![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_1575317431cf6bb218d1789cccd6e0ea.svg) | Quizartinib | IC50 | 39.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_c8494007663098abb5d227cb27cc738b.svg) | Sorafenib | IC50 | 33.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_7de5848be93196a6906eba944a298431.svg) | Sunitinib | IC50 | 9.9 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_9a52b202d60d4e94b9b65b18a6931448.svg) | N-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-4-(thieno[2,3-d]pyrimidin-4-ylamino)-1H-pyrazole-5-carboxamide | IC50 | 1.85 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_4ee8632c180d42f14a1148faf37622c7.svg) | Tandutinib | IC50 | 102.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_1154e00f808447364900da7327ac72d1.svg) | 4-[(2-Methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)amino]-N-(4-piperazin-1-ylphenyl)-1H-pyrazole-5-carboxamide | IC50 | 8.74 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_4e38800d1c310079b3b3e65c5db78d0d.svg) | Linifanib | IC50 | 7.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_5bf6e56bbc335740215e09fe8aeecee1.svg) | 3-[1-[3-(Dimethylamino)propyl]pyrazol-4-yl]-7-(1H-pyrazol-4-yl)-5H-indeno[1,2-b]indol-10-one | IC50 | 4.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_34ec291e290db2e13648ccc8dee7e3a5.svg) | Cabozantinib | IC50 | 6.0 [1], 11.3 [2], 25.0 [3], 7500.0 [4] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_2060f6287083a28c9ead968a2460ede5.svg) | Tozasertib | IC50 | 30.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_2060f6287083a28c9ead968a2460ede5.svg) | Tozasertib | Ki | 30.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_d5b9a5aa59f0f55db22a25d2e6011f3c.svg) | Lestaurtinib | IC50 | 1.5 [1], 2.5 [2], 2.6 [3], 5.0 [4], 8.2 [5] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_173905a1d8206fe6271a8ee9486c99d9.svg) | Foretinib | IC50 | 3.6 [1], 5.58 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_62c354bc824a18213dbbccfcb95a065a.svg) | 3-N-[4-(4-Morpholin-4-ylcyclohexyl)phenyl]-1-pyridin-2-yl-1,2,4-triazole-3,5-diamine | IC50 | 1.3 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_62c354bc824a18213dbbccfcb95a065a.svg) | 3-N-[4-(4-Morpholin-4-ylcyclohexyl)phenyl]-1-pyridin-2-yl-1,2,4-triazole-3,5-diamine | Ki | 0.17 [1], 2.0 [2], 5.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_5c152aca39bcabd0fbf040aca395c590.svg) | 1-[4-Chloro-3-(trifluoromethyl)phenyl]-3-[4-(1H-pyrazolo[3,4-d]pyrimidin-4-yloxy)phenyl]urea | IC50 | 1.0 [1], 3.0 [2], 4.0 [3], 39.0 [4] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_a43a739a10eb2a01ac6e315a0c33b8da.svg) | 1-(5-Ethyl-1,2-oxazol-3-yl)-3-[4-[2-[[6-(4-ethylpiperazin-1-yl)-2-methylpyrimidin-4-yl]amino]-1,3-thiazol-5-yl]phenyl]urea | IC50 | 10.0 [1], 38.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_fe739739798d5a426922dc4c74a41375.svg) | (4S,6Z,9S,10S)-9,10,18-Trihydroxy-16-methoxy-4-methyl-3-oxabicyclo[12.4.0]octadeca-1(14),6,15,17-tetraene-2,8-dione | IC50 | 1.59 [1], 11.0 [2], 36.0 [3], 62.0 [4] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_ac9e30b723e2c9bf1debc2a45966acbb.svg) | 3-(1H-Indol-3-yl)-4-(3,4,5-trimethoxyphenyl)pyrrole-2,5-dione | IC50 | 18.0 [1], 166.0 [2], 270.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_55619603be8f6245d7236aed5771fc57.svg) | Flt-3 Inhibitor II | IC50 | 33.0 [1], 40.0 [2], 100.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_ba5a8e5214016d7ee25d82822d4987e5.svg) | 1-[(5,6-Dimethyl-2-thiophen-2-ylthieno[2,3-d]pyrimidin-4-yl)amino]-3-methylpyrrole-2,5-dione | IC50 | 11.38 [1], 13.68 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_ad5ee8a0243e92c9a1c5708abac9fbc1.svg) | 1-[[6-(Hydroxymethyl)-5-methyl-2-thiophen-2-ylthieno[2,3-d]pyrimidin-4-yl]amino]-3-methylpyrrole-2,5-dione | IC50 | 91.23 [1], 112.0 [2], 156.0 [3], 175.0 [4] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_d82fab1028f4e0de22d7e5370ed8f8b9.svg) | 4-N-(3,5-Dimethoxyphenyl)-4-N-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-1-N-propan-2-ylcyclohexane-1,4-diamine | IC50 | 3801.89 [1], 5370.32 [2], 8511.38 [3], 10000.0 [4] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_e46c2aed0fe6a75bbf9f67ad96920326.svg) | 3-Methyl-1-[[5-methyl-6-[4-[2-(methylamino)ethoxy]phenyl]-2-thiophen-2-ylthieno[2,3-d]pyrimidin-4-yl]amino]pyrrole-2,5-dione | IC50 | 8.03 [1], 10.15 [2], 11.1 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_b0aae8da0213ea09e5fa4e2429d9e2e7.svg) | Palbociclib | IC50 | 3000.0 [1], 3480.0 [2], 10000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_34f4790e2343c1a554bba4bf5edc6ba5.svg) | Midostaurin | IC50 | 13.0 [1], 15.0 [2], 37.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_c38cbdee4404993837adfc282c860ec1.svg) | Nvp-tae 684 | IC50 | 3.0 [1], 554.0 [2], 3000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_21b312da3a0ca2e00016eafda80097df.svg) | Bemcentinib | IC50 | 0.9 [1], 2.0 [2], 6.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_2de598172b9c7c6d2c3bb7d3509db05c.svg) | (16E)-14-Methyl-20-oxa-5,7,14,27-tetrazatetracyclo[19.3.1.12,6.18,12]heptacosa-1(25),2(27),3,5,8,10,12(26),16,21,23-decaene | IC50 | 21.0 [1], 42.0 [2], 56.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_a2d32a1f7c79660a88d646bbda5ee232.svg) | 4-Methyl-5-(2-((4-morpholinophenyl)amino)-pyrimidin-4-yl)thiazol-2-amine | IC50 | 25.12 [1], 88.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_a2d32a1f7c79660a88d646bbda5ee232.svg) | 4-Methyl-5-(2-((4-morpholinophenyl)amino)-pyrimidin-4-yl)thiazol-2-amine | Ki | 44.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_473fafde5f65865ea7207466037e5614.svg) | 4-[2-(Butylamino)-5-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 0.35 [1], 0.8 [2], 14.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_7cab6c6a39b70d94e7351afdd4bac5b6.svg) | Amg-925 | IC50 | 1.0 [1], 1.5 [2], 5.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_1b4e021e73e18c4d77e61a14bc0121f0.svg) | 4-[5-[4-[(4-Methyl-1,4-diazepan-1-yl)methyl]phenyl]-2-[[(2S)-pentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 2.5 [1], 39.0 [2], 70.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_2da2a4adb73557432dd9443d0e23f9f9.svg) | Flt3-IN-3 | IC50 | 3.0 [1], 8.0 [2], 13.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_a412c971baf636a384fa53e9f26decf0.svg) | 2-N-(4-Aminocyclohexyl)-9-cyclopentyl-6-N-(4-morpholin-4-ylphenyl)purine-2,6-diamine | IC50 | 2.0 [1], 7.0 [2], 21.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_5b587fbf3c1f97125b8ebd4d0d5f15d5.svg) | Propan-2-yl 2-hydroxy-4-methoxy-6-[(E)-3-(prop-2-enoylamino)prop-1-enyl]benzoate | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_52ffb2bafcaf260cf2564f177ef35b65.svg) | Propan-2-yl 4-[2-(4-fluorophenyl)ethoxy]-2-hydroxy-6-[(E)-3-(prop-2-enoylamino)prop-1-enyl]benzoate | IC50 | 8310.0 [1], 30000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_70947d0e5fd859b6eb1c3a5c9c3a9db4.svg) | Propan-2-yl 2-hydroxy-4-(3-morpholin-4-ylpropoxy)-6-[(E)-3-(prop-2-enoylamino)prop-1-enyl]benzoate | IC50 | 500.0 [1], 2810.0 [2], 9610.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_3a97978024dda0074bc093125b9fea3d.svg) | Propan-2-yl 2-[(E)-3-[[(E)-4-(diethylamino)but-2-enoyl]amino]prop-1-enyl]-4-[2-(4-fluorophenyl)ethoxy]-6-hydroxybenzoate | IC50 | 1110.0 [1], 30000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_f0184d3cd9595acb7ae60a8a3f75ab4e.svg) | Propan-2-yl 2-[(E)-3-(ethenylsulfonylamino)prop-1-enyl]-6-hydroxy-4-methoxybenzoate | IC50 | 2250.0 [1], 10820.0 [2], 12030.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_e7da067858ad859958103c5e7a14294c.svg) | Propan-2-yl 2-[3-(ethenylsulfonylamino)propyl]-6-hydroxy-4-(2-morpholin-4-ylethoxy)benzoate | IC50 | 4230.0 [1], 18590.0 [2], 30000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_a20baa4afcfe03aa85dc1829f5db4b7b.svg) | (4-Bromophenyl)methyl 2-[(E)-3-(ethenylsulfonylamino)prop-1-enyl]-6-hydroxy-4-methoxybenzoate | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_c602265891dda1d13acf8355e31271eb.svg) | (4-Fluorophenyl)methyl 2-[(E)-3-(ethenylsulfonylamino)prop-1-enyl]-6-hydroxy-4-methoxybenzoate | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_73532b6d2befe930d6c54863d276b3ed.svg) | Cyclohexylmethyl 2-[(E)-3-(ethenylsulfonylamino)prop-1-enyl]-6-hydroxy-4-methoxybenzoate | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_3973affcb0079621455b11a866f995b8.svg) | 2-Phenylpropyl 2-[(E)-3-(ethenylsulfonylamino)prop-1-enyl]-6-hydroxy-4-methoxybenzoate | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_ce53d802a61c5df3adca231b6dca221a.svg) | Propan-2-yl 2-acetyloxy-6-[(E)-3-(2,5-dioxopyrrol-1-yl)prop-1-enyl]-4-methoxybenzoate | IC50 | 3370.0 [1], 3610.0 [2], 21800.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_3aaaf8a85787f1b86e04645e70869194.svg) | Propan-2-yl 2-[(E)-3-(2,5-dioxopyrrol-1-yl)prop-1-enyl]-6-hydroxy-4-methoxybenzoate | IC50 | 540.0 [1], 1340.0 [2], 9790.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_50bd749f6f5eb770e1fcc63b59653470.svg) | Propan-2-yl 2-[3-(2,5-dioxopyrrol-1-yl)propyl]-6-hydroxy-4-methoxybenzoate | IC50 | 430.0 [1], 3030.0 [2], 13180.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_931df31577ac3d4d2e300a7189a84242.svg) | Propan-2-yl 2-[(E)-3-(2,5-dioxopyrrol-1-yl)prop-1-enyl]-6-hydroxy-4-(3-morpholin-4-ylpropoxy)benzoate | IC50 | 150.0 [1], 940.0 [2], 980.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_14b9eba81e4f8b75b513560d47029a00.svg) | Propan-2-yl 2-[3-(2,5-dioxopyrrol-1-yl)propyl]-6-hydroxy-4-(2-morpholin-4-ylethoxy)benzoate | IC50 | 580.0 [1], 810.0 [2], 8870.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_d387566544303e59df08fc796e37fb3c.svg) | (4-Bromophenyl)methyl 2-[(E)-3-(2,5-dioxopyrrol-1-yl)prop-1-enyl]-6-hydroxy-4-methoxybenzoate | IC50 | 1740.0 [1], 1900.0 [2], 30000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_c5762f29ea41617d122187f9e4e63897.svg) | (4-Fluorophenyl)methyl 2-[(E)-3-(2,5-dioxopyrrol-1-yl)prop-1-enyl]-6-hydroxy-4-methoxybenzoate | IC50 | 950.0 [1], 1640.0 [2], 30000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_6e6e8625407fe89c988efcbc317865d2.svg) | Cyclohexylmethyl 2-[(E)-3-(2,5-dioxopyrrol-1-yl)prop-1-enyl]-6-hydroxy-4-methoxybenzoate | IC50 | 2100.0 [1], 2690.0 [2], 30000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_0f270530e5cf6838f253c75eeb5cfeed.svg) | 2-Phenylpropyl 2-[(E)-3-(2,5-dioxopyrrol-1-yl)prop-1-enyl]-6-hydroxy-4-methoxybenzoate | IC50 | 3010.0 [1], 5200.0 [2], 30000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_16dc2d11b5b0c36c40c2295f2ea6e947.svg) | Propan-2-yl 2-[(E)-3-[[(E)-but-2-enoyl]amino]prop-1-enyl]-6-hydroxy-4-methoxybenzoate | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_61cb9b4a5865b586be03c31f4efc95f5.svg) | Propan-2-yl 2-[(E)-3-[[(E)-but-2-enoyl]amino]prop-1-enyl]-4-[2-(4-fluorophenyl)ethoxy]-6-hydroxybenzoate | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_7258ad0b0f41be9fe9f68b6952f49097.svg) | [(2S)-3-Methylbutan-2-yl] 2-hydroxy-4-methoxy-6-[(E)-3-(prop-2-enoylamino)prop-1-enyl]benzoate | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_eafa65673632ba3dfab124e4491e3e59.svg) | [(2S)-3-Methylbutan-2-yl] 2-[(E)-3-[[(E)-4-(diethylamino)but-2-enoyl]amino]prop-1-enyl]-6-hydroxy-4-methoxybenzoate | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_24c66235e711ba44f63918dd534d0597.svg) | 2-N-(5-Aminopentyl)-9-cyclopentyl-6-N-[4-(morpholin-4-ylmethyl)phenyl]purine-2,6-diamine | IC50 | 5.0 [1], 25.0 [2], 65.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_9fab6b2add9b790e78d9c162dfe1aa9d.svg) | 2-N-(4-Aminocyclohexyl)-9-cyclopentyl-6-N-(4-pyrrolidin-1-ylphenyl)purine-2,6-diamine | IC50 | 3.0 [1], 11.0 [2], 21.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_7d54d0066eda8d11cb4cb75917cfaff2.svg) | 2-N-(4-Aminobutyl)-9-cyclopentyl-6-N-(4-morpholin-4-ylphenyl)purine-2,6-diamine | IC50 | 4.0 [1], 7.0 [2], 23.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_33fddaae2b44f56dc4a092db995fd577.svg) | 2-N-(6-Aminohexyl)-9-cyclopentyl-6-N-[4-(morpholin-4-ylmethyl)phenyl]purine-2,6-diamine | IC50 | 10.0 [1], 21.0 [2], 69.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_30d5424edff1427f29fa738ec7c2af5f.svg) | 2-N-(4-Aminobutyl)-9-cyclopentyl-6-N-[4-(morpholin-4-ylmethyl)phenyl]purine-2,6-diamine | IC50 | 1.0 [1], 5.0 [2], 6.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_f61de99a5a6e0088b291b23c7245c4b7.svg) | 1-(Cyclopentylmethyl)-N-methyl-3-[6-(4-methylpiperazin-1-yl)pyridin-3-yl]pyrazolo[3,4-d]pyrimidin-6-amine | IC50 | 8.0 [1], 12.0 [2], 30.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_de10835b408d1a3225272d91f6124fbd.svg) | 2-N-Benzyl-9-cyclopentyl-6-N-[4-(morpholin-4-ylmethyl)phenyl]purine-2,6-diamine | IC50 | 26.0 [1], 83.0 [2], 624.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_fb7e1444d0095289928e9bf275b495bc.svg) | 2-N-(4-Aminobutyl)-9-cyclopentyl-6-N-[4-(4-ethylpiperazin-1-yl)phenyl]purine-2,6-diamine | IC50 | 1.0 [1], 3.0 [2], 13.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_accea8a38b341a6dfbd42231f4ee1e19.svg) | 1-(Cyclopentylmethyl)-N-methyl-3-[4-(4-methylpiperazin-1-yl)phenyl]pyrazolo[3,4-d]pyrimidin-6-amine | IC50 | 1.4 [1], 4.0 [2], 11.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_458e0fbda926923da1736178630182b6.svg) | 2-N-(4-Aminocyclohexyl)-9-cyclopentyl-6-N-[4-(2-oxa-6-azaspiro[3.3]heptan-6-yl)phenyl]purine-2,6-diamine | IC50 | 4.0 [1], 13.0 [2], 28.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_8b0fecf7a4be4bd132100a115c34c877.svg) | 2-N-(4-Aminocyclohexyl)-6-N-(4-bromophenyl)-9-cyclopentylpurine-2,6-diamine | IC50 | 4.0 [1], 16.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_0c1c48d6a1fb5d1ae68880d28c6457f7.svg) | 2-N-(4-Aminocyclohexyl)-9-cyclopentyl-6-N-[4-(4-ethylpiperazin-1-yl)phenyl]purine-2,6-diamine | IC50 | 2.0 [1], 3.0 [2], 10.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_03e0d1a2e88126708ed3a73e7e36755b.svg) | N-[5-[6-(Methylamino)pyrazin-2-yl]-2-oxo-1H-pyridin-3-yl]-4-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]benzamide | Ki | 20.0 [1], 1000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_cad00bfc972060df433644e94524c467.svg) | 5-Fluoro-3-[[4-[2-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]ethoxy]-3-methylazulen-1-yl]methylidene]-1H-indol-2-one | IC50 | 67.0 [1], 70.0 [2], 98.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_f24a27aabd40d91f43493e56a7da4ba1.svg) | N-[5-[4-[[(5-Tert-butyl-1,2-oxazol-3-yl)carbamoylamino]methyl]phenyl]-1H-pyrazol-3-yl]-4-(2-morpholin-4-ylethoxy)benzamide | IC50 | 1.0 [1], 18.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_8edb893ba88c5700603edef201da4265.svg) | Nintedanib | IC50 | 26.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_295456cbf7462dfb1eaccb88d6610904.svg) | Ceritinib | IC50 | 60.0 [1], 3143.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_47d151d561f848592c41ab2966c047a4.svg) | Dovitinib | IC50 | 1.0 [1], 3.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_b9eaaf091dbd9cf8d3bb931a4b80c14f.svg) | Pexidartinib | IC50 | 5.0 [1], 130.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_e98e38f8f3edf8be20fec1223eba919f.svg) | 6,7-Dimethyl-2-phenylquinoxaline | IC50 | 1100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_1369612825d9c926449f3546840889ff.svg) | Crenolanib | IC50 | 3.0 [1], 4.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_e7ecb06887875f4d78baf892d82c33a5.svg) | Bms-777607 | IC50 | 16.0 [1], 18.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_fa37ae125bcd4e6df1af4be57fbea491.svg) | 1-Cyclopropyl-3-(3-(5-(morpholinomethyl)-1H-benzo[d]imidazol-2-yl)-1H-pyrazol-4-yl)urea | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_2cf324237228e1f753214eb9a2ce619a.svg) | Erdafitinib | IC50 | 5.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_5a195f14ee440a5b4ba476435d82989d.svg) | KW-2449 | IC50 | 13.1 [1], 14.8 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_4e8b5202a71aafe003ab207cc4576058.svg) | 3-(1H-Indol-5-yl)-5-(4-((4-methylpiperazin-1-yl)methyl)phenyl)-1H-pyrrolo[2,3-b]pyridine | IC50 | 4.0 [1], 560.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_5c51c2370d44a47470f8106e240be0b9.svg) | JNJ-28312141 free base | IC50 | 21.0 [1], 30.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_02cf835f99d3cd203b60d49cf2af128d.svg) | Flt-3 inhibitor | IC50 | 42.0 [1], 2900.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_eafced04fef738ebffddbab9151e6f26.svg) | CID 44545852 | IC50 | 134.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_81451b6325bdc51ecc91d525cf1e5a78.svg) | Mivavotinib | IC50 | 4.6 [1], 22.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_3ee7568a09840225cd8af9a1f5126d5a.svg) | Tafetinib | IC50 | 1.3 [1], 5.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_7ba2c79d04a961439347046220210c11.svg) | 2-(4-((6,7-Dimethoxyquinazolin-4-yl)oxy)phenyl)-N-(1-isopropyl-1H-pyrazol-4-yl)acetamide | IC50 | 7.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_020a881748307fc93e2c40bec206b4bc.svg) | 11-(2-Pyrrolidin-1-ylethoxy)-14,19-dioxa-5,7,27-triazatetracyclo[19.3.1.12,6.18,12]heptacosa-1(24),2(27),3,5,8(26),9,11,16,21(25),22-decaene | IC50 | 6.0 [1], 22.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_6796b3172393b6fe2a8eec6cf8639fd1.svg) | 2-(6,7-Dimethoxyquinazolin-4-yl)sulfanyl-1,3-thiazole | IC50 | 7.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_66ee537084332a28fb4fd921d6adf367.svg) | CID 56673651 | IC50 | 11.0 [1], 13.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_a3bb3a5f0dd6cc174d624dfab74909ff.svg) | 2-[4-[(6,7-Dimethoxyquinazolin-4-yl)amino]phenyl]-N-(1-propan-2-ylpyrazol-4-yl)acetamide | IC50 | 20.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_4ccde7f7c200706c01de15dc0bb3d959.svg) | N-Phenyl-1H-indazole-3-carboxamide | IC50 | 350.0 [1], 417.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_7c37f197a24ee22101cd0cdabb3b7082.svg) | 2-[[4-[4-Amino-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]amino]acetic acid | IC50 | 28.0 [1], 32.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_7f169650bc883b9a2002ab81188c57b7.svg) | (2S)-2-[[4-[4-Amino-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]amino]-4-methylpentanoic acid | IC50 | 14.0 [1], 23.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-receptor-flt3_6fa3b0a74a6da88ea2b85feb2b54c0d3.svg) | 3-Methyl-1-[(6-methyl-2-thiophen-2-ylthieno[2,3-d]pyrimidin-4-yl)amino]pyrrole-2,5-dione | IC50 | 14.66 [1], 16.78 [2] |