![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_6fb2b7740ad7c1642c73ba72caccec4d.svg) | Losartan | IC50 | 0.33 [1], 8.0 [2], 28.0 [3], 88.0 [4] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_6fb2b7740ad7c1642c73ba72caccec4d.svg) | Losartan | Ki | 12.0 [1], 17.0 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_5e73a1ef8d0e8c863280cb26b68ae8b5.svg) | Telmisartan | IC50 | 3.0 [1], 150.0 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_a2b6ca4b5cfddd7af28200040231e2e7.svg) | Saralasin | IC50 | 0.57 [1], 1.0 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_a2b6ca4b5cfddd7af28200040231e2e7.svg) | Saralasin | Ki | 0.22 [1], 0.33 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_c54686e7ba1b8f8a75fa8e6b4047c4d0.svg) | Irbesartan | IC50 | 0.9 [1], 20.8 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_c54686e7ba1b8f8a75fa8e6b4047c4d0.svg) | Irbesartan | Ki | 0.8 [1], 1.1 [2], 2.0 [3] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_9564fc2936faf5c4d42425d06ed470d0.svg) | Angiotensin II | IC50 | 0.72 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_9564fc2936faf5c4d42425d06ed470d0.svg) | Angiotensin II | Ki | 0.16 [1], 0.5 [2], 0.9 [3] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_545242164eb50221116b0ed84ae6f48e.svg) | Candesartan | IC50 | 0.69 [1], 10.72 [2], 110.0 [3] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_545242164eb50221116b0ed84ae6f48e.svg) | Candesartan | Ki | 10.4 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_25289f60ca2c0eabf86761712245c2b3.svg) | Butyl 3-(4-((1H-imidazol-1-yl)methyl)phenyl)-5-isobutylthiophen-2-ylsulfonylcarbamate | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_8caaf26cfbf2a8f0ff8e60cab756856b.svg) | Bms-248360 | IC50 | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_8caaf26cfbf2a8f0ff8e60cab756856b.svg) | Bms-248360 | Ki | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_ada53fb3ad72124bc2a88caa4590199d.svg) | Valsartan | IC50 | 2.7 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_ada53fb3ad72124bc2a88caa4590199d.svg) | Valsartan | Ki | 3.0 [1], 4700.0 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_3fd92c249001e0afb8d96d0db7dac9eb.svg) | 2-Ethyl-7-methyl-5-(2-methylpropyl)-3-[(1S)-5-[2-(2H-tetrazol-5-yl)phenyl]-2,3-dihydro-1H-inden-1-yl]imidazo[4,5-b]pyridine | IC50 | 1.6 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_3fd92c249001e0afb8d96d0db7dac9eb.svg) | 2-Ethyl-7-methyl-5-(2-methylpropyl)-3-[(1S)-5-[2-(2H-tetrazol-5-yl)phenyl]-2,3-dihydro-1H-inden-1-yl]imidazo[4,5-b]pyridine | Ki | 0.69 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_0f59871ecb15db8adac75e71b018a2a3.svg) | Angiotensin IV | Ki | 407.38 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_ef95aae72ddf9503168c657c7427dce1.svg) | Eprosartan | IC50 | 2.0 [1], 7.3 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_3a7c4cf2d6d4342eb7ddaaf10e131e9c.svg) | Tasosartan | IC50 | 32.0 [1], 38.0 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_95a2fd905b8ec00b6e3753c9f3480601.svg) | 2-Ethyl-5,7-dimethyl-3-((4-(2-(2H-tetrazol-5-yl)phenyl)phenyl)methyl)imidazo(4,5-b)pyridine | IC50 | 0.3 [1], 2.7 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_568398354ee28fedcb9bb28f9ee726f3.svg) | (1,1'-Biphenyl)-2-sulfonamide, N-(3,4-dimethyl-5-isoxazolyl)-4'-(2-oxazolyl)- | Ki | 0.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_75056e08a400a6daaac2fad41d416d4d.svg) | Sparsentan | Ki | 0.8 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_c4d4329d072cdea638d99f43afce3401.svg) | Butyl N-[2-[4-[(2-ethyl-5,7-dimethylimidazo[4,5-b]pyridin-3-yl)methyl]phenyl]-4-propylphenyl]sulfonylcarbamate | IC50 | 1.5 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_3334c5ad0ff8c1c805cbec3ed2099700.svg) | N-[4-Oxo-2-propyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]quinazolin-6-yl]-N-pentylbenzamide | IC50 | 1.7 [1], 7.0 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_e5598a6334ea9c395efbe7bc91403185.svg) | N-[2-[4-[[3-Butyl-5-oxo-1-[2-(trifluoromethyl)phenyl]-1,2,4-triazol-4-yl]methyl]phenyl]phenyl]sulfonylbenzamide | IC50 | 2.5 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_e5598a6334ea9c395efbe7bc91403185.svg) | N-[2-[4-[[3-Butyl-5-oxo-1-[2-(trifluoromethyl)phenyl]-1,2,4-triazol-4-yl]methyl]phenyl]phenyl]sulfonylbenzamide | Ki | 1.7 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_84905401227ffbd1286ee6bad3a58f99.svg) | 3-Butyl-2-[2'-(1H-tetrazole-5-yl)-4-biphenylylmethyl]-2,3-diazaspiro[4.4]nonane-1,4-dione | Ki | 25.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_754dbedc8eba554ef3ab4179d3bfa1bd.svg) | 7-Methyl-N-(2-phenylpropyl)-2-propyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]benzimidazole-5-carboxamide | IC50 | 0.9 [1], 16.7 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_1be5db3868901a2107aa0a020d9c3edb.svg) | Tert-butyl N-[2-[4-[[1-[2-bromo-5-(pentanoylamino)phenyl]-3-ethyl-5-oxo-1,2,4-triazol-4-yl]methyl]-3-fluorophenyl]phenyl]sulfonylcarbamate | IC50 | 0.2 [1], 3.5 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_e1432e7d40c2480c2c48d696a2e64fc4.svg) | Unii-A9T9wvah03 | IC50 | 1.2 [1], 31.0 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_a9f1eee02242c037dd658180ca95ed8e.svg) | 2,4-Bis(hydroxymethyl)-8-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]pyrido[2,3-d]pyrimidin-7-one | IC50 | 44.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_2f5f1aa2216fe8f82b37d88a09f778c2.svg) | 2-[4-[[4-Methyl-6-(2-phenylethylcarbamoyl)-2-propylbenzimidazol-1-yl]methyl]phenyl]benzoic acid | IC50 | 3.0 [1], 23.1 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_c81e2c19c603cc7dfc6d6dce159ba95d.svg) | 4-Methyl-7-oxo-8-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]-5,6-dihydropyrido[2,3-d]pyrimidine-2-carboxylic acid | IC50 | 11.0 [1], 23.0 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_0b1f799f3124796b33261f949f3ed517.svg) | 2-(1,3-Benzodioxol-5-yl)-2-[4-[(2-ethyl-5,7-dimethylimidazo[4,5-b]pyridin-3-yl)methyl]-2-propylphenoxy]-N-(4-propan-2-ylphenyl)sulfonylacetamide | IC50 | 13.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_3218ef0df658334051d7b60b6f885845.svg) | 2-Propyl-5-[(4-pyridin-2-ylpiperazin-1-yl)methyl]-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazole-4-carboxylic acid | IC50 | 4.2 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_643e71f949ee1a4555bf57532192af27.svg) | Tert-butyl N-[2-[4-[[3-butyl-1-[2-chloro-5-[(2-ethoxyacetyl)amino]phenyl]-5-oxo-1,2,4-triazol-4-yl]methyl]-3-fluorophenyl]phenyl]sulfonylcarbamate | IC50 | 0.38 [1], 0.56 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_763b548108fb470a10c42aa01a718baf.svg) | Tert-butyl N-[2-[4-[[3-butyl-5-oxo-1-[5-(pentanoylamino)-2-(trifluoromethyl)phenyl]-1,2,4-triazol-4-yl]methyl]-3-fluorophenyl]phenyl]sulfonylcarbamate | IC50 | 0.41 [1], 0.9 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_b2a00b53c3be3ffd48fd85cfec301eaa.svg) | N-[2-[4-[[3-Butyl-5-oxo-1-[5-(propanoylamino)-2-(trifluoromethyl)phenyl]-1,2,4-triazol-4-yl]methyl]-3-fluorophenyl]phenyl]sulfonyl-2-chlorobenzamide | IC50 | 0.25 [1], 0.43 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_bf05f2323bc74f74b4ff131bd08c07b8.svg) | 3-[2-[4-[[2-Butyl-6-oxo-4-propan-2-yl-5-(2-pyrrolidin-1-yl-2-sulfanylideneethyl)pyrimidin-1-yl]methyl]phenyl]phenyl]-4H-1,2,4-oxadiazol-5-one | IC50 | 2.2 [1], 10.5 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_9f9c54dccf36917b5705db0d926abdf2.svg) | (2S)-2-[N-(4-Hydroxypentanoyl)-4-[2-(2H-tetrazol-5-yl)phenyl]anilino]-3-methylbutanoic acid | IC50 | 0.47 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_9f9c54dccf36917b5705db0d926abdf2.svg) | (2S)-2-[N-(4-Hydroxypentanoyl)-4-[2-(2H-tetrazol-5-yl)phenyl]anilino]-3-methylbutanoic acid | Ki | 370.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_c8a68ce0b38f705751b0a01375a26cdf.svg) | [Sar1,Bpa2]AngII | Ki | 0.6 [1], 18.3 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_e3d58861553e149f95fcb906190a5034.svg) | (2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-3-(4-Benzoylphenyl)-2-[[(2S)-2-[[(2S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[2-(methylamino)acetyl]amino]pentanoyl]amino]-3-methylbutanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]pyrrolidine-2-carbonyl]amino]-3-phenylpropanoic acid | Ki | 0.7 [1], 250.0 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_1a875ea4a96cfa7234e2b90fe5b7d733.svg) | (2S)-2-[[(2S)-1-[(2S)-3-(4-Benzoylphenyl)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[2-(methylamino)acetyl]amino]pentanoyl]amino]-3-methylbutanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-3-phenylpropanoic acid | Ki | 31.6 [1], 500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_89c00e26cd755ed823179d09b708e852.svg) | (2S)-2-[[(2S)-3-(4-Benzoylphenyl)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[2-(methylamino)acetyl]amino]pentanoyl]amino]-3-methylbutanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]propanoyl]amino]-3-phenylpropanoic acid | Ki | 12.8 [1], 500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_d0c95acc3dab5c83f5a9e81955995264.svg) | [Tdf1]AngII | Ki | 0.7 [1], 26.4 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_a5d3b5e21f416fb86399818977a7d13e.svg) | [Sar1,Tdf2]AngII | Ki | 0.4 [1], 24.7 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_ee7714d1358890bed01701131e1d26ce.svg) | [Sar1,Tdf3]AngII | Ki | 0.3 [1], 1.3 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_890bcf5788e7d68c294defa4def42c41.svg) | (2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-5-(Diaminomethylideneamino)-2-[[2-(methylamino)acetyl]amino]pentanoyl]amino]-3-methylbutanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-[4-[3-(trifluoromethyl)diazirin-3-yl]phenyl]propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]pyrrolidine-2-carbonyl]amino]-3-phenylpropanoic acid | Ki | 0.5 [1], 250.0 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_e5d0ac96dbae9b6aa85a31a7b9c6f536.svg) | (2S)-2-[[(2S)-1-[(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-5-(Diaminomethylideneamino)-2-[[2-(methylamino)acetyl]amino]pentanoyl]amino]-3-methylbutanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-3-[4-[3-(trifluoromethyl)diazirin-3-yl]phenyl]propanoyl]pyrrolidine-2-carbonyl]amino]-3-phenylpropanoic acid | Ki | 58.2 [1], 500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_f291bb1938b02a3f2fb5ee2067ef9279.svg) | (2S)-2-[[(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-5-(Diaminomethylideneamino)-2-[[2-(methylamino)acetyl]amino]pentanoyl]amino]-3-methylbutanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-[4-[3-(trifluoromethyl)diazirin-3-yl]phenyl]propanoyl]amino]-3-phenylpropanoic acid | Ki | 3.8 [1], 500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_6a987ec29aeaaca2a4bd54baa1e965b7.svg) | [Bpa1]AngII | Ki | 0.8 [1], 19.4 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_524ba92d3d1c782963eb0ed6bbc921f2.svg) | [Sar1,Bpa3]AngII | Ki | 0.4 [1], 0.7 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_5f715cb64ec67aece75f1bfca3f37339.svg) | (2S)-2-[[(2S)-1-[(2S)-2-[[(2S,3S)-2-[[(2S)-3-(4-Benzoylphenyl)-2-[[(2S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[2-(methylamino)acetyl]amino]pentanoyl]amino]-3-methylbutanoyl]amino]propanoyl]amino]-3-methylpentanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]pyrrolidine-2-carbonyl]amino]-3-phenylpropanoic acid | Ki | 250.0 [1], 500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_6239b2b7bd3f93f9c443c2eba45908e4.svg) | (2S)-2-[[(2S)-1-[(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-5-(Diaminomethylideneamino)-2-[[2-(methylamino)acetyl]amino]pentanoyl]amino]-3-methylbutanoyl]amino]-3-[4-[3-(trifluoromethyl)diazirin-3-yl]phenyl]propanoyl]amino]-3-methylpentanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]pyrrolidine-2-carbonyl]amino]-3-phenylpropanoic acid | Ki | 250.0 [1], 500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_39e082c44d310010ae1b9ad8168a02fd.svg) | [Sar1,Bpa8]AngII | Ki | 0.6 [1], 0.8 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_5682aaf5b53e1d61f05f883ebe8f86d2.svg) | [Sar1,Tdf8]AngII | Ki | 0.7 [1], 0.9 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_ed324d438f9fa7eca521d50105ec11c8.svg) | 2-Butyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]-2,3-diazaspiro[4.4]nonane-6,9-dione | IC50 | 22.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_ed324d438f9fa7eca521d50105ec11c8.svg) | 2-Butyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]-2,3-diazaspiro[4.4]nonane-6,9-dione | Ki | 25.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_08222d03155c65bd61f0fadc369ed8bd.svg) | N-[2-[4-[(2-Butyl-6,9-dioxo-2,3-diazaspiro[4.4]nonan-3-yl)methyl]phenyl]phenyl]sulfonylbenzamide | IC50 | 12.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_08222d03155c65bd61f0fadc369ed8bd.svg) | N-[2-[4-[(2-Butyl-6,9-dioxo-2,3-diazaspiro[4.4]nonan-3-yl)methyl]phenyl]phenyl]sulfonylbenzamide | Ki | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_c78fa8acda4e712727b6f929e1c171be.svg) | (2-Benzoylphenyl)methyl 5-ethyl-3-[[2-fluoro-4-[2-(3-methylbutoxycarbonylsulfamoyl)phenyl]phenyl]methyl]-2-propylimidazole-4-carboxylate | IC50 | 0.5 [1], 570.0 [2] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_c70f5b79af37726016ec15cea0b55e94.svg) | Propranolol | IC50 | 5011.87 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_2d2c9357fb3c1c3e7cf2db26f14cf2f7.svg) | Losartan potassium | IC50 | 5.5 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_ec4f5e4970bd2d5895f7bf4f28866c74.svg) | Fimasartan | IC50 | 4.5 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_510ba2be80daf2c348f2583453fa9822.svg) | CID 121879 | IC50 | 3600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_09cf7047fac7d9415e9f827755923623.svg) | ZD 7155 hydrochloride | Ki | 0.5 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_e39e3bc989cee0b1a0a409acf38c8621.svg) | Cipargamin | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_dbb221ce910b0892ca283424422f354f.svg) | Piboserod | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_73e8353dd9415f963e941d5d863a68c8.svg) | Butyl N-[3-[4-[(2-ethyl-5,7-dimethylimidazo[4,5-b]pyridin-3-yl)methyl]phenyl]-5-(2-methylpropyl)thiophen-2-yl]sulfonylcarbamate | IC50 | 1.1 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_1ea30b92b55abd50c8b325a1854f3a68.svg) | Forasartan | IC50 | 6.9 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_220156a362868d0a368cd411c5e46918.svg) | (Sar1,Ile8)-Angiotensin II | Ki | 0.65 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_0287f832ae1adfacc5542f4dbc729a09.svg) | Zolasartan | Ki | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_1dc8dc1d6c90b5b09e7479f8cf836e92.svg) | Ripisartan | Ki | 24.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_6e6be4b817165180ec99c703597fa9b8.svg) | Edonentan | Ki | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_c0bfbc1c06145e9e5f88a50750f35b14.svg) | Potassium;2-[[5-ethyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]-1,3,4-thiadiazol-2-ylidene]carbamoyl]cyclopentene-1-carboxylate | IC50 | 0.4 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_b754a269c42e3ecd3ab65087c1e70ef1.svg) | (6S)-1-[(4-Amino-3-methylphenyl)methyl]-5-(2,2-diphenylacetyl)-6,7-dihydro-4H-imidazo[4,5-c]pyridine-6-carboxylic acid | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_82d5cc0cd6cdc72a5070bfcba2a2cca7.svg) | 3-((2'-(Benzoylaminosulfonyl)biphenyl-4-yl)methyl)-2-ethyl-5,7-dimethyl-3H-imidazo(4,5-b)pyridine | IC50 | 0.2 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_ac81d37dbe35e8ea96db7ce049de2c04.svg) | 4-Ethyl-2-propyl-1-(2'-(1H-tetrazol-5-yl)biphenyl-4-yl)methylimidazole-5-carboxylic acid | IC50 | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_0a163ab5b45981e4ee6693ccd4e9accc.svg) | 4-Oxo-6-((pyrimidin-2-ylthio)methyl)-4H-pyran-3-yl 4-nitrobenzoate | IC50 | 79000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_55ea42d2e8df72f19704f5b51e68a407.svg) | 2-[4-[[2-Butyl-6-(cyclohexylcarbamoylamino)benzimidazol-1-yl]methyl]phenyl]benzoic acid | Ki | 29.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_0c080142c8a9f1144feac996e630c566.svg) | 2-[[4-[[2-Butyl-6-[methylcarbamoyl(pentyl)amino]benzimidazol-1-yl]methyl]phenyl]carbamoyl]-3,6-dichlorobenzoic acid | Ki | 20.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_1aa28ab844f3ba78680172f2f918e147.svg) | CID 5311416 | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_401c2d481c22d184e88431fe37f72ca0.svg) | 6-(((4-Methylpyrimidin-2-yl)thio)methyl)-4-oxo-4H-pyran-3-yl furan-2-carboxylate | IC50 | 79000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_fbfa1a09b13c7444d81e84de68f2e78a.svg) | 6-(((4-Methylpyrimidin-2-yl)thio)methyl)-4-oxo-4H-pyran-3-yl 2-chloro-5-nitrobenzoate | IC50 | 79000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_f82f7c0d921f26658e7dd1b389389d56.svg) | Butyl N-[2-[4-[(2-ethyl-5,7-dimethylimidazo[4,5-b]pyridin-3-yl)methyl]phenyl]-4-[(3-methoxyphenyl)methyl]phenyl]sulfonylcarbamate | IC50 | 1.4 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_9ff6a01bd51ddc6431a161043f0021f8.svg) | Butyl N-[2-[4-[(2-ethyl-5,7-dimethylimidazo[4,5-b]pyridin-3-yl)methyl]phenyl]-4-(2-methylpropyl)phenyl]sulfonylcarbamate | IC50 | 2.1 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_9bafab5d3914382ee7eefd7636949a89.svg) | 6-(((4-Methylpyrimidin-2-yl)thio)methyl)-4-oxo-4H-pyran-3-yl 4-(pyrrolidin-1-ylsulfonyl)benzoate | IC50 | 79000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_9d2c6131a923980a41d4efdc3ed7f01a.svg) | [6-[(4-Methylpyrimidin-2-yl)sulfanylmethyl]-4-oxopyran-3-yl] 4-chloro-3-nitrobenzoate | IC50 | 79000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_8ac7bbcc279f5b470d023f4097f4339a.svg) | [4-Oxo-6-(pyrimidin-2-ylsulfanylmethyl)pyran-3-yl] 4-(dimethylsulfamoyl)benzoate | IC50 | 79000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_b1773636375d2bab83045e9e4fae5cbc.svg) | 6-(((4-Methylpyrimidin-2-yl)thio)methyl)-4-oxo-4H-pyran-3-yl benzoate | IC50 | 79000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_a0fd2c9114ed238be9470d82de8beb4d.svg) | 4-Oxo-6-((pyrimidin-2-ylthio)methyl)-4H-pyran-3-yl 3-nitrobenzoate | IC50 | 79000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_06aaac731fa253276c4f13d60e300af7.svg) | Butyl N-[3-[3-(imidazol-1-ylmethyl)phenyl]-5-(2-methylpropyl)thiophen-2-yl]sulfonylcarbamate | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_57e05013148c57b46d848b2f5fe110bc.svg) | 3-[2-Butyl-4-oxo-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]quinazolin-6-yl]-1-methyl-1-propan-2-ylurea | IC50 | 0.1 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_dd3a5beab83edecdbd6cec36f0bed973.svg) | (E)-3-[2-Butyl-1-(2-chlorobenzyl)-1H-imidazol-5-yl]-2-(2-thienylmethyl)acrylic acid | IC50 | 4530.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_2683c1538a375699bb214b8b73cbb95c.svg) | (2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-1-[2-[[(2S)-6-Amino-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-5-amino-2-[[(2S)-5-carbamimidamido-2-[[(2S)-5-carbamimidamido-2-[[(2S)-2-[[(2S)-2,6-diaminohexanoyl]amino]-3-phenylpropanoyl]amino]pentanoyl]amino]pentanoyl]amino]-5-oxopentanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]-5-carbamimidamidopentanoyl]amino]-4-methylpentanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]hexanoyl]amino]acetyl]pyrrolidine-2-carbonyl]amino]-4-methylsulfanylbutanoyl]pyrrolidine-2-carbonyl]amino]-3-phenylpropanoic acid | Ki | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_0e104614a10f27a7ddad898a78021692.svg) | 4-Oxo-6-((pyrimidin-2-ylthio)methyl)-4H-pyran-3-yl 4-(pyrrolidin-1-ylsulfonyl)benzoate | IC50 | 79000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/type-1-angiotensin-ii-receptor_f108ed5721652d30b693371176eb44ae.svg) | [4-Oxo-6-(pyrimidin-2-ylsulfanylmethyl)pyran-3-yl] 4-(diethylsulfamoyl)benzoate | IC50 | 79000.0 [1] |