UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	N-[4-(4-Naphthalen-2-yltriazol-1-yl)phenyl]acetamide	IC50	66700.0 [1]
	N-[4-(4-Naphthalen-2-yltriazol-1-yl)phenyl]acetamide	Ki	28600.0 [1], 59800.0 [2]
	N-[4-[4-(4-Phenylphenyl)triazol-1-yl]phenyl]acetamide	IC50	139000.0 [1]
	N-[4-[4-(4-Phenylphenyl)triazol-1-yl]phenyl]acetamide	Ki	92000.0 [1], 310000.0 [2]
	Phenyl 5-chloro-2-oxobenzo[d]oxazole-3(2H)-carboxylate	IC50	10000.0 [1]
	6-[[1-[[(2R,3S,4R,5R)-5-(2,4-Dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl]triazol-4-yl]methyl]-N-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]pyridine-2-carboxamide	IC50	340000.0 [1]
	6-[[1-[[(2R,3S,4R,5R)-5-(2,4-Dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl]triazol-4-yl]methyl]-N-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]pyridine-2-carboxamide	Ki	420000.0 [1]
	Alloxan	IC50	100000.0 [1]
	Uridine-5'-diphosphate	IC50	1800.0 [1]
	2-Benzoxazolinone	IC50	11900.0 [1]
	2-Ethynylnaphthalene	IC50	4000000.0 [1]
	4-Ethynyl-1,1'-biphenyl	IC50	1000000.0 [1]
	1,1-Diphenyl-2-propyn-1-ol	IC50	1964000.0 [1]
	N-(4-Azidophenyl)acetamide	IC50	4000000.0 [1]
	1-(2-Thienyl)-3-(4-cyanobenzylthio)-5,6,7,8-tetrahydroisoquinoline-4-carboxylic acid	IC50	100000.0 [1]
	N-(4-Azidophenyl)-2-iodoacetamide	IC50	865000.0 [1]
	2-Chloro-N-[4-(4-naphthalen-2-yltriazol-1-yl)phenyl]acetamide	IC50	71700.0 [1]
	2-Chloro-N-[4-[4-(4-phenylphenyl)triazol-1-yl]phenyl]acetamide	IC50	91200.0 [1]
	2-Chloro-N-[4-[4-[hydroxy(diphenyl)methyl]triazol-1-yl]phenyl]acetamide	IC50	89300.0 [1]
	N-[4-[4-[Hydroxy(diphenyl)methyl]triazol-1-yl]phenyl]acetamide	IC50	1001000.0 [1]
	CID 21340782	IC50	3967000.0 [1]
	(2S)-8-[5-[(2S)-5,7-Dihydroxy-4-oxo-2,3-dihydrochromen-2-yl]-2-hydroxyphenyl]-5,7-dihydroxy-2-(4-hydroxyphenyl)-2,3-dihydrochromen-4-one	IC50	22000.0 [1]
	[(2R,3R,4R,5S,6R)-3-Acetamido-4,5-dihydroxy-6-(hydroxymethyl)oxan-2-yl]sulfanyl-[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxyphosphinic acid	Ki	93000.0 [1]
	[[(2S,3R,4R,5S,6R)-3-Acetamido-4,5-dihydroxy-6-(hydroxymethyl)oxan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl hydrogen phosphate	IC50	5000000.0 [1]
	3-(1-Adamantylmethyl)-2-(4-chlorophenyl)imino-4-oxo-1,3-thiazinane-6-carboxylic acid	IC50	53000.0 [1]
	(2S)-N-[(2S,3R)-1-[[(2S)-1-Amino-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]-2-[[(2S)-2-[[(2S)-1-[(2S,3R)-2-[[(2S)-2-[[(2R)-2-amino-3-sulfanylpropanoyl]amino]-3-methylbutanoyl]amino]-3-hydroxybutanoyl]pyrrolidine-2-carbonyl]amino]-3-methylbutanoyl]amino]-N'-[2-[2-[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy]ethoxy]ethyl]pentanediamide	IC50	493000.0 [1]
	(2S)-N-[(2S)-1-[[(2S)-1-[[(2S,3R)-1-[[(2S)-1-Amino-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]-1-[(2S,3R)-2-[[(2S)-2-[[(2R)-2-amino-3-sulfanylpropanoyl]amino]-3-methylbutanoyl]amino]-3-hydroxybutanoyl]pyrrolidine-2-carboxamide	IC50	385000.0 [1]
	N-[[4-[[(5S)-6-[[(2S,3R)-1-[[(2S)-1-Amino-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-5-[[(2S)-2-[[(2S)-1-[(2S,3R)-2-[[(2S)-2-[[(2R)-2-amino-3-sulfanylpropanoyl]amino]-3-methylbutanoyl]amino]-3-hydroxybutanoyl]pyrrolidine-2-carbonyl]amino]-3-methylbutanoyl]amino]-6-oxohexyl]carbamoyl]phenyl]methyl]-2-oxo-1H-quinoline-4-carboxamide	IC50	117000.0 [1]
	(2S)-N-[(2S,3R)-1-[[(2S)-1-Amino-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]-2-[[(2S)-2-[[(2S)-1-[(2S,3R)-2-[[(2S)-2-[[(2R)-2-amino-3-sulfanylpropanoyl]amino]-3-methylbutanoyl]amino]-3-hydroxybutanoyl]pyrrolidine-2-carbonyl]amino]-3-methylbutanoyl]amino]-N'-[2-[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy]ethyl]pentanediamide	IC50	1000000.0 [1]
	(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-Amino-5-(diaminomethylideneamino)pentanoyl]amino]-3-methylbutanoyl]pyrrolidine-2-carbonyl]amino]-3-hydroxypropanoyl]amino]-5-[2-[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy]ethylamino]-5-oxopentanoyl]amino]-N-[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]pentanediamide	IC50	1000000.0 [1]
	(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-Amino-5-(diaminomethylideneamino)pentanoyl]amino]-3-methylbutanoyl]pyrrolidine-2-carbonyl]amino]-3-hydroxypropanoyl]amino]propanoyl]amino]-N-[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]pentanediamide	IC50	193000.0 [1]
	(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-Amino-5-(diaminomethylideneamino)pentanoyl]amino]-3-methylbutanoyl]pyrrolidine-2-carbonyl]amino]-3-hydroxypropanoyl]amino]-5-[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methylamino]-5-oxopentanoyl]amino]-N-[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]pentanediamide	IC50	1000000.0 [1]
	(2S)-N-[(2S,3R)-1-[[(2S)-1-Amino-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]-2-[[(2S)-2-[[(2S)-1-[(2S,3R)-2-[[(2S)-2-[[(2R)-2-amino-3-sulfanylpropanoyl]amino]-3-methylbutanoyl]amino]-3-hydroxybutanoyl]pyrrolidine-2-carbonyl]amino]-3-methylbutanoyl]amino]-N'-[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl]pentanediamide	IC50	297000.0 [1]
	[(2S,3R,4R,5S,6R)-3-Acetamido-4,5-dihydroxy-6-(hydroxymethyl)thian-2-yl] [[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate	Ki	8000.0 [1]
	1-[(2R,3R,4S,5R)-5-[[4-(6-Bromopyridin-2-yl)triazol-1-yl]methyl]-3,4-dihydroxyoxolan-2-yl]pyrimidine-2,4-dione	IC50	710000.0 [1]
	1-[(2R,3R,4S,5R)-3,4-Dihydroxy-5-[[4-[6-[1-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]triazol-4-yl]pyridin-2-yl]triazol-1-yl]methyl]oxolan-2-yl]pyrimidine-2,4-dione	IC50	1600000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 36 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/udp-n-acetylglucosamine-peptide-n-acetylglucosaminyltransferase-110-kda-subunit-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, November 21). Quest Database™ UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/udp-n-acetylglucosamine-peptide-n-acetylglucosaminyltransferase-110-kda-subunit-inhibitors-ic50-ki.
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