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Transient receptor potential cation channel subfamily A member 1 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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2-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetrahydro-7H-purin-7-yl)-N-(4-isopropylphenyl)acetamideIC505300.0 [1]
4-Methyl-N-[2,2,2-trichloro-1-(4-nitro-phenylsulfanyl)-ethyl]-benzamideIC50850.0 [1]
4-(4-Chlorophenyl)-3-methylbut-3-EN-2-oximeIC502200.0 [1], 2800.0 [2], 3100.0 [3]
4-Methoxy-N-[2,2,2-trichloro-1-(4-chloro-phenylsulfanyl)-ethyl]-benzamideIC5029.0 [1], 91.0 [2], 260.0 [3]
4-Nitro-N-{2,2,2-trichloro-1-[(4-chlorophenyl)sulfanyl]ethyl}benzamideIC5035.0 [1], 105.0 [2], 167.0 [3]
4-Bromo-N-[2,2,2-trichloro-1-(4-chloro-phenylsulfanyl)-ethyl]-benzamideIC5028.0 [1], 51.0 [2], 252.0 [3]
4-[3-(3-Methoxypropoxy)phenyl]-2-sulfanylidene-3,4-dihydro-1H-indeno[1,2-d]pyrimidin-5-oneIC505.61 [1], 30.0 [2], 50.0 [3]
4-(3-Methoxyphenyl)-2-sulfanylidene-3,4-dihydro-1H-indeno[1,2-d]pyrimidin-5-oneIC50128.0 [1], 130.0 [2], 1500.0 [3]
1-(4-Chlorophenyl)-N-[2-[4-hydroxy-4-(trifluoromethyl)piperidin-1-yl]-3-phenylpropyl]cyclopentane-1-carboxamideIC501.0 [1], 17.0 [2], 374.0 [3]
N-(3,4-Difluorophenyl)-6-(trifluoromethoxy)-1H-pyrazolo[4,3-b]pyridin-3-amineIC5020.0 [1], 330.0 [2], 16000.0 [3]
N-[2-[4-(Difluoromethoxy)phenyl]ethyl]-2-(8-methyl-4-oxoquinazolin-3-yl)acetamideIC50685.0 [1], 6270.0 [2], 25000.0 [3]
N-[2,2,2-Trichloro-1-(4-chlorophenyl)sulfanylethyl]benzamideIC507.0 [1], 21.0 [2], 120.0 [3]
1-(4-Chlorophenyl)-N-[(2R)-2-[4-hydroxy-4-(trifluoromethyl)piperidin-1-yl]-3-phenylpropyl]cyclopentane-1-carboxamideIC500.7 [1], 0.72 [2], 1578.0 [3]
ResveratrolIC50750.0 [1], 30000.0 [2]
(1e,3e)-1-(4-Fluorophenyl)-2-methylpent-1-en-3-one oximeIC5074.0 [1], 98.44 [2]
D-CamphorIC50400000.0 [1], 660000.0 [2]
Chembridge-5861528IC5014300.0 [1], 18700.0 [2]
2-[(E)-2-Phenylethenyl]phenolIC501700.0 [1], 30000.0 [2]
1-((3-(4-Chlorophenethyl)-1,2,4-oxadiazol-5-yl)methyl)-7-methyl-1H-purin-6(7H)-oneIC5020.0 [1], 131.0 [2]
(4R)-4-[3-(3-Methoxypropoxy)phenyl]-2-sulfanylidene-3,4-dihydro-1H-indeno[1,2-d]pyrimidin-5-oneIC5013.0 [1], 26.0 [2]
1-(4-Chlorophenyl)-N-[2-[4-hydroxy-4-(trifluoromethyl)piperidin-1-yl]-3-phenylpropyl]cyclopropane-1-carboxamideIC5014.0 [1], 73.0 [2]
1-[[3-[(E)-2-(4-Chlorophenyl)prop-1-enyl]-1,2,4-oxadiazol-5-yl]methyl]-7-methylpurin-6-oneIC5063.0 [1], 71.0 [2]
3-[[5-[2-(4-Chlorophenyl)ethyl]-1,2,4-oxadiazol-3-yl]methyl]pyrido[2,3-d]pyrimidin-4-oneIC50156.0 [1], 1580.0 [2]
3-[[3-[2-(4-Chlorophenyl)ethyl]-1,2,4-oxadiazol-5-yl]methyl]pyrido[2,3-d]pyrimidin-4-oneIC5041.0 [1], 376.0 [2]
3-[[3-[2-(4-Chlorophenyl)-2-hydroxyethyl]-1,2,4-oxadiazol-5-yl]methyl]pyrido[2,3-d]pyrimidin-4-oneIC5058.0 [1], 251.0 [2]
3-[[5-[(E)-2-(4-Chlorophenyl)prop-1-enyl]-1,2,4-oxadiazol-3-yl]methyl]pyrido[2,3-d]pyrimidin-4-oneIC5085.0 [1], 116.0 [2]
4-[6-(Trifluoromethoxy)-1H-indazol-3-yl]benzonitrileIC50686.0 [1], 10000.0 [2]
N-[3-Methyl-1-(4-nitrophenyl)-1-oxobutan-2-yl]benzamideIC50251.19 [1], 316.23 [2]
N-[1-(4-Fluorophenyl)-3-methyl-1-oxobutan-2-yl]benzamideIC505011.87 [1], 7943.28 [2]
5-Chloro-N-[1-(4-cyanophenyl)-3-methyl-1-oxobutan-2-yl]-2-(trifluoromethyl)benzamideIC50316.23 [1], 398.11 [2]
N-[1-(4-Cyanophenyl)-3-methyl-1-oxobutan-2-yl]-3-methyl-5-phenyl-1,2-oxazole-4-carboxamideIC503981.07 [1], 7943.28 [2]
N-[1-(4-Cyanophenyl)-3-methyl-1-oxobutan-2-yl]-1-methylindole-2-carboxamideIC501584.89 [1], 3981.07 [2]
N-[1-(4-Cyanophenyl)-3-methyl-1-oxobutan-2-yl]decanamideIC501000.0 [1], 1995.26 [2]
Tert-butyl N-[1-(4-chlorophenyl)-3-methyl-1-oxobutan-2-yl]carbamateIC50794.33 [1], 1000.0 [2]
N-[1-(4-Cyanophenyl)-3-methyl-1-oxobutan-2-yl]-2-(trifluoromethyl)benzamideIC503162.28 [1], 5011.87 [2]
N-[1-(4-Cyanophenyl)-3-methyl-1-oxobutan-2-yl]-3-methyl-5-propan-2-yl-1,2-oxazole-4-carboxamideIC501584.89 [1], 1995.26 [2]
N-[1-(4-Cyanophenyl)-3-methyl-1-oxobutan-2-yl]-3,4-dihydro-1H-isoquinoline-2-carboxamideIC505011.87 [1]
N-[1-(4-Chlorophenyl)-3,3-dimethyl-1-oxobutan-2-yl]benzamideIC50398.11 [1], 1000.0 [2]
1-Tert-butyl-3-[1-(4-chlorophenyl)-3-methyl-1-oxobutan-2-yl]-1-methylureaIC50251.19 [1], 630.96 [2]
Tert-butyl N-[1-(4-cyano-3-fluorophenyl)-3-methyl-1-oxobutan-2-yl]carbamateIC501258.93 [1], 1995.26 [2]
N-[1-(4-Bromophenyl)-3-methyl-1-oxobutan-2-yl]benzamideIC501258.93 [1], 7943.28 [2]
N-[1-(4-Cyanophenyl)-3-methyl-1-oxobutan-2-yl]-4-methoxybenzamideIC506309.57 [1], 12589.25 [2]
2,4-Dichloro-N-[1-(4-cyanophenyl)-3-methyl-1-oxobutan-2-yl]benzamideIC502511.89 [1], 5011.87 [2]
4-Chloro-N-[1-(4-cyanophenyl)-3-methyl-1-oxobutan-2-yl]-2-fluorobenzamideIC503162.28 [1], 3981.07 [2]
Tert-butyl N-[1-(4-cyanophenyl)-3-methyl-1-oxobutan-2-yl]carbamateIC502511.89 [1], 6309.57 [2]
N-[2-(4-Chlorophenyl)-1-cyclopropyl-2-oxoethyl]benzamideIC501995.26 [1]
5-Tert-butyl-N-[1-(4-cyanophenyl)-3-methyl-1-oxobutan-2-yl]-1,2-oxazole-4-carboxamideIC50501.19 [1], 1000.0 [2]
1-Tert-butyl-3-[1-(4-chlorophenyl)-3-methyl-1-oxobutan-2-yl]ureaIC501995.26 [1], 2511.89 [2]
Tert-butyl N-[1-(5-chloropyridin-2-yl)-3-methyl-1-oxobutan-2-yl]carbamateIC505011.87 [1], 15848.93 [2]
N-(6-Chloropyridin-3-yl)-6-(trifluoromethyl)-1H-indazol-3-amineIC50550.0 [1], 2500.0 [2]
3-ButylidenephthalideIC5023000.0 [1]
DihydroresveratrolIC5030000.0 [1]
(1E,3E)-1-(4-Fluorophenyl)-2-methyl-1-penten-3-one oximeIC50701.0 [1]
7-Bromo-N-(1-phenylcyclopropyl)-3-[(4-piperidin-1-ylpiperidin-1-yl)methyl]-2-[3-(trifluoromethyl)phenyl]quinoline-4-carboxamideIC5025000.0 [1]
N,N'-DibenzylthioureaIC5010000.0 [1]
2-Thioxo-4-phenyl-1,2,3,4,7,8-hexahydroquinazoline-5(6H)-oneIC5010000.0 [1]
4,6-Diphenyl-1,2,3,4-tetrahydropyrimidine-2-thioneIC5010000.0 [1]
trans-3,3',5-TrihydroxystilbeneIC5030000.0 [1]
4-Phenyl-3,4-dihydro-2H-indeno[1,2-d]pyrimidine-2,5(1H)-dioneIC5010000.0 [1]
8-Benzylidene-4-phenyl-3,4,5,6,7,8-hexahydro-2(1H)-quinazolinethioneIC5010000.0 [1]
2-MethoxystilbeneIC501700.0 [1]
P-MethoxystilbeneIC5012100.0 [1]
4-Phenyl-3,4,5,6-tetrahydrobenzo[h]quinazoline-2(1H)-thioneIC5010000.0 [1]
4-Phenyl-2-thioxo-1,2,3,4-tetrahydro-5H-indeno[1,2-d]pyrimidin-5-oneIC501800.0 [1]
CID 49783953IC5010000.0 [1]
3-Methyl-4-phenyl-but-3-en-2-one oximeIC502700.0 [1]
[2-(4-Chloro-2-fluoroanilino)-5-methyl-1,3-thiazol-4-yl]-[(2S,3S)-2,3-dimethylpiperidin-1-yl]methanoneIC5025000.0 [1]
N-[4-(4-Bromophenyl)-1,3-thiazol-2-yl]-2-(1,3-dimethyl-2,6-dioxopurin-7-yl)acetamideIC501000.0 [1]
5-[(1E)-2-(4-Chlorophenyl)ethenyl]-1,3-BenzenediolIC5030000.0 [1]
2,6-Dibromo-4-[(E)-2-(4-hydroxyphenyl)ethenyl]phenolIC5016100.0 [1]
1,3-Dichloro-5-[(1E)-2-(4-chlorophenyl)ethenyl]-benzeneIC5030000.0 [1]
2-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetrahydro-7H-purin-7-yl)-N-(4-phenyl-1,3-thiazol-2-yl)acetamideIC501000.0 [1]
(2S,4R)-4-Fluoro-1-(4-fluorophenyl)sulfonyl-N-[[6-[6-(trifluoromethyl)pyridin-3-yl]pyrimidin-4-yl]methyl]pyrrolidine-2-carboxamideIC501200.0 [1]
(2S,4S)-4-Fluoro-1-(4-fluorophenyl)sulfonyl-N-[[6-[6-(trifluoromethyl)pyridin-3-yl]pyrimidin-4-yl]methyl]pyrrolidine-2-carboxamideIC504400.0 [1]
(2S,4R,5S)-4-Fluoro-1-(4-fluorophenyl)sulfonyl-5-methyl-N-[[2-[2-(trifluoromethyl)pyrimidin-5-yl]pyridin-4-yl]methyl]pyrrolidine-2-carboxamideIC5069.0 [1]
(2S,5R)-1-(4-Fluorophenyl)sulfonyl-5-methyl-N-[[6-[6-(trifluoromethyl)pyridin-3-yl]pyrimidin-4-yl]methyl]pyrrolidine-2-carboxamideIC50239.0 [1]
(2S)-1-(4-Fluorophenyl)sulfonyl-N-[[6-[6-(trifluoromethyl)pyridin-3-yl]pyrimidin-4-yl]methyl]azetidine-2-carboxamideIC501500.0 [1]
(2S,5S)-1-(4-Fluorophenyl)sulfonyl-5-methyl-N-[[6-[6-(trifluoromethyl)pyridin-3-yl]pyrimidin-4-yl]methyl]pyrrolidine-2-carboxamideIC5013.0 [1]
N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-N-[(1R)-1-(3,5-difluorophenyl)ethyl]benzamideIC5030000.0 [1]
N-[3-(Thiophen-2-ylmethylamino)-5-(trifluoromethyl)phenyl]thiophene-2-carboxamideIC502700.0 [1]
N-[3-(Benzylamino)-5-(trifluoromethyl)phenyl]thiophene-2-carboxamideIC502900.0 [1]
N-[3-(2-Phenylethylamino)-5-(trifluoromethyl)phenyl]thiophene-2-carboxamideIC503900.0 [1]
Methyl N-[3-(thiophene-2-carbonylamino)-5-(trifluoromethyl)phenyl]carbamateIC502300.0 [1]
N-[3-(Dipropylamino)-5-(trifluoromethyl)phenyl]thiophene-2-carboxamideIC5032000.0 [1]
N-[3-(3-Methylbutan-2-ylamino)-5-(trifluoromethyl)phenyl]thiophene-2-carboxamideIC501300.0 [1]
N-[3-(2-Methylpropylamino)-5-(trifluoromethyl)phenyl]thiophene-2-carboxamideIC50790.0 [1]
N-[3-(Propylamino)-5-(trifluoromethyl)phenyl]thiophene-2-carboxamideIC50390.0 [1]
N-[3-(Propan-2-ylamino)-5-(trifluoromethyl)phenyl]thiophene-2-carboxamideIC50290.0 [1]
N-[3-(Propylamino)-5-(trifluoromethyl)phenyl]benzamideIC50200.0 [1]
N-[3-(Propylamino)-5-(trifluoromethyl)phenyl]pyridine-2-carboxamideIC5032000.0 [1]
N-[3-(Propylamino)-5-(trifluoromethyl)phenyl]pyridine-3-carboxamideIC50940.0 [1]
N-[3-(Propylamino)-5-(trifluoromethyl)phenyl]pyridine-4-carboxamideIC502600.0 [1]
4-Fluoro-N-[3-(propylamino)-5-(trifluoromethyl)phenyl]benzamideIC501400.0 [1]
3,4-Difluoro-N-[3-(propylamino)-5-(trifluoromethyl)phenyl]benzamideIC501200.0 [1]
2,6-Difluoro-N-[3-(propylamino)-5-(trifluoromethyl)phenyl]benzamideIC50110.0 [1]
3-N-Propyl-5-(trifluoromethyl)benzene-1,3-diamineIC5032000.0 [1]
N-[3-(Ethylamino)-5-(trifluoromethyl)phenyl]-2,6-difluorobenzamideIC5074.0 [1]
2,6-Difluoro-N-[3-(propan-2-ylamino)-5-(trifluoromethyl)phenyl]benzamideIC5091.0 [1]
2,6-Difluoro-N-[3-[methyl(propyl)amino]-5-(trifluoromethyl)phenyl]benzamideIC5032000.0 [1]
2,6-Difluoro-N-[3-propoxy-5-(trifluoromethyl)phenyl]benzamideIC5032000.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Transient receptor potential cation channel subfamily A member 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/transient-receptor-potential-cation-channel-subfamily-a-member-1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 20). Quest Database™ Transient receptor potential cation channel subfamily A member 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/transient-receptor-potential-cation-channel-subfamily-a-member-1-inhibitors-ic50-ki.
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