![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_34ec291e290db2e13648ccc8dee7e3a5.svg) | Cabozantinib | IC50 | 7.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_c77eb69f87d46b4d00314a6bfb851cf8.svg) | Crizotinib | IC50 | 1.0 [1], 100.0 [2], 294.0 [3], 300.0 [4] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_b5f9e60dc2b2b7e76e07307c1d8f7888.svg) | Bosutinib | IC50 | 174.0 [1], 340.0 [2], 560.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_21b312da3a0ca2e00016eafda80097df.svg) | Bemcentinib | IC50 | 0.7 [1], 14.0 [2], 30.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_473fafde5f65865ea7207466037e5614.svg) | 4-[2-(Butylamino)-5-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 1.65 [1], 14.0 [2], 122.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_0f4a04984ecf34abfddd13f4de2d16f4.svg) | 1-[(trans-4-Aminocyclohexyl)methyl]-N-Butyl-3-(4-Fluorophenyl)-1h-Pyrazolo[3,4-D]pyrimidin-6-Amine | IC50 | 37.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_1b4e021e73e18c4d77e61a14bc0121f0.svg) | 4-[5-[4-[(4-Methyl-1,4-diazepan-1-yl)methyl]phenyl]-2-[[(2S)-pentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 12.1 [1], 80.0 [2], 859.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 3.0 [1], 40.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_7de5848be93196a6906eba944a298431.svg) | Sunitinib | IC50 | 9.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_173905a1d8206fe6271a8ee9486c99d9.svg) | Foretinib | IC50 | 11.0 [1], 100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_e7ecb06887875f4d78baf892d82c33a5.svg) | Bms-777607 | IC50 | 1.1 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_3439230493a724d9f3f294065e2b89fc.svg) | Merestinib | IC50 | 2.0 [1], 11.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_5c51c2370d44a47470f8106e240be0b9.svg) | JNJ-28312141 free base | IC50 | 12.0 [1], 2600.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_176ecd1fb7b7bdf4a5a7674cda633952.svg) | c-FMS inhibitor | IC50 | 6.4 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_26823f4b402d0ef34901e1d6fee64cb6.svg) | CID 46194178 | IC50 | 10.0 [1], 500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_3675ea77fc19d393771a33a213dcb993.svg) | Exelixis | IC50 | 7.0 [1], 42.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_f35e91676c97c13abc32ca78f6dc0d85.svg) | CID 49870909 | IC50 | 7.0 [1], 56.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_a8c912344fec9d9cdfd3916574a57d57.svg) | CID 46870258 | IC50 | 58.0 [1], 1000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_b9bacc89876e00377722328a91c61513.svg) | 1-[(4-Aminocyclohexyl)methyl]-N-methyl-3-(4-piperazin-1-ylphenyl)pyrazolo[3,4-d]pyrimidin-6-amine | IC50 | 14.0 [1], 140.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_e0841b3388fd1dc0d3a8bcf12203d5a6.svg) | 6-[6-Amino-5-[(1R)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]pyridin-3-yl]-1'-methylspiro[1H-indole-3,4'-piperidine]-2-one | IC50 | 28.9 [1], 300000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_6a63a58acb1ce160573a1db1434b1f6d.svg) | 1-[(4-Aminocyclohexyl)methyl]-N-methyl-3-phenylpyrazolo[3,4-d]pyrimidin-6-amine | IC50 | 81.0 [1], 370.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_ffde2368846e99fcfbf9ca2c88012152.svg) | 4-[[6-(Methylamino)-3-phenylpyrazolo[3,4-d]pyrimidin-1-yl]methyl]cyclohexan-1-ol | IC50 | 83.0 [1], 190.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_2016e1fb48c552930d228a3e7f6e1433.svg) | Quercetin | IC50 | 960.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_0a83b01cf93719a90ccaeda771089c43.svg) | Doramapimod | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_6ce223fbd5241efea172edc836e9b6c1.svg) | Sotrastaurin | IC50 | 9100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_a257c791d1de1df5d4a1fa04612f9c76.svg) | Nvp-aew541 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_7e037c210cad9a24b0c9ce116fb5b97c.svg) | CID 53469448 | IC50 | 2705.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_d9312d16977155a14b08c6bd8c8b0132.svg) | Gilteritinib | IC50 | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_b9bd2d98b11bb07c7703bd6ad3510bbb.svg) | Amuvatinib | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_ad2e213c6bc5eb972596bba5a265d460.svg) | 1-(3-Chlorophenyl)-3-{5-[2-(Thieno[3,2-D]pyrimidin-4-Ylamino)ethyl]-1,3-Thiazol-2-Yl}urea | IC50 | 84.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_e0e66b7329f74ac9e778459370265f14.svg) | Norlichexanthone | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_5c7de9754b7b236c50ae4b7c0056fee4.svg) | TP-0903 | IC50 | 27.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_fe739739798d5a426922dc4c74a41375.svg) | (4S,6Z,9S,10S)-9,10,18-Trihydroxy-16-methoxy-4-methyl-3-oxabicyclo[12.4.0]octadeca-1(14),6,15,17-tetraene-2,8-dione | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_836d58634120a742d63c1602f26addff.svg) | CID 59604787 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_5fdad235d88d47467d429d2ef1d29e33.svg) | CID 44155856 | IC50 | 3.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_792fb9fb89419c9228e5974ac890efb7.svg) | Unii-T7755XP5Y6 | IC50 | 85.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_8fb35f27122721b8a0a25b7d7119f63d.svg) | 4-[[2-(Butylamino)-5-[5-(morpholin-4-ylmethyl)pyridin-2-yl]pyrimidin-4-yl]amino]cyclohexan-1-ol | IC50 | 270.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_c681437902b1c5f81123d723cc9476e0.svg) | R428 (BGB324; Bemcentinib) | IC50 | 14.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_da0d3b5102a55b7b2a2359d0105d93cb.svg) | CID 56847486 | IC50 | 19.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_5a8e321781069aee089dcc439066b321.svg) | 2,3,6,8-Tetrahydroxy-1-methylxanthone | IC50 | 6600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_5803643fba2a49f1581ea6790292d883.svg) | Epicoccolide B | IC50 | 220.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_d936f3dbad41727bd0deb9f9d3361e5f.svg) | 4-(5-Phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | IC50 | 182.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_62c354bc824a18213dbbccfcb95a065a.svg) | 3-N-[4-(4-Morpholin-4-ylcyclohexyl)phenyl]-1-pyridin-2-yl-1,2,4-triazole-3,5-diamine | Ki | 40.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_d72e6a5f6bda112109d526c400d3a392.svg) | Astrogorgiadiol B | IC50 | 16900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_d99325f173e26d7db80592089b850e5b.svg) | 2-(Butylamino)-4-[(4-hydroxycyclohexyl)amino]-N-[(4-imidazol-1-ylphenyl)methyl]pyrimidine-5-carboxamide | IC50 | 360.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_e24a6ef90b6dda81406d577957bafbf2.svg) | (1S,9R)-5,6,12,13,14-Pentahydroxy-4,11-dimethyl-16-oxo-8,17-dioxatetracyclo[7.7.1.02,7.010,15]heptadeca-2(7),3,5,10,12,14-hexaene-3-carbaldehyde | IC50 | 160.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_8547ec1c061a6923170866cf54d1c0d4.svg) | (1R,3As,4S,5R,7aR)-4-[2-(5-hydroxy-2-methylphenyl)ethyl]-7a-methyl-1-[(2R)-6-methyl-5-methylideneheptan-2-yl]-1,2,3,3a,4,5,6,7-octahydroinden-5-ol | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_9f0649c0af7300504c89d15a04caf360.svg) | Calicoferol B | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_628e796c331326ac7d59e9f8e229eaa5.svg) | 6,6-Dimethyl-8-[1-(oxan-4-ylmethyl)piperidin-4-yl]-11-oxo-5H-benzo[b]carbazole-3-carbonitrile | IC50 | 170.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_89f93b41ac7e8a2307bd8fc1d9fad8a4.svg) | Calicoferol E | IC50 | 32600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_3e70e51b426b206601dadb33b22bbf88.svg) | 2-Amino-N-[3-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]phenyl]acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_f64ae507fb96828f441cbfe1c221da9b.svg) | 1-[5-Amino-4-(3,4-dichlorophenyl)-3-methylpyrazol-1-yl]ethanone | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_f046ae8812a77e5cb35fd8b53bebf05d.svg) | Ripk1-IN-7 | IC50 | 35.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_dbc9774b4a10efc12e4d4309ee79f133.svg) | (13R,15S)-13-Methyl-16-oxa-8,9,12,22,24-pentazahexacyclo[15.6.2.16,9.112,15.02,7.021,25]heptacosa-1(24),2,4,6,17,19,21(25)-heptaene-23,27-dione | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_ec2afc1757433395b635cd30b7f7c89c.svg) | 8-(2,3-Dihydro-1H-inden-5-yl)-2-[4-(4-methylpiperazin-1-yl)anilino]-5-oxopyrido[2,3-d]pyrimidine-6-carboxamide | IC50 | 300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_9802efc27e72e36737af7825b3a8eda1.svg) | 8-(2,3-Dihydro-1H-inden-5-yl)-2-[4-[2-(4-methylpiperazin-1-yl)ethyl]anilino]-5-oxopyrido[2,3-d]pyrimidine-6-carboxamide | IC50 | 500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_ffa491388720238076ac7eccd6da397d.svg) | Methyl 1H-pyrrolo[2,3-b]pyridine-3-carboxylate | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_482caccce5577424472b4f30ef45663d.svg) | [6-Chloro-4-methyl-3-[[3-(methylsulfamoylamino)phenyl]methyl]-2-oxochromen-7-yl] N,N-dimethylcarbamate | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_826e6b90b3093494f22f4135571e56ab.svg) | 1-(2,6-Dichlorophenyl)-3-(6-(4-(2-(diethylamino)ethoxy)phenylamino)pyrimidin-4-yl)urea | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_a058bbc7d0f80bfd4a2414688d763f71.svg) | 3-Hydroxy-N-(2-hydroxy-1-methyl-ethyl)-5-(4-phenylamino-phenylamino)-isothiazole-4-carboxamidine | IC50 | 389.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_34a7749fa0ae5593ff30d6c21331df71.svg) | 3-(4-(1H-Tetrazol-5-yl)phenyl)-5-phenyl-1H-pyrrolo[2,3-b]pyridine | IC50 | 524.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_4af080018fcfdd3453abbbc05a2c39a3.svg) | N-[4-(6,7-Dimethoxyquinolin-4-yl)oxy-3-fluorophenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_400786f64062ecb5f10a9d3b11455207.svg) | 1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_bd7ab61fd74e87578c2dfefbcc47d031.svg) | 7,8-Dichloro-9-methyl-1-oxospiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_0f76e681b91255e37ea799fd5e965847.svg) | N-[5-[(Z)-(5-Fluoro-2-oxo-1H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrol-3-yl]-3-(4-methylpiperazin-1-yl)propanamide | Ki | 63.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_83e923e2811f5cd4e194d29630f84fbc.svg) | 3,5-Diphenyl-1H-pyrrolo[2,3-b]pyridine | IC50 | 4060.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_5c1c042b05f26ce92f172346c957e7d0.svg) | N-(7-Methoxyquinolin-6-yl)thieno[3,2-d]pyrimidine-7-carboxamide | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_0ca3e879b155ef6af0c4654d7cf4d922.svg) | 4-(Cyclopentylamino)-2-[(2-methoxyphenyl)methylamino]-N-[3-(2-oxopyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide | IC50 | 5700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_be6f7f8b06f86a492aec83c8596cec64.svg) | 4-(Cyclopentylamino)-2-[(2,5-dichlorophenyl)methylamino]-N-[3-(2-oxopyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide | IC50 | 3200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_25dd0b4f2746e9aaee1e0d2ca0362bc9.svg) | 4-(Cyclopentylamino)-2-[(2,5-dichlorophenyl)methylamino]-N-[3-(2-oxo-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide | IC50 | 3990.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_77f4b74dc836b9bdb4b558af6f5da27f.svg) | 6-(6-Fluoroindol-1-yl)-2-[2-[7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxyethyl]pyridazin-3-one | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_b48ec436f5a292f18e8fde779fde6c11.svg) | (7S)-7-Amino-N-[(4-fluorophenyl)methyl]-8-oxo-2,9,16,18,21-pentazabicyclo[15.3.1]henicosa-1(21),17,19-triene-20-carboxamide | IC50 | 120.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_f5abe3234d4b41fad1784bb6b6683e98.svg) | 5-[1-(Cyclopropylmethyl)-5-[(1R,5S)-3-(oxetan-3-yl)-3-azabicyclo[3.1.0]hexan-6-yl]pyrazol-3-yl]-3-(trifluoromethyl)pyridin-2-amine | IC50 | 448.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_70b0d2cbc054446af80b12d3d42fd894.svg) | (8S,16S)-3,16-Dihydroxy-9,10-seco-1,3,5(10)-cholestatrien-9-one | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_c67b754da3023ab057380dedf2f5a397.svg) | Calicoferol A | IC50 | 14700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_3ba3cfff437203d3cd5cef3fe6f6283a.svg) | (1R,3As,4S,7aR)-4-[2-(5-hydroxy-2-methylphenyl)ethyl]-7a-methyl-1-[(2R)-6-methyl-5-methylideneheptan-2-yl]-2,3,3a,4,6,7-hexahydro-1H-inden-5-one | IC50 | 20200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_744944dff0e05dbecbc6d3433ce3e640.svg) | 5-Phenyl-1H-pyrrolo[2,3-b]pyridine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_0b37fcadf8f90dc3bf2f29ca0be2a519.svg) | Methyl 3-[[(1R,2S,4aR,8aS)-1,2,4a,5-tetramethyl-2,3,4,7,8,8a-hexahydronaphthalen-1-yl]methyl]-4,5-dihydroxybenzoate | IC50 | 13100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_e79b9d9c36df2b44452606bd5a26f115.svg) | N-(1H-Pyrazol-5-yl)-1H-pyrrolo[2,3-b]pyridine-3-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_b9860f72a51c84f28c0f16192c41b8e7.svg) | N-Pyridin-3-yl-1H-pyrrolo[2,3-b]pyridine-3-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_617e98907525b08572f43e6444cefbb8.svg) | 5-Cyano-N-[2-(cyclohexen-1-yl)-4-[1-(2-methylsulfonylethyl)piperidin-4-yl]phenyl]-1H-imidazole-2-carboxamide | IC50 | 16.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_ec6b9c1a0d333fcceedfca28b3c6ddd2.svg) | 5-Cyano-N-[2-(cyclohexen-1-yl)-4-[1-(2-morpholin-4-ylethyl)piperidin-4-yl]phenyl]-1H-imidazole-2-carboxamide | IC50 | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_ca08212b911ff77e7266240517191aaf.svg) | 4-[5-[4-(Morpholin-4-ylmethyl)phenyl]-2-[[(2S)-pentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 218.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_f0a37a03c0093e032226113e49c1a05e.svg) | 4-[5-[3-[(4-Methylpiperazin-1-yl)methyl]phenyl]-2-[[(2S)-pentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 213.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_71c7e087d633f4e19f7daec405e54563.svg) | 4-[2-(Butylamino)-5-[4-(piperidin-4-ylamino)phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 42.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_0d98b4b226593ed7c0a8defd998755d1.svg) | 4-[5-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-2-[[(2R)-pentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 560.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_e392d737a0df7005ece96281df7cbe82.svg) | 4-[5-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-2-(pentan-2-ylamino)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 125.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_3f6518b869b2986e22f8da030a770263.svg) | 4-[2-[[(2S)-Heptan-2-yl]amino]-5-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 81.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_69b40bac9011556cd6dce5403e2715b4.svg) | 4-[5-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-2-[[(2S)-pentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 118.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_9c7d6e0a23eb7bfa3e5ed7b31b6be340.svg) | 4-[5-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-2-[[(2S)-1,1,1-trifluoropentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 11037.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_d05db671c729e40f8875ed38981dee9f.svg) | 4-[2-(2-Methylbutylamino)-5-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_07ab18d3db5057f9358cde6058c8e247.svg) | 4-[2-(2-Ethylbutylamino)-5-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 206.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_fcc4aed6b7459f36c0512afd232a74e6.svg) | 4-[5-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-2-[[(2R)-1,1,1-trifluoropentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 2543.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_ec209bc088d0fb656e0f2c34c5fe1073.svg) | 4-[2-[[(2S)-Hexan-2-yl]amino]-5-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 64.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_fb29fb1dee00965bf330db406b7e4be1.svg) | 4-[5-[4-[[2-(Diethylamino)ethylamino]methyl]phenyl]-2-[[(2S)-pentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 80.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_f8f0852d6a47a15276fb53b646bc7a21.svg) | 4-[2-[[(2S)-Pentan-2-yl]amino]-5-[4-(piperidin-4-ylamino)phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 206.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_448f1b5de31eb90a36c6fc2eb55d6cc9.svg) | 4-[5-[4-(Cyclohexylamino)phenyl]-2-[[(2S)-pentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 7356.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_97d47df88b3c08bf705bee1b72f3a8b2.svg) | 4-[5-[4-(7-Azabicyclo[2.2.1]heptan-7-ylmethyl)phenyl]-2-[[(2S)-pentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 84.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-ufo_d828f8c0f29b9de121301416f4615bf1.svg) | 4-[5-[2-Fluoro-4-(4-methylpiperazin-1-yl)sulfonylphenyl]-2-[[(2S)-pentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 191.0 [1] |