UDP-glucuronosyltransferase 1-1 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Levothyroxine	IC50	4900.0 [1], 5600.0 [2]
	Ethinyl estradiol	IC50	21000.0 [1], 44000.0 [2]
	Ketoconazole	IC50	13000.0 [1], 27000.0 [2]
	Ritonavir	IC50	1700.0 [1], 3000.0 [2]
	Carvedilol	IC50	12000.0 [1], 27000.0 [2]
	Daidzein	IC50	7300.0 [1], 120000.0 [2]
	Riluzole	IC50	160000.0 [1], 180000.0 [2]
	Baicalein	IC50	4400.0 [1], 7000.0 [2]
	Raltegravir	IC50	170000.0 [1], 190000.0 [2]
	4-Methylumbelliferone	IC50	100000.0 [1]
	1-Naphthol	IC50	240000.0 [1], 280000.0 [2]
	Niflumic acid	IC50	13000.0 [1], 53000.0 [2]
	Farnesol	IC50	40000.0 [1], 47000.0 [2]
	5-(4-Hydroxyphenyl)-5-phenylimidazolidine-2,4-dione	IC50	110000.0 [1], 120000.0 [2]
	2,6-Dihydroxyanthraquinone	IC50	3600.0 [1], 4000.0 [2]
	Irilone	Ki	8500.0 [1], 14100.0 [2]
	3-[5-(4-Cyclopentyloxy-2-hydroxybenzoyl)-2-[(3-oxo-1,2-benzoxazol-6-yl)methoxy]phenyl]propanoic acid	Ki	1540.0 [1], 4670.0 [2]
	Diclofenac	Ki	52000.0 [1]
	7-Ethyl-10-hydroxycamptothecin	IC50	360000.0 [1]
	Probenecid	Ki	221000.0 [1]
	Dolutegravir	IC50	100000.0 [1]
	Scutellarin	Ki	96600.0 [1]
	3-(5-Chloropyridin-2-yl)-5-(2-hydroxypropan-2-yl)-N-[(1R)-1-[1-oxido-6-(trifluoromethyl)pyridin-1-ium-3-yl]ethyl]benzamide	IC50	20000.0 [1]
	N-[(1R)-1-(5-Fluoropyridin-2-yl)ethyl]-3-(5-methylpyridin-2-yl)-5-[(5S)-5-pyridin-2-yl-4,5-dihydro-1,2-oxazol-3-yl]benzamide	IC50	1000.0 [1]
	(1S,4R,6S,7E,18S)-18-[7-Methoxy-8-methyl-2-[4-(trifluoromethyl)-1,3-thiazol-2-yl]quinolin-4-yl]oxy-13-methyl-N-(1-methylcyclopropyl)sulfonyl-2,14-dioxo-3,13,15-triazatricyclo[13.4.0.04,6]nonadec-7-ene-4-carboxamide	IC50	10000.0 [1]
	(Z)-4-[5-[(3,5-Difluorophenyl)methyl]-1-[(2-fluorophenyl)methyl]-2-oxopyridin-3-yl]-4-hydroxy-1-[4-(4-pyrrol-1-ylphenyl)piperazin-1-yl]but-3-ene-1,2-dione	IC50	300000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 26 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ UDP-glucuronosyltransferase 1-1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Nov. 2024, https://www.aatbio.com/data-sets/udp-glucuronosyltransferase-1-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, November 20). Quest Database™ UDP-glucuronosyltransferase 1-1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/udp-glucuronosyltransferase-1-1-inhibitors-ic50-ki.
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