UDP-glucuronosyltransferase 2B7 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Mycophenolic acid	Ki	1500.0 [1]
	Zidovudine	Ki	150000.0 [1], 200000.0 [2]
	6-Methyl-3,4-dihydro-2H-chromen-4-ol	Ki	113000.0 [1], 258000.0 [2]
	6-Methyl-2,3-dihydro-1H-inden-1-ol	Ki	301000.0 [1], 624000.0 [2]
	5,7-Dimethyltetralin-1-ol	Ki	101000.0 [1], 192000.0 [2]
	(R)-Phenyl-[(1R,2S,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]methanol	IC50	47.0 [1]
	(R)-Phenyl-[(1R,2S,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]methanol	Ki	18.4 [1]
	Valproic acid	Ki	1600000.0 [1]
	Haloperidol	Ki	590000.0 [1]
	Epiestriol	Ki	162000.0 [1]
	Isolongifolol	IC50	100.0 [1]
	(1R,2S,7S,8S,9S)-3,3,7-Trimethyltricyclo[5.4.0.02,9]undecane-8-carboxylic acid	IC50	2000.0 [1]
	(1S)-3-Diethoxyphosphoryl-1-[(1R,2R,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]propan-1-ol	IC50	4000.0 [1]
	(1R)-2-Diethoxyphosphoryl-1-[(1R,2R,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]ethanol	IC50	10000.0 [1]
	(1R)-3-Diethoxyphosphoryl-1-[(1R,2R,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]propan-1-ol	IC50	5000.0 [1]
	(1S)-1-[(1R,2S,7S,8S,9S)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]propan-1-ol	IC50	500.0 [1]
	(1S)-1-[(1R,2S,7S,8S,9S)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]prop-2-en-1-ol	IC50	600.0 [1]
	(1S)-1-[(1R,2S,7S,8S,9S)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]but-3-en-1-ol	IC50	200.0 [1]
	(1R)-2-Methyl-1-[(1R,2S,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]propan-1-ol	IC50	400.0 [1]
	(1S)-2,2-Dimethyl-1-[(1R,2S,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]propan-1-ol	IC50	200.0 [1]
	(S)-Phenyl-[(1R,2S,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]methanol	IC50	900.0 [1]
	2-[(1R,2S,7R,8S,9R)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]ethanol	IC50	500.0 [1]
	4-[(1R,2S,7R,8S,9R)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]butan-1-ol	IC50	3000.0 [1]
	4-[(1R,2S,7R,8S,9R)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]butanoic acid	IC50	16000.0 [1]
	3-[(1R,2S,7R,8S,9R)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]propylphosphonic acid	IC50	32000.0 [1]
	(E)-3-[(1R,2S,7S,8S,9S)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]prop-2-en-1-ol	IC50	800.0 [1]
	(Z)-3-[(1R,2S,7S,8S,9S)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]prop-2-enoic acid	IC50	3000.0 [1]
	(3R)-3-Hydroxy-3-[(1R,2S,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]propanoic acid	IC50	900.0 [1]
	Ethyl (3R)-3-hydroxy-3-[(1R,2S,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]propanoate	IC50	400.0 [1]
	[(2S)-2-Hydroxy-2-[(1R,2S,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]ethyl]phosphonic acid	IC50	18000.0 [1]
	(1S)-2-Diethoxyphosphoryl-1-[(1R,2S,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]ethanol	IC50	10000.0 [1]
	[(3S)-3-Hydroxy-3-[(1R,2S,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]propyl]phosphonic acid	IC50	18000.0 [1]
	(1S)-3-Dimethoxyphosphoryl-1-[(1R,2S,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]propan-1-ol	IC50	4000.0 [1]
	(1S)-1-[(1R,2S,7S,8S,9S)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]propane-1,3-diol	IC50	300.0 [1]
	(1R)-1-[(1R,2S,7S,8S,9S)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]propan-1-ol	IC50	500.0 [1]
	(1R)-1-[(1R,2S,7S,8S,9S)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]prop-2-en-1-ol	IC50	300.0 [1]
	(1R)-1-[(1R,2S,7S,8S,9S)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]but-3-en-1-ol	IC50	400.0 [1]
	(1S)-2-Methyl-1-[(1R,2S,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]propan-1-ol	IC50	400.0 [1]
	(1R)-2,2-Dimethyl-1-[(1R,2S,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]propan-1-ol	IC50	800.0 [1]
	3-[(1R,2S,7R,8S,9R)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]propan-1-ol	IC50	900.0 [1]
	(Z)-3-[(1R,2S,7S,8S,9S)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]prop-2-en-1-ol	IC50	700.0 [1]
	3-[(1R,2S,7R,8S,9R)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]propanoic acid	IC50	2000.0 [1]
	(E)-3-[(1R,2S,7S,8S,9S)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]prop-2-enoic acid	IC50	3000.0 [1]
	2-[(1R,2S,7R,8S,9R)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]ethylphosphonic acid	IC50	12000.0 [1]
	[(E)-2-[(1R,2S,7S,8R,9S)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]ethenyl]phosphonic acid	IC50	8000.0 [1]
	[(E)-3-[(1R,2S,7R,8S,9R)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]prop-1-enyl]phosphonic acid	IC50	41000.0 [1]
	(3S)-3-Hydroxy-3-[(1R,2S,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]propanoic acid	IC50	1000.0 [1]
	Ethyl (3S)-3-hydroxy-3-[(1R,2S,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]propanoate	IC50	300.0 [1]
	[(2R)-2-Hydroxy-2-[(1R,2S,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]ethyl]phosphonic acid	IC50	13000.0 [1]
	[(3R)-3-Hydroxy-3-[(1R,2S,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]propyl]phosphonic acid	IC50	28000.0 [1]
	(1R)-3-Dimethoxyphosphoryl-1-[(1R,2S,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]propan-1-ol	IC50	3000.0 [1]
	(1R)-1-[(1R,2S,7S,8S,9S)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]propane-1,3-diol	IC50	200.0 [1]
	(1S)-2-Chloro-1-[(1R,2S,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]ethanol	IC50	200.0 [1]
	(1R)-2-Chloro-1-[(1R,2S,7S,8S,9S)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]ethanol	IC50	200.0 [1]
	(1R)-1-[(1R,2S,7S,8S,9S)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]ethanol	IC50	500.0 [1]
	(1S)-1-[(1R,2S,7S,8S,9S)-3,3,7-Trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]ethanol	IC50	700.0 [1]
	N,N-Dimethyl-2-[(1R,2S,7R,8S,9R)-3,3,7-trimethyl-8-tricyclo[5.4.0.02,9]undecanyl]ethanamine;hydrochloride	IC50	5000.0 [1]
	(Z)-4-[5-[(3,5-Difluorophenyl)methyl]-1-[(2-fluorophenyl)methyl]-2-oxopyridin-3-yl]-4-hydroxy-1-[4-(4-pyrrol-1-ylphenyl)piperazin-1-yl]but-3-ene-1,2-dione	IC50	300000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

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References

This online tool may be cited as follows

MLA	"Quest Database™ UDP-glucuronosyltransferase 2B7 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Nov. 2024, https://www.aatbio.com/data-sets/udp-glucuronosyltransferase-2b7-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, November 20). Quest Database™ UDP-glucuronosyltransferase 2B7 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/udp-glucuronosyltransferase-2b7-inhibitors-ic50-ki.
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