![](https://images.aatbio.com/dataset/ic50/translocator-protein_a8643c8f051557f676a3e85676e53d0c.svg) | 1-(2-Chlorophenyl)-N-methyl-N-(1-methylpropyl)-3-isoquinolinecarboxamide | IC50 | 1.1 [1], 2.5 [2], 490.0 [3] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_a8643c8f051557f676a3e85676e53d0c.svg) | 1-(2-Chlorophenyl)-N-methyl-N-(1-methylpropyl)-3-isoquinolinecarboxamide | Ki | 4.5 [1], 7.11 [2], 29.2 [3], 36.0 [4] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_fc0496b8d36d46964b874f3e0b854916.svg) | N,N-Diethyl-2-(2-(4-methoxyphenyl)-5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)acetamide | Ki | 6.68 [1], 8.2 [2], 19.5 [3], 98.8 [4] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_dc8536536605297a019f3ac76a6b897a.svg) | N-(2,5-Dimethoxybenzyl)-N-(5-fluoro-2-phenoxyphenyl)acetamide | Ki | 0.19 [1], 0.2 [2], 0.24 [3] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_cc1f83fd1f2e9b39555e45d437032b92.svg) | 2-[1-Methyl-2-(4-nitrophenyl)indol-3-yl]-2-oxo-N,N-dipropylacetamide | Ki | 1.57 [1], 1.82 [2], 9.53 [3] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_35bdc0b4fd731443ba4656e0b73a705b.svg) | Emapunil | Ki | 6.4 [1], 31.3 [2] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_e74adad61b13a7c71288dfbff078ee32.svg) | N,N-Diethyl-2-[2-(4-methoxyphenyl)-4,6-dimethylindol-1-yl]acetamide | Ki | 28.13 [1], 806.0 [2] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_8326890c7f510fae96e292b75b077e25.svg) | N,N-Diethyl-2-[2-(4-methoxyphenyl)-4,6-dimethylbenzimidazol-1-yl]acetamide | Ki | 224.46 [1], 398.18 [2] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_ed7c1a35d6eb0784dd0248d8f7d19940.svg) | N,N-Diethyl-2-[2-(4-methoxyphenyl)-5,7-dimethylimidazo[4,5-b]pyridin-3-yl]acetamide | Ki | 29.11 [1], 144.33 [2] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_12a9eda48ec5a1c66f8f7da82d8d3a55.svg) | N,N-Diethyl-2-[8-(4-methoxyphenyl)-2,6-dimethylpurin-9-yl]acetamide | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_aa97c32bb623b0bc042fb018bbfd40bf.svg) | 9H-Carbazole-9-acetamide, N,N-diethyl- | Ki | 30.1 [1], 176.6 [2] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_f0e8c8d306ed21ecc421fe826db8b191.svg) | N,N-Diethyl-2-[3-(4-methoxyphenyl)carbazol-9-yl]acetamide | Ki | 28.9 [1], 93.4 [2] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_2c4982416b4571f2503a9450b30a9cfd.svg) | N,N-Diethyl-2-[3-(2-methoxyphenyl)carbazol-9-yl]acetamide | Ki | 25.4 [1], 137.3 [2] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_1383ab490feee399a7bcde7f69022c6f.svg) | N-Benzyl-2-(3-bromocarbazol-9-yl)-N-ethylacetamide | Ki | 54.3 [1], 123.4 [2] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_ab1ebc5e49f509b505a51d3af9e0486a.svg) | N-Benzyl-2-carbazol-9-yl-N-ethylacetamide | Ki | 91.6 [1], 459.6 [2] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_ac4a14991179b9f01ef1ed0f62f20799.svg) | 2-(3-Bromocarbazol-9-yl)-N,N-diethylacetamide | Ki | 31.5 [1], 160.9 [2] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_ddcbbd1a2e4366a8cab5ada8ba2e7a24.svg) | N,N-Diethyl-2-(3-phenylcarbazol-9-yl)acetamide | Ki | 31.6 [1], 159.8 [2] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_7903bd2d1c6893b8465dc90acb9c0c40.svg) | Diazepam | IC50 | 123594743.3 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_981dad8026c15b69be26950695255dcf.svg) | Lorazepam | IC50 | 285759054.3 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_8c17699dd6a8601a97ee28fed7c9da3c.svg) | Clonazepam | IC50 | 555904257.3 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_5172f44ff113535835c74fffc2a5e8e3.svg) | Flunitrazepam | IC50 | 263026799.2 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_91102e83cc9dd60b3164e96fbd589fcf.svg) | Oxazepam | IC50 | 55590425.73 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_8fe2951674d6ff418f204dfa134a6493.svg) | Nitrazepam | IC50 | 100000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_bf85d85b6f14b2d05c2d3de0f6a66e86.svg) | Temazepam | IC50 | 62517269.28 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_6fbf89047e841f2d4d5e6f8692f4ccba.svg) | Nordazepam | IC50 | 106414301.8 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_d5507dad6c930f3c681f3c5de8c8eb70.svg) | N,N-Dihexyl-2-(4-fluorophenyl)indole-3-acetamide | Ki | 3.25 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_8aa2b399c0b5a9cf98b338ace0ef292e.svg) | Delorazepam | IC50 | 555904257.3 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_5e3aa3f832dd7f1a480c7a61693500d9.svg) | N-(2-Methoxybenzyl)-N-(4-phenoxypyridin-3-yl)acetamide | Ki | 2.5 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_613bd559e314252ec76ed0cdf79b77e9.svg) | 5-(4-Chlorophenyl)-N-(3,5-dimethoxyphenyl)furan-2-carboxamide | IC50 | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_ee141607af93a358db77b0d8a34a6843.svg) | Halazepam | IC50 | 10864256.24 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_94e2af914e71d49c420e40f9d0827604.svg) | 7-Aminoflunitrazepam | IC50 | 15381546.4 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_a19f65871dd99f97e92a4af09e55d209.svg) | Norfludiazepam | IC50 | 500034535.0 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_3bab44928a53e01431ed8a69ba906c19.svg) | 2H-1,4-Benzodiazepin-2-one, 5-(2-chlorophenyl)-1,3-dihydro-3-methyl-7-nitro-, (R)- | IC50 | 833681184.6 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_662c13b3b9490582947b1b21cfa77389.svg) | Acetamide, N-(5-fluoro-2-phenoxyphenyl)-N-((2-methoxy-5-(methoxy-11C)phenyl)methyl)- | Ki | 0.24 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_07487c5e665021df1bca2b6d240ebfc7.svg) | 7-Aminoclonazepam | IC50 | 13335214.32 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_7c854c775864706e5cde169db2af5de0.svg) | Unii-FS47vof3O7 | Ki | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_25f5e25b0dad5fba18d7a0a972a7ad5f.svg) | Naluzotan | Ki | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_eb53007d6577a48a848a6104edb8b626.svg) | Norflunitrazepam | IC50 | 666806769.2 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_f856ffa14c789a520a930bc242dcea97.svg) | 1,3-Dihydro-5-phenyl-2H-1,4-benzodiazepin-2-one | IC50 | 2857590.54 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_0d535489c082e3234d0bcf5b1986f469.svg) | 7-Aminonitrazepam | IC50 | 2588212.92 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_fe2a7f7190df5d8ca99a0e10d7f06041.svg) | 5-(2-Chlorophenyl)-1,3-dihydro-1-methyl-7-nitro-2H-1,4-benzodiazepin-2-one | IC50 | 454988060.2 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_de238d6a3f9e5815e11c1fceea47087d.svg) | Mivebresib | IC50 | 800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_909b723f602749274a62bb67630edeed.svg) | (3r)-5-(2-Fluorophenyl)-1,3-dimethyl-7-nitro-1,3-dihydro-2h-1,4-benzodiazepin-2-one | IC50 | 142889395.9 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_9a7501b8d54fc088a2b0754525d5045f.svg) | 1H-1,4-Benzodiazepine-7-carbonitrile, 2,3-dihydro-1-methyl-2-oxo-5-phenyl- | IC50 | 2630267.99 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_d0ae2ec628d684735ce55c7d92a514ce.svg) | 5-(2-Fluorophenyl)-1,3-dihydro-1-methyl-2H-1,4-benzodiazepin-2-one | IC50 | 71449632.61 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_efbfe59fd9f8e2c2ce283f8f560ea2c2.svg) | 2H-1,4-Benzodiazepin-2-one, 1,3-dihydro-5-phenyl-7-(trifluoromethyl)- | IC50 | 76913044.03 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_dfcd84a39fc5d27d8d25680abeaaada3.svg) | 7-Fluoro-5-phenyl-1,3-dihydro-2h-1,4-benzodiazepin-2-one | IC50 | 25003453.62 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_11b55eed32c71b3b673e6538f9e8799b.svg) | N-(4-Chloro-2-phenoxyphenyl)-N-(2-isopropoxybenzyl)acetamide | IC50 | 0.92 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_4768ae2bbe8b8a3c0149c958a4c64132.svg) | N-(3-(3,6-Dibromo-9H-carbazol-9-yl)-2-fluoropropyl)-3-methoxyaniline | IC50 | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_2d9206eaa55133bca6c881f42a85ddf0.svg) | CID 53245590 | Ki | 2540.0 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_6bf1e297fe3834ef6cf0823e04938d43.svg) | 5-(2-Fluorophenyl)-7-iodo-1-methyl-1,3-dihydro-2h-1,4-benzodiazepin-2-one | IC50 | 345143739.3 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_bea075376079d3748f077dca44922efe.svg) | 1,3-Dihydro-7-nitro-5-(alpha,alpha,alpha-trifluoro-o-tolyl)2H-1,4-benzodiazepin-2-one | IC50 | 285759054.3 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_684d5b39fdc0e4bbc7ea2a3c82b1ddc8.svg) | 7-Fluoro-5-(2-fluorophenyl)-1-methyl-3H-1,4-benzodiazepin-2-one | IC50 | 195884467.4 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_4fef376dde1307167afaf1af8568177f.svg) | 5-Acetyl-6-(2-chloro-4-phenylmethoxyphenyl)-1-hydroxy-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one | IC50 | 30000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_6ad24065afc05f37260044c6a396328b.svg) | N-(6-Fluoro-4-phenoxypyridin-3-yl)-N-[(2-methoxyphenyl)methyl]acetamide | Ki | 1.19 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_acba5eee759773dd0e0debb3b3e84498.svg) | 7-Chloro-5-(2,6-dichlorophenyl)-1-methyl-1H-benzo[e][1,4]diazepin-2(3H)-one | IC50 | 181970085.9 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_a061257f9e36cd3e639308594ba0a64f.svg) | 5-(2-Fluorophenyl)-7,8-dichloro-1H-1,4-benzodiazepin-2(3H)-one | IC50 | 277971326.8 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_cbad55800e205e03b07097fcf19dcfa3.svg) | 7-Chloro-5-(2,6-dichlorophenyl)-1,3-dihydro-1,4-benzodiazepin-2-one | IC50 | 142889395.9 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_790b2f102547e621280a8cafcb1217cb.svg) | 5-Phenyl-7-ethenyl-1H-1,4-benzodiazepin-2(3H)-one | IC50 | 41686938.35 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_2ba7269daca0986fd48d7886701b4ff2.svg) | 7,8-Dichloro-1-methyl-5-phenyl-3H-1,4-benzodiazepin-2-one | IC50 | 25003453.62 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_28d74f767daa3700044875978faba54c.svg) | 5-(2-Fluorophenyl)-8-chloro-7-methyl-1H-1,4-benzodiazepin-2(3H)-one | IC50 | 71449632.61 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_1ef2cbf6584c3b10b408824a6c1748c3.svg) | 2H-1,4-Benzodiazepin-2-one, 7-chloro-1-(1,1-dimethylethyl)-1,3-dihydro-5-phenyl- | IC50 | 1614358.56 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_a3f5233318be480c8026d3d121f57187.svg) | Motrazepam | IC50 | 2328091.26 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_a685853812d1619d29f1808292eec4ab.svg) | 7-Ethyl-5-phenyl-1,3-dihydro-1,4-benzodiazepin-2-one | IC50 | 27797132.68 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_3d09ab23796b3585eae73b18d74ef8ee.svg) | 5-(2-Chlorophenyl)-1-methyl-3H-1,4-benzodiazepin-2-one | IC50 | 263026799.2 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_a7589375cd013885f6bf32c7329b1f6d.svg) | (6-Chloro-1,3-benzodioxol-5-yl)methyl 4-(2-oxo-3H-benzimidazol-1-yl)piperidine-1-carboxylate | IC50 | 1040.0 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_0726f23084804a91982ee5278b06529e.svg) | N,N-Dibutyl-2-[6,8-dichloro-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-3-yl]acetamide | Ki | 2.68 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_907352035a912f7d2d8f9bbe9766bff2.svg) | Unii-82MI0GT75Z | Ki | 2.47 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_0c2ce483efe4fbc3d387b73a18e41061.svg) | 2-[4-[4-(3-Methoxyphenyl)piperazin-1-yl]butyl]-4-methyl-1,2,4-triazine-3,5-dione | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_8077712111cba3239d33b40dbaca0eb4.svg) | 1,3-Dihydro-5-(2-fluorophenyl)-2H-1,4-benzodiazepin-2-one | IC50 | 47643098.68 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_1604fa54f37dce19a4c798c394eb43d0.svg) | 7-Bromo-5-(2,6-difluorophenyl)-1-methyl-3H-1,4-benzodiazepin-2-one | IC50 | 416869383.5 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_c626b7cfa61f855f83dfb50a8184cca9.svg) | 2H-1,4-Benzodiazepin-2-one, 5-(2-fluorophenyl)-1,3-dihydro-7-(hydroxyamino)-1-methyl- | IC50 | 10423174.29 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_a50eb5ed185a886aacfad8a9222f0066.svg) | 4-Fluoro-N-methyl-N-(4-(6-(methylamino)pyrimidin-4-yl)-1,3-thiazol-2-yl)benzamide | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_ac98602e4d6dc70935439dd59c0ee661.svg) | 5-(2-Fluorophenyl)-1-methyl-2-oxo-3H-1,4-benzodiazepine-7-carbonitrile | IC50 | 33342641.28 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_d344523f90173552a37ef82d09ab4a4c.svg) | 7-Amino-1-methyl-5-phenyl-1,3-dihydro-2H-1,4-benzodiazepin-2-one | IC50 | 2172701.18 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_663de5ef803d63c650218d1d54191ad8.svg) | 8-Chloro-5-(2,6-difluorophenyl)-1,3-dihydro-2H-1,4-benzodiazepine-2-one | IC50 | 35727283.82 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_f1ca47169afd93e6704a85b828edfd19.svg) | 7-Chloro-5-(2,6-difluorophenyl)-1H-benzo[e][1,4]diazepin-2(3H)-one | IC50 | 625172692.8 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_e00e0297e0f9490227b10dbc9a38b762.svg) | 7-Acetyl-5-(2-fluorophenyl)-1,3-dihydro-2H-1,4-benzodiazepine-2-one | IC50 | 55590425.73 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_3165a243ad66b766d5fca35e28b8d662.svg) | 2H-1,4-Benzodiazepin-2-one, 1,3-dihydro-7-chloro-5-(2-fluorophenyl)-1-(2-hydroxyethyl)- | IC50 | 40831938.63 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_ae72352f36ae9a30ed219a680fd136a5.svg) | 2-Oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepine-7-carbaldehyde | IC50 | 23280912.58 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_07f2bbf4ca5e25877efba9df07c26a30.svg) | 7-Fluoro-5-(2-fluorophenyl)-1,3-dihydro-1,4-benzodiazepin-2-one | IC50 | 135207256.3 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_34a66849dec8bbfed96c5929cf2a6a06.svg) | 3,7-Dichloro-5-(2-fluorophenyl)-1,3-dihydro-1,4-benzodiazepin-2-one | IC50 | 188799134.9 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_fd9f458559c31db207c6d9cd8780c1b4.svg) | 1,7-Dichloro-3-methyl-5-phenyl-3H-1,4-benzodiazepin-2-one | IC50 | 20417379.45 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_fad572126f403ef020fd9e385d485faa.svg) | 5-(2-Fluorophenyl)-8-methyl-1,3-dihydro-1,4-benzodiazepin-2-one | IC50 | 52601726.64 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_45289ba8a0e68555573c3a4a8648b297.svg) | 1-Tert-butyl-5-(2-fluorophenyl)-7-nitro-3H-1,4-benzodiazepin-2-one | IC50 | 3334264.13 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_615864cb852215ebe62950a06952e9a5.svg) | 7-Fluoro-1-methyl-5-phenyl-3H-1,4-benzodiazepin-2-one | IC50 | 58884365.54 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_755aae8338556c56d96e3796c29457eb.svg) | 7-Chloro-5-(2-chloro-6-fluorophenyl)-1,3-dihydro-1,4-benzodiazepin-2-one | IC50 | 333426412.8 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_6049405974dd9e8fe97c449b7e0f3814.svg) | 7-Azido-5-(2-fluorophenyl)-1,3-dihydro-1,4-benzodiazepin-2-one | IC50 | 188799134.9 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_ca5542ab57ac317962251546429bfee0.svg) | 7-Chloro-5-(2,6-difluorophenyl)-1-methyl-1H-benzo[e][1,4]diazepin-2(3H)-one | IC50 | 243781081.8 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_d1bc89cf4542b8d1dff0a4df27e0b4a0.svg) | 5-(2,6-Difluorophenyl)-1,3-dihydro-1,4-benzodiazepin-2-one | IC50 | 52601726.64 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_af26f03bcfe348aa699d199dac691c7c.svg) | N-[(2,5-Dimethoxyphenyl)methyl]-N-(4-fluoro-2-phenoxyphenyl)acetamide | IC50 | 1.6 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_7656a45c616371fb0920f7a5679e1ed9.svg) | (111C)Methyl 2-[(N-acetyl-2-phenoxyanilino)methyl]benzoate | Ki | 1.4 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_8d4bf4c5e0ded6a575c2023e3c25db5c.svg) | (4S)-N,N-Diethyl-9-(2-fluoroethyl)-1,2,3,4-tetrahydrocarbazole-4-carboxamide | Ki | 0.87 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_6aed6fa0d6ef71d2f3ed4ababe554f9e.svg) | 18,19-Dimethoxy-13-methyl-15-phenyl-5,7-dioxa-13-azapentacyclo[10.7.1.02,10.04,8.016,20]icosa-1(20),2,4(8),9,16,18-hexaene | Ki | 2897.0 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_9ff23b3a020dd643ba849b995ccaf566.svg) | 19-[(4-Bromophenyl)methoxy]-18-methoxy-13-methyl-5,7-dioxa-13-azapentacyclo[10.7.1.02,10.04,8.016,20]icosa-1(20),2,4(8),9,16,18-hexaene | Ki | 900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_636f3ed209486d614db3bcf7caa8baac.svg) | N-[(2S)-Butan-2-yl]-1-(2-chlorophenyl)-N-(111C)methylisoquinoline-3-carboxamide | Ki | 4.5 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_e210a60082be53ced3b9631de0ef5be4.svg) | Ethyl (1S,2R,3S,4R,5S)-4-[2-chloro-6-(dicyclopropylmethylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate | Ki | 2100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_e5594886890ed7f32e48d5e5cf26a8d5.svg) | Propyl (1S,2R,3S,4R,5S)-4-[2-chloro-6-(dicyclopropylmethylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate | Ki | 2200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_d52dec49c6a95097b1281472835f36f0.svg) | N-(2-Aminoethyl)-3-[(21S,22S)-16-ethenyl-11-ethyl-4-hydroxy-12,17,21,26-tetramethyl-7,23,24,25-tetrazahexacyclo[18.2.1.15,8.110,13.115,18.02,6]hexacosa-1,4,6,8(26),9,11,13(25),14,16,18(24),19-undecaen-22-yl]propanamide | IC50 | 5600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/translocator-protein_d01558b0c81e7476226af252630b4caf.svg) | N-[6-[3-[(21S,22S)-16-Ethenyl-11-ethyl-4-hydroxy-12,17,21,26-tetramethyl-7,23,24,25-tetrazahexacyclo[18.2.1.15,8.110,13.115,18.02,6]hexacosa-1,4,6,8(26),9,11,13(25),14,16,18(24),19-undecaen-22-yl]propanoylamino]hexyl]-1-(2-iodophenyl)isoquinoline-3-carboxamide | IC50 | 310.0 [1] |