![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_024d4bdd32ee0fe9aad0dd505da4bd7a.svg) | (2R)-2-[[3-Fluoro-6-[4-(trifluoromethyl)cyclohexyl]pyridin-2-yl]methylamino]-3-methylbutan-1-ol | IC50 | 290.0 [1], 310.0 [2], 340.0 [3] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_4acd1b5710e169ef307270f0b01b3162.svg) | 3-[(S)-Hydroxy(pyridin-2-yl)methyl]-1-methyl-3-[4-(trifluoromethyl)pyridin-2-yl]cyclobutan-1-ol | IC50 | 380.0 [1], 930.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_e1021feab62fc1c8885c4150d544a0b3.svg) | 1-(8-Methyl-3,4-dihydro-2H-quinolin-1-yl)-2-[5-(trifluoromethyl)pyridin-2-yl]sulfanylethanone | IC50 | 200.0 [1], 500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_f6525ac136cc05ebb30e726a9813f278.svg) | 2-[3-Chloro-5-(trifluoromethyl)pyridin-2-yl]sulfanyl-1-(8-methyl-3,4-dihydro-2H-quinolin-1-yl)ethanone | IC50 | 200.0 [1], 500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_c068fd6e827a160cd815542e6d2784f7.svg) | 2-(3-Chloro-pyridin-2-ylsulfanyl)-1-(8-methyl-3,4-dihydro-2H-quinolin-1-yl)-ethanone | IC50 | 200.0 [1], 1000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_3e9ce218f5b7558703ced128093e3c91.svg) | 2-(5-Chloro-pyridin-2-ylsulfanyl)-1-(8-methyl-3,4-dihydro-2H-quinolin-1-yl)-ethanone | IC50 | 500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_196f7f130a3fc05d83b0ca4bb9f48d9b.svg) | 1-(8-Methyl-3,4-dihydro-2H-quinolin-1-yl)-2-[3-(trifluoromethyl)pyridin-2-yl]sulfanylethanone | IC50 | 1000.0 [1], 5000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_a16a0f3d3e635205490765eaeae09a3e.svg) | 1-(3,4-Dihydro-2H-quinolin-1-yl)-2-[5-(trifluoromethyl)pyridin-2-yl]sulfanylethanone | IC50 | 1000.0 [1], 5000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_8542e1e9367796ed3ffd7923f49e9cda.svg) | 1-(8-Methyl-3,4-dihydro-2H-quinolin-1-yl)-2-pyridin-2-ylsulfanylethanone | IC50 | 5000.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_0ff5bf646acd0931fb79136274ec825f.svg) | 2-(5-Chloropyridin-2-yl)sulfanyl-1-(3,4-dihydro-2H-quinolin-1-yl)ethanone | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_56520dc0e151d6a709ebb9b75a5d1d37.svg) | 1-(8-Methyl-3,4-dihydro-2H-quinolin-1-yl)-2-(5-methylpyridin-2-yl)sulfanylethanone | IC50 | 5000.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_e16692eb1d58a8131aea5b6061eaab93.svg) | 6-[2-(8-Methyl-3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]sulfanylpyridine-3-carbonitrile | IC50 | 5000.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_59cb41e914b29dbf1f7534daa824c2f6.svg) | 2-[3-Fluoro-5-(trifluoromethyl)pyridin-2-yl]sulfanyl-1-(8-methyl-3,4-dihydro-2H-quinolin-1-yl)ethanone | IC50 | 200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_559d27f8bc8e0f39f8a90f05e2560ebc.svg) | 2-(3,5-Dichloropyridin-2-yl)sulfanyl-1-(8-methyl-3,4-dihydro-2H-quinolin-1-yl)ethanone | IC50 | 200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_8e2b2d433d6c77b8f57ab261c9606566.svg) | 2-[2-(8-Methyl-3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]sulfanylpyridine-3-carbonitrile | IC50 | 500.0 [1], 1000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_2a14eead92d88975250022132477ad32.svg) | 2-[2-(8-Methyl-3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]sulfanylpyridine-4-carbonitrile | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_034501e544f936ffaa222faab3d939eb.svg) | 2-(3-Chloropyridin-2-yl)sulfanyl-1-(8-methoxy-3,4-dihydro-2H-quinolin-1-yl)ethanone | IC50 | 500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_623866af6f6e63c5e867276116f2951c.svg) | 2-(3,4-Dimethylpyridin-2-yl)sulfanyl-1-(8-methyl-3,4-dihydro-2H-quinolin-1-yl)ethanone | IC50 | 1000.0 [1], 5000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_eb87550649ad00326e5accc6430373d0.svg) | 2-(4,5-Dimethylpyridin-2-yl)sulfanyl-1-(8-methyl-3,4-dihydro-2H-quinolin-1-yl)ethanone | IC50 | 200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_4500d425893295a7ebb523fdc58d87d1.svg) | 2-(5-Bromopyridin-2-yl)sulfanyl-1-(8-methyl-3,4-dihydro-2H-quinolin-1-yl)ethanone | IC50 | 500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_bb786143ec1711c17142ecedef3a4009.svg) | 2-[3-Ethyl-5-(trifluoromethyl)pyridin-2-yl]sulfanyl-1-(8-methyl-3,4-dihydro-2H-quinolin-1-yl)ethanone | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_eb6c485649d0d69819dab7645fa59340.svg) | Methyl 5-chloro-6-[2-(8-methyl-3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]sulfanylpyridine-3-carboxylate | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_4c05926d5ee65b1a2488e4715d630b32.svg) | 2-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetrahydro-7H-purin-7-yl)-N-(4-isopropylphenyl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_a170766a13421b500d531de7cca1ed1b.svg) | (1e,3e)-1-(4-Fluorophenyl)-2-methylpent-1-en-3-one oxime | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_d33ec2b41b84fafe803d97bde6190274.svg) | N-[2-Methyl-3-[[4-[4-[[4-(trifluoromethoxy)phenyl]methoxy]piperidin-1-yl]-1,3,5-triazin-2-yl]amino]phenyl]acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_8c0f69451571d53b87466f5412a0bb13.svg) | CID 121513880 | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_1d226f0717081ae918932605a0972ba7.svg) | (R)-8-{5-[3-Methyl-4-(trifluoromethyl)phenyl]oxazol-2-ylamino}-1,2,3,4-tetrahydronaphthalen-2-ol | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_49c3c24301c59374b5a41fb82201154f.svg) | 4-[3-(3-Methoxypropoxy)phenyl]-2-sulfanylidene-3,4-dihydro-1H-indeno[1,2-d]pyrimidin-5-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_2232b95e8a4b104b8e5c49e7d90dd33e.svg) | N-[2-[4-(Difluoromethoxy)phenyl]ethyl]-2-(8-methyl-4-oxoquinazolin-3-yl)acetamide | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_f47107dd1a290f5d23ff15724fa3fcc2.svg) | 6-[[(S)-(3-Fluoropyridin-2-yl)-[3-fluoro-4-(trifluoromethoxy)phenyl]methyl]carbamoyl]pyridine-3-carboxylic acid | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_71e649856a43295bf3899dabbfe4b67e.svg) | 5-[2-(Trifluoromethyl)phenyl]-1H-indazole | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_37c2d307d957fd1847f42a31adde17ad.svg) | 6-Chloro-5-[2-(trifluoromethyl)phenyl]-1H-indazole | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_6ab0fa8b8e8548d2c5ce42cbf8dd5202.svg) | 6-Methyl-5-[2-(trifluoromethyl)phenyl]-1H-indazole | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_ec4cab99f8253e22d2190100af238a9d.svg) | 6-Methoxy-5-[2-(trifluoromethyl)phenyl]-1H-indazole | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_7eeb5e806b5a6bf3f40bbe00ba83b941.svg) | 6-(Cyclopropylmethoxy)-5-[2-(trifluoromethyl)phenyl]-1H-indazole | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_b9c4ec0e06b2cf15e9cffc8f38153cc5.svg) | 6-(Trifluoromethoxy)-5-[2-(trifluoromethyl)phenyl]-1H-indazole | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_ee6b044f92e387fba11f05b9ac85efe4.svg) | 2-(1,3-Dimethyl-2,4-dioxoquinazolin-5-yl)-N-[4-[4-(2-methylpropoxy)phenyl]-1,3-thiazol-2-yl]acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_3450a15c568f696a41c2348692d78940.svg) | N-[4-[3,5-Difluoro-4-(3,3,3-trifluoropropyl)phenyl]-1,3-thiazol-2-yl]-2-(1,3-dimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_57f2a8118b55392b954664bc05b815c2.svg) | N-[4-(4-Bromophenyl)-1,3-thiazol-2-yl]-2-(5-methyl-4-oxo-7,8-dihydroimidazo[2,1-b]purin-3-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_a58d86b0fdfe0d31a0b33daa0a6c3a35.svg) | N-[4-(4-Tert-butylphenyl)-1,3-thiazol-2-yl]-2-(5-methyl-4-oxo-7,8-dihydroimidazo[2,1-b]purin-3-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_7673004507e9423f522602ccb44ae063.svg) | 2-(6-Chlorospiro[3,4-dihydrochromene-2,1'-cyclobutane]-4-yl)-N-[(2-cyclopentyloxy-3-methoxyphenyl)methyl]acetamide | IC50 | 725.3 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_545e361f6d2cd395bf1606a49621175e.svg) | N-[4-(5-Chloro-2-fluorophenyl)-1,3-thiazol-2-yl]-2-(1,3-dimethyl-2,4-dioxoquinazolin-5-yl)acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_06316a71d820ab6924308fb982add803.svg) | N-[4-(3,4-Dichlorophenyl)-1,3-thiazol-2-yl]-2-(1,3-dimethyl-2,4-dioxoquinazolin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_75962d516f3e6b9e2de47491b5ef10b2.svg) | N-[4-(3-Chloro-2-fluorophenyl)-1,3-thiazol-2-yl]-2-(1,3-dimethyl-2,4-dioxoquinazolin-5-yl)acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_590a954b5606c59c78d24ae20e14d7a0.svg) | N-[4-(3-Chloro-4-fluorophenyl)-1,3-thiazol-2-yl]-2-(1,3-dimethyl-2,4-dioxoquinazolin-5-yl)acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_625379b813d6c5fda546721d14ea0e16.svg) | N-[4-[3,5-Difluoro-4-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]-2-(1,3-dimethyl-2,4-dioxoquinazolin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_480887728cf28aba5aed941ec118612e.svg) | N-[4-[2,4-Difluoro-3-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]-2-(1,3-dimethyl-2,4-dioxoquinazolin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_0c7756ae4277a0d3ccfb71c3580ac38c.svg) | N-[4-[2,3-Difluoro-4-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]-2-(1,3-dimethyl-2,4-dioxoquinazolin-5-yl)acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_a4619a3e3091c61e49708f9c55739636.svg) | N-[4-[3,5-Difluoro-4-(2,2,2-trifluoroethoxy)phenyl]-1,3-thiazol-2-yl]-2-(1,3-dimethyl-2,4-dioxoquinazolin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_663d533efdfe105df613e1c8a6c0e043.svg) | 2-(1,3-Dimethyl-2,4-dioxoquinazolin-5-yl)-N-[4-[4-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_da1ebfe652c529799c60a8a226cbf2cf.svg) | N-[1-(4-Chlorophenyl)pyrazol-3-yl]-2-(1,3-dimethyl-2,4-dioxoquinazolin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_f6d31d19757ce59f878e3c460716e063.svg) | N-[4-(3-Chlorophenyl)-1,3-thiazol-2-yl]-2-(1,3-dimethyl-2,4-dioxoquinazolin-5-yl)acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_2a1976d86e525d47bd6effceba46da75.svg) | 2-(1,3-Dimethyl-2,4-dioxoquinazolin-5-yl)-N-[4-(4-iodophenyl)-1,3-thiazol-2-yl]acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_ef18f9d2544f0cbde63ca487514a1c96.svg) | 2-(1,3-Dimethyl-2,4-dioxoquinazolin-5-yl)-N-[1-[3-(trifluoromethyl)phenyl]pyrazol-3-yl]acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_29f82da444e05ece0a9d8220a7f6666e.svg) | N-[4-(4-Bromophenyl)-1,3-thiazol-2-yl]-2-(1,3-dimethyl-2,4-dioxoquinazolin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_68b2afc7f4a3ccd37128d14be88b30de.svg) | 2-(1,3-Dimethyl-2,4-dioxoquinazolin-5-yl)-N-[4-[3-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]acetamide | IC50 | 2100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_acc64978c82c95e4446260cf70b955f2.svg) | N-[4-(4-Cyclohexylphenyl)-1,3-thiazol-2-yl]-2-(1,3-dimethyl-2,4-dioxoquinazolin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_48b28d67705e7a2bd7f87094bb07a414.svg) | 2-(1,3-Dimethyl-2,4-dioxoquinazolin-5-yl)-N-[4-[3-(trifluoromethoxy)phenyl]-1,3-thiazol-2-yl]acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_d15880effa792e4ae95ed7a886787f5c.svg) | N-[4-(4-Tert-butylphenyl)-1,3-thiazol-2-yl]-2-(1,3-dimethyl-2,4-dioxoquinazolin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_2c82e0976175bf8903cd58cc26330a56.svg) | 2-(1,3-Dimethyl-2,4-dioxoquinazolin-5-yl)-N-[4-[4-(3-methylbutoxy)phenyl]-1,3-thiazol-2-yl]acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_8909e28e5f07c5ffcf273b1ec9b476dd.svg) | N-[4-(2,4-Difluorophenyl)-1,3-thiazol-2-yl]-2-(1,3-dimethyl-2,4-dioxoquinazolin-5-yl)acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_be55f44508210aa41ff3a5e672ae5a0e.svg) | 2-(1,3-Dimethyl-2,4-dioxoquinazolin-5-yl)-N-[4-(4-methylphenyl)-1,3-thiazol-2-yl]acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_dcc0985e865bb5decef0d20aa94571d9.svg) | 2-(1,3-Dimethyl-2,4-dioxoquinazolin-5-yl)-N-[4-(4-propan-2-ylphenyl)-1,3-thiazol-2-yl]acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_26529edbb2e0055218f7bcbb3acb7447.svg) | N-[4-(2,3-Difluorophenyl)-1,3-thiazol-2-yl]-2-(1,3-dimethyl-2,4-dioxoquinazolin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_db80cf7b6ed9178cce01826dcc033247.svg) | 2-(1,3-Dimethyl-2,4-dioxoquinazolin-5-yl)-N-[4-[3-fluoro-4-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_8f6f4b1bc5d172a7bce6976ed2a4abdb.svg) | 2-(1,3-Dimethyl-2,4-dioxoquinazolin-5-yl)-N-[4-[4-fluoro-3-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_1da14af78ab9bf541b4f289aedcdd1fd.svg) | 2-(1,3-Dimethyl-2,4-dioxoquinazolin-5-yl)-N-[4-[2-fluoro-4-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_c79e5738a095f900bfacd44baa81317e.svg) | N-[4-[4-Chloro-3-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]-2-(1,3-dimethyl-2,4-dioxoquinazolin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_6ab2f51001ebd3f212d82b01d9f7287d.svg) | N-[4-[3,5-Dichloro-4-(2,2-dimethylpropoxy)phenyl]-1,3-thiazol-2-yl]-2-(4,6-dimethyl-5,7-dioxopyrazolo[4,3-d]pyrimidin-1-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_a8f8fc36daa348d71e12774af80f51cb.svg) | 2-(5,7-Dimethyl-4,6-dioxo-[1,2]thiazolo[5,4-d]pyrimidin-3-yl)-N-[4-[3-fluoro-5-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_0f0a70700767490d50bb6030154e5f1b.svg) | 2-(1,3-Dimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)-N-[4-[3-fluoro-4-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_40f40db4a453117ba6289a1a32f7a313.svg) | 2-(1,3-Dimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)-N-[4-[4-fluoro-3-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_f715ae989fadd114ad600b6e0e31ffa7.svg) | 2-(1,3-Dimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)-N-[4-[2-fluoro-3-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_9f54116f254b510df7406449fa93a465.svg) | 2-(1,3-Dimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)-N-[4-[3-fluoro-5-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_43c39a5e55e1a894d31ec9c9a902b580.svg) | N-[4-[3,5-Dichloro-4-(2,2,2-trifluoroethoxy)phenyl]-1,3-thiazol-2-yl]-2-(1,3-dimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_a5897e14171f28da17e50d7f5fa76c78.svg) | N-[4-[3-Chloro-5-fluoro-4-(2,2,2-trifluoroethoxy)phenyl]-1,3-thiazol-2-yl]-2-(1,3-dimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_3fb2b9a754126b05582e8de8b707ed41.svg) | N-[4-[3,5-Difluoro-4-(2-methylpropoxy)phenyl]-1,3-thiazol-2-yl]-2-(1,3-dimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_9d09e5ff846628d74f280dc130776dfb.svg) | N-[4-[4-Fluoro-3-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]-2-(1,3,6-trimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_66fa8c44d193f62b6f663a1c252a437e.svg) | N-[4-[2-Fluoro-4-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]-2-(1,3,6-trimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_e72ffe804d78da59512a6ce2ab46fd3c.svg) | N-[4-[2-Fluoro-3-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]-2-(1,3,6-trimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_e2115fe6036e253da28c041e2ab0b65b.svg) | N-[4-[3-Fluoro-5-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]-2-(1,3,6-trimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_b241c5bff96c437df2d2e5b13bb89484.svg) | N-[4-[4-Chloro-3-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]-2-(1,3,6-trimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_c137b273ed1e972cc3343649d091c1bc.svg) | N-[4-[3-Fluoro-4-(trifluoromethoxy)phenyl]-1,3-thiazol-2-yl]-2-(1,3,6-trimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_812be28b7454cfda33d08e0dc013b525.svg) | N-[4-[4-Fluoro-3-(trifluoromethoxy)phenyl]-1,3-thiazol-2-yl]-2-(1,3,6-trimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_379c3e0374412b43a38cfdb580fb624d.svg) | N-[4-[4-Chloro-3-(trifluoromethoxy)phenyl]-1,3-thiazol-2-yl]-2-(1,3,6-trimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_01906e189960c435af40fa93dfe6bd59.svg) | N-[4-[3-Chloro-4-(trifluoromethoxy)phenyl]-1,3-thiazol-2-yl]-2-(1,3,6-trimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 4450.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_5d1f248b6cea196305aef49e2fb46bb3.svg) | N-[4-[3-Chloro-4-(2,2,2-trifluoroethoxy)phenyl]-1,3-thiazol-2-yl]-2-(1,3,6-trimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_25aed614c209f6bbc9f16bae5dda3619.svg) | N-[4-[4-(2,2-Dimethylpropoxy)-3,5-difluorophenyl]-1,3-thiazol-2-yl]-2-(1,3,6-trimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_474ce8d59fa96381ed40609c7a807ec5.svg) | N-[4-[3,5-Dichloro-4-(2-methylpropoxy)phenyl]-1,3-thiazol-2-yl]-2-(1,3,6-trimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_ab60bde3288daf6aa3c21901770a76d1.svg) | N-[4-[2,4-Difluoro-3-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]-2-(1,3,6-trimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_d37b0beae2cc822036f8528f1535692e.svg) | N-[4-[3,5-Difluoro-4-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]-2-(1,3,6-trimethyl-2,4-dioxofuro[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_b5e70870a12f197720728602d551a122.svg) | N-[4-[2,4-Difluoro-3-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]-2-(1,3-dimethyl-2,4-dioxothieno[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_f5ce10e462ac25f7a41d5adaf1d6a581.svg) | 2-(6-Ethyl-1,3-dimethyl-2,4-dioxothieno[2,3-d]pyrimidin-5-yl)-N-[4-[3-fluoro-4-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_3bfe3da11501c60cdd55c9db334ab92c.svg) | N-[4-[4-(Difluoromethoxy)-3,5-difluorophenyl]-1,3-thiazol-2-yl]-2-(6-ethyl-1,3-dimethyl-2,4-dioxothieno[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_6d9767edeec047695fee2445d1dc500e.svg) | 2-(1,3-Dimethyl-2,4-dioxo-6-propan-2-ylthieno[2,3-d]pyrimidin-5-yl)-N-[4-[3-fluoro-4-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_b3111eee2420480dc12ed853e70d3547.svg) | N-[4-(3,4-Dichlorophenyl)-1,3-thiazol-2-yl]-2-(1,3,6-trimethyl-2,4-dioxothieno[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_ee017368e91ce47d456b371fa787ca9c.svg) | N-[4-[3,5-Difluoro-4-(2,2,2-trifluoroethoxy)phenyl]-1,3-thiazol-2-yl]-2-(6-ethyl-1,3-dimethyl-2,4-dioxothieno[2,3-d]pyrimidin-5-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_34ac24c05ecff47cedff4aa879708f68.svg) | N-[4-[3-Chloro-4-(trifluoromethoxy)phenyl]-1,3-thiazol-2-yl]-2-(5,7-dimethyl-4,6-dioxo-[1,2]thiazolo[5,4-d]pyrimidin-3-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_4841b0c4f448c46d08043f4ec9dfe541.svg) | N-[4-[2,4-Difluoro-3-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]-2-(5,7-dimethyl-4,6-dioxo-[1,2]thiazolo[5,4-d]pyrimidin-3-yl)acetamide | IC50 | 1770.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-v-member-3_4fbf628d2dabc6b7a961019feb053d91.svg) | N-[4-[2,3-Difluoro-4-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]-2-(5,7-dimethyl-4,6-dioxo-[1,2]thiazolo[5,4-d]pyrimidin-3-yl)acetamide | IC50 | 2830.0 [1] |