![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_1b4ef0d9148634ae24bca565168a335c.svg) | CID 16095384 | IC50 | 4.0 [1], 160.0 [2], 190.0 [3] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_afc740352ad46086513c07d55f0d1636.svg) | Menthol | IC50 | 19000.0 [1], 92000.0 [2], 520000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_55a7d57ce9c848a2ae7c233a49d58f5f.svg) | 4-({[4-Fluoro-3-(trifluoromethyl)phenyl]methyl}(3-methyl-1-benzothiophen-2-yl)sulfamoyl)benzoic acid | IC50 | 4.0 [1], 5.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_dbb67602db744b0f86fd55c9a4b416b6.svg) | 5-Methoxytryptamine | IC50 | 11600.0 [1], 12400.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_7e3e6f52432e393cb82af4575833e227.svg) | Bctc | IC50 | 475.0 [1], 800.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_9e841b26436884b87d30ee562e8c3272.svg) | 5-Fluorotryptamine | IC50 | 12300.0 [1], 13100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_2ee404c25cd73701f83ae5379b2af6fe.svg) | 5-Benzyloxytryptamine | IC50 | 340.0 [1], 660.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_525b581ac6f7a94edf0df42582cabb33.svg) | 5-Chlorotryptamine | IC50 | 21500.0 [1], 32200.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_2078c8f152ad9cf653a3862fb974e6a5.svg) | 5-Bromotryptamine | IC50 | 22700.0 [1], 30400.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_f133aa240b161f2f4ae6eebadf466492.svg) | 3-[4-(Trifluoromethyl)-6-[2-(trifluoromethyl)phenyl]-1H-benzimidazol-2-yl]-1-oxa-2-azaspiro[4.5]dec-2-ene | IC50 | 0.41 [1], 3.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_815ea42af187fc11d3ec5512e380a68e.svg) | 7-Benzyloxytryptamine | IC50 | 3340.0 [1], 8930.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_9af6d8882cb8143dc7e5f025ca087dd0.svg) | 1H-Indole-3-ethanamine, N,N'-dimethyl-5-(phenylmethoxy)- | IC50 | 5630.0 [1], 5960.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_9ca616945d9bc539db1e007810c5ae2c.svg) | CID 60195662 | IC50 | 103.0 [1], 181.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_7884fbef047fedd8518f2446cd39b4aa.svg) | Ethyl {2-[5-(benzyloxy)-1H-indol-3-yl]ethyl}carbamate | IC50 | 21600.0 [1], 28800.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_e4d8ef6ff72854033e15a20580fc8b9e.svg) | 2-(5-Benzyloxy-2-methyl-1H-indol-3-yl)-ethylamine | IC50 | 1500.0 [1], 2360.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_2d71f0b8c8b4f61dcf19c68c1aaeebfe.svg) | 4-[(3-Methyl-1-benzothiophen-2-yl)-[[4-(trifluoromethoxy)phenyl]methyl]sulfamoyl]benzoic acid | IC50 | 1.4 [1], 1.8 [2] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_90de930cbc88fc4d289f538755fdc916.svg) | Capsazepine | IC50 | 18000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_4c05926d5ee65b1a2488e4715d630b32.svg) | 2-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetrahydro-7H-purin-7-yl)-N-(4-isopropylphenyl)acetamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_de6e155f8ff8d9b4ce06aca7e7507d0f.svg) | N-(p-Amylcinnamoyl)anthranilic acid | IC50 | 3900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_fdf921beff8ce7a71de0eab04f245344.svg) | 7-Bromo-N-(1-phenylcyclopropyl)-3-[(4-piperidin-1-ylpiperidin-1-yl)methyl]-2-[3-(trifluoromethyl)phenyl]quinoline-4-carboxamide | IC50 | 25000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_d33ec2b41b84fafe803d97bde6190274.svg) | N-[2-Methyl-3-[[4-[4-[[4-(trifluoromethoxy)phenyl]methoxy]piperidin-1-yl]-1,3,5-triazin-2-yl]amino]phenyl]acetamide | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_8c0f69451571d53b87466f5412a0bb13.svg) | CID 121513880 | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_670d192c1b4ab8bd7b14601ec118eaa5.svg) | CID 49783953 | IC50 | 8.3 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_743cf494aabf4b4791b5357c7ec770c1.svg) | (8R)-8-[4-(Trifluoromethyl)phenyl]-N-[(2S)-1,1,1-trifluoropropan-2-yl]-6,8-dihydro-5H-1,7-naphthyridine-7-carboxamide | IC50 | 25.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_1d226f0717081ae918932605a0972ba7.svg) | (R)-8-{5-[3-Methyl-4-(trifluoromethyl)phenyl]oxazol-2-ylamino}-1,2,3,4-tetrahydronaphthalen-2-ol | IC50 | 44000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_e919a302d7ec9afeff48324f4926963c.svg) | (1R)-N-(4-Fluorophenyl)-1-[4-(trifluoromethyl)phenyl]-3,4-dihydro-1H-isoquinoline-2-carboxamide | IC50 | 36.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_17ded7d13509f3179d0da7193df93afd.svg) | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(3-methylphenyl)methyl]benzamide | IC50 | 870.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_15edf8a322671dba8be2f440b0ccc473.svg) | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[[3-(trifluoromethyl)phenyl]methyl]benzamide | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_61bb054a0298bc17fbc68a83cfebf251.svg) | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1R)-1-(3-methoxyphenyl)ethyl]benzamide | IC50 | 240.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_0e809749e581351c240338b1a08846b7.svg) | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1R)-1-(3-chlorophenyl)ethyl]benzamide | IC50 | 400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_58b12812d29addc9b68dc237cc732ad0.svg) | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1S)-1-(3-methoxyphenyl)ethyl]benzamide | IC50 | 43000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_35e26bb838a99a0382ab92353068c87a.svg) | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1R)-1-phenylpropyl]benzamide | IC50 | 19000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_3e045d48b1eab55d8024f90b7630e851.svg) | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1R)-1-(3,5-difluorophenyl)ethyl]benzamide | IC50 | 80.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_59f6a469a02f957aabc3b6f413d7e92a.svg) | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(2-chlorophenyl)methyl]benzamide | IC50 | 5600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_c7a0c567343d44f1a8cedab11dec0412.svg) | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(4-chlorophenyl)methyl]benzamide | IC50 | 28000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_873d4f93914622a4a5543878ab429291.svg) | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1R)-1-(3-chlorophenyl)ethyl]-2-hydroxybenzamide | IC50 | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_7e239a0978b184cb075028deef38447e.svg) | (2R)-2-[(3-Methoxyphenyl)methyl-(2-phenylacetyl)amino]-2-phenylacetamide | IC50 | 19000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_c0ca81bdfc62351eb4df3207eeae43b7.svg) | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(3-fluorophenyl)methyl]benzamide | IC50 | 8100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_ce471a2e7c44a29504a900d100b364c3.svg) | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-benzylbenzamide | IC50 | 11000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_0bfda88e0ead1fca99c1144d3ba0abf3.svg) | N-[(1R)-2-Amino-2-oxo-1-pyridin-3-ylethyl]-N-[(1R)-1-(3-chlorophenyl)ethyl]benzamide | IC50 | 4100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_c52bf05f6c8a1418ac2166c7dea90ca7.svg) | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1R)-1-(3-chlorophenyl)ethyl]-3-methylbenzamide | IC50 | 2100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_c370e67db7749e20d42e2024b2cce35e.svg) | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1R)-1-(3-chlorophenyl)ethyl]-4-methylbenzamide | IC50 | 850.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_034f2a5d2a2e32b1f560cc8e54b92c4f.svg) | N-[(2R)-1-Amino-1-oxo-3-phenylpropan-2-yl]-N-[(3-methoxyphenyl)methyl]thiophene-2-carboxamide | IC50 | 37000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_7b0719be771afdb161a9dc0b0d9340d2.svg) | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(3-methoxyphenyl)methyl]thiophene-2-carboxamide | IC50 | 1700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_dd4dc380f1fa600ea7600472c8ab3c2d.svg) | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[[3-(trifluoromethoxy)phenyl]methyl]benzamide | IC50 | 4700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_b9967f65fc88a5a1bf69f22179462879.svg) | N-[(1S)-2-Amino-2-oxo-1-phenylethyl]-N-[(3-methoxyphenyl)methyl]thiophene-2-carboxamide | IC50 | 54000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_ffa0bf6a3ac0f97a15d0f72f576450ec.svg) | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1R)-1-(3-chlorophenyl)ethyl]-2-methylbenzamide | IC50 | 390.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_9037ae2e2ca56c61d3d09935d0944c08.svg) | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(3-chlorophenyl)methyl]benzamide | IC50 | 3000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_91853a438e783dd123583d575552e81b.svg) | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1R)-1-(3-chloro-5-fluorophenyl)ethyl]benzamide | IC50 | 180.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_690b132fecf46acfc30646f41b5e1d1c.svg) | 2-[Benzyl-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]sulfamoyl]benzoic acid | IC50 | 15974.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_ad4f4f8052303769020e2172e11215cc.svg) | 4-[Benzyl-(3-chloro-5-cyanopyridin-2-yl)sulfamoyl]benzoic acid | IC50 | 23782.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_41b7b0aa1f819e98724f1a8a75b2d71e.svg) | 4-[Benzyl-[3-cyano-5-(trifluoromethyl)pyridin-2-yl]sulfamoyl]benzoic acid | IC50 | 2472.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_bb4a6097883e4568e6886412803fbd13.svg) | 4-[Benzyl-[5-chloro-3-(trifluoromethyl)pyridin-2-yl]sulfamoyl]benzoic acid | IC50 | 1562.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_0f6bb05d9117db8cde3d91803b8a64d9.svg) | 4-[(4-Acetamidophenyl)methyl-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]sulfamoyl]benzoic acid | IC50 | 18216.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_d20ab9e7e3ab704ce860636156f7cbab.svg) | 3-[[[2-(3-Chlorophenyl)acetyl]-[(1R)-1-(4-fluorophenyl)ethyl]amino]methyl]benzoic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_840c732b7e7f8dbd4ba10b9c5550ffe6.svg) | 3-[[[(1R)-1-(4-Fluorophenyl)ethyl]-(3-phenylbenzoyl)amino]methyl]benzoic acid | IC50 | 837.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_3dcb9c1a19db410a8ebccdcb06484280.svg) | 3-[[[(1R)-1-(4-Fluorophenyl)ethyl]-(1H-pyrrolo[2,3-c]pyridine-5-carbonyl)amino]methyl]benzoic acid | IC50 | 951.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_b514051d0a7fa76bb9220a2de86e4c53.svg) | 3-[[Cinnoline-3-carbonyl-[(1R)-1-(4-fluorophenyl)ethyl]amino]methyl]benzoic acid | IC50 | 340.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_1ad3c22c3cca5eea6c1648c2d87e853d.svg) | 3-[[[(1R)-1-(4-Fluorophenyl)ethyl]-(imidazo[1,2-a]pyridine-2-carbonyl)amino]methyl]benzoic acid | IC50 | 307.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_e82439a80a28993969c86801b91d1d4b.svg) | 3-[[[(1R)-1-(4-Fluorophenyl)ethyl]-(4-phenoxybenzoyl)amino]methyl]benzoic acid | IC50 | 6166.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_e7d906f53b1c2e1675824f4ceeecb650.svg) | 5-[[[(1R)-1-(4-Fluorophenyl)ethyl]-(quinoline-3-carbonyl)amino]methyl]-2-methylbenzoic acid | IC50 | 7820.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_fdba7b64ba7ff50750034a1974ffc642.svg) | 2-[3-[[[(1R)-1-(4-Fluorophenyl)ethyl]-(quinoline-3-carbonyl)amino]methyl]phenyl]acetic acid | IC50 | 3249.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_681e774966fc4fef1bf2b8956f42ee4a.svg) | N-[(1R)-1-(4-Fluorophenyl)ethyl]-N-[[3-(2H-tetrazol-5-yl)phenyl]methyl]quinoline-3-carboxamide | IC50 | 1613.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_f2f6788cb2ff33e0307cd07d502c790e.svg) | 3-[[(4-Fluorophenyl)methyl-(quinoline-3-carbonyl)amino]methyl]benzoic acid | IC50 | 9356.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_e2d39117fa1fda0bbaf05cf72f447373.svg) | 3-[[[(1S)-2-Hydroxy-1-phenylethyl]-(quinoline-3-carbonyl)amino]methyl]benzoic acid | IC50 | 6863.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_ee98556e4ff1766621b6fb906a5344d2.svg) | 3-[[[(1R)-1-(2,4-Difluorophenyl)ethyl]-(quinoline-3-carbonyl)amino]methyl]benzoic acid | IC50 | 288.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_9e0ac831ec1ae60ee4d8d0b73113b1f2.svg) | 3-[[2-(4-Fluorophenyl)propan-2-yl-(quinoline-3-carbonyl)amino]methyl]benzoic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_4705e160eb96ab0d7401046557df5054.svg) | 3-[[1-(4-Methoxyphenyl)ethyl-(quinoline-3-carbonyl)amino]methyl]benzoic acid | IC50 | 6104.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_a1251e4a39bc5270f5d0c75a0a973194.svg) | 6-[[[(1R)-1-(2,4-Difluorophenyl)ethyl]-(isoquinoline-3-carbonyl)amino]methyl]pyridine-2-carboxylic acid | IC50 | 190.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_598e6cae054ea60e13b795bf471b8c0f.svg) | (2S,4R,5S)-4-Fluoro-1-(4-fluorophenyl)sulfonyl-N-[[5-fluoro-2-[2-(trifluoromethyl)pyrimidin-5-yl]pyridin-4-yl]methyl]-5-methylpyrrolidine-2-carboxamide | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_ae4d1fc664b83e73af8381513ba5eb9d.svg) | 2-Amino-N-[(1R)-2-amino-2-oxo-1-phenylethyl]-N-[(1R)-1-(3-chlorophenyl)ethyl]benzamide | IC50 | 420.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_7202d15335cbaeab5d901975233af89d.svg) | 2-[Benzoyl-[(3-methoxyphenyl)methyl]amino]-2-phenylacetic acid | IC50 | 59000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_af97979b069a8635a4eaa2f46ba1eb28.svg) | N-[(1R)-2-(Dimethylamino)-2-oxo-1-phenylethyl]-N-[(3-methoxyphenyl)methyl]benzamide | IC50 | 86000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_7cf1b3335539e04fb7eec931531ed2d8.svg) | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1R)-1-(3-chlorophenyl)ethyl]pyridine-3-carboxamide | IC50 | 2500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_73ebc0c64bd1494b316e0b79cf521e47.svg) | N-[(2R)-1-Amino-1-oxopropan-2-yl]-N-[(3-methoxyphenyl)methyl]benzamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_40feb7d008fc63cefbefbaf6c5ffb7db.svg) | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[[4-[(4-fluorophenyl)methoxy]-3-methoxyphenyl]methyl]thiophene-2-carboxamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_656bd3f5a1cc7e774fbeaa4ff2514849.svg) | N-(2-Amino-2-oxoethyl)-N-[[4-[(4-fluorophenyl)methoxy]-3-methoxyphenyl]methyl]thiophene-2-carboxamide | IC50 | 9100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_8272880ac9cd74ba9fd39ccdb62a10ac.svg) | N-[(3-Methoxyphenyl)methyl]-N-[(1R)-2-(methylamino)-2-oxo-1-phenylethyl]benzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_648ece7b7776412e94c22582607d0e52.svg) | Methyl (2R)-2-[benzoyl-[(3-methoxyphenyl)methyl]amino]-2-phenylacetate | IC50 | 210.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_5022f7729dde6785cadadbeb2b57e139.svg) | 4-[(3S,4R)-1-(2,4-Dichlorophenyl)sulfonyl-4-hydroxy-4-(hydroxymethyl)pyrrolidin-3-yl]oxy-2-fluorobenzonitrile | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_a5f80e0071a3ac21be7645cac39ae0be.svg) | N-[(S)-(2-Methylphenyl)-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamide | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_31cd25eae44d5060827bbbd9ff4c57d4.svg) | N-[(R)-1,3-Thiazol-2-yl-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_945dbe7997817252488b35683dbfa22a.svg) | N-[(S)-Pyridin-2-yl-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_510fded7edce253f97691e1224f2bf50.svg) | Quinolin-6-yl-[(1R)-1-[4-(trifluoromethyl)phenyl]-3,4-dihydro-1H-isoquinolin-2-yl]methanone | IC50 | 390.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_8e7b96c98eeb70a41eecec57d61a3925.svg) | N-[(S)-[3-Fluoro-4-(trifluoromethyl)phenyl]-[2-(trifluoromethyl)phenyl]methyl]quinoline-7-carboxamide | IC50 | 109.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_91d8be15fc142038a38c27665f79c33b.svg) | N-[(S)-Cyclohexyl-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamide | IC50 | 301.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_7da78cad454545659cb019ea1b08cfb9.svg) | N-[(S)-[4-(Trifluoromethyl)phenyl]-[4-(trifluoromethyl)pyridin-3-yl]methyl]quinoline-7-carboxamide | IC50 | 311.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_c208fd9ef34db1047a5f4ac41e3dfbe8.svg) | N-[(1S)-2-Phenyl-1-[3-(trifluoromethyl)pyridin-2-yl]ethyl]quinoline-7-carboxamide | IC50 | 1140.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_b508876e63d55e2c10bfc656ce26d747.svg) | (5R)-N-(4-Fluorophenyl)-5-[4-(trifluoromethyl)phenyl]-7,8-dihydro-5H-1,6-naphthyridine-6-carboxamide | IC50 | 391.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_12dbb0e225374bbe1142d7d1ee6ccdfc.svg) | (8R)-N-(4-Fluorophenyl)-8-[4-(trifluoromethyl)phenyl]-6,8-dihydro-5H-1,7-naphthyridine-7-carboxamide | IC50 | 14.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_5b6119190c87cd6f4080d1463ee2c342.svg) | (8R)-N-Pyridin-3-yl-8-[4-(trifluoromethyl)phenyl]-6,8-dihydro-5H-1,7-naphthyridine-7-carboxamide | IC50 | 24.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_54d1e5cc47abf12a9223d9e2c8c9e0af.svg) | (5R)-N-(4-Fluorophenyl)-5-[4-(trifluoromethyl)phenyl]-7,8-dihydro-5H-pyrido[3,4-b]pyrazine-6-carboxamide | IC50 | 200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_b3ed79fc4a7010b99228ee346160f08d.svg) | N-(4-Fluorophenyl)-1-[4-(trifluoromethyl)phenyl]-3,4-dihydro-1H-2,6-naphthyridine-2-carboxamide | IC50 | 1262.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_2ebb8071e56c79b41c0a2c14d7086750.svg) | N-(4-Fluorophenyl)-1-[4-(trifluoromethyl)phenyl]-3,4-dihydro-1H-2,7-naphthyridine-2-carboxamide | IC50 | 463.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_7302e61177041f86138e94156e8358ce.svg) | N-(4-Fluorophenyl)-8-[4-(trifluoromethyl)phenyl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carboxamide | IC50 | 786.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_76712777fc9fe5cb45782b77990f1142.svg) | N-Benzyl-N-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]benzenesulfonamide | IC50 | 183.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_4fb1241398c305625526f3f2d787c6af.svg) | (1R)-1-[4-(Trifluoromethyl)phenyl]-N-[(2R)-1,1,1-trifluoropropan-2-yl]-3,4-dihydro-1H-isoquinoline-2-carboxamide | IC50 | 52.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_3b88028bddc6f1d6669f95179ffa217d.svg) | (1R)-N-Pyridin-2-yl-1-[4-(trifluoromethyl)phenyl]-3,4-dihydro-1H-isoquinoline-2-carboxamide | IC50 | 171.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_e08bb59abd6e602a34307c7e8031c502.svg) | (8R)-8-[3-Fluoro-4-(trifluoromethyl)phenyl]-N-[(2S)-1,1,1-trifluoropropan-2-yl]-6,8-dihydro-5H-1,7-naphthyridine-7-carboxamide | IC50 | 12.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transient-receptor-potential-cation-channel-subfamily-m-member-8_0b574f785958af2ae66101ee13476b69.svg) | 8-Bromo-N-[4-(trifluoromethyl)phenyl]spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide | IC50 | 18.9 [1] |