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Transcription initiation factor IIA alpha and bTranscription initiation factor IIA alpha and beta chains Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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(2R)-2-(Benzylsulfonylamino)-N-[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]-5-phenylpentanamideKi240.0 [1]
(2R)-2-(Benzylsulfonylamino)-N-[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]-5-pyridin-4-ylpentanamideKi1200.0 [1]
(2R)-2-(Benzylsulfonylamino)-N-[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]-5-(tetrazol-1-yl)pentanamideKi4700.0 [1]
(2S)-2-[[(2R)-2-(Benzylsulfonylamino)-2-phenylacetyl]amino]-N-[(4-carbamimidoylphenyl)methyl]-4-piperidin-4-ylbutanamideKi1700.0 [1]
(2S)-2-[[(2R)-2-(Benzylsulfonylamino)-4-pyridin-4-ylbutanoyl]amino]-N-[(4-carbamimidoylphenyl)methyl]-4-piperidin-4-ylbutanamideKi3900.0 [1]
(2S)-2-[[(2R)-2-(Benzylsulfonylamino)-4-(1-oxidopyridin-1-ium-4-yl)butanoyl]amino]-N-[(4-carbamimidoylphenyl)methyl]-4-piperidin-4-ylbutanamideKi9000.0 [1]
Methyl 3-[[(2R)-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]amino]-1-oxo-5-phenylpentan-2-yl]sulfamoylmethyl]benzoateKi920.0 [1]
3-[[(2R)-1-[[(2S)-1-[(4-Carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]amino]-1-oxo-5-phenylpentan-2-yl]sulfamoylmethyl]benzoic acidKi4400.0 [1]
(2S)-2-[[(2R)-4-(1-Acetylpiperidin-4-yl)-2-(benzylsulfonylamino)butanoyl]amino]-N-[(4-carbamimidoylphenyl)methyl]-4-piperidin-4-ylbutanamideKi8000.0 [1]
Methyl 4-[(3R)-3-(benzylsulfonylamino)-4-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]amino]-4-oxobutyl]piperidine-1-carboxylateKi13000.0 [1]
(2S)-2-[[(2R)-2-(Benzylsulfonylamino)-4-[1-(2-methoxyacetyl)piperidin-4-yl]butanoyl]amino]-N-[(4-carbamimidoylphenyl)methyl]-4-piperidin-4-ylbutanamideKi4500.0 [1]
4-[(3R)-3-(Benzylsulfonylamino)-4-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]amino]-4-oxobutyl]-N-methylpiperidine-1-carboxamideKi4800.0 [1]
4-[(3R)-3-(Benzylsulfonylamino)-4-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]amino]-4-oxobutyl]-N,N-dimethylpiperidine-1-carboxamideKi13000.0 [1]
(2S)-2-[[(2R)-2-(Benzylsulfonylamino)-4-[1-(cyclopropanecarbonyl)piperidin-4-yl]butanoyl]amino]-N-[(4-carbamimidoylphenyl)methyl]-4-piperidin-4-ylbutanamideKi8500.0 [1]
(2S)-2-[[(2R)-2-(Benzylsulfonylamino)-4-(1-butanoylpiperidin-4-yl)butanoyl]amino]-N-[(4-carbamimidoylphenyl)methyl]-4-piperidin-4-ylbutanamideKi5500.0 [1]
(2S)-2-[[(2R)-2-(Benzylsulfonylamino)-4-[1-(2-methylpropanoyl)piperidin-4-yl]butanoyl]amino]-N-[(4-carbamimidoylphenyl)methyl]-4-piperidin-4-ylbutanamideKi13000.0 [1]
(2R)-2-(Benzylsulfonylamino)-N-[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]-5-piperidin-4-ylpentanamideKi800.0 [1]
(2R)-5-(1-Acetylpiperidin-4-yl)-2-(benzylsulfonylamino)-N-[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]pentanamideKi3800.0 [1]
Methyl 4-[(4R)-4-(benzylsulfonylamino)-5-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]amino]-5-oxopentyl]piperidine-1-carboxylateKi3600.0 [1]
(2S)-2-[[(2R)-2-(Benzylsulfonylamino)-4-(1-propanoylpiperidin-4-yl)butanoyl]amino]-N-[(4-carbamimidoylphenyl)methyl]-4-piperidin-4-ylbutanamideKi5600.0 [1]
(2S)-2-[[(2R)-2-(Benzylsulfonylamino)-4-piperidin-4-ylbutanoyl]amino]-N-[(4-carbamimidoylphenyl)methyl]-4-piperidin-4-ylbutanamideKi4200.0 [1]
(2R)-2-(Benzylsulfonylamino)-N-[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]-5-(1-oxidopyridin-1-ium-4-yl)pentanamideKi4900.0 [1]
Items per page: 1 - 10 of 22
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References

This online tool may be cited as follows

MLA

"Quest Database™ Transcription initiation factor IIA alpha and bTranscription initiation factor IIA alpha and beta chains Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/transcription-initiation-factor-iia-alpha-and-btranscription-initiation-factor-iia-alpha-and-beta-chains-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ Transcription initiation factor IIA alpha and bTranscription initiation factor IIA alpha and beta chains Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/transcription-initiation-factor-iia-alpha-and-btranscription-initiation-factor-iia-alpha-and-beta-chains-inhibitors-ic50-ki.
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