![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_01384179eb1c1c1ef001bfbf31bfa500.svg) | Ibrutinib | IC50 | 2.3 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_6c38560dee3540f939fdaa0ff2c01d1d.svg) | N-(2-Chloro-6-methylphenyl)-2-[(2,6-dimethylpyrimidin-4-yl)amino]-1,3-thiazole-5-carboxamide | IC50 | 0.8 [1], 1.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_9c61c33e381bf2745dcd4e2fb5de136b.svg) | N-[4-[4-Amino-7-[(E)-3-[(4-aminocyclohexyl)amino]prop-1-enyl]thieno[3,2-c]pyridin-3-yl]-2-methoxyphenyl]-1-methylindole-2-carboxamide | IC50 | 17900.0 [1], 21700.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_9dd6da7cb57ea869429d2bb32c1c121c.svg) | 2-PropenaMide, N-[cis-4-[4-aMino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyriMidin-1-yl]cyclohexyl]- | IC50 | 0.4 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_c77eb69f87d46b4d00314a6bfb851cf8.svg) | Crizotinib | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_b5f9e60dc2b2b7e76e07307c1d8f7888.svg) | Bosutinib | IC50 | 1.1 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_295456cbf7462dfb1eaccb88d6610904.svg) | Ceritinib | IC50 | 1947.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_0a83b01cf93719a90ccaeda771089c43.svg) | Doramapimod | IC50 | 8500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_4e38800d1c310079b3b3e65c5db78d0d.svg) | Linifanib | IC50 | 500000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_0161179f2c7cfb11abb7ada9cb7db29a.svg) | Apitolisib | IC50 | 697.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_abf993ccf8ddfbd4e938356e627022d7.svg) | 1,4-Diaminoanthraquinone | IC50 | 24000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_6218d7660845b31fc510a0466313fd99.svg) | Amg-458 | IC50 | 328.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_f16bb71c80d20af237a458b33f574231.svg) | CID 44462758 | IC50 | 81.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_fa6bb23d0a45b7ba93e3c09b9d34e672.svg) | A-770041 | IC50 | 14100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_468407cc322128f69875c7ebf3453330.svg) | 3-[[2-[3-(Morpholin-4-ylmethyl)phenyl]thieno[3,2-b]pyridin-7-yl]amino]phenol | IC50 | 3.7 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_20ab18b8c16e5f284f7c3ab51a4a7a8f.svg) | N-Cyclopropyl-6-[(6,7-dimethoxyquinolin-4-yl)oxy]naphthalene-1-carboxamide | IC50 | 396.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_edc84196e7f0496a1c21e674ea92f53d.svg) | Unii-8FX9DP2Y1W | IC50 | 2.8 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_f046ae8812a77e5cb35fd8b53bebf05d.svg) | Ripk1-IN-7 | IC50 | 470.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_b7a1121a044d870d75dc38e0ca856330.svg) | N-[2-[3-(Dimethylamino)propyl-methylamino]-5-(trifluoromethyl)phenyl]-2-fluoro-5-[3-[4-(methylamino)-1,3,5-triazin-2-yl]pyridin-2-yl]oxybenzamide | IC50 | 8300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_420c640ab3d9d5b9acd6e7f999ac08f0.svg) | CID 27666048 | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_a7ee75d4a7ce2e8d7ffa73cb444c324f.svg) | 5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_771f17b91df724779a9947844c5b6f74.svg) | Unii-7N5LJ2Z26C | IC50 | 33.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_400786f64062ecb5f10a9d3b11455207.svg) | 1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_3e5e956fd3311d2f1725fa72559e89d1.svg) | CID 59627005 | IC50 | 2.2 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_ea5eb9d28ea73c1459251ec3ca29dbf2.svg) | 8-(4-Ethylphenyl)-5-Methyl-2,5-Dihydropyrazolo[4,3-C][2,1]benzothiazine 4,4-Dioxide | IC50 | 1900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_fb2996a255e5f9696d221b04a92bff1c.svg) | 1-Ethyl-8-(4-Ethylphenyl)-5-Methyl-1,5-Dihydropyrazolo[4,3-C][2,1]benzothiazine 4,4-Dioxide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_96d4b3c732c98defe38ea0a9f92d354f.svg) | N-[4-[4-Amino-7-[(E)-3-(4-hydroxypiperidin-1-yl)prop-1-enyl]thieno[3,2-c]pyridin-3-yl]-2-methoxyphenyl]-1-methylindole-2-carboxamide | IC50 | 37900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_b6faf72dfa81ac6f5cbbee7518dcb7f6.svg) | 4-[6-(Benzylamino)imidazo[1,2-B]pyridazin-3-Yl]benzonitrile | IC50 | 6400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_5d7901f03aa52a959c119b7fc87d0b0c.svg) | 6-[(2r)-2-(3-Fluorophenyl)pyrrolidin-1-Yl]-3-(Pyridin-2-Yl)imidazo[1,2-B]pyridazine | IC50 | 8700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_07f245678e6fcc2d52455f8c1a6544d0.svg) | 2-[4-[4-[6-[(2R)-2-(3-Fluorophenyl)pyrrolidin-1-yl]imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl]piperazin-1-yl]acetic acid | IC50 | 2800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_cadcfe40c75731fb4d071e8664de359c.svg) | 1-[4-[6-[(2R)-2-(3-Fluorophenyl)pyrrolidin-1-yl]imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl]piperidin-4-ol | IC50 | 5900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_9d109cefe6f21cc70e74499a7c9999ec.svg) | 3-(5-Cyclopropyl-1,2-oxazol-3-yl)-1-propan-2-ylpyrazolo[3,4-d]pyrimidin-4-amine | IC50 | 65.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_15b2f8cea2dcdba2c171894aaa9d8511.svg) | 4-[8-Amino-3-[(3R)-1-(2-methylpropanoyl)piperidin-3-yl]imidazo[1,5-a]pyrazin-1-yl]-3-fluoro-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide | IC50 | 203.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_748741d33d31d55972c10ed41fd023a8.svg) | 4-[8-Amino-3-[(2R)-4-(oxan-4-yl)morpholin-2-yl]imidazo[1,5-a]pyrazin-1-yl]-3-fluoro-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide | IC50 | 39.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_323e92cefd36d9d14a85ead4b64a3427.svg) | 4-[8-Amino-3-[(3R)-1-(oxan-4-yl)piperidin-3-yl]imidazo[1,5-a]pyrazin-1-yl]-3-fluoro-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide | IC50 | 22.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_14d6c4d8b5472476bb7332aacbc27d0e.svg) | 4-[8-Amino-3-[(2R)-4-(2-methylpropanoyl)morpholin-2-yl]imidazo[1,5-a]pyrazin-1-yl]-3-fluoro-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide | IC50 | 268.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_c009120ca19478ba69924ce16dc2791c.svg) | 5-(1,3-Benzodioxol-5-yl)-7-[[(2R)-1-ethenylsulfonylpyrrolidin-2-yl]methyl]pyrrolo[2,3-d]pyrimidin-4-amine | IC50 | 133.3 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_4ef2a0837fb3397010c52d8323e1a689.svg) | 5-[2-(2-Aminopyrimidin-5-yl)ethynyl]-N-[2-[(3S)-3-(dimethylamino)piperidin-1-yl]-5-(trifluoromethyl)phenyl]-2-fluorobenzamide | IC50 | 43.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_345d0ac5a70d97c558fac8afc930fc66.svg) | N-[4-[4-Amino-7-[(E)-3-(piperidin-4-ylamino)prop-1-enyl]thieno[3,2-c]pyridin-3-yl]-2-methoxyphenyl]-1-methylindole-2-carboxamide | IC50 | 26500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_f622a3713bfdad386a6b0dc08fa37bad.svg) | N-[4-[4-Amino-7-[(E)-3-(diethylamino)prop-1-enyl]thieno[3,2-c]pyridin-3-yl]-2-methoxyphenyl]-1-methylindole-2-carboxamide | IC50 | 14100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_fba488180963c8946f3c38122b79401f.svg) | N-[6-Fluoro-2-methyl-3-[5-[(5-methyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-2-yl)amino]-6-oxo-1H-pyridazin-3-yl]phenyl]-1-benzothiophene-2-carboxamide | IC50 | 1033.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_f53592583ff8163cade38a09145190a2.svg) | 4-[8-Amino-3-[(3R)-1-(2-methoxyacetyl)piperidin-3-yl]imidazo[1,5-a]pyrazin-1-yl]-3-fluoro-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide | IC50 | 28.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_61a22fc74231ad66bd487ef394e94197.svg) | 4-[8-Amino-3-[(2R)-4-(2-methoxyacetyl)morpholin-2-yl]imidazo[1,5-a]pyrazin-1-yl]-3-fluoro-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide | IC50 | 69.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-fgr_5711133ca718b66fa0cee0f039b3b462.svg) | 4-Amino-8-(5-Methyl-1h-Indazol-6-Yl)cinnoline-3-Carboxamide | IC50 | 41.0 [1] |