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Transmembrane protease serine 11D Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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▼
N-(Benzylsulfonyl)seryl-N~1~-{4-[(Z)-amino(imino)methyl]benzyl}serinamideKi78.0 [1]
CID 46899577Ki19.0 [1]
N-(Benzylsulfonyl)-3-Cyclohexyl-D-Alanyl-N-(4-Carbamimidoylbenzyl)-L-ProlinamideKi108.0 [1]
N-(Benzylsulfonyl)-D-Valyl-N-(4-Carbamimidoylbenzyl)-L-ProlinamideKi76.0 [1]
N-(Benzylsulfonyl)-D-Leucyl-N-(4-Carbamimidoylbenzyl)-L-ProlinamideKi120.0 [1]
Inhibitor 1 [Colombo et al., 2012]Ki8.4 [1]
(2S)-2-[[(2S)-2-[[(2S)-5-Amino-2-[[(2S)-2-[(2-aminobenzoyl)amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-oxopentanoyl]amino]-3-carboxypropanoyl]amino]-5-(diaminomethylideneamino)pentanoic acidKi54.3 [1]
(2S)-6-Amino-2-[[(2S)-2-[[(2S)-5-amino-2-[[(2S)-2-[(2-aminobenzoyl)amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-oxopentanoyl]amino]-3-carboxypropanoyl]amino]hexanoic acidKi112.3 [1]
(2S)-1-[(2R)-6-Amino-2-(benzylsulfonylamino)hexanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamideKi40.0 [1]
N~2~-(Benzylsulfonyl)-D-Arginyl-N-(4-Carbamimidoylbenzyl)glycinamideKi430.0 [1]
Benzyl N-[(5S)-5-[[(2R)-2-(benzylsulfonylamino)-3-hydroxypropanoyl]amino]-6-[(4-carbamimidoylphenyl)methylamino]-6-oxohexyl]carbamateKi51.0 [1]
(2S)-1-[(2R)-2-(Benzylsulfonylamino)-3-phenylpropanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamideKi98.0 [1]
(2S)-1-[(2R)-2-(Benzylsulfonylamino)-4-phenylbutanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamideKi63.0 [1]
Benzyl N-[(5R)-5-(benzylsulfonylamino)-6-[(2S)-2-[(4-carbamimidoylphenyl)methylcarbamoyl]pyrrolidin-1-yl]-6-oxohexyl]carbamateKi53.0 [1]
(2S)-1-[(2R)-2-(Benzylsulfonylamino)-6-(diaminomethylideneamino)hexanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamideKi13.0 [1]
(2S)-1-[(2R)-2-(Benzylsulfonylamino)-3-(4-cyanophenyl)propanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamideKi311.0 [1]
(2S)-1-[(2R)-2-(Benzylsulfonylamino)-3-(4-carbamimidoylphenyl)propanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamideKi168.0 [1]
(2S)-1-[(2R)-2-(Benzylsulfonylamino)-5-oxo-5-(4-pyrimidin-2-ylpiperazin-1-yl)pentanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamideKi17.0 [1]
Benzyl 4-[(3R)-3-(benzylsulfonylamino)-4-[(2S)-2-[(4-carbamimidoylphenyl)methylcarbamoyl]pyrrolidin-1-yl]-4-oxobutanoyl]piperazine-1-carboxylateKi135.0 [1]
(2S)-1-[(2R)-2-(Benzylsulfonylamino)-4-[4-[3-(dimethylamino)propyl]piperazin-1-yl]-4-oxobutanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamideKi149.0 [1]
4-[[[(2S,4R)-4-(Benzylsulfonylamino)-7-(diaminomethylideneamino)-3-oxoheptan-2-yl]amino]methyl]benzenecarboximidamideKi30.0 [1]
4-[[[(2S,4R)-4-(Benzylsulfonylamino)-7-(diaminomethylideneamino)-3-oxo-1-phenylheptan-2-yl]amino]methyl]benzenecarboximidamideKi57.0 [1]
(3S,5R)-5-(Benzylsulfonylamino)-3-[(4-carbamimidoylphenyl)methylamino]-8-(diaminomethylideneamino)-4-oxooctanoic acidKi422.0 [1]
(2S)-1-[(2R)-4-(4-Benzylpiperazin-1-yl)-2-(benzylsulfonylamino)-4-oxobutanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamideKi158.0 [1]
(2S)-1-[(2R)-2-(Benzylsulfonylamino)-4-oxo-4-(4-propan-2-ylpiperazin-1-yl)butanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamideKi221.0 [1]
4-[[[(4S,6R)-6-(Benzylsulfonylamino)-9-(diaminomethylideneamino)-5-oxononan-4-yl]amino]methyl]benzenecarboximidamideKi15.0 [1]
(2S)-1-[(2R)-2-(Benzylsulfonylamino)-4-[4-(2,5-dimethylphenyl)piperazin-1-yl]-4-oxobutanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamideKi73.0 [1]
(2S)-1-[(2R)-2-(Benzylsulfonylamino)-4-[4-(2-hydroxyethyl)piperazin-1-yl]-4-oxobutanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamideKi210.0 [1]
Benzyl N-[(5S,7R)-7-(benzylsulfonylamino)-5-[(4-carbamimidoylphenyl)methylamino]-10-(diaminomethylideneamino)-6-oxodecyl]carbamateKi34.0 [1]
4-[[[(4S,6R)-6-(Benzylsulfonylamino)-9-(diaminomethylideneamino)-2-methyl-5-oxononan-4-yl]amino]methyl]benzenecarboximidamideKi47.0 [1]
Tert-butyl (4R)-4-(benzylsulfonylamino)-5-[(2S)-2-[(4-carbamimidoylphenyl)methylcarbamoyl]pyrrolidin-1-yl]-5-oxopentanoateKi36.0 [1]
(3R)-3-(Benzylsulfonylamino)-4-[(2S)-2-[(4-carbamimidoylphenyl)methylcarbamoyl]pyrrolidin-1-yl]-4-oxobutanoic acidKi1425.0 [1]
4-[[[(3S,5R)-5-(Benzylsulfonylamino)-8-(diaminomethylideneamino)-2-methyl-4-oxooctan-3-yl]amino]methyl]benzenecarboximidamideKi22.0 [1]
4-[[[(2S,4R)-4-(Benzylsulfonylamino)-7-(diaminomethylideneamino)-1-hydroxy-3-oxoheptan-2-yl]amino]methyl]benzenecarboximidamideKi34.0 [1]
Tert-butyl (3S,5R)-5-(benzylsulfonylamino)-3-[(4-carbamimidoylphenyl)methylamino]-8-(diaminomethylideneamino)-4-oxooctanoateKi512.0 [1]
Tert-butyl (3R)-3-(benzylsulfonylamino)-4-[(2S)-2-[(4-carbamimidoylphenyl)methylcarbamoyl]pyrrolidin-1-yl]-4-oxobutanoateKi38.0 [1]
(2S)-1-[(2R)-2-(Benzylsulfonylamino)-5-oxo-5-piperazin-1-ylpentanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamideKi68.0 [1]
4-[[[(5R)-5-(Benzylsulfonylamino)-8-(diaminomethylideneamino)-4-oxooctan-3-yl]amino]methyl]benzenecarboximidamideKi14.0 [1]
4-[[[(3S,4S,6R)-6-(Benzylsulfonylamino)-9-(diaminomethylideneamino)-3-methyl-5-oxononan-4-yl]amino]methyl]benzenecarboximidamideKi23.0 [1]
Benzyl 4-[(4R)-4-(benzylsulfonylamino)-5-[(2S)-2-[(4-carbamimidoylphenyl)methylcarbamoyl]pyrrolidin-1-yl]-5-oxopentanoyl]piperazine-1-carboxylateKi38.0 [1]
(2S)-1-[(2R)-2-(Benzylsulfonylamino)-4-oxo-4-(4-pyrimidin-2-ylpiperazin-1-yl)butanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamideKi43.0 [1]
(2S)-1-[(2R)-2-(Benzylsulfonylamino)-4-morpholin-4-yl-4-oxobutanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamideKi183.0 [1]
(2S)-1-[(2R)-2-(Benzylsulfonylamino)-4-oxo-4-piperazin-1-ylbutanoyl]-N-[(4-carbamimidoylphenyl)methyl]pyrrolidine-2-carboxamideKi202.0 [1]
4-[[[(4S,6R)-6-(Benzylsulfonylamino)-1,9-bis(diaminomethylideneamino)-5-oxononan-4-yl]amino]methyl]benzenecarboximidamideKi457.0 [1]
Items per page: 1 - 10 of 44
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References

This online tool may be cited as follows

MLA

"Quest Database™ Transmembrane protease serine 11D Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/transmembrane-protease-serine-11d-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, November 21). Quest Database™ Transmembrane protease serine 11D Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/transmembrane-protease-serine-11d-inhibitors-ic50-ki.
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