Transient receptor potential cation channel subfamily M member 2 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	N-(p-Amylcinnamoyl)anthranilic acid	IC50	320.0 [1], 1700.0 [2], 4500.0 [3]
	Adenosine monophosphate	IC50	70000.0 [1]
	2-Aminoethyl diphenylborinate	IC50	1000.0 [1]
	Clotrimazole	IC50	3000.0 [1]
	Mefenamic acid	IC50	124000.0 [1]
	Flufenamic acid	IC50	70000.0 [1]
	Niflumic acid	IC50	149000.0 [1]
	Econazole	IC50	3000.0 [1]
	3,4-Dihydro-5-(4-(1-piperidinyl)butoxy)-1(2H)-isoquinolinone	IC50	600.0 [1]
	Salicyl-AMS	IC50	100000.0 [1]
	N-(3-Methylphenyl)anthranilic acid	IC50	76000.0 [1]
	4-[(3S,4R)-1-(2,4-Dichlorophenyl)sulfonyl-4-hydroxy-4-(hydroxymethyl)pyrrolidin-3-yl]oxy-2-fluorobenzonitrile	IC50	10000.0 [1]
	6-Bromo-8-methyl-2-(5-phenyl-1H-pyrazol-4-yl)-2,3-dihydro-1H-quinazolin-4-one	IC50	4600.0 [1]
	6-Chloro-8-methyl-2-(5-phenyl-1H-pyrazol-4-yl)-2,3-dihydro-1H-quinazolin-4-one	IC50	5100.0 [1]
	6-Chloro-8-methyl-2-(5-naphthalen-1-yl-1H-pyrazol-4-yl)-2,3-dihydro-1H-quinazolin-4-one	IC50	4000.0 [1]
	6-Bromo-8-methyl-2-(5-naphthalen-1-yl-1H-pyrazol-4-yl)-2,3-dihydro-1H-quinazolin-4-one	IC50	3700.0 [1]
	2-(Dimethylamino)-N-(6-oxo-5H-phenanthridin-2-yl)acetamide;hydrate;hydrochloride	IC50	25.0 [1]
	[[(2R,3S,4R,5R)-5-(6-Amino-8-bromopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3S,4R)-3,4,5-trihydroxyoxolan-2-yl]methyl hydrogen phosphate	IC50	300000.0 [1]
	[[(2R,3S,4R,5R)-5-(6-Amino-8-phenylpurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] cyclopentyl hydrogen phosphate	IC50	15000.0 [1]
	[4-(6-Aminopurin-9-yl)butoxy-hydroxyphosphoryl] [(2R,3S,4R)-3,4,5-trihydroxyoxolan-2-yl]methyl hydrogen phosphate	IC50	100000.0 [1]
	[[(2R,3S,4R,5R)-5-(6-Amino-8-phenylpurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3S,4R)-3,4,5-trihydroxyoxolan-2-yl]methyl hydrogen phosphate	IC50	11000.0 [1]
	2-Amino-3-[4-[6-amino-9-[(2R,3R,4S,5R)-3,4-dihydroxy-5-(phosphonooxymethyl)oxolan-2-yl]purin-8-yl]phenyl]propanoic acid	IC50	100000.0 [1]
	[[(2R,3S,5R)-5-(6-Amino-8-phenylpurin-9-yl)-3-hydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3S,4R)-3,4,5-trihydroxyoxolan-2-yl]methyl hydrogen phosphate	IC50	3000.0 [1]
	[[(2R,3S,4R,5R)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] cyclopentyl hydrogen phosphate	IC50	900000.0 [1]
	[[(2R,3S,4R,5R)-5-(6-Amino-8-thiophen-3-ylpurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3S,4R)-3,4,5-trihydroxyoxolan-2-yl]methyl hydrogen phosphate	IC50	51000.0 [1]
	[[(2R,3S,4R,5R)-5-[8-(3-Acetylphenyl)-6-aminopurin-9-yl]-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3S,4R)-3,4,5-trihydroxyoxolan-2-yl]methyl hydrogen phosphate	IC50	49000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

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References

This online tool may be cited as follows

MLA	"Quest Database™ Transient receptor potential cation channel subfamily M member 2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Feb. 2025, https://www.aatbio.com/data-sets/transient-receptor-potential-cation-channel-subfamily-m-member-2-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, February 21). Quest Database™ Transient receptor potential cation channel subfamily M member 2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/transient-receptor-potential-cation-channel-subfamily-m-member-2-inhibitors-ic50-ki.
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