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Transcription intermediary factor 1-alpha Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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▼
4-[(2s,4r)-1-Acetyl-4-[(4-Chlorophenyl)amino]-2-Methyl-1,2,3,4-Tetrahydroquinolin-6-Yl]benzoic AcidIC5010000.0 [1], 15848.93 [2]
CID 91827373IC501600.0 [1], 10000.0 [2]
N-[6-(4-Methoxyphenoxy)-1,3-Dimethyl-2-Oxo-2,3-Dihydro-1h-Benzimidazol-5-Yl]benzenesulfonamideIC50730.0 [1], 1500.0 [2]
Sgc-cbp30IC5020000.0 [1]
N-(1,3-Dimethyl-2-oxo-2,3-dihydro-1H-benzimidazol-5-yl)-4-methoxybenzenesulfonamideIC509300.0 [1]
N-(1,3-Dimethyl-2-oxo-2,3-dihydro-1H-benzimidazol-5-yl)-5,6,7,8-tetrahydro-2-naphthalenesulfonamideIC506170.0 [1]
N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)benzenesulfonamideIC5023000.0 [1]
N,2-Dimethyl-5-(3-methyl[1,2,4]triazolo[3,4-a]phthalazin-6-yl)benzenesulfonamideIC50100000.0 [1]
3-Cyano-N-(6-methoxy-1,3-dimethyl-2-oxobenzimidazol-5-yl)benzenesulfonamideIC5010000.0 [1]
3,4-Dimethoxy-N-[6-(4-methoxyphenoxy)-1,3-dimethyl-2-oxobenzimidazol-5-yl]benzenesulfonamideIC50430.0 [1]
N-[3-(3-Methyl-4-Oxo-4,5,6,7-Tetrahydro-2h-Isoindol-1-Yl)-4-Phenoxyphenyl]methanesulfonamideIC5010000.0 [1]
1-[2-(2,4-Difluorophenoxy)-5-methylsulfonylphenyl]-3-methyl-2,5,6,7-tetrahydropyrrolo[3,4-c]pyridin-4-oneIC5010000.0 [1]
N-[6-[3-(6-Aminohexoxy)-5-propoxyphenoxy]-1,3-dimethyl-2-oxobenzimidazol-5-yl]-1-methylimidazole-4-sulfonamideIC5010.0 [1]
N-[6-[3-(4-Aminobutoxy)-5-propoxyphenoxy]-1,3-dimethyl-2-oxobenzimidazol-5-yl]-1-methylimidazole-4-sulfonamideIC507.9 [1]
N-[6-[3-(3-Methoxypropoxy)phenoxy]-1,3-dimethyl-2-oxobenzimidazol-5-yl]-1,2-dimethylimidazole-4-sulfonamideIC50130.0 [1]
N-[1,3-Dimethyl-2-oxo-6-(3-phenylmethoxyphenoxy)benzimidazol-5-yl]-1-methylimidazole-4-sulfonamideIC50220.0 [1]
N-[1,3-Dimethyl-6-[3-(2-methylpropoxy)phenoxy]-2-oxobenzimidazol-5-yl]cyclopropanesulfonamideIC50110.0 [1]
N-[6-[3-(6-Aminohexoxy)-5-propoxyphenoxy]-1,3-dimethyl-2-oxobenzimidazol-5-yl]-3,4-dimethoxybenzenesulfonamideIC5013.0 [1]
N-[6-(3-Butoxyphenoxy)-1,3-dimethyl-2-oxobenzimidazol-5-yl]-1,2-dimethylimidazole-4-sulfonamideIC50160.0 [1]
N-[6-[3-(4-Aminobutoxy)-5-propoxyphenoxy]-1,3-dimethyl-2-oxobenzimidazol-5-yl]-3,4-dimethoxybenzenesulfonamideIC508.3 [1]
N-[1,3-Dimethyl-2-oxo-6-[3-(oxolan-3-ylmethoxy)phenoxy]benzimidazol-5-yl]-1-methylimidazole-4-sulfonamideIC50100.0 [1]
N-[1,3-Dimethyl-2-oxo-6-(3-phenylmethoxyphenoxy)benzimidazol-5-yl]-1,2-dimethylimidazole-4-sulfonamideIC50270.0 [1]
N-[6-[3-(3-Aminopropoxy)-5-propoxyphenoxy]-1,3-dimethyl-2-oxobenzimidazol-5-yl]-3,4-dimethoxybenzenesulfonamideIC5013.0 [1]
N-[6-[3-(5-Aminopentoxy)-5-propoxyphenoxy]-1,3-dimethyl-2-oxobenzimidazol-5-yl]-1-methylimidazole-4-sulfonamideIC5011.0 [1]
N-[6-[3-(6-Hydroxyhexoxy)-5-propoxyphenoxy]-1,3-dimethyl-2-oxobenzimidazol-5-yl]-1-methylimidazole-4-sulfonamideIC5060.0 [1]
N-[6-(3-Ethoxyphenoxy)-1,3-dimethyl-2-oxobenzimidazol-5-yl]-1,2-dimethylimidazole-4-sulfonamideIC50180.0 [1]
N-[1,3-Dimethyl-2-oxo-6-(3-propoxyphenoxy)benzimidazol-5-yl]-1,2-dimethylimidazole-4-sulfonamideIC5053.0 [1]
N-[1,3-Dimethyl-2-oxo-6-(3-propoxyphenoxy)benzimidazol-5-yl]-3,4-dimethoxybenzenesulfonamideIC5043.0 [1]
Tert-butyl N-[6-[3-[1,3-dimethyl-6-[(1-methylimidazol-4-yl)sulfonylamino]-2-oxobenzimidazol-5-yl]oxy-5-propoxyphenoxy]hexyl]carbamateIC50160.0 [1]
N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-2,2-dimethyl-3,4-dihydrochromene-6-sulfonamideIC503690.0 [1]
(2S)-N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-2,3-dimethoxy-2,3-dimethyl-1,4-benzodioxine-6-sulfonamideIC5010000.0 [1]
N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-3,4-dihydro-2H-chromene-6-sulfonamideIC504630.0 [1]
N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-2-methylbenzenesulfonamideIC502620.0 [1]
N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-3-methoxybenzenesulfonamideIC502380.0 [1]
N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-5,6,7,8-tetrahydronaphthalene-2-sulfonamideIC5010000.0 [1]
N-(1-Methyl-2-oxo-3H-indol-5-yl)-4-methylsulfanylbenzenesulfonamideIC5017000.0 [1]
N-(1-Methyl-2-oxo-3,4-dihydroquinolin-6-yl)-4-methylsulfanylbenzenesulfonamideIC504800.0 [1]
N-[6-[3-[4-(Dimethylamino)butoxy]phenoxy]-1,3-dimethyl-2-oxobenzimidazol-5-yl]-3,4-dimethoxybenzenesulfonamideIC50270.0 [1]
4-Cyclohexyl-N-(1-methyl-2-oxo-3,4-dihydroquinolin-6-yl)benzenesulfonamideIC502800.0 [1]
N-(7-Methoxy-1-methyl-2-oxo-3,4-dihydroquinolin-6-yl)benzenesulfonamideIC5036000.0 [1]
N-(1-Methyl-2-oxo-3,4-dihydroquinolin-7-yl)-4-methylsulfanylbenzenesulfonamideIC5014000.0 [1]
1,3-Dimethyl-5-[3-(2-methylpropoxy)phenoxy]benzimidazol-2-oneIC502400.0 [1]
N-[1,3-Dimethyl-2-oxo-6-(4-phenylmethoxyphenoxy)benzimidazol-5-yl]-1-methylimidazole-4-sulfonamideIC502000.0 [1]
3-[(1-Acetyl-5-methoxyindole-3-carbonyl)amino]-5-(furan-2-yl)benzoic acidIC5020000.0 [1]
3-[(1-Acetyl-5-methoxyindole-3-carbonyl)amino]-4-fluoro-5-(1-methylpyrazol-4-yl)benzoic acidIC5020000.0 [1]
3-[(1-Acetylindole-3-carbonyl)amino]-4-fluorobenzoic acidIC5020000.0 [1]
3-[(1-Acetylindole-3-carbonyl)amino]benzoic acidIC5020000.0 [1]
3-[(1-Acetylindole-3-carbonyl)amino]-5-(oxan-2-yloxymethyl)benzoic acidIC5020000.0 [1]
3-[(1-Acetyl-5-methoxyindole-3-carbonyl)amino]-5-(1-methylpyrazol-4-yl)benzoic acidIC5020000.0 [1]
3-[(1-Acetylindole-3-carbonyl)amino]-5-(furan-2-yl)benzoic acidIC5010440.0 [1]
N,N,2-Trimethyl-5-(3-methyl-[1,2,4]triazolo[3,4-a]phthalazin-6-yl)benzenesulfonamideIC50100000.0 [1]
2,4-Dimethoxy-N-(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl)benzenesulfonamideIC502500.0 [1]
4-Cyclohexyl-N-(1,3-dimethyl-2-oxo-2,3-dihydro-1H-benzimidazol-5-yl)benzenesulfonamideIC501700.0 [1]
N-(1-Methyl-2-oxo-3,4-dihydroquinolin-6-yl)-4-(2-methylpropoxy)benzenesulfonamideIC503700.0 [1]
N-[2-Methyl-5-(3-methyl[1,2,4]triazolo[3,4-a]phthalazin-6-yl)phenyl]methanesulfonamideIC50100000.0 [1]
N-[2-Methyl-5-(3-methyl[1,2,4]triazolo[3,4-a]phthalazin-6-yl)phenyl]propanamideIC50100000.0 [1]
N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-4-(2-methylpropoxy)benzenesulfonamideIC504000.0 [1]
N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-3-fluoro-4-methylbenzenesulfonamideIC5010000.0 [1]
N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-4-propan-2-ylbenzenesulfonamideIC503450.0 [1]
N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-2,3-dihydro-1H-indene-5-sulfonamideIC5010000.0 [1]
4-Chloro-N-(1,3-dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)benzenesulfonamideIC501560.0 [1]
N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-3,4-dimethoxybenzenesulfonamideIC50480.0 [1]
N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-3,4-dimethylbenzenesulfonamideIC504770.0 [1]
N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-4-methoxybenzenesulfonamideIC50740.0 [1]
N-[6-(4-Methoxyphenoxy)-1,3-dimethyl-2-oxobenzimidazol-5-yl]-2-methylbenzenesulfonamideIC501470.0 [1]
N-[6-(4-Methoxyphenoxy)-1,3-dimethyl-2-oxobenzimidazol-5-yl]-4-propoxybenzenesulfonamideIC508400.0 [1]
4-Chloro-N-(1,3-dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-2-methylbenzenesulfonamideIC502450.0 [1]
N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-5-fluoro-2-methylbenzenesulfonamideIC503420.0 [1]
N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-3-fluoro-4-methylbenzenesulfonamideIC502700.0 [1]
N-[6-(4-Methoxyphenoxy)-1,3-dimethyl-2-oxobenzimidazol-5-yl]-4-methylbenzenesulfonamideIC502700.0 [1]
4-Methoxy-N-[6-(4-methoxyphenoxy)-1,3-dimethyl-2-oxobenzimidazol-5-yl]benzenesulfonamideIC50770.0 [1]
N-(1,3-Dimethyl-2-oxo-6-phenoxy-2,3-dihydro-1H-benzimidazol-5-yl)-4-methylbenzenesulfonamideIC501270.0 [1]
N-(1,3-Dimethyl-2-oxo-2,3-dihydro-1H-benzimidazol-5-yl)-4-(methylsulfanyl)benzenesulfonamideIC504900.0 [1]
3-[2-(2,4-Difluorophenoxy)-5-methylsulfonylphenyl]-1-methyl-6H-pyrrolo[2,3-c]pyridin-7-oneIC5010000.0 [1]
N-[1,3-Dimethyl-2-oxo-6-(3-phenylmethoxyphenoxy)benzimidazol-5-yl]-3,4-dimethoxybenzenesulfonamideIC50140.0 [1]
N-[1,3-Dimethyl-6-[3-(2-methylpropoxy)phenoxy]-2-oxobenzimidazol-5-yl]-1,2-dimethylimidazole-4-sulfonamideIC5057.0 [1]
N-[6-[3-[4-(Dimethylamino)butoxy]-5-propoxyphenoxy]-1,3-dimethyl-2-oxobenzimidazol-5-yl]-3,4-dimethoxybenzenesulfonamideIC507.6 [1]
1-Methyl-5-(2-Methyl-1,3-Thiazol-4-Yl)-1,3-Dihydro-2h-Indol-2-OneIC508500.0 [1]
Items per page: 1 - 10 of 78
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References

This online tool may be cited as follows

MLA

"Quest Database™ Transcription intermediary factor 1-alpha Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 22 Dec. 2024, https://www.aatbio.com/data-sets/transcription-intermediary-factor-1-alpha-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 22). Quest Database™ Transcription intermediary factor 1-alpha Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/transcription-intermediary-factor-1-alpha-inhibitors-ic50-ki.
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