| 3-Aminoquinoxalin-2(1H)-one | Ki | 20.8 [1] |
| 2-[[12-(3,5-Dimethylpiperidin-1-yl)-8-oxo-15-oxa-14-azatetracyclo[7.6.1.02,7.013,16]hexadeca-1(16),2,4,6,9,11,13-heptaen-10-yl]amino]benzoic acid | IC50 | 10000.0 [1] |
| 6,12-Dihydroquinoxalino[2,3-b][1,4]benzodiazepin-13-one | Ki | 1.33 [1] |
| 2-[(1R,4S,7S,13S,19S,22S,25S,28S,31R,34S,40S,43R,49S)-25-(4-Aminobutyl)-49-benzyl-4,19-bis[(2S)-butan-2-yl]-34-[3-(diaminomethylideneamino)propyl]-28-[(1R)-1-hydroxyethyl]-22-(hydroxymethyl)-3,6,12,18,21,24,27,30,33,36,39,42,48,51-tetradecaoxo-53,54-dithia-2,5,11,17,20,23,26,29,32,35,38,41,47,50-tetradecazapentacyclo[29.20.4.07,11.013,17.043,47]pentapentacontan-40-yl]acetic acid | Ki | 500000.0 [1] |
| 3-(1H-Benzimidazol-2-yl)-1-(1H-benzimidazol-2-ylmethyl)-5-phenylpyrrol-2-amine | Ki | 0.0 [1] |
| 6-(1H-Benzimidazol-2-ylmethyl)-11H-quinoxalino[2,3-b][1,4]benzodiazepin-13-one | Ki | 0.01 [1] |
| 2-Amino-1-(1H-benzimidazol-2-ylmethyl)-5-phenyl-pyrrole-3-carbonitrile | Ki | 0.0 [1] |
| 3-(1H-Benzimidazol-2-yl)-5-phenyl-1-(2-pyridyl)pyrrol-2-amine | Ki | 0.01 [1] |
| 3-(1H-Benzimidazol-2-yl)-1-(3-chlorophenyl)-5-phenylpyrrol-2-amine | Ki | 0.0 [1] |
| 6-[(1-Prop-2-enylbenzimidazol-2-yl)methyl]-11H-quinoxalino[2,3-b][1,4]benzodiazepin-13-one | Ki | 0.0 [1] |
| 2-Amino-1-(1H-benzimidazol-2-yl)-5-phenyl-pyrrole-3-carbonitrile | Ki | 0.0 [1] |
| 3-(1H-Benzimidazol-2-yl)-5-phenyl-1-(4-pyridyl)pyrrol-2-amine | Ki | 0.0 [1] |
| 3-(1H-Benzimidazol-2-yl)-1-(4-bromophenyl)-5-phenyl-pyrrol-2-amine | Ki | 0.01 [1] |
| Ethyl 2-[2-[(13-oxo-11H-quinoxalino[2,3-b][1,4]benzodiazepin-6-yl)methyl]benzimidazol-1-yl]acetate | Ki | 0.0 [1] |
| 3-(1H-Benzimidazol-2-yl)-1-(3-bromophenyl)-5-phenyl-pyrrol-2-amine | Ki | 0.01 [1] |
| 1,3-Bis(1H-benzimidazol-2-yl)-5-phenyl-pyrrol-2-amine | Ki | 0.0 [1] |
| 3-(1H-Benzimidazol-2-yl)-1-(4-chlorophenyl)-5-phenylpyrrol-2-amine | Ki | 0.0 [1] |
| 2-Amino-1-(4-chlorophenyl)-5-phenylpyrrole-3-carbonitrile | Ki | 0.0 [1] |
| 2-Amino-1-(3-chlorophenyl)-5-phenylpyrrole-3-carbonitrile | Ki | 0.0 [1] |
| 2-Amino-1-(4-bromophenyl)-5-phenylpyrrole-3-carbonitrile | Ki | 0.0 [1] |
| 3-[[12-(3-Ethoxycarbonylpiperidin-1-yl)-8-oxo-15-oxa-14-azatetracyclo[7.6.1.02,7.013,16]hexadeca-1(16),2,4,6,9,11,13-heptaen-10-yl]amino]propanoic acid | IC50 | 51000.0 [1] |
| 4-[[12-(3-Methylpiperidin-1-yl)-8-oxo-15-oxa-14-azatetracyclo[7.6.1.02,7.013,16]hexadeca-1(16),2,4,6,9,11,13-heptaen-10-yl]amino]butanoic acid | IC50 | 20000.0 [1] |
| 4-[[12-(3,5-Dimethylpiperidin-1-yl)-8-oxo-15-oxa-14-azatetracyclo[7.6.1.02,7.013,16]hexadeca-1(16),2,4,6,9,11,13-heptaen-10-yl]amino]butanoic acid | IC50 | 36000.0 [1] |
| 3-[[12-(3-Methylpiperidin-1-yl)-8-oxo-15-oxa-14-azatetracyclo[7.6.1.02,7.013,16]hexadeca-1(16),2,4,6,9,11,13-heptaen-10-yl]amino]propanoic acid | IC50 | 24000.0 [1] |
| 2-[(8-Oxo-12-pyrrolidin-1-yl-15-oxa-14-azatetracyclo[7.6.1.02,7.013,16]hexadeca-1(16),2,4,6,9,11,13-heptaen-10-yl)amino]benzoic acid | IC50 | 21000.0 [1] |
| 3-[[12-(3-Methylpiperidin-1-yl)-8-oxo-15-oxa-14-azatetracyclo[7.6.1.02,7.013,16]hexadeca-1(16),2,4,6,9,11,13-heptaen-10-yl]amino]benzoic acid | IC50 | 7000.0 [1] |
| 3-[[12-(2-Methylpiperidin-1-yl)-8-oxo-15-oxa-14-azatetracyclo[7.6.1.02,7.013,16]hexadeca-1(16),2,4,6,9,11,13-heptaen-10-yl]amino]benzoic acid | IC50 | 10000.0 [1] |
| 3-[[12-(3,5-Dimethylpiperidin-1-yl)-8-oxo-15-oxa-14-azatetracyclo[7.6.1.02,7.013,16]hexadeca-1(16),2,4,6,9,11,13-heptaen-10-yl]amino]benzoic acid | IC50 | 5000.0 [1] |
| (2S)-4-Amino-2-[[(3S,6R,9S,12R,15S,18R,21S,26S,29R)-21-amino-3,18-bis(2-amino-2-oxoethyl)-6-(3-amino-3-oxopropyl)-15-(2-carboxyethyl)-9-(1H-imidazol-5-ylmethyl)-12-(2-methylpropyl)-2,5,8,11,14,17,20,28-octaoxo-23,24-dithia-1,4,7,10,13,16,19,27-octazabicyclo[27.3.0]dotriacontane-26-carbonyl]amino]-4-oxobutanoic acid | IC50 | 30000.0 [1] |
| (2S)-4-Amino-2-[[(3S,6R,9S,12R,15R,18R,21S,26S,29R)-21-amino-15-(4-aminobutyl)-18-(2-amino-2-oxoethyl)-6-(3-amino-3-oxopropyl)-9-(1H-imidazol-5-ylmethyl)-12-(2-methylpropyl)-2,5,8,11,14,17,20,28-octaoxo-3-propan-2-yl-23,24-dithia-1,4,7,10,13,16,19,27-octazabicyclo[27.3.0]dotriacontane-26-carbonyl]amino]-4-oxobutanoic acid | IC50 | 30000.0 [1] |
| (2S)-4-Amino-2-[[(3S,6R,9S,12R,15S,18S,21S,26S,29R)-21-amino-18-(2-amino-2-oxoethyl)-6-(3-amino-3-oxopropyl)-15-(2-carboxyethyl)-9-(1H-imidazol-5-ylmethyl)-12-(2-methylpropyl)-2,5,8,11,14,17,20,28-octaoxo-3-propan-2-yl-23,24-dithia-1,4,7,10,13,16,19,27-octazabicyclo[27.3.0]dotriacontane-26-carbonyl]amino]-4-oxobutanoic acid | IC50 | 30000.0 [1] |
| (2S)-4-Amino-2-[[(3S,6R,9S,12R,15S,18R,21S,26S,29R)-21-amino-18-(2-amino-2-oxoethyl)-6-(3-amino-3-oxopropyl)-15-(2-carboxyethyl)-9-(1H-imidazol-5-ylmethyl)-12-(2-methylpropyl)-2,5,8,11,14,17,20,28-octaoxo-3-propan-2-yl-23,24-dithia-1,4,7,10,13,16,19,27-octazabicyclo[27.3.0]dotriacontane-26-carbonyl]amino]-4-oxobutanoic acid | IC50 | 900.0 [1] |
| (3S,6R,9S,12R,15S,18R,21S,27S,32S,35R,38S,41R)-27-Amino-18,35-bis(2-amino-2-oxoethyl)-6-(3-amino-3-oxopropyl)-15-(2-carboxyethyl)-21,38-bis(hydroxymethyl)-9-(1H-imidazol-5-ylmethyl)-12-(2-methylpropyl)-2,5,8,11,14,17,20,23,26,34,37,40-dodecaoxo-3-propan-2-yl-29,30-dithia-1,4,7,10,13,16,19,22,25,33,36,39-dodecazabicyclo[39.3.0]tetratetracontane-32-carboxylic acid | IC50 | 700.0 [1] |
| (2S)-4-Amino-2-[[(3S,6R,9S,12R,15S,18R,21R,26R,29R)-21-amino-18-(2-amino-2-oxoethyl)-6-(3-amino-3-oxopropyl)-15-(2-carboxyethyl)-9-(1H-imidazol-5-ylmethyl)-12-(naphthalen-2-ylmethyl)-2,5,8,11,14,17,20,28-octaoxo-3-propan-2-yl-23,24-dithia-1,4,7,10,13,16,19,27-octazabicyclo[27.3.0]dotriacontane-26-carbonyl]amino]-4-oxobutanoic acid | IC50 | 80.0 [1] |
| (2S)-4-Amino-2-[[(3S,6R,9S,12R,15S,18R,21R,26R,29R)-21-amino-18-(2-amino-2-oxoethyl)-6-(3-amino-3-oxopropyl)-15-(2-carboxyethyl)-9-(1H-imidazol-5-ylmethyl)-12-(naphthalen-1-ylmethyl)-2,5,8,11,14,17,20,28-octaoxo-3-propan-2-yl-23,24-dithia-1,4,7,10,13,16,19,27-octazabicyclo[27.3.0]dotriacontane-26-carbonyl]amino]-4-oxobutanoic acid | IC50 | 50.0 [1] |
| (2S)-4-Amino-2-[[(3S,6R,9S,12R,15S,18R,21R,26R,29R)-21-amino-18-(2-amino-2-oxoethyl)-6-(3-amino-3-oxopropyl)-15-butyl-9-(1H-imidazol-5-ylmethyl)-12-(2-methylpropyl)-2,5,8,11,14,17,20,28-octaoxo-3-propan-2-yl-23,24-dithia-1,4,7,10,13,16,19,27-octazabicyclo[27.3.0]dotriacontane-26-carbonyl]amino]-4-oxobutanoic acid | IC50 | 60.0 [1] |
| (3S,6R,9S,12R,15S,18R,21S,27R,32S,35R,38S,41R)-27-Amino-18,35-bis(2-amino-2-oxoethyl)-6-(3-amino-3-oxopropyl)-15-(2-carboxyethyl)-21,38-bis(hydroxymethyl)-9-(1H-imidazol-5-ylmethyl)-12-(2-methylpropyl)-2,5,8,11,14,17,20,23,26,34,37,40-dodecaoxo-3-propan-2-yl-29,30-dithia-1,4,7,10,13,16,19,22,25,33,36,39-dodecazabicyclo[39.3.0]tetratetracontane-32-carboxylic acid | IC50 | 200.0 [1] |
| (2S)-4-Amino-2-[[(3S,6R,9S,12R,15S,18R,21R,26R,29R)-21-amino-18-(2-amino-2-oxoethyl)-6-(3-amino-3-oxopropyl)-15-(2-carboxyethyl)-9-(1H-imidazol-5-ylmethyl)-12-(2-methylpropyl)-2,5,8,11,14,17,20,28-octaoxo-3-propan-2-yl-23,24-dithia-1,4,7,10,13,16,19,27-octazabicyclo[27.3.0]dotriacontane-26-carbonyl]amino]-4-oxobutanoic acid | IC50 | 40.0 [1] |
| (2S)-4-Amino-2-[[(3S,6S,9S,12R,15S,18R,21S,26S,29R)-21-amino-18-(2-amino-2-oxoethyl)-15-(2-carboxyethyl)-6-(hydroxymethyl)-9-(1H-imidazol-5-ylmethyl)-12-(2-methylpropyl)-2,5,8,11,14,17,20,28-octaoxo-3-propan-2-yl-23,24-dithia-1,4,7,10,13,16,19,27-octazabicyclo[27.3.0]dotriacontane-26-carbonyl]amino]-4-oxobutanoic acid | IC50 | 30000.0 [1] |
| 3-[[12-(3,5-Dimethylpiperidin-1-yl)-8-oxo-15-oxa-14-azatetracyclo[7.6.1.02,7.013,16]hexadeca-1(16),2,4,6,9,11,13-heptaen-10-yl]amino]propanoic acid | IC50 | 18000.0 [1] |
| 4-[[8-Oxo-12-(4-oxopiperidin-1-yl)-15-oxa-14-azatetracyclo[7.6.1.02,7.013,16]hexadeca-1(16),2,4,6,9,11,13-heptaen-10-yl]amino]benzoic acid | IC50 | 100000.0 [1] |
| 4-[[[3-(1,3-Benzodioxol-5-yl)-4-phenylbutyl]amino]methyl]-N,N-dimethylaniline | Ki | 20000.0 [1] |
| 2-Phenacylpropanedinitrile | Ki | 0.3 [1] |
| Methyl 3-[[12-(azepan-1-yl)-8-oxo-15-oxa-14-azatetracyclo[7.6.1.02,7.013,16]hexadeca-1(16),2,4,6,9,11,13-heptaen-10-yl]amino]benzoate | IC50 | 100000.0 [1] |
| 3-[(3-Bromo-4-hydroxy-6,7-dimethyl-9,10-dioxoanthracen-1-yl)amino]benzoic acid | IC50 | 67000.0 [1] |
| 2-Amino-5-phenyl-1-pyridin-4-ylpyrrole-3-carbonitrile | Ki | 0.01 [1] |
| 3-[(3-Bromo-9,10-dioxo-4-propan-2-yloxyanthracen-1-yl)amino]benzoic acid | IC50 | 30000.0 [1] |
| 3-[(3-Bromo-4-hydroxy-6-methyl-9,10-dioxoanthracen-1-yl)amino]benzoic acid | IC50 | 146000.0 [1] |
| 2-Amino-5-phenyl-1-pyridin-2-ylpyrrole-3-carbonitrile | Ki | 0.03 [1] |
| 3-[(3-Bromo-9,10-dioxo-4-phenylmethoxyanthracen-1-yl)amino]benzoic acid | IC50 | 30000.0 [1] |
| 4-[[12-(3-Methylpiperidin-1-yl)-8-oxo-15-oxa-14-azatetracyclo[7.6.1.02,7.013,16]hexadeca-1(16),2,4,6,9,11,13-heptaen-10-yl]methyl]benzoic acid | IC50 | 11000.0 [1] |
| 2-Amino-1-(3-bromophenyl)-5-phenylpyrrole-3-carbonitrile | Ki | 0.0 [1] |
| 2-[[12-[(3S,5S)-3,5-Dimethylpiperidin-1-yl]-8-oxo-15-oxa-14-azatetracyclo[7.6.1.02,7.013,16]hexadeca-1(16),2,4,6,9,11,13-heptaen-10-yl]amino]benzoic acid | IC50 | 10000.0 [1] |