![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_52d89a2fc69d21765248014dedd86d63.svg) | CID 71605047 | IC50 | 1.0 [1], 2.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_3da15cae02e23edfbc9cbb5a47e328e3.svg) | N-[3-(2-Imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methylphenyl]-4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)benzamide | IC50 | 8.0 [1], 39.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_1d4a25fd962c8dfe261f24e70e2cff46.svg) | 1-[5-(2-Imidazo[1,2-a]pyrazin-5-ylethynyl)-1-methylpyrazol-3-yl]-3-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]urea | IC50 | 11.0 [1], 15.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_18a7adbed3e765c6b234321bb359b7f6.svg) | 1-[5-(2-Imidazo[1,2-a]pyrazin-3-ylethynyl)-1-methylpyrazol-3-yl]-3-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]urea | IC50 | 3.0 [1], 10.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_58c945c089c809d7e9aa3266c2a3508f.svg) | 1-[5-(2-Imidazo[1,2-b]pyridazin-3-ylethynyl)-1-methylpyrazol-3-yl]-3-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]urea | IC50 | 6.0 [1], 47.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_58d2243e6df61bdf4b3ebd94b634f0a2.svg) | N-[3-[2-(5-Anilinopyrimidin-2-yl)ethynyl]-4-methylphenyl]-4-(imidazol-1-ylmethyl)-3-(trifluoromethyl)benzamide | IC50 | 298.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_de616ea00f663554114acce8d8c9f2a2.svg) | 1-[5-(2-Imidazo[1,2-a]pyridin-3-ylethynyl)-1-methylpyrazol-3-yl]-3-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]urea | IC50 | 12.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_4519beed3cf9e9bf3e7f9f9c7b5bebe7.svg) | 1-[4-[(4-Methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-3-[1-methyl-5-(2-pyridin-3-ylethynyl)pyrazol-3-yl]urea | IC50 | 14.0 [1], 66.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_8b9e932f133afa4723d9177a2044be1d.svg) | 1-[5-[2-(6-Aminopyridin-3-yl)ethynyl]-1-methylpyrazol-3-yl]-3-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]urea | IC50 | 36.0 [1], 67.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_8babcafcaa23b01885fa6b59f5b92f72.svg) | 4-[[4-(2-Hydroxyethyl)piperazin-1-yl]methyl]-N-[3-(2-imidazo[1,2-a]pyridin-3-ylethynyl)-4-methylphenyl]-3-(trifluoromethyl)benzamide | IC50 | 18.0 [1], 41.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_a787dc6765a28dc767ae132efe2d2ba3.svg) | 4-(Imidazol-1-ylmethyl)-N-[4-methyl-3-(2-pyrimidin-5-ylethynyl)phenyl]-3-(trifluoromethyl)benzamide | IC50 | 40.0 [1], 163.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_b2d54f313fd6fae3559ad99a1d264705.svg) | Imatinib | IC50 | 272.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 75.9 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_b5f9e60dc2b2b7e76e07307c1d8f7888.svg) | Bosutinib | IC50 | 0.5 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_0a83b01cf93719a90ccaeda771089c43.svg) | Doramapimod | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_836d58634120a742d63c1602f26addff.svg) | CID 59604787 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_f046ae8812a77e5cb35fd8b53bebf05d.svg) | Ripk1-IN-7 | IC50 | 306.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_dbc9774b4a10efc12e4d4309ee79f133.svg) | (13R,15S)-13-Methyl-16-oxa-8,9,12,22,24-pentazahexacyclo[15.6.2.16,9.112,15.02,7.021,25]heptacosa-1(24),2,4,6,17,19,21(25)-heptaene-23,27-dione | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_a7ee75d4a7ce2e8d7ffa73cb444c324f.svg) | 5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_400786f64062ecb5f10a9d3b11455207.svg) | 1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_0f76e681b91255e37ea799fd5e965847.svg) | N-[5-[(Z)-(5-Fluoro-2-oxo-1H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrol-3-yl]-3-(4-methylpiperazin-1-yl)propanamide | Ki | 180.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_dc5ff7b87d06ec962585df9a614f5950.svg) | 6-[4-[(5-Tert-butyl-1,2-oxazol-3-yl)carbamoylamino]phenyl]-N-[3-(dimethylamino)propyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_04588a23ef4514c75cdc02ecc45743ea.svg) | N-[(4-Methoxyphenyl)methyl]-[1]benzofuro[2,3-b]pyridin-4-amine | Ki | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_e499a579d43efadfe258c451837bf054.svg) | 4-Fluoro-N-[4-[(6-oxo-5H-benzo[c][1,8]naphthyridin-1-yl)amino]phenyl]-2-(trifluoromethyl)benzamide | IC50 | 863.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tyrosine-protein-kinase-abl2_ad946fa32618a037eb1c316583993f21.svg) | 9-[[8-Fluoro-6-(1-methylpyrazol-4-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]sulfanyl]-4-methyl-[1,4]oxazino[3,2-c]quinolin-3-one | IC50 | 30000.0 [1] |