-Tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,7,10,12-hexaen-3-yl)-3-[4-(trifluoromethyl)phenyl]ureaIC503980.0 [1]
1-(4,6,8,9-Tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,7,10,12-hexaen-3-yl)-3-[3-(trifluoromethyl)phenyl]ureaIC50251.0 [1]
1-(3-Nitrophenyl)-3-(4,6,8,9-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,7,10,12-hexaen-3-yl)ureaIC5010000.0 [1]
1-(4-Bromophenyl)-3-(4,6,8,9-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,7,10,12-hexaen-3-yl)ureaIC503980.0 [1]
Vandetanib hydrochlorideIC5060.0 [1]
1,6-Naphthyridine deriv. 20IC5037.0 [1]
Anilinoquinazoline deriv. 21IC50300.0 [1]
Anilinoquinazoline deriv. 22IC5050.0 [1]
Anilinoquinazoline deriv. 28IC50200.0 [1]
3-(5-Thien-3-ylpyridin-3-yl)-1Hindole 3fIC50328.0 [1]
2,4-Disubstituted Pyrimidine 2dIC5019.0 [1]
Pyrazolo[1,5-a]pyrimidine 4aIC5022.0 [1]
Pyrazolo[1,5-a]pyrimidine 4gIC5029.0 [1]
N-[4-[2-(3-Tert-butylanilino)-1-methylbenzimidazol-5-yl]oxypyridin-2-yl]acetamideIC502.0 [1]
2-Methyl-5-(pyrrolo[2,1-f][1,2,4]triazin-4-ylamino)-phenolIC50360000.0 [1]
4-Bromo-2-chloro-N-(4-chlorophenyl)sulfonylbenzamideIC50200.0 [1]
2-Methyl-5-(6-methyl-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino)-phenolIC50213000.0 [1]
2-Methyl-5-(7-methyl-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino)-phenolIC50477000.0 [1]
5-(5,6-Dimethyl-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino)-2-methyl-phenolIC50310000.0 [1]
3-Piperidin-1-ylpropyl N-[4-[2,4-difluoro-5-(methoxycarbamoyl)anilino]-5-propan-2-ylpyrrolo[2,1-f][1,2,4]triazin-6-yl]carbamateIC5062.0 [1]
5-[[6-[5-(Cyclopropylmethyl)-1,3,4-oxadiazol-2-yl]-5-propan-2-ylpyrrolo[2,1-f][1,2,4]triazin-4-yl]amino]-2,4-difluoro-N-methoxybenzamideIC504.0 [1]
N-(4-Chlorophenyl)sulfonyl-4-(dimethylamino)benzamideIC5016000.0 [1]
2,4-Dichloro-N-(4-methoxyphenyl)sulfonylbenzamideIC50350.0 [1]
2,4-Dichloro-N-(3-methoxyphenyl)sulfonylbenzamideIC50910.0 [1]
3-Chloro-N-(4-chlorophenyl)sulfonylbenzamideIC5014000.0 [1]
2,4-Dichloro-N-(3-chloro-4-fluorophenyl)sulfonylbenzamideIC50410.0 [1]
2,5-Dichloro-N-(4-chlorophenyl)sulfonylbenzamideIC5013000.0 [1]
4-Chloro-N-(4-chlorophenyl)sulfonyl-2-propylbenzamideIC501300.0 [1]
2,4-Dibromo-N-(4-chlorophenyl)sulfonylbenzamideIC50250.0 [1]
4-Chloro-N-(4-chlorophenyl)sulfonyl-2-nitrobenzamideIC505900.0 [1]
2,4-Dichloro-N-(3,4-dimethoxyphenyl)sulfonylbenzamideIC503900.0 [1]
2,4-Dichloro-N-(3,5-dichlorophenyl)sulfonylbenzamideIC501400.0 [1]
4-Bromo-N-(4-chlorophenyl)sulfonyl-2-methylbenzamideIC50610.0 [1]
N-(3-Bromophenyl)sulfonyl-2,4-dichlorobenzamideIC50250.0 [1]
N-(4-Acetylphenyl)sulfonyl-2,4-dichlorobenzamideIC50560.0 [1]
2,4-Dichloro-N-[4-(dimethylamino)phenyl]sulfonylbenzamideIC50930.0 [1]
2,4-Dichloro-N-(3-nitrophenyl)sulfonylbenzamideIC50910.0 [1]
N-(4-Chlorophenyl)sulfonyl-2-nitro-4-(trifluoromethyl)benzamideIC5011000.0 [1]
N-(2-Methoxyphenyl)-5-phenyl-1,3-oxazol-2-amine;hydrochlorideIC503260.0 [1]
4-Chloro-N-(4-chlorophenyl)sulfonyl-2-methoxybenzamideIC502000.0 [1]
2-Chloro-N-(4-chlorophenyl)sulfonyl-4-nitrobenzamideIC50620.0 [1]
N-(3,4-Dimethoxyphenyl)-5-phenyl-1,3-oxazol-2-amine;hydrochlorideIC501130.0 [1]
2,4-Dichloro-N-(4-methylphenyl)sulfonylbenzamideIC50210.0 [1]
2,4-Dichloro-N-(3-chlorophenyl)sulfonylbenzamideIC50440.0 [1]
3-Bromo-N-(4-chlorophenyl)sulfonylbenzamideIC5015000.0 [1]
2,4-Dichloro-N-(3-chloro-4-methylphenyl)sulfonylbenzamideIC50360.0 [1]
2,4-Dichloro-N-(3,4-dibromophenyl)sulfonylbenzamideIC50910.0 [1]
4-Chloro-N-(4-chlorophenyl)sulfonyl-2-ethylbenzamideIC50630.0 [1]
N-(4-Chlorophenyl)sulfonyl-2-methylbenzamideIC5015000.0 [1]
N-(4-Chlorophenyl)sulfonyl-2,4-dimethoxybenzamideIC5020000.0 [1]
N-(3-Chloro-4-fluorophenyl)-7-methylpyrrolo[2,1-f][1,2,4]triazin-4-amineIC502500000.0 [1]
N-(2-Bromo-4-methylphenyl)sulfonyl-2,4-dichlorobenzamideIC5020000.0 [1]
N-(4-Chlorophenyl)sulfonyl-2,4-dinitrobenzamideIC5013000.0 [1]
2-Amino-4-chloro-N-(4-chlorophenyl)sulfonylbenzamideIC503200.0 [1]
2,4-Dichloro-N-(2-chlorophenyl)sulfonylbenzamideIC5014000.0 [1]
Ethyl N-[4-[2,4-difluoro-5-(methoxycarbamoyl)anilino]-5-propan-2-ylpyrrolo[2,1-f][1,2,4]triazin-6-yl]carbamateIC5031.0 [1]
(1-Methylpiperidin-4-yl) N-[4-[2,4-difluoro-5-(methoxycarbamoyl)anilino]-5-propan-2-ylpyrrolo[2,1-f][1,2,4]triazin-6-yl]carbamateIC5019.0 [1]
2,4-Difluoro-N-methoxy-5-[[6-(5-methyl-1H-1,2,4-triazol-3-yl)-5-propan-2-ylpyrrolo[2,1-f][1,2,4]triazin-4-yl]amino]benzamideIC5050.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Vascular endothelial growth factor receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 22 Dec. 2024, https://www.aatbio.com/data-sets/vascular-endothelial-growth-factor-receptor-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 22). Quest Database™ Vascular endothelial growth factor receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/vascular-endothelial-growth-factor-receptor-inhibitors-ic50-ki.
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