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Tyrosine-protein kinase FYN Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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▼
StaurosporineIC5015.0 [1]
Rosmarinic acidIC5017000.0 [1]
Rosmarinic acidKi7500.0 [1], 10200.0 [2]
DoramapimodIC501000.0 [1], 20000.0 [2], 24000.0 [3], 30000.0 [4]
4-[(3-Bromophenyl)amino]-6-acrylamidoquinazolineIC501.0 [1], 42.0 [2], 420.0 [3], 300000.0 [4]
N-(4-Phenylamino-Quinazolin-6-Yl)-AcrylamideIC505.0 [1], 6.0 [2], 1100.0 [3], 3700.0 [4]
N-(4-(4-Tert-Butylphenylamino)quinazolin-6-yl)acrylamideIC5024.0 [1], 900.0 [2], 8400.0 [3], 300000.0 [4]
N-(4-(4-Bromophenylamino)quinazolin-6-yl)acrylamideIC5019.0 [1], 34.0 [2], 4650.0 [3], 300000.0 [4]
N-[4-(4-Phenylanilino)quinazolin-6-yl]prop-2-enamideIC50107.0 [1], 760.0 [2], 9700.0 [3], 300000.0 [4]
N-(4-(4-Isopropylphenylamino)quinazolin-6-yl)acrylamideIC5032.0 [1], 340.0 [2], 2200.0 [3], 300000.0 [4]
N-(4-(Naphthalen-2-ylamino)quinazolin-6-yl)acrylamideIC503.0 [1], 32.0 [2], 1800.0 [3], 18100.0 [4]
N-(4-(Naphthalen-1-ylamino)quinazolin-6-yl)acrylamideIC5030.0 [1], 670.0 [2], 2100.0 [3], 16300.0 [4]
N-(4-((Naphthalen-1-yl)methylamino)quinazolin-6-yl)acrylamideIC50150.0 [1], 1500.0 [2], 1700.0 [3], 32000.0 [4]
N-(4-(Phenethylamino)quinazolin-6-yl)acrylamideIC5088.0 [1], 1400.0 [2], 3800.0 [3], 40000.0 [4]
N-(4-(4-Tert-Butylphenylamino)quinazolin-6-yl)propionamideIC50540.0 [1], 1500.0 [2], 300000.0 [3]
BosutinibIC501.8 [1], 410.0 [2]
7-[cis-4-(4-Methylpiperazin-1-Yl)cyclohexyl]-5-(4-Phenoxyphenyl)-7h-Pyrrolo[2,3-D]pyrimidin-4-AmineIC500.3 [1], 59.0 [2], 2030.0 [3]
DasatinibIC500.2 [1], 0.5 [2]
IbrutinibIC5095.6 [1]
1-(Tert-Butyl)-3-(p-tolyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amineIC5010.0 [1], 27.0 [2]
PDGF Receptor Tyrosine Kinase Inhibitor IVIC50378.0 [1]
1-(Tert-Butyl)-3-(naphthalen-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amineIC50600.0 [1]
1-[4-Amino-7-(3-hydroxypropyl)-5-(4-methylphenyl)-7H-pyrrolo[2,3-d]pyrimidin-6-yl]-2-fluoroethanoneIC501.0 [1], 4000000.0 [2]
N-(2-Chloro-6-methylphenyl)-2-[(2,6-dimethylpyrimidin-4-yl)amino]-1,3-thiazole-5-carboxamideIC501.0 [1]
1-(4-Amino-7-(3-hydroxypropyl)-5-(p-tolyl)-7h-pyrrolo[2,3-d]pyrimidin-6-yl)-2-chloroethanoneIC50100.0 [1], 4000000.0 [2]
N-[4-[4-Amino-7-[(E)-3-[(4-aminocyclohexyl)amino]prop-1-enyl]thieno[3,2-c]pyridin-3-yl]-2-methoxyphenyl]-1-methylindole-2-carboxamideIC5025900.0 [1], 26300.0 [2]
1-(2,2-Diethoxyethyl)-3-(1H-pyrrolo[2,3-b]pyridin-5-yl)pyrazolo[3,4-d]pyrimidin-4-amineIC501226.0 [1], 1230.0 [2]
2-PropenaMide, N-[cis-4-[4-aMino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyriMidin-1-yl]cyclohexyl]-IC507.1 [1]
DopamineIC50100000.0 [1]
GenisteinIC5058180.0 [1]
CrizotinibIC5010000.0 [1]
HarmineIC50250000.0 [1]
1-Tert-butyl-3-(4-chlorophenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amineIC5010.0 [1]
PalbociclibIC5010000.0 [1]
Su6656IC50170.0 [1]
SotrastaurinIC505500.0 [1]
1H-Inden-2-amine, 2,3-dihydro-5,6-dimethoxy-N,N-dipropyl-IC50100000.0 [1]
Lfm-a13IC50240000.0 [1]
Pyridone 6IC50500.0 [1]
(5e)-5-(Quinolin-6-Ylmethylidene)-2-[(Thiophen-2-Ylmethyl)amino]-1,3-Thiazol-4(5h)-OneKi2000.0 [1]
(5Z)-5-(Quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5H)-oneKi2000.0 [1]
4-[2-(Dipropylamino)ethyl]benzene-1,2-diolIC50100000.0 [1]
Raf265(chir-265)IC5010000.0 [1]
(3Z)-3-[(2,4,6-Trimethoxyphenyl)methylidene]-1H-indol-2-oneIC50100000.0 [1]
4-Amino-5-(4-Phenoxyphenyl)-7h-Pyrrolo[2,3-D]pyrimidin-7-Yl-CyclopentaneIC50126.0 [1]
1-Tert-butyl-3-(naphthalen-1-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amineIC501000.0 [1]
LY-3009120IC5091.0 [1]
3-((4-Bromo-2,6-difluorobenzyl)oxy)-5-(3-(4-(pyrrolidin-1-yl)butyl)ureido)isothiazole-4-carboxamideIC50161.0 [1]
CID 6918852Ki5000.0 [1]
A-770041IC5044100.0 [1]
CID 44219749IC5050000.0 [1]
JNK Inhibitor VIIIKi810.0 [1]
6-(Dipropylamino)-5,6,7,8-tetrahydronaphthalene-2,3-diolIC5050000.0 [1]
Bms-509744IC501100.0 [1]
IlorasertibIC50110.0 [1]
CID 56649281IC5011.09 [1]
N-Benzyl-1-(2-chloro-2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amineKi3500.0 [1]
4-[(2,4-Dichlorophenyl)amino]-6,7-dimethoxy-3-quinolinecarbonitrileIC5010000.0 [1]
CID 44814409IC5010000.0 [1]
Unii-mbe6kwv0QIKi100.0 [1]
7-(2,6-Dimethylphenyl)-5-methyl-N-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-1,2,4-benzotriazin-3-amineIC5023.0 [1]
4-[2-(3-Tert-butylanilino)-1-methylbenzimidazol-5-yl]oxy-N-methylpyridine-2-carboxamideIC505.0 [1]
N-Acetyl-O-phosphono-Tyr-Glu-Glu-Ile-GluIC501100.0 [1]
1-(2-Chloro-2-phenylethyl)-6-(2-morpholin-4-ylethylsulfanyl)-N-phenylpyrazolo[3,4-d]pyrimidin-4-amineKi7500.0 [1]
(2R)-2-[(2S)-4-[3-Chloro-5-fluoro-6-(2H-pyrazolo[3,4-b]pyridin-3-yl)pyridin-2-yl]piperazin-2-yl]-3-methylbutan-2-olKi1000.0 [1]
Unii-8FX9DP2Y1WIC505.0 [1]
N-(2-Chloro-6-methylphenyl)-2-[(cyclopropylcarbonyl)amino]-1,3-thiazole-5-carboxamideIC5071.0 [1]
N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)acetamideKi810.0 [1]
4-Amino-5-chloro-6-ethoxy-pyridine-2-carboxylic acid 4-methanesulfonyl-benzylamideIC50810.0 [1]
1-(2,6-Dichlorophenyl)-5-(2,4-difluorophenyl)-7-(4-piperidinyl)-1,2,3,4-tetrahydroquinazoline-2-oneIC5010000.0 [1]
(3Z)-N-Methyl-3-[[3-[3-(4-methylpiperazin-1-yl)propyl]-4,5,6,7-tetrahydro-1H-indol-2-yl]methylidene]-2-oxo-1H-indole-5-sulfonamideIC50800.0 [1]
7-Chloro-3-oxo-8-(1,3-thiazol-5-ylmethylamino)-11,16-dioxa-2,4,19,21-tetrazatricyclo[15.3.1.05,10]henicosa-1(20),5,7,9,17(21),18-hexaene-18-carbonitrileKi809.0 [1]
1-({4-[(3,4-Dichlorophenyl)methoxy]phenyl}methyl)azetidine-3-carboxylic acidIC5010000.0 [1]
1-(2-Chloro-2-phenyl-ethyl)-6-(2-morpholinoethylsulfanyl)-N-propyl-pyrazolo[3,4-d]pyrimidin-4-amineKi8150.0 [1]
1-(2-Chloro-2-phenylethyl)-N-[(4-fluorophenyl)methyl]-6-(2-morpholin-4-ylethylsulfanyl)pyrazolo[3,4-d]pyrimidin-4-amineKi15500.0 [1]
4-Phenylamino-3-quinolinecarbonitrile deriv. 25IC503200.0 [1]
7-Chloro-8-(3-hydroxypropoxy)-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5,7,9,18(22),19-hexaene-19-carbonitrileKi10000.0 [1]
7-Chloro-8-(3-hydroxypropyl)-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5(10),6,8,18(22),19-hexaene-19-carbonitrileKi10000.0 [1]
N-(7-Chloro-19-cyano-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5,7,9,18(22),19-hexaen-8-yl)methanesulfonamideKi10000.0 [1]
N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)-2-(2,5-dimethoxy-4-methylsulfonylphenyl)acetamideKi810.0 [1]
cis-3-(3-Azetidin-1-ylmethylcyclobutyl)-1-(2-phenylquinolin-7-yl)imidazo[1,5-a]pyrazin-8-ylamineIC5010000.0 [1]
1-[4-(3-Amino-1-methylpyrazolo[3,4-c]pyridin-4-yl)phenyl]-3-(3-methylphenyl)ureaIC5012500.0 [1]
3-[5-[3-(2-Methoxyethoxy)prop-1-ynyl]thiophen-3-yl]-7-(1,2,4-triazol-1-ylmethyl)-1,4-dihydroindeno[1,2-c]pyrazoleIC5050000.0 [1]
N-(4-Amino-5-chloro-6-ethoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamideKi810.0 [1]
N-(4-Amino-5-cyano-6-isopropoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamideKi810.0 [1]
N-(4-Amino-5-cyano-6-phenylpyridin-2-yl)acetamideKi810.0 [1]
Tert-butyl N-[4-[4-amino-1-[2-[4-(dimethylamino)piperidin-1-yl]ethyl]pyrazolo[3,4-d]pyrimidin-3-yl]-2-methoxyphenyl]carbamateIC502.1 [1]
2-(Dipropylamino)-2,3-dihydro-1H-inden-5-olIC50100000.0 [1]
2-[[N-[2-[3-Ethylsulfonyl-4-(4-methylpiperazin-1-yl)anilino]-5-fluoropyrimidin-4-yl]-5-(hydroxymethyl)-2-methylanilino]methyl]benzonitrileIC5045.0 [1]
Ripk1-IN-7IC50187.0 [1]
3-{[(1R)-1-Phenylethyl]amino}-4-(pyridin-4-ylamino)cyclobut-3-ene-1,2-dioneIC5050000.0 [1]
N-(2-Chloro-6-fluorobenzyl)-5-(furan-2-yl)-2H-1,2,4-triazol-3-amineIC50600.0 [1]
N-Propyl-4-({4-[(2,2,2-trifluoroethyl)amino]-1H-pyrrolo[2,3-d]pyrimidin-2-yl}amino)benzamideIC501030.0 [1]
6-[(4-Methylpiperazin-1-yl)methyl]-3-[5-(3-phenoxyprop-1-ynyl)thiophen-3-yl]-1,4-dihydroindeno[1,2-c]pyrazoleIC5027300.0 [1]
2-Methoxy-12-(2-hydroxyethyl)-13,14-dihydronaphthol[2,1-a]pyrrolo[3,4-c]carbazole-5-oneIC503400.0 [1]
[6-Chloro-4-methyl-3-[[3-(methylsulfamoylamino)phenyl]methyl]-2-oxochromen-7-yl] N,N-dimethylcarbamateIC5050000.0 [1]
N-(3-(2-(Pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl)phenyl)-3-(trifluoromethyl)benzamideIC5050000.0 [1]
CID 25207521IC5050000.0 [1]
7-Fluoro-1-methyl-9H-pyrido[3,4-b]indoleIC50250000.0 [1]
1-(5-Methyl-1H-imidazol-4-yl)-9H-beta-carbolineIC50250000.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Tyrosine-protein kinase FYN Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/tyrosine-protein-kinase-fyn-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ Tyrosine-protein kinase FYN Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/tyrosine-protein-kinase-fyn-inhibitors-ic50-ki.
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