 | Telotristat | IC50 | 16.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-(3-methylpyrazol-1-yl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 26.0 [1] |
 | 4-(4-Amino-6-{[(1R)-1-naphthalen-2-ylethyl]amino}-1,3,5-triazin-2-yl)-L-phenylalanine | IC50 | 26.0 [1] |
 | (2S)-2-Amino-3-[4-[4-amino-6-(naphthalen-2-ylmethylamino)-1,3,5-triazin-2-yl]phenyl]propanoic acid | IC50 | 24.0 [1] |
 | 4-Chloro-L-phenylalanine | IC50 | 100000.0 [1] |
 | Rodatristat | IC50 | 33.0 [1] |
 | 8-[2-Amino-6-[(1R)-1-[4-chloro-2-(3-methylpyrazol-1-yl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 55.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-2,2,2-trifluoro-1-[4-(1-methylindazol-5-yl)phenyl]ethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 30.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-[3-(2-oxopyrrolidin-1-yl)phenyl]phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 77.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-(3,4-dimethylphenyl)-2-(3-methylpyrazol-1-yl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 20.0 [1] |
 | 8-[4-Amino-6-[(1R)-1-[4-chloro-2-(3-methylpyrazol-1-yl)phenyl]-2,2,2-trifluoroethoxy]-1,3,5-triazin-2-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 2266.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-(3-fluorophenyl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 32.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-(3-chloro-5-fluorophenyl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 35.0 [1] |
 | 8-[6-[(1R)-1-[4-Chloro-2-(3-methylpyrazol-1-yl)phenyl]-2,2,2-trifluoroethoxy]-2-(cyclohexylamino)pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 79.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-(4-sulfamoylphenyl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 1125.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-(3-methylsulfonylphenyl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 14.0 [1] |
 | 3-[2-Amino-6-[(1R)-1-[4-chloro-2-(3-methylpyrazol-1-yl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-3,9-diazaspiro[5.5]undecane-10-carboxylic acid | IC50 | 949.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-(3-chlorophenyl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 30.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-2,2,2-trifluoro-1-(4-isoquinolin-6-ylphenyl)ethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 25.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-2,2,2-trifluoro-1-[4-(2-methyl-1-oxo-3,4-dihydroisoquinolin-6-yl)phenyl]ethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 39.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-2,2,2-trifluoro-1-[4-(2-oxo-3,4-dihydro-1H-quinolin-6-yl)phenyl]ethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 28.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[2-(3-carbamoylphenyl)-4-chlorophenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 40.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-(3-methylphenyl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 26.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-[3-(methanesulfonamido)phenyl]phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 51.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-2,2,2-trifluoro-1-[4-(4-methoxyphenyl)-2-(3-methylpyrazol-1-yl)phenyl]ethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 23.0 [1] |
 | 8-[6-[(1R)-1-[4-Chloro-2-(3-methylpyrazol-1-yl)phenyl]-2,2,2-trifluoroethoxy]-2-phenoxypyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 128.0 [1] |
 | (3R)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-(3-methylpyrazol-1-yl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 1787.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-(4-chloro-3-methylphenyl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 62.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-(1,3-dimethylindazol-6-yl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 32.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-(3-sulfamoylphenyl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 11.0 [1] |
 | 8-[4-[(1R)-1-[4-Chloro-2-(3-methylpyrazol-1-yl)phenyl]-2,2,2-trifluoroethoxy]pyridin-2-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 211.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-[3-(trifluoromethyl)phenyl]phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 21.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-[3-(dimethylsulfamoyl)phenyl]phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 53.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-(3-chloro-4-ethoxyphenyl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 207.0 [1] |
 | 8-[6-[(1R)-1-[4-Chloro-2-(3-methylpyrazol-1-yl)phenyl]-2,2,2-trifluoroethoxy]-2-methylpyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 65.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-2,2,2-trifluoro-1-[4-(2-methylsulfanylquinolin-6-yl)phenyl]ethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 26.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-(6-methylpyridin-2-yl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 73.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-(2,3-dimethylindazol-6-yl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 37.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-(4-chloro-2-pyridin-3-ylphenyl)-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 65.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[2-(3-tert-butylphenyl)-4-chlorophenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 23.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-2,2,2-trifluoro-1-[4-(3-fluoroquinolin-6-yl)phenyl]ethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 40.0 [1] |
 | 8-[5-[(1R)-1-[4-Chloro-2-(3-methylpyrazol-1-yl)phenyl]-2,2,2-trifluoroethoxy]pyridazin-3-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 5930.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-(4-methylsulfonylphenyl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 885.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-(3,4-difluorophenyl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 35.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-(4-chlorophenyl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 53.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-2,2,2-trifluoro-1-[4-(1H-indazol-5-yl)phenyl]ethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 32.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-(3-methoxyphenyl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 19.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-(3-cyanophenyl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 30.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-(3,4-dichlorophenyl)-2-(3-methylpyrazol-1-yl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 22.0 [1] |
 | (3S)-8-[2-Amino-6-[(1R)-1-[4-chloro-2-(3,5-difluorophenyl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid | IC50 | 22.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[(2-piperidin-1-ylphenyl)methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 22.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-(2-chlorophenoxy)-6-piperidin-1-ylphenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 15.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[(2-methoxy-6-piperidin-1-ylphenyl)methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 18.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[(2-pyrrolidin-1-ylphenyl)methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 32.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[(2-cyclohexyloxy-6-piperidin-1-ylphenyl)methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 30.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[2-(2-phenylphenyl)ethyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 61.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[(3-methoxy-2-piperidin-1-ylphenyl)methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 35.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-piperidin-1-yl-5-(1,3-thiazol-2-yl)phenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 7.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[(4-phenylphenyl)methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 2200.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[(5-chloro-2-piperidin-1-ylphenyl)methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 16.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[3-(2-phenylphenyl)propyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 599.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-(4-benzylpiperidin-1-yl)phenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 38.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-piperidin-1-yl-6-[3-(trifluoromethyl)phenoxy]phenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 14.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[(4-chloro-2-piperidin-1-ylphenyl)methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 74.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[(3-chloro-2-piperidin-1-ylphenyl)methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 66.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-piperidin-1-yl-6-(trifluoromethyl)phenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 11.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-(3-methylpiperidin-1-yl)phenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 20.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-(diethylamino)phenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 99.0 [1] |
 | (2S)-2-Amino-3-[4-[(N'-benzylcarbamimidoyl)carbamoyl]phenyl]propanoic acid | IC50 | 11036.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-(4-methylphenoxy)-6-piperidin-1-ylphenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 15.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[(2-phenoxy-6-piperidin-1-ylphenyl)methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 26.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[(5-methoxy-2-piperidin-1-ylphenyl)methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 22.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-piperidin-1-yl-6-[2-(trifluoromethyl)phenoxy]phenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 10.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-(3-methylphenoxy)-6-piperidin-1-ylphenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 8.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[(2-thiomorpholin-4-ylphenyl)methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 58.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-(4-hydroxypiperidin-1-yl)phenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 106.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-(3,5-dimethylpiperidin-1-yl)phenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 25.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[(3-phenylphenyl)methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 405.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[(4-methoxy-2-piperidin-1-ylphenyl)methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 61.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-piperidin-1-yl-6-[4-(trifluoromethyl)phenoxy]phenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 6.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[(3-methyl-2-piperidin-1-ylphenyl)methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 46.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[(5-methyl-2-piperidin-1-ylphenyl)methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 25.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-(3-methoxyphenoxy)-6-piperidin-1-ylphenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 6.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[(2-phenylphenyl)methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 165.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-(4-chlorophenoxy)-6-piperidin-1-ylphenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 11.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[(2-ethoxy-6-piperidin-1-ylphenyl)methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 43.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-(azetidin-1-yl)phenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 129.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[(2-piperidin-1-yl-6-propan-2-yloxyphenyl)methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 28.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-(2-azabicyclo[2.2.1]heptan-2-yl)phenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 11.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-(2-methylphenoxy)-6-piperidin-1-ylphenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 11.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-(4-methoxyphenoxy)-6-piperidin-1-ylphenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 16.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[(2-morpholin-4-ylphenyl)methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 106.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-(4-methoxypiperidin-1-yl)phenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 33.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-(1,2,4-triazol-1-yl)phenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 1844.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-(3-chlorophenoxy)-6-piperidin-1-ylphenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 6.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-(azepan-1-yl)phenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 16.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-(azepan-1-yl)-6-phenoxyphenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 13.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-(2-methylpiperidin-1-yl)phenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 15.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[[2-(3-methylpyrazol-1-yl)phenyl]methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 666.0 [1] |
 | (2S)-2-Amino-3-[4-[[N'-[(2-chloro-6-piperidin-1-ylphenyl)methyl]carbamimidoyl]carbamoyl]phenyl]propanoic acid | IC50 | 33.0 [1] |