Trace amine-associated receptor 1 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Epptb	IC50	7490.0 [1]
	Epptb	Ki	5000.0 [1]
	N-(3-Methoxyphenyl)-4-(4-methylpiperidin-1-yl)-3-nitrobenzamide	IC50	3790.0 [1]
	N-(3-Methoxyphenyl)-4-(4-methylpiperidin-1-yl)-3-nitrobenzamide	Ki	20000.0 [1]
	4-(3,5-Dimethylpiperidin-1-yl)sulfonyl-3-fluoro-N-(3-methoxyphenyl)benzamide	IC50	10000.0 [1]
	4-(3,5-Dimethylpiperidin-1-yl)sulfonyl-3-fluoro-N-(3-methoxyphenyl)benzamide	Ki	20000.0 [1]
	Tolazoline	Ki	1640.0 [1]
	2-Benzyl-1h-imidazole	Ki	400.0 [1]
	1H-Imidazole, 2-[(2,6-dichlorophenyl)methyl]-4,5-dihydro-	Ki	500.0 [1]
	2-(2,6-Dimethyl-benzyl)-4,5-dihydro-1H-imidazole	Ki	82.0 [1]
	4-Benzyl-1H-imidazole	Ki	20.0 [1]
	N-Benzyl-N-(1H-imidazol-5-ylmethyl)aniline	Ki	32.0 [1]
	(1h-Imidazol-2-ylmethyl)phenylamine	Ki	4250.0 [1]
	1H-Imidazole, 5-(2-phenylethyl)-	Ki	2.0 [1]
	N-(1H-Imidazol-4-ylmethyl)aniline	Ki	65.0 [1]
	2-[(2,6-Dimethylphenyl)methyl]-1H-imidazole	Ki	36.0 [1]
	4-Chloro-N-(1H-imidazol-2-ylmethyl)-N-propan-2-ylaniline	Ki	138.0 [1]
	1H-Imidazole, 2-[(2,6-dichlorophenyl)methyl]-	Ki	1390.0 [1]
	3,5-Dichloro-N-(1H-imidazol-5-ylmethyl)-N-propan-2-ylaniline	Ki	4.0 [1]
	2-(2,6-Diethyl-benzyl)-4,5-dihydro-1H-imidazole	Ki	300.0 [1]
	2-(2,6-Diethyl-benzyl)-1H-imidazole	Ki	24.0 [1]
	3-Chloro-N-(1H-imidazol-2-ylmethyl)-N-propan-2-ylaniline	Ki	68.0 [1]
	Ethyl-(3H-imidazol-4-ylmethyl)-phenyl-amine	Ki	48.0 [1]
	Methyl-(3h-imidazol-4-ylmethyl)-phenyl-amine	Ki	11.0 [1]
	N-(1H-Imidazol-5-ylmethyl)-N-propan-2-ylaniline	Ki	22.0 [1]
	(3-Chloro-phenyl)-(3h-imidazol-4-ylmethyl)-methyl-amine	Ki	11.0 [1]
	3-Chloro-N-(1H-imidazol-5-ylmethyl)-N-propan-2-ylaniline	Ki	4.0 [1]
	N-(1H-Imidazol-5-ylmethyl)-3-methoxy-N-propan-2-ylaniline	Ki	5.0 [1]
	4-Chloro-N-(1H-imidazol-5-ylmethyl)-N-propan-2-ylaniline	Ki	6.0 [1]
	3,4-Dichloro-N-(1H-imidazol-5-ylmethyl)-N-propan-2-ylaniline	Ki	4.0 [1]
	4-Fluoro-N-(1H-imidazol-5-ylmethyl)-N-propan-2-ylaniline	Ki	13.0 [1]
	(3-Chloro-phenyl)-ethyl-(1h-imidazol-4-ylmethyl)-amine	Ki	2.0 [1]
	1-(1H-Imidazol-4-ylmethyl)-1,2,3,4-tetrahydro-quinoline	Ki	12.0 [1]
	1H-Indole, 2,3-dihydro-1-(1H-imidazol-5-ylmethyl)-	Ki	35.0 [1]
	2-(2,6-Bis-trifluoromethyl-benzyl)-4,5-dihydro-1H-imidazole	Ki	43000.0 [1]
	2-(2,6-Diisopropyl-benzyl)-1H-imidazole	Ki	630.0 [1]
	2-(2,6-Diisopropyl-benzyl)-4,5-dihydro-1H-imidazole	Ki	825.0 [1]
	(1H-Imidazol-2-ylmethyl)-isopropyl-phenyl-amine	Ki	470.0 [1]
	(1h-Imidazol-2-ylmethyl)-methyl-phenyl-amine	Ki	1270.0 [1]
	2-Chloro-N-(1H-imidazol-5-ylmethyl)-N-propan-2-ylaniline	Ki	40.0 [1]
	N-(1H-Imidazol-5-ylmethyl)-4-methoxy-N-propan-2-ylaniline	Ki	80.0 [1]
	Ethyl-(3H-imidazol-5-ylmethyl)-(4-methoxypyrimidin-2-yl)amine	Ki	84.0 [1]
	N-(1H-Imidazol-5-ylmethyl)-6-methoxy-N-propan-2-ylpyridin-2-amine	Ki	12.0 [1]
	N-(1H-Imidazol-5-ylmethyl)-N-phenylaniline	Ki	69.0 [1]
	3-Fluoro-N-(1H-imidazol-5-ylmethyl)-N-propan-2-ylaniline	Ki	12.0 [1]
	N-Cyclopropyl-N-(1H-imidazol-5-ylmethyl)aniline	Ki	100.0 [1]
	(3h-Imidazol-4-ylmethyl)-isopropyl-pyridin-2-yl-amine	Ki	195.0 [1]
	4-Chloro-N-(1H-imidazol-5-ylmethyl)-N-propan-2-ylpyrimidin-2-amine	Ki	100.0 [1]
	N-(1H-Imidazol-5-ylmethyl)-3-methylsulfonyl-N-propan-2-ylaniline	Ki	128.0 [1]
	2-Fluoro-N-(1H-imidazol-5-ylmethyl)-N-propan-2-ylaniline	Ki	18.0 [1]
	N-Tert-butyl-3-chloro-N-(1H-imidazol-5-ylmethyl)aniline	Ki	33.0 [1]
	CID 66552052	Ki	710.0 [1]
	2-[[2,6-Bis(trifluoromethyl)phenyl]methyl]-1H-imidazole	Ki	13300.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 53 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Trace amine-associated receptor 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Feb. 2025, https://www.aatbio.com/data-sets/trace-amine-associated-receptor-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, February 21). Quest Database™ Trace amine-associated receptor 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/trace-amine-associated-receptor-1-inhibitors-ic50-ki.
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