Transcription activator BRG1 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	4-[(2-Amino-4-hydroxy-5-methylphenyl)diazenyl]-N-pyridin-2-ylbenzenesulfonamide	Ki	7970.0 [1]
	4-[(2-Amino-3-chloro-4-hydroxy-5-methylphenyl)diazenyl]-N-pyridin-2-ylbenzenesulfonamide	Ki	6560.0 [1]
	N-[3-(3-Methyl-4-Oxo-4,5,6,7-Tetrahydro-2h-Isoindol-1-Yl)-4-Phenoxyphenyl]methanesulfonamide	IC50	1000.0 [1]
	(3E)-3-(Piperidin-1-ylmethylidene)-1,2-dihydropyrrolo[1,2-a]quinazolin-5-one	IC50	6200.0 [1]
	(3E)-3-(Pyrrolidin-1-ylmethylidene)-1,2-dihydropyrrolo[1,2-a]quinazolin-5-one	IC50	9600.0 [1]
	(3E)-3-(Dimethylaminomethylidene)-1,2-dihydropyrrolo[1,2-a]quinazolin-5-one	IC50	11000.0 [1]
	(3E)-3-[(4-Ethylpiperazin-1-yl)methylidene]-1,2-dihydropyrrolo[1,2-a]quinazolin-5-one	IC50	6900.0 [1]
	(3E)-3-[(4-Methylpiperazin-1-yl)methylidene]-1,2-dihydropyrrolo[1,2-a]quinazolin-5-one	IC50	7300.0 [1]
	(3E)-3-[(4-Methyl-1,4-diazepan-1-yl)methylidene]-1,2-dihydropyrrolo[1,2-a]quinazolin-5-one	IC50	22000.0 [1]
	1-(2-Chloropyridin-4-yl)-3-pyridin-2-ylurea	IC50	1700.0 [1]
	4-[(E)-(4-Hydroxy-3,5-Dimethylphenyl)diazenyl]-N-(Pyridin-2-Yl)benzenesulfonamide	Ki	6560.0 [1]
	4-[(E)-(2-Amino-4-Hydroxy-3,5-Dimethylphenyl)diazenyl]-N-(Pyridin-2-Yl)benzenesulfonamide	Ki	6560.0 [1]
	BRM/BRG1 ATP Inhibitor-1	IC50	5.0 [1]
	1-(2-Chloropyridin-4-yl)-3-[3-(difluoromethyl)-1,2-thiazol-5-yl]urea	IC50	6.0 [1]
	1-(2-Chloropyridin-4-yl)-3-(4-methyl-1,3-thiazol-2-yl)urea	IC50	570.0 [1]
	1-(5-Amino-2-fluoropyridin-4-yl)-3-[3-(difluoromethyl)-1,2-thiazol-5-yl]urea	IC50	5.0 [1]
	1-(2-Chloropyridin-4-yl)-3-(2-methylpyridin-4-yl)urea	IC50	150.0 [1]
	1-[2-Chloro-5-(hydroxymethyl)pyridin-4-yl]-3-[3-(difluoromethyl)-1,2-thiazol-5-yl]urea	IC50	5.0 [1]
	1-(2-Chloropyridin-4-yl)-3-pyridin-4-ylurea	IC50	770.0 [1]
	1-(2-Chloropyridin-4-yl)-3-[2-(trifluoromethyl)pyridin-4-yl]urea	IC50	30.0 [1]
	1-(2-Chloropyridin-4-yl)-3-(3-methyl-1,2-thiazol-5-yl)urea	IC50	30.0 [1]
	1-(5-Amino-2-chloropyridin-4-yl)-3-[3-(difluoromethyl)-1,2-thiazol-5-yl]urea	IC50	5.0 [1]
	1-(2-Chloropyridin-4-yl)-3-[3-(trifluoromethyl)-1,2-thiazol-5-yl]urea	IC50	10.0 [1]
	3-[2-(2,4-Difluorophenoxy)-5-methylsulfonylphenyl]-1-methyl-6H-pyrrolo[2,3-c]pyridin-7-one	IC50	1000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 24 ⟨⟩

---

---

References

This online tool may be cited as follows

MLA	"Quest Database™ Transcription activator BRG1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/transcription-activator-brg1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, December 21). Quest Database™ Transcription activator BRG1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/transcription-activator-brg1-inhibitors-ic50-ki.
BibTeX	EndNote	RefMan