![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_473fafde5f65865ea7207466037e5614.svg) | 4-[2-(Butylamino)-5-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 5.83 [1], 17.0 [2], 301.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_c77eb69f87d46b4d00314a6bfb851cf8.svg) | Crizotinib | IC50 | 100.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_21b312da3a0ca2e00016eafda80097df.svg) | Bemcentinib | IC50 | 17.0 [1], 700.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_0f4a04984ecf34abfddd13f4de2d16f4.svg) | 1-[(trans-4-Aminocyclohexyl)methyl]-N-Butyl-3-(4-Fluorophenyl)-1h-Pyrazolo[3,4-D]pyrimidin-6-Amine | IC50 | 48.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_1b4e021e73e18c4d77e61a14bc0121f0.svg) | 4-[5-[4-[(4-Methyl-1,4-diazepan-1-yl)methyl]phenyl]-2-[[(2S)-pentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 3.1 [1], 9.1 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_c12c46d9f2e802f216d4a0500732451d.svg) | 3-Amino-N-(5-hydroxy-2-adamantyl)-6-[3-(1-methylpyrazol-4-yl)phenyl]pyrazine-2-carboxamide | IC50 | 20.0 [1], 40.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_0ca3e879b155ef6af0c4654d7cf4d922.svg) | 4-(Cyclopentylamino)-2-[(2-methoxyphenyl)methylamino]-N-[3-(2-oxopyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide | IC50 | 400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_be6f7f8b06f86a492aec83c8596cec64.svg) | 4-(Cyclopentylamino)-2-[(2,5-dichlorophenyl)methylamino]-N-[3-(2-oxopyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide | IC50 | 355.0 [1], 360.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_25dd0b4f2746e9aaee1e0d2ca0362bc9.svg) | 4-(Cyclopentylamino)-2-[(2,5-dichlorophenyl)methylamino]-N-[3-(2-oxo-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide | IC50 | 70.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_6a63a58acb1ce160573a1db1434b1f6d.svg) | 1-[(4-Aminocyclohexyl)methyl]-N-methyl-3-phenylpyrazolo[3,4-d]pyrimidin-6-amine | IC50 | 1400.0 [1], 4800.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_ffde2368846e99fcfbf9ca2c88012152.svg) | 4-[[6-(Methylamino)-3-phenylpyrazolo[3,4-d]pyrimidin-1-yl]methyl]cyclohexan-1-ol | IC50 | 2800.0 [1], 3500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_41ee610ec2a21757478bc91cf14f93d4.svg) | 3-Amino-N-(5-hydroxy-2-adamantyl)-6-[3-(methanesulfonamido)phenyl]pyrazine-2-carboxamide | IC50 | 380.0 [1], 650.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_bf3b0bcf96d03b37d07e0c6ba7fb7151.svg) | 3-Amino-N-(5-hydroxy-2-adamantyl)-6-[3-[1-(2-hydroxyethyl)pyrazol-4-yl]phenyl]pyrazine-2-carboxamide | IC50 | 60.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_88bce5b05668d6d00e4cd2797c4d73c1.svg) | 3-Amino-N-(5-hydroxy-2-adamantyl)-6-(1H-indazol-6-yl)pyrazine-2-carboxamide | IC50 | 100.0 [1], 180.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_b64412e385e07c34c480c0fc0075695b.svg) | 3-Amino-6-[3-(1-ethylpyrazol-4-yl)phenyl]-N-(5-hydroxy-2-adamantyl)pyrazine-2-carboxamide | IC50 | 20.0 [1], 30.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 48.99 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_e7ecb06887875f4d78baf892d82c33a5.svg) | Bms-777607 | IC50 | 4.3 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_836d58634120a742d63c1602f26addff.svg) | CID 59604787 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_68edb09c1caa9b3c2f0a46eeb28fe9e7.svg) | 2-{[(3r,4r)-3-Aminotetrahydro-2h-Pyran-4-Yl]amino}-4-[(4-Methylphenyl)amino]pyrimidine-5-Carboxamide | IC50 | 40.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_792fb9fb89419c9228e5974ac890efb7.svg) | Unii-T7755XP5Y6 | IC50 | 60.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_8fb35f27122721b8a0a25b7d7119f63d.svg) | 4-[[2-(Butylamino)-5-[5-(morpholin-4-ylmethyl)pyridin-2-yl]pyrimidin-4-yl]amino]cyclohexan-1-ol | IC50 | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_d99325f173e26d7db80592089b850e5b.svg) | 2-(Butylamino)-4-[(4-hydroxycyclohexyl)amino]-N-[(4-imidazol-1-ylphenyl)methyl]pyrimidine-5-carboxamide | IC50 | 250.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_628e796c331326ac7d59e9f8e229eaa5.svg) | 6,6-Dimethyl-8-[1-(oxan-4-ylmethyl)piperidin-4-yl]-11-oxo-5H-benzo[b]carbazole-3-carbonitrile | IC50 | 71.9 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_21aa752395444707db3d7c65ae53dc35.svg) | 1-({4-[(3,4-Dichlorophenyl)methoxy]phenyl}methyl)azetidine-3-carboxylic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_b076cdaba7bb8b7d9a4e8120c86a34a8.svg) | N-Propyl-4-({4-[(2,2,2-trifluoroethyl)amino]-1H-pyrrolo[2,3-d]pyrimidin-2-yl}amino)benzamide | IC50 | 1030.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_b9bacc89876e00377722328a91c61513.svg) | 1-[(4-Aminocyclohexyl)methyl]-N-methyl-3-(4-piperazin-1-ylphenyl)pyrazolo[3,4-d]pyrimidin-6-amine | IC50 | 260.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_ac2ac44cc6c324cb845a2c77f9c11dd1.svg) | CID 71553154 | IC50 | 0.7 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_77f4b74dc836b9bdb4b558af6f5da27f.svg) | 6-(6-Fluoroindol-1-yl)-2-[2-[7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxyethyl]pyridazin-3-one | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_b48ec436f5a292f18e8fde779fde6c11.svg) | (7S)-7-Amino-N-[(4-fluorophenyl)methyl]-8-oxo-2,9,16,18,21-pentazabicyclo[15.3.1]henicosa-1(21),17,19-triene-20-carboxamide | IC50 | 220.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_5b5057f07ba36d969b42e83280bc9205.svg) | 2-[3-(3-Piperidin-4-ylpropoxy)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_61551f1612b1d03b33f689e3fdae85ae.svg) | 2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_ca08212b911ff77e7266240517191aaf.svg) | 4-[5-[4-(Morpholin-4-ylmethyl)phenyl]-2-[[(2S)-pentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_f0a37a03c0093e032226113e49c1a05e.svg) | 4-[5-[3-[(4-Methylpiperazin-1-yl)methyl]phenyl]-2-[[(2S)-pentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 29.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_71c7e087d633f4e19f7daec405e54563.svg) | 4-[2-(Butylamino)-5-[4-(piperidin-4-ylamino)phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 34.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_0d98b4b226593ed7c0a8defd998755d1.svg) | 4-[5-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-2-[[(2R)-pentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 13.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_e392d737a0df7005ece96281df7cbe82.svg) | 4-[5-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-2-(pentan-2-ylamino)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 6.7 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_3f6518b869b2986e22f8da030a770263.svg) | 4-[2-[[(2S)-Heptan-2-yl]amino]-5-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 6.9 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_69b40bac9011556cd6dce5403e2715b4.svg) | 4-[5-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-2-[[(2S)-pentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 12.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_9c7d6e0a23eb7bfa3e5ed7b31b6be340.svg) | 4-[5-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-2-[[(2S)-1,1,1-trifluoropentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 151.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_d05db671c729e40f8875ed38981dee9f.svg) | 4-[2-(2-Methylbutylamino)-5-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 12.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_07ab18d3db5057f9358cde6058c8e247.svg) | 4-[2-(2-Ethylbutylamino)-5-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 6.7 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_fcc4aed6b7459f36c0512afd232a74e6.svg) | 4-[5-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-2-[[(2R)-1,1,1-trifluoropentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 99.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_ec209bc088d0fb656e0f2c34c5fe1073.svg) | 4-[2-[[(2S)-Hexan-2-yl]amino]-5-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 4.3 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_fb29fb1dee00965bf330db406b7e4be1.svg) | 4-[5-[4-[[2-(Diethylamino)ethylamino]methyl]phenyl]-2-[[(2S)-pentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 4.4 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_f8f0852d6a47a15276fb53b646bc7a21.svg) | 4-[2-[[(2S)-Pentan-2-yl]amino]-5-[4-(piperidin-4-ylamino)phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 26.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_448f1b5de31eb90a36c6fc2eb55d6cc9.svg) | 4-[5-[4-(Cyclohexylamino)phenyl]-2-[[(2S)-pentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 850.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_97d47df88b3c08bf705bee1b72f3a8b2.svg) | 4-[5-[4-(7-Azabicyclo[2.2.1]heptan-7-ylmethyl)phenyl]-2-[[(2S)-pentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 3.4 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_d828f8c0f29b9de121301416f4615bf1.svg) | 4-[5-[2-Fluoro-4-(4-methylpiperazin-1-yl)sulfonylphenyl]-2-[[(2S)-pentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 33.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_cb5f0d1b2973f214dbee47024fa34cd7.svg) | 4-[2-(Butylamino)-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 1662.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_397f9163ba8122b083e9cbde37ddfde5.svg) | 4-[2-(Butylamino)-5-[4-(4-methylpiperazin-1-yl)phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 22.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_0d0dd40987e4500a15c5e6b21d467eea.svg) | 2-Fluoro-4-[8-fluoro-3-(quinolin-6-ylmethyl)imidazo[1,2-a]pyridin-6-yl]-N-methylbenzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_07f245678e6fcc2d52455f8c1a6544d0.svg) | 2-[4-[4-[6-[(2R)-2-(3-Fluorophenyl)pyrrolidin-1-yl]imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl]piperazin-1-yl]acetic acid | IC50 | 5200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_cadcfe40c75731fb4d071e8664de359c.svg) | 1-[4-[6-[(2R)-2-(3-Fluorophenyl)pyrrolidin-1-yl]imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl]piperidin-4-ol | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_574a45544e8cb1fe403e1c65b194818e.svg) | 6-(1-Methylpyrazol-4-yl)-2-[[3-[[5-(1-methylpyrazol-4-yl)pyrimidin-2-yl]amino]phenyl]methyl]pyridazin-3-one | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_e021781d73f737111b72f54323b55bbc.svg) | 6-[Difluoro-[6-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b][1,2,4]triazin-3-yl]methyl]quinoline | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_f321563f2050b22443b36ad392046691.svg) | 18-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-1,13,15,21-tetrazatricyclo[12.5.2.017,20]henicosa-14,16,18,20-tetraen-5-ol | IC50 | 25.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_9c21d098deec5e6c52185677ffff5b57.svg) | 19-Pyridin-2-yl-1,14,16,22-tetrazatricyclo[13.5.2.018,21]docosa-15,17,19,21-tetraen-6-ol | IC50 | 690.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_6efa5aa571be54c31c8f10827b6a796b.svg) | 19-(4-Fluorophenyl)-1,14,16,22-tetrazatricyclo[13.5.2.018,21]docosa-15,17,19,21-tetraen-6-ol | IC50 | 1300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_99e4e4fd9611f62be4f84ef6cfbabe51.svg) | (6S)-6-Amino-20-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]-1,8,15,17,23-pentazatricyclo[14.5.2.019,22]tricosa-16,18,20,22-tetraen-7-one | IC50 | 13.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_3d9e0bc8095fe13405486889dde3d844.svg) | 19-(4-Methoxyphenyl)-1,14,16,22-tetrazatricyclo[13.5.2.018,21]docosa-15,17,19,21-tetraen-6-ol | IC50 | 940.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_89097c210eadebcd7eba31bc2ccf5b2a.svg) | 19-Pyridin-3-yl-1,14,16,22-tetrazatricyclo[13.5.2.018,21]docosa-15,17,19,21-tetraen-6-ol | IC50 | 210.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_5e3b26f4e6680b624c8728fb2dda19b2.svg) | 19-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-1,14,16,22-tetrazatricyclo[13.5.2.018,21]docosa-15,17,19,21-tetraen-6-ol | IC50 | 31.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_391d72f717d1d073f621f054573b77ee.svg) | 17-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-1,12,14,20-tetrazatricyclo[11.5.2.016,19]icosa-13,15,17,19-tetraen-6-ol | IC50 | 170.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_4cdc999f5b9a5c71f981787f87466777.svg) | 19-(Oxan-4-yl)-1,14,16,22-tetrazatricyclo[13.5.2.018,21]docosa-15,17,19,21-tetraen-6-ol | IC50 | 1200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_84406f33252ba2ecee2f206a4d3b48c0.svg) | N-[4-(6-Hydroxy-1,14,16,22-tetrazatricyclo[13.5.2.018,21]docosa-15,17,19,21-tetraen-19-yl)phenyl]morpholine-4-carboxamide | IC50 | 300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_e573219e22075aec56611920b5c1c117.svg) | 19-(3-Methoxyphenyl)-1,14,16,22-tetrazatricyclo[13.5.2.018,21]docosa-15,17,19,21-tetraen-6-ol | IC50 | 1200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_9e0d110e5c3728402277601f01fe0aaf.svg) | [4-(6-Hydroxy-1,14,16,22-tetrazatricyclo[13.5.2.018,21]docosa-15,17,19,21-tetraen-19-yl)phenyl]-morpholin-4-ylmethanone | IC50 | 78.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_efa67826d549f5fe42a8ebb13f352ae3.svg) | 19-Phenyl-1,14,16,22-tetrazatricyclo[13.5.2.018,21]docosa-15,17,19,21-tetraen-6-ol | IC50 | 1800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_e07833fb6bbcb26e09796569c62bc2e4.svg) | 18-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-1,13,15,21-tetrazatricyclo[12.5.2.017,20]henicosa-14,16,18,20-tetraen-6-ol | IC50 | 94.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_874118ef07efeb184a8861f8f7d18e0d.svg) | 19-(2-Methoxyphenyl)-1,14,16,22-tetrazatricyclo[13.5.2.018,21]docosa-15,17,19,21-tetraen-6-ol | IC50 | 1100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_d31156660b9b5f8aa1f68804b0626304.svg) | 19-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-1,14,16,22-tetrazatricyclo[13.5.2.018,21]docosa-15,17,19,21-tetraen-5-ol | IC50 | 54.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_5df64f7da6b5bea0970c7d60f44e71a7.svg) | 16-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-1,11,13,19-tetrazatricyclo[10.5.2.015,18]nonadeca-12,14,16,18-tetraen-5-ol | IC50 | 53.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_db2462e9c8f772c42accf349f478e852.svg) | 20-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-1,15,17,23-tetrazatricyclo[14.5.2.019,22]tricosa-16,18,20,22-tetraen-7-ol | IC50 | 38.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_7dca3992f1283c1998a2e8f1d7ec33fb.svg) | 16-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-1,6,11,13,19-pentazatricyclo[10.5.2.015,18]nonadeca-12,14,16,18-tetraen-5-one | IC50 | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_3d38eb673c9fa6ac01e8313ea9ebded9.svg) | 18-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-1,13,15,21-tetrazatricyclo[12.5.2.017,20]henicosa-14,16,18,20-tetraen-7-ol | IC50 | 57.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_e7e8a8958ceeb49a12a0397911119dd5.svg) | (5S)-5-Amino-19-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]-1,7,14,16,22-pentazatricyclo[13.5.2.018,21]docosa-15,17,19,21-tetraen-6-one | IC50 | 110.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_0d80a24a326a4d5dd49de22a3d6d640c.svg) | (6S)-6-Amino-22-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]-1,8,17,19,25-pentazatricyclo[16.5.2.021,24]pentacosa-18,20,22,24-tetraen-7-one | IC50 | 7.5 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_8d8cdd392f695ffe9ce576a2d6eefba2.svg) | 19-(4-Morpholin-4-ylsulfonylphenyl)-1,14,16,22-tetrazatricyclo[13.5.2.018,21]docosa-15,17,19,21-tetraen-6-ol | IC50 | 190.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_17db2c37dfbad193b3bd234483028eec.svg) | 20-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-1,15,17,23-tetrazatricyclo[14.5.2.019,22]tricosa-16,18,20,22-tetraen-6-ol | IC50 | 22.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_27b3197f55bd51b87a4126e1783b01fa.svg) | (5S)-5-Amino-21-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]-1,7,16,18,24-pentazatricyclo[15.5.2.020,23]tetracosa-17,19,21,23-tetraen-6-one | IC50 | 170.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_3adff58e1156e561ea64212ac12f244c.svg) | 19-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-1,14,16,22-tetrazatricyclo[13.5.2.018,21]docosa-15,17,19,21-tetraen-7-ol | IC50 | 44.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_cf7f65cf2823fea5bcf2a041ee50e9ca.svg) | (5S)-5-Amino-17-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]-1,7,12,14,20-pentazatricyclo[11.5.2.016,19]icosa-13,15,17,19-tetraen-6-one | IC50 | 39.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_b169db42fb55af1f5a47349db18a5a0c.svg) | 19-Pyridin-4-yl-1,14,16,22-tetrazatricyclo[13.5.2.018,21]docosa-15,17,19,21-tetraen-6-ol | IC50 | 170.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_3bed95974bc0edfb9c2376508c466b84.svg) | 19-(4-Morpholin-4-ylphenyl)-1,14,16,22-tetrazatricyclo[13.5.2.018,21]docosa-15,17,19,21-tetraen-6-ol | IC50 | 350.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_31517cda861ad2049c104298c694fd0b.svg) | (6S)-6-Amino-18-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]-1,8,13,15,21-pentazatricyclo[12.5.2.017,20]henicosa-14,16,18,20-tetraen-7-one | IC50 | 130.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_3e74bebfa448350f2468a9aad41e906d.svg) | 17-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-1,12,14,20-tetrazatricyclo[11.5.2.016,19]icosa-13,15,17,19-tetraen-5-ol | IC50 | 60.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_9c0c4c88aa4aa3f9529e1e9a6f7fe825.svg) | 19-[4-(Morpholin-4-ylmethyl)phenyl]-1,14,16,22-tetrazatricyclo[13.5.2.018,21]docosa-15,17,19,21-tetraen-6-ol | IC50 | 300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_05314cc548e3f5af464447b495d5aaa7.svg) | 21-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-1,16,18,24-tetrazatricyclo[15.5.2.020,23]tetracosa-17,19,21,23-tetraen-7-ol | IC50 | 49.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_25be3fc7aeabe3f032b08a388602acce.svg) | 4-Chloro-2-[5-[[(1R)-2-hydroxy-1-phenylethyl]amino]-3-isoquinolin-6-ylpyridin-2-yl]phenol | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_0b43927816ebbc9be13e6e44e4f9f2e1.svg) | 5,5-Dimethyl-8-[[4-(2,2,2-trifluoroethylamino)furo[3,2-d]pyrimidin-2-yl]amino]-1H-4,1-benzoxazepin-2-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_68cbe63d62204863632720dd1e248b65.svg) | 4-Fluoro-2-[5-[[(1R)-2-hydroxy-1-phenylethyl]amino]-3-(3-methyl-2H-indazol-5-yl)pyridin-2-yl]phenol | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_5dfd7bf06ab62aaaef4955ebb4ab716c.svg) | 5-Fluoro-2-[5-[[(1R)-2-hydroxy-1-phenylethyl]amino]-3-(3-methyl-2H-indazol-5-yl)pyridin-2-yl]phenol | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_bfd6b87cf089aa6a697f222ce580e253.svg) | 4-Chloro-2-[5-[[(1R)-2-hydroxy-1-phenylethyl]amino]-3-(3-methyl-2H-indazol-5-yl)pyridin-2-yl]phenol | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_99e2c6cd0c29fa0c48ca6f47857abde2.svg) | 4-[2-[[(2R)-1-Hydroxyhexan-2-yl]amino]-5-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 143.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_6225554c86e626355502b672461bd8e7.svg) | 1-(Cyclopentylmethyl)-3-[6-(4-ethylpiperazin-1-yl)pyridin-3-yl]-N-methylpyrazolo[3,4-d]pyrimidin-6-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_804245a07134eab2aa9f2f49b61841f9.svg) | 1-[(1-Benzyltriazol-4-yl)methyl]-N-methyl-3-(4-piperazin-1-ylphenyl)pyrazolo[3,4-d]pyrimidin-6-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_6d6b86df4ac117182e566deac77d9c71.svg) | 1-(Cyclopentylmethyl)-N-methyl-3-(6-piperazin-1-ylpyridin-3-yl)pyrazolo[3,4-d]pyrimidin-6-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_6e59ddd56e164ec59ff518b6817be23b.svg) | 1-[(1-Benzyltriazol-4-yl)methyl]-N-methyl-3-(6-piperazin-1-ylpyridin-3-yl)pyrazolo[3,4-d]pyrimidin-6-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-tyro3_f61de99a5a6e0088b291b23c7245c4b7.svg) | 1-(Cyclopentylmethyl)-N-methyl-3-[6-(4-methylpiperazin-1-yl)pyridin-3-yl]pyrazolo[3,4-d]pyrimidin-6-amine | IC50 | 3670.0 [1] |