![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_cc13628645c821a4d949b6b2e0576a37.svg) | 4-[(2s,4r)-1-Acetyl-4-[(4-Chlorophenyl)amino]-2-Methyl-1,2,3,4-Tetrahydroquinolin-6-Yl]benzoic Acid | IC50 | 10000.0 [1], 15848.93 [2] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_ce0ddc17b1983393b9e28f7597d2378a.svg) | CID 91827373 | IC50 | 1600.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_23e00f2017c211b736ed0d885021ef97.svg) | N-[6-(4-Methoxyphenoxy)-1,3-Dimethyl-2-Oxo-2,3-Dihydro-1h-Benzimidazol-5-Yl]benzenesulfonamide | IC50 | 730.0 [1], 1500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_44d1a6e5980820d01a8d1ca3b47b75c3.svg) | Sgc-cbp30 | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_68023d26d55a3c14e04fd49649cda015.svg) | N-(1,3-Dimethyl-2-oxo-2,3-dihydro-1H-benzimidazol-5-yl)-4-methoxybenzenesulfonamide | IC50 | 9300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_449b621332acf235c11cb177ebea19ae.svg) | N-(1,3-Dimethyl-2-oxo-2,3-dihydro-1H-benzimidazol-5-yl)-5,6,7,8-tetrahydro-2-naphthalenesulfonamide | IC50 | 6170.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_36e135db85f03efa4c2e6260ffeb3db0.svg) | N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)benzenesulfonamide | IC50 | 23000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_72013193af36cf2fbb8c74b5e81239a2.svg) | N,2-Dimethyl-5-(3-methyl[1,2,4]triazolo[3,4-a]phthalazin-6-yl)benzenesulfonamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_cfa6ca57a967b08a70060b04d35b1641.svg) | 3-Cyano-N-(6-methoxy-1,3-dimethyl-2-oxobenzimidazol-5-yl)benzenesulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_8a03d2f948782f0a967dd9e9aceae8de.svg) | 3,4-Dimethoxy-N-[6-(4-methoxyphenoxy)-1,3-dimethyl-2-oxobenzimidazol-5-yl]benzenesulfonamide | IC50 | 430.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_ba6c458cef44ebde344a4c0e58953eb6.svg) | N-[3-(3-Methyl-4-Oxo-4,5,6,7-Tetrahydro-2h-Isoindol-1-Yl)-4-Phenoxyphenyl]methanesulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_e4b62e86226ef3a7c2e14d821455cc8f.svg) | 1-[2-(2,4-Difluorophenoxy)-5-methylsulfonylphenyl]-3-methyl-2,5,6,7-tetrahydropyrrolo[3,4-c]pyridin-4-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_780671bd435b12876f806ef7c7d02f6c.svg) | N-[6-[3-(6-Aminohexoxy)-5-propoxyphenoxy]-1,3-dimethyl-2-oxobenzimidazol-5-yl]-1-methylimidazole-4-sulfonamide | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_e186de024153f93186adb3e1f84e9378.svg) | N-[6-[3-(4-Aminobutoxy)-5-propoxyphenoxy]-1,3-dimethyl-2-oxobenzimidazol-5-yl]-1-methylimidazole-4-sulfonamide | IC50 | 7.9 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_0cfbc23460a7051101520f63a4bf63a5.svg) | N-[6-[3-(3-Methoxypropoxy)phenoxy]-1,3-dimethyl-2-oxobenzimidazol-5-yl]-1,2-dimethylimidazole-4-sulfonamide | IC50 | 130.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_109719eb1173edeac519beb62c2bf957.svg) | N-[1,3-Dimethyl-2-oxo-6-(3-phenylmethoxyphenoxy)benzimidazol-5-yl]-1-methylimidazole-4-sulfonamide | IC50 | 220.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_1834beddd0df14a180bc031c8b836f99.svg) | N-[1,3-Dimethyl-6-[3-(2-methylpropoxy)phenoxy]-2-oxobenzimidazol-5-yl]cyclopropanesulfonamide | IC50 | 110.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_b0712c980ddade123f3616aeba06eca8.svg) | N-[6-[3-(6-Aminohexoxy)-5-propoxyphenoxy]-1,3-dimethyl-2-oxobenzimidazol-5-yl]-3,4-dimethoxybenzenesulfonamide | IC50 | 13.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_e55562345500eedbb86d363fef426c3a.svg) | N-[6-(3-Butoxyphenoxy)-1,3-dimethyl-2-oxobenzimidazol-5-yl]-1,2-dimethylimidazole-4-sulfonamide | IC50 | 160.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_0017e3e7373de757575a36645e8ce720.svg) | N-[6-[3-(4-Aminobutoxy)-5-propoxyphenoxy]-1,3-dimethyl-2-oxobenzimidazol-5-yl]-3,4-dimethoxybenzenesulfonamide | IC50 | 8.3 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_f279c8bc563150a48e94d25d651db05b.svg) | N-[1,3-Dimethyl-2-oxo-6-[3-(oxolan-3-ylmethoxy)phenoxy]benzimidazol-5-yl]-1-methylimidazole-4-sulfonamide | IC50 | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_928d4d175be4bca4fec66cc287e203ad.svg) | N-[1,3-Dimethyl-2-oxo-6-(3-phenylmethoxyphenoxy)benzimidazol-5-yl]-1,2-dimethylimidazole-4-sulfonamide | IC50 | 270.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_acb5deb5b010362f5a6d3d6cc30ca72e.svg) | N-[6-[3-(3-Aminopropoxy)-5-propoxyphenoxy]-1,3-dimethyl-2-oxobenzimidazol-5-yl]-3,4-dimethoxybenzenesulfonamide | IC50 | 13.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_4b0498f41c05012a5f708b2f0bd90045.svg) | N-[6-[3-(5-Aminopentoxy)-5-propoxyphenoxy]-1,3-dimethyl-2-oxobenzimidazol-5-yl]-1-methylimidazole-4-sulfonamide | IC50 | 11.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_8f215dc3a47edea8e56d188ebf0cf951.svg) | N-[6-[3-(6-Hydroxyhexoxy)-5-propoxyphenoxy]-1,3-dimethyl-2-oxobenzimidazol-5-yl]-1-methylimidazole-4-sulfonamide | IC50 | 60.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_e60326288933bf03fe30a932b7fd49aa.svg) | N-[6-(3-Ethoxyphenoxy)-1,3-dimethyl-2-oxobenzimidazol-5-yl]-1,2-dimethylimidazole-4-sulfonamide | IC50 | 180.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_ab220effacf7b2d656d630857b185f72.svg) | N-[1,3-Dimethyl-2-oxo-6-(3-propoxyphenoxy)benzimidazol-5-yl]-1,2-dimethylimidazole-4-sulfonamide | IC50 | 53.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_d2d82eb07eddfa76ced7077e95b232b5.svg) | N-[1,3-Dimethyl-2-oxo-6-(3-propoxyphenoxy)benzimidazol-5-yl]-3,4-dimethoxybenzenesulfonamide | IC50 | 43.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_af7dd7ae33ca37a0dc74117a3b2dac52.svg) | Tert-butyl N-[6-[3-[1,3-dimethyl-6-[(1-methylimidazol-4-yl)sulfonylamino]-2-oxobenzimidazol-5-yl]oxy-5-propoxyphenoxy]hexyl]carbamate | IC50 | 160.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_370f0c39e7ac0dbc09bbcd0d59f2d6cb.svg) | N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-2,2-dimethyl-3,4-dihydrochromene-6-sulfonamide | IC50 | 3690.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_99088a6129ee89d599103e8e372f6d12.svg) | (2S)-N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-2,3-dimethoxy-2,3-dimethyl-1,4-benzodioxine-6-sulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_952c2c150b3e9d80991ba6ef9fc74a9c.svg) | N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-3,4-dihydro-2H-chromene-6-sulfonamide | IC50 | 4630.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_a5f7b33710f9ae61446c32b889073a47.svg) | N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-2-methylbenzenesulfonamide | IC50 | 2620.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_5a3176ed16c92446719eb1c51b5a4121.svg) | N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-3-methoxybenzenesulfonamide | IC50 | 2380.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_ea25b48ae4d7c175ab40c77c14e31d22.svg) | N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-5,6,7,8-tetrahydronaphthalene-2-sulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_a56c83168d617f15a6fcd8fee5c3be86.svg) | N-(1-Methyl-2-oxo-3H-indol-5-yl)-4-methylsulfanylbenzenesulfonamide | IC50 | 17000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_c883f4d3a040517dede5f3793e2f73c9.svg) | N-(1-Methyl-2-oxo-3,4-dihydroquinolin-6-yl)-4-methylsulfanylbenzenesulfonamide | IC50 | 4800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_bb33b1a22f45e94731e3fe7b5170b896.svg) | N-[6-[3-[4-(Dimethylamino)butoxy]phenoxy]-1,3-dimethyl-2-oxobenzimidazol-5-yl]-3,4-dimethoxybenzenesulfonamide | IC50 | 270.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_d33cf436d7e427605eb276d559c15779.svg) | 4-Cyclohexyl-N-(1-methyl-2-oxo-3,4-dihydroquinolin-6-yl)benzenesulfonamide | IC50 | 2800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_a8032af441b2ab31530bf98ba47d9754.svg) | N-(7-Methoxy-1-methyl-2-oxo-3,4-dihydroquinolin-6-yl)benzenesulfonamide | IC50 | 36000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_36baeb8f8c1db0cbc238eb86b0425216.svg) | N-(1-Methyl-2-oxo-3,4-dihydroquinolin-7-yl)-4-methylsulfanylbenzenesulfonamide | IC50 | 14000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_1fce7a083e4ea1994b073e0be3ed0b9c.svg) | 1,3-Dimethyl-5-[3-(2-methylpropoxy)phenoxy]benzimidazol-2-one | IC50 | 2400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_4d0e99ea030bf3730ff36902529f4f45.svg) | N-[1,3-Dimethyl-2-oxo-6-(4-phenylmethoxyphenoxy)benzimidazol-5-yl]-1-methylimidazole-4-sulfonamide | IC50 | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_fcf2ce514f07459050b4e8676eb35a45.svg) | 3-[(1-Acetyl-5-methoxyindole-3-carbonyl)amino]-5-(furan-2-yl)benzoic acid | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_ee19c44fe23cd63eeebe483bf602cc25.svg) | 3-[(1-Acetyl-5-methoxyindole-3-carbonyl)amino]-4-fluoro-5-(1-methylpyrazol-4-yl)benzoic acid | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_fa44b72275df2582692739dd72425d01.svg) | 3-[(1-Acetylindole-3-carbonyl)amino]-4-fluorobenzoic acid | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_85a2956dc90c939e22fb6420e5725771.svg) | 3-[(1-Acetylindole-3-carbonyl)amino]benzoic acid | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_56ee0082ae60186b992a0a052290c2c2.svg) | 3-[(1-Acetylindole-3-carbonyl)amino]-5-(oxan-2-yloxymethyl)benzoic acid | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_c3bca8b0ac250821aa58a99065eab07a.svg) | 3-[(1-Acetyl-5-methoxyindole-3-carbonyl)amino]-5-(1-methylpyrazol-4-yl)benzoic acid | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_f1f088cd6f5b8224786003ec91f0b1a5.svg) | 3-[(1-Acetylindole-3-carbonyl)amino]-5-(furan-2-yl)benzoic acid | IC50 | 10440.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_9d2256befb487ba98b8f539225685dcb.svg) | N,N,2-Trimethyl-5-(3-methyl-[1,2,4]triazolo[3,4-a]phthalazin-6-yl)benzenesulfonamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_30f1fac2238e636582b032b911835e15.svg) | 2,4-Dimethoxy-N-(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl)benzenesulfonamide | IC50 | 2500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_0848becdf3ce4ae50b0621703c5d640d.svg) | 4-Cyclohexyl-N-(1,3-dimethyl-2-oxo-2,3-dihydro-1H-benzimidazol-5-yl)benzenesulfonamide | IC50 | 1700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_4ce3171cb6798fcab00556c2305c566e.svg) | N-(1-Methyl-2-oxo-3,4-dihydroquinolin-6-yl)-4-(2-methylpropoxy)benzenesulfonamide | IC50 | 3700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_7ad22cf31a99e547f3d6f423a77b40a4.svg) | N-[2-Methyl-5-(3-methyl[1,2,4]triazolo[3,4-a]phthalazin-6-yl)phenyl]methanesulfonamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_b9456135d3548ae476ba7b50ec0687e7.svg) | N-[2-Methyl-5-(3-methyl[1,2,4]triazolo[3,4-a]phthalazin-6-yl)phenyl]propanamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_10a53bf654e88ece0ded582932cccacd.svg) | N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-4-(2-methylpropoxy)benzenesulfonamide | IC50 | 4000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_0ff07a0195ed837ab5ed5e529c6751a7.svg) | N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-3-fluoro-4-methylbenzenesulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_fcbdbe202ff3348984b89c043fd665eb.svg) | N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-4-propan-2-ylbenzenesulfonamide | IC50 | 3450.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_d6d595a715c9a80836b15015a7e5770e.svg) | N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-2,3-dihydro-1H-indene-5-sulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_4384396157302e7ce13acab8a3aa86a2.svg) | 4-Chloro-N-(1,3-dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)benzenesulfonamide | IC50 | 1560.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_a4cd6a63e595207501e83673179e6ee3.svg) | N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-3,4-dimethoxybenzenesulfonamide | IC50 | 480.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_9cf1545bf1ef8d7c96c434c23bbaea4c.svg) | N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-3,4-dimethylbenzenesulfonamide | IC50 | 4770.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_0b6bd54dea7ac0a81090612c1ebc8ca4.svg) | N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-4-methoxybenzenesulfonamide | IC50 | 740.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_42fe3e73d7e22259210e76aa76ca670d.svg) | N-[6-(4-Methoxyphenoxy)-1,3-dimethyl-2-oxobenzimidazol-5-yl]-2-methylbenzenesulfonamide | IC50 | 1470.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_c3fe9bcee3abbf74eeef0d94f4433d41.svg) | N-[6-(4-Methoxyphenoxy)-1,3-dimethyl-2-oxobenzimidazol-5-yl]-4-propoxybenzenesulfonamide | IC50 | 8400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_298d60d02de722ab353bfcd3c2653c55.svg) | 4-Chloro-N-(1,3-dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-2-methylbenzenesulfonamide | IC50 | 2450.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_cc127e869d00ca793329f348c212181b.svg) | N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-5-fluoro-2-methylbenzenesulfonamide | IC50 | 3420.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_7b08236e14745a48413f1baff40fe388.svg) | N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-3-fluoro-4-methylbenzenesulfonamide | IC50 | 2700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_0e3df27b5bdbc9511144f285eb97b0a3.svg) | N-[6-(4-Methoxyphenoxy)-1,3-dimethyl-2-oxobenzimidazol-5-yl]-4-methylbenzenesulfonamide | IC50 | 2700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_236f04cf725b031c367f3704feb28f83.svg) | 4-Methoxy-N-[6-(4-methoxyphenoxy)-1,3-dimethyl-2-oxobenzimidazol-5-yl]benzenesulfonamide | IC50 | 770.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_7c008dcd1d3473b98ce425a403a612f2.svg) | N-(1,3-Dimethyl-2-oxo-6-phenoxy-2,3-dihydro-1H-benzimidazol-5-yl)-4-methylbenzenesulfonamide | IC50 | 1270.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_2f47841b05b4795be157fce34188622c.svg) | N-(1,3-Dimethyl-2-oxo-2,3-dihydro-1H-benzimidazol-5-yl)-4-(methylsulfanyl)benzenesulfonamide | IC50 | 4900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_dc562a7b4f1d2c7d72c7eea3aa94fcab.svg) | 3-[2-(2,4-Difluorophenoxy)-5-methylsulfonylphenyl]-1-methyl-6H-pyrrolo[2,3-c]pyridin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_3d12e7b513805e2a68b054c7c869a048.svg) | N-[1,3-Dimethyl-2-oxo-6-(3-phenylmethoxyphenoxy)benzimidazol-5-yl]-3,4-dimethoxybenzenesulfonamide | IC50 | 140.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_47f19ada64beb54ddf5dc4f7aac43dad.svg) | N-[1,3-Dimethyl-6-[3-(2-methylpropoxy)phenoxy]-2-oxobenzimidazol-5-yl]-1,2-dimethylimidazole-4-sulfonamide | IC50 | 57.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_7d3de1cf87b580c7efa34a9e02c56d56.svg) | N-[6-[3-[4-(Dimethylamino)butoxy]-5-propoxyphenoxy]-1,3-dimethyl-2-oxobenzimidazol-5-yl]-3,4-dimethoxybenzenesulfonamide | IC50 | 7.6 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-intermediary-factor-1-alpha_3c24d53268a8db254d114742feb07841.svg) | 1-Methyl-5-(2-Methyl-1,3-Thiazol-4-Yl)-1,3-Dihydro-2h-Indol-2-One | IC50 | 8500.0 [1] |