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Tyrosine-protein phosphatase non-receptor type 5 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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▼
Standard Values (in nM)
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▼
8-(Trifluoromethyl)-1,2,3,4,5-benzopentathiepin-6-amine;hydrochlorideIC5024.6 [1], 8800.0 [2]
8-(Trifluoromethyl)-1,2,3,4,5-benzopentathiepin-6-amine;hydrochlorideKi115.0 [1]
2,2,2-Trifluoro-N-[8-(trifluoromethyl)-1,2,3,4,5-benzopentathiepin-6-yl]acetamideIC5024.0 [1], 15000.0 [2]
2,2,2-Trifluoro-N-[8-(trifluoromethyl)-1,2,3,4,5-benzopentathiepin-6-yl]acetamideKi235.0 [1]
N-[8-(Trifluoromethyl)-1,2,3,4,5-benzopentathiepin-6-yl]acetamideIC5049.0 [1], 24000.0 [2]
N-[8-(Trifluoromethyl)-1,2,3,4,5-benzopentathiepin-6-yl]acetamideKi123.0 [1]
N-Ethyl-8-(trifluoromethyl)-1,2,3,4,5-benzopentathiepin-6-amineIC5059.0 [1], 50000.0 [2]
N-Ethyl-8-(trifluoromethyl)-1,2,3,4,5-benzopentathiepin-6-amineKi230.0 [1]
N-Benzyl-8-(trifluoromethyl)-1,2,3,4,5-benzopentathiepin-6-amineIC5078.0 [1], 27000.0 [2]
N-Benzyl-8-(trifluoromethyl)-1,2,3,4,5-benzopentathiepin-6-amineKi175.0 [1]
4-Nitro-6-(trifluoromethyl)-1,2,3-benzotrithioleIC50145.0 [1], 34000.0 [2]
4-Nitro-6-(trifluoromethyl)-1,2,3-benzotrithioleKi210.0 [1]
7-(Trifluoromethyl)-1,2,3,4,5-benzopentathiepineIC5010.0 [1], 17000.0 [2]
7-(Trifluoromethyl)-1,2,3,4,5-benzopentathiepineKi109.0 [1]
8-Methyl-1,2,3,4,5-benzopentathiepin-6-amineIC5025.0 [1], 17000.0 [2]
8-Methyl-1,2,3,4,5-benzopentathiepin-6-amineKi116.0 [1]
1,2,3,4,5-Benzopentathiepin-6-amineIC5032.0 [1], 33000.0 [2]
1,2,3,4,5-Benzopentathiepin-6-amineKi183.0 [1]
8,17-Bis(trifluoromethyl)-2,3,4,11,12,13-hexathiatricyclo[12.4.0.05,10]octadeca-1(18),5,7,9,14,16-hexaene-6,15-diamineIC5033.0 [1], 20000.0 [2]
8,17-Bis(trifluoromethyl)-2,3,4,11,12,13-hexathiatricyclo[12.4.0.05,10]octadeca-1(18),5,7,9,14,16-hexaene-6,15-diamineKi124.0 [1]
[[4-[3-[(3,4-Dichlorophenyl)methyl]phenyl]phenyl]-difluoromethyl]phosphonic acidKi9600.0 [1]
[[4-[3-[(3,4-Dichlorophenyl)-hydroxymethyl]phenyl]phenyl]-difluoromethyl]phosphonic acidKi16000.0 [1]
5,7-Dichloro-4-((3-(4-methoxyphenylthio)benzyl)(methyl)amino)quinoline-2-carboxylic acidIC5060600.0 [1]
Biphenyl-4-yldifluoromethylphosphonic acidKi120000.0 [1]
3-Biphenylyldifluoromethylphosphonic acidKi337000.0 [1]
[[3-(3-Cyclohexyl-2-hydroxyphenyl)phenyl]-difluoromethyl]phosphonic acidKi20000.0 [1]
[(S)-[4-[3-[(R)-(3,4-Dichlorophenyl)-hydroxymethyl]phenyl]phenyl]-hydroxymethyl]phosphonic acidKi8900.0 [1]
[(S)-[4-[3-[(S)-(3,4-Dichlorophenyl)-hydroxymethyl]phenyl]phenyl]-hydroxymethyl]phosphonic acidKi7800.0 [1]
4-[[4-[(E)-[5-[4-(Dimethylamino)phenyl]-6-ethoxycarbonyl-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-2-ylidene]methyl]phenoxy]methyl]benzoic acidIC5016600.0 [1]
2-Hydroxy-4-[1-(cyclohexylcarbamoyl)pentyloxy]-5-[2-(trifluoromethoxy)phenylethynyl]benzoic acidIC5050000.0 [1]
[(R)-[4-[2-Fluoro-3-[(2,4,5-trichlorophenyl)methyl]phenyl]phenyl]-hydroxymethyl]phosphonic acidKi15000.0 [1]
[Difluoro-[4-[2-fluoro-3-[(2,4,5-trichlorophenyl)methyl]phenyl]phenyl]methyl]phosphonic acidKi2400.0 [1]
[2-Cyclohexyl-1-fluoro-1-[4-[2-fluoro-3-[(2,4,5-trichlorophenyl)methyl]phenyl]phenyl]-2-oxoethyl]phosphonic acidKi1000.0 [1]
[Difluoro-[4-[3-[(2,4,5-trichlorophenyl)methyl]phenyl]phenyl]methyl]phosphonic acidKi4700.0 [1]
[(S)-[4-[2-Fluoro-3-[(2,4,5-trichlorophenyl)methyl]phenyl]phenyl]-hydroxymethyl]phosphonic acidKi2600.0 [1]
[1-Fluoro-1-[4-[2-fluoro-3-[(2,4,5-trichlorophenyl)methyl]phenyl]phenyl]-2-oxo-2-piperidin-1-ylethyl]phosphonic acidKi3000.0 [1]
[2-(Dimethylamino)-1-[4-[2-fluoro-3-[(2,4,5-trichlorophenyl)methyl]phenyl]phenyl]-2-oxoethyl]phosphonic acidKi2400.0 [1]
[Fluoro-[4-[2-fluoro-3-[(2,4,5-trichlorophenyl)methyl]phenyl]phenyl]-morpholin-4-ylsulfonylmethyl]phosphonic acidKi110.0 [1]
[[4-[2-Fluoro-3-[(2,4,5-trichlorophenyl)methyl]phenyl]phenyl]-morpholin-4-ylsulfonylmethyl]phosphonic acidKi430.0 [1]
[1-[4-[2-Fluoro-3-[(2,4,5-trichlorophenyl)methyl]phenyl]phenyl]-2-(methylamino)-2-oxoethyl]phosphonic acidKi6800.0 [1]
[[4-[3-[(4,5-Dichloro-2-fluorophenyl)-hydroxymethyl]phenyl]phenyl]-difluoromethyl]phosphonic acidKi14000.0 [1]
[1-Fluoro-1-[4-[2-fluoro-3-[(2,4,5-trichlorophenyl)methyl]phenyl]phenyl]-2-oxo-2-phenylethyl]phosphonic acidKi540.0 [1]
[[4-[3-[(2-Bromo-4,5-dichlorophenyl)methyl]phenyl]phenyl]-difluoromethyl]phosphonic acidKi3700.0 [1]
[Difluoro-[4-[3-[hydroxy-(2,4,5-trichlorophenyl)methyl]phenyl]phenyl]methyl]phosphonic acidKi10000.0 [1]
[1-[4-[2-Fluoro-3-[(2,4,5-trichlorophenyl)methyl]phenyl]phenyl]-2-oxo-2-piperidin-1-ylethyl]phosphonic acidKi2700.0 [1]
[1-[4-[2-Fluoro-3-[(2,4,5-trichlorophenyl)methyl]phenyl]phenyl]-2-morpholin-4-yl-2-oxoethyl]phosphonic acidKi1700.0 [1]
[Fluoro-[4-[2-fluoro-3-[(2,4,5-trichlorophenyl)methyl]phenyl]phenyl]methyl]phosphonic acidKi1500.0 [1]
[[4-[3-[(4,5-Dichloro-2-fluorophenyl)methyl]phenyl]phenyl]-difluoromethyl]phosphonic acidKi5600.0 [1]
2-[[6-(1,3-Dioxoisoindol-2-yl)-1,3-benzothiazol-2-yl]sulfanyl]-N-[5-[(3-methylphenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]acetamideIC5096040.0 [1]
4-({4-[(E)-(1-Ethyl-2,5-dioxoimidazolidin-4-ylidene)methyl]-2-iodophenoxy}methyl)benzoic acidIC50100000.0 [1]
N-(4-Fluoro-1,3-benzothiazol-2-yl)-5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-amineIC50100000.0 [1]
[Difluoro-[3-(4-methylphenyl)phenyl]methyl]phosphonic acidKi205000.0 [1]
[Difluoro-[3-(4-propan-2-ylphenyl)phenyl]methyl]phosphonic acidKi222000.0 [1]
[Difluoro-[3-(3-methylphenyl)phenyl]methyl]phosphonic acidKi137000.0 [1]
[Difluoro-[3-(3-propan-2-ylphenyl)phenyl]methyl]phosphonic acidKi81000.0 [1]
[Difluoro-[3-(2-hydroxyphenyl)phenyl]methyl]phosphonic acidKi168000.0 [1]
[Difluoro-[3-(2-methoxyphenyl)phenyl]methyl]phosphonic acidKi271000.0 [1]
[Difluoro-[3-(2-hydroxy-3-propan-2-ylphenyl)phenyl]methyl]phosphonic acidKi69000.0 [1]
[Difluoro-[3-(2-hydroxy-5-propan-2-ylphenyl)phenyl]methyl]phosphonic acidKi95000.0 [1]
[[3-(3-Ethyl-2-hydroxyphenyl)phenyl]-difluoromethyl]phosphonic acidKi124000.0 [1]
[[3-(3-Tert-butyl-2-hydroxyphenyl)phenyl]-difluoromethyl]phosphonic acidKi63000.0 [1]
[[3-(3-Cyclobutyl-2-hydroxyphenyl)phenyl]-difluoromethyl]phosphonic acidKi45000.0 [1]
[[3-(3-Cyclopentyl-2-hydroxyphenyl)phenyl]-difluoromethyl]phosphonic acidKi25000.0 [1]
[[3-(3-Cycloheptyl-2-hydroxyphenyl)phenyl]-difluoromethyl]phosphonic acidKi62000.0 [1]
[[3-(3-Cyclohexyl-2-hydroxyphenyl)phenyl]-hydroxymethyl]phosphonic acidKi36000.0 [1]
[[4-(2-Cyanophenyl)phenyl]-difluoromethyl]phosphonic acidKi375000.0 [1]
[[4-(3-Cyanophenyl)phenyl]-difluoromethyl]phosphonic acidKi400000.0 [1]
[[4-(4-Cyanophenyl)phenyl]-difluoromethyl]phosphonic acidKi617000.0 [1]
[Difluoro-[4-(3-propan-2-yloxyphenyl)phenyl]methyl]phosphonic acidKi200000.0 [1]
[Difluoro-[4-(4-propan-2-yloxyphenyl)phenyl]methyl]phosphonic acidKi231000.0 [1]
[Difluoro-[4-(3-propan-2-ylphenyl)phenyl]methyl]phosphonic acidKi132000.0 [1]
[Difluoro-[4-(4-propan-2-ylphenyl)phenyl]methyl]phosphonic acidKi185000.0 [1]
[Difluoro-[4-[2-(methanesulfonamido)phenyl]phenyl]methyl]phosphonic acidKi673000.0 [1]
[Difluoro-[4-[3-(methanesulfonamido)phenyl]phenyl]methyl]phosphonic acidKi113000.0 [1]
[Difluoro-[4-[3-(1-hydroxyethyl)phenyl]phenyl]methyl]phosphonic acidKi88000.0 [1]
[Difluoro-[4-[4-(1-hydroxyethyl)phenyl]phenyl]methyl]phosphonic acidKi450000.0 [1]
[[4-(3-Anilinophenyl)phenyl]-difluoromethyl]phosphonic acidKi112000.0 [1]
[Difluoro-[4-[3-[(4-fluorophenyl)methyl]phenyl]phenyl]methyl]phosphonic acidKi35000.0 [1]
[[4-[3-[(4-Chlorophenyl)methyl]phenyl]phenyl]-difluoromethyl]phosphonic acidKi19000.0 [1]
[[4-[3-[(3,4-Dichlorophenyl)methyl]phenyl]phenyl]-hydroxymethyl]phosphonic acidKi8300.0 [1]
[[4-(3-Benzylphenyl)phenyl]-difluoromethyl]phosphonic acidKi73000.0 [1]
[(R)-[4-[3-[(R)-(3,4-Dichlorophenyl)-hydroxymethyl]phenyl]phenyl]-hydroxymethyl]phosphonic acidKi88000.0 [1]
[(R)-[4-[3-[(S)-(3,4-Dichlorophenyl)-hydroxymethyl]phenyl]phenyl]-hydroxymethyl]phosphonic acidKi93000.0 [1]
[4-[3-[(3,4-Dichlorophenyl)-hydroxymethyl]phenyl]phenyl]methylphosphonic acidKi97000.0 [1]
6-Hydroxy-3-iodo-1-methyl-2-[3-[[2-oxo-2-(4-thiophen-3-ylanilino)acetyl]amino]phenyl]indole-5-carboxylic acidIC504000.0 [1]
Items per page: 1 - 10 of 85
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References

This online tool may be cited as follows

MLA

"Quest Database™ Tyrosine-protein phosphatase non-receptor type 5 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/tyrosine-protein-phosphatase-non-receptor-type-5-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, November 21). Quest Database™ Tyrosine-protein phosphatase non-receptor type 5 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/tyrosine-protein-phosphatase-non-receptor-type-5-inhibitors-ic50-ki.
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