![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_706b94c9e6ddb96fa5f00a1e011bdd19.svg) | 4-[(2-Amino-4-hydroxy-5-methylphenyl)diazenyl]-N-pyridin-2-ylbenzenesulfonamide | Ki | 7970.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_20a5468b26c48166284cfe2bfe6dfcdb.svg) | 4-[(2-Amino-3-chloro-4-hydroxy-5-methylphenyl)diazenyl]-N-pyridin-2-ylbenzenesulfonamide | Ki | 6560.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_ba6c458cef44ebde344a4c0e58953eb6.svg) | N-[3-(3-Methyl-4-Oxo-4,5,6,7-Tetrahydro-2h-Isoindol-1-Yl)-4-Phenoxyphenyl]methanesulfonamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_78158b41d3ba30afab4c7131b658e4ab.svg) | (3E)-3-(Piperidin-1-ylmethylidene)-1,2-dihydropyrrolo[1,2-a]quinazolin-5-one | IC50 | 6200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_e0d47f74704a19ff8747b92f04f3bb9e.svg) | (3E)-3-(Pyrrolidin-1-ylmethylidene)-1,2-dihydropyrrolo[1,2-a]quinazolin-5-one | IC50 | 9600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_76ea439d01964febde383f1c3a0f313f.svg) | (3E)-3-(Dimethylaminomethylidene)-1,2-dihydropyrrolo[1,2-a]quinazolin-5-one | IC50 | 11000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_14efdce93e11b1d9375a199a7e7fc809.svg) | (3E)-3-[(4-Ethylpiperazin-1-yl)methylidene]-1,2-dihydropyrrolo[1,2-a]quinazolin-5-one | IC50 | 6900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_8914b473c2244bc556a54a497a75e4ed.svg) | (3E)-3-[(4-Methylpiperazin-1-yl)methylidene]-1,2-dihydropyrrolo[1,2-a]quinazolin-5-one | IC50 | 7300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_4dccdc0627e500fdbec4234c8ba52c05.svg) | (3E)-3-[(4-Methyl-1,4-diazepan-1-yl)methylidene]-1,2-dihydropyrrolo[1,2-a]quinazolin-5-one | IC50 | 22000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_792128385a0dc40815074af547cea702.svg) | 1-(2-Chloropyridin-4-yl)-3-pyridin-2-ylurea | IC50 | 1700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_ab373dda620d78d6b6bdab256bb2a3af.svg) | 4-[(E)-(4-Hydroxy-3,5-Dimethylphenyl)diazenyl]-N-(Pyridin-2-Yl)benzenesulfonamide | Ki | 6560.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_5986419096142a2bb95e35881e46f18f.svg) | 4-[(E)-(2-Amino-4-Hydroxy-3,5-Dimethylphenyl)diazenyl]-N-(Pyridin-2-Yl)benzenesulfonamide | Ki | 6560.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_8cafb34395c07cdd2a7b01a10b410568.svg) | BRM/BRG1 ATP Inhibitor-1 | IC50 | 5.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_8b9d4ffc0c2de396b4535d1b90747393.svg) | 1-(2-Chloropyridin-4-yl)-3-[3-(difluoromethyl)-1,2-thiazol-5-yl]urea | IC50 | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_830e83c688ed4f380269c48f82f05373.svg) | 1-(2-Chloropyridin-4-yl)-3-(4-methyl-1,3-thiazol-2-yl)urea | IC50 | 570.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_62d4853ac5ca8e65099b7128626eb332.svg) | 1-(5-Amino-2-fluoropyridin-4-yl)-3-[3-(difluoromethyl)-1,2-thiazol-5-yl]urea | IC50 | 5.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_f75a2282e55702f84af6b89a39019dd7.svg) | 1-(2-Chloropyridin-4-yl)-3-(2-methylpyridin-4-yl)urea | IC50 | 150.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_c647bd0fb449300a2e1878e9a87a582b.svg) | 1-[2-Chloro-5-(hydroxymethyl)pyridin-4-yl]-3-[3-(difluoromethyl)-1,2-thiazol-5-yl]urea | IC50 | 5.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_06c57bd03550785bde5617556a1c096a.svg) | 1-(2-Chloropyridin-4-yl)-3-pyridin-4-ylurea | IC50 | 770.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_e4d662c88b463b1fae647fc4c016596d.svg) | 1-(2-Chloropyridin-4-yl)-3-[2-(trifluoromethyl)pyridin-4-yl]urea | IC50 | 30.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_2062c622ba20f9f2fa839b8c3be197a6.svg) | 1-(2-Chloropyridin-4-yl)-3-(3-methyl-1,2-thiazol-5-yl)urea | IC50 | 30.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_9a7b901cecb5d045fd87fc0211299a57.svg) | 1-(5-Amino-2-chloropyridin-4-yl)-3-[3-(difluoromethyl)-1,2-thiazol-5-yl]urea | IC50 | 5.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_a0007e04916623c2063c2b1535c77392.svg) | 1-(2-Chloropyridin-4-yl)-3-[3-(trifluoromethyl)-1,2-thiazol-5-yl]urea | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/transcription-activator-brg1_dc562a7b4f1d2c7d72c7eea3aa94fcab.svg) | 3-[2-(2,4-Difluorophenoxy)-5-methylsulfonylphenyl]-1-methyl-6H-pyrrolo[2,3-c]pyridin-7-one | IC50 | 1000.0 [1] |