Thyroid stimulating hormone receptor Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	1-Acetyl-2,2,4-trimethyl-4-phenyl-3H-quinoline-6-carboxamide	IC50	88.0 [1]
	N-(1-Acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)-3-thiophen-2-ylpropanamide	IC50	100.0 [1]
	1-(1-Acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)-3-[(4-chlorophenyl)methyl]urea	IC50	100.0 [1]
	N-(1-Acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)-3-(4-chlorophenyl)propanamide	IC50	100.0 [1]
	[(2S)-3-Methylbutan-2-yl] N-(1-acetyl-4-methyl-4-phenyl-2,3-dihydroquinolin-6-yl)carbamate	IC50	100.0 [1]
	[(1S,2S)-2-Bicyclo[2.2.1]heptanyl] N-(1-acetyl-4-methyl-4-phenyl-2,3-dihydroquinolin-6-yl)carbamate	IC50	100.0 [1]
	N-(1-Acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)-3-[3-(trifluoromethyl)phenyl]propanamide	IC50	100.0 [1]
	N-(1-Acetyl-4-methyl-4-phenyl-2,3-dihydroquinolin-6-yl)-2-(3-chloro-4-fluorophenyl)acetamide	IC50	100.0 [1]
	1-(1-Acetyl-4-methyl-4-phenyl-2,3-dihydroquinolin-6-yl)-3-[(3-chlorophenyl)methyl]urea	IC50	100.0 [1]
	N-[(4R)-1-Acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl]-3-(3-chlorophenyl)propanamide	IC50	100.0 [1]
	N-[(4R)-1-Acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl]-3-[3-(trifluoromethyl)phenyl]propanamide	IC50	100.0 [1]
	Cyclopentyl N-[(4S)-1-acetyl-4-methyl-4-phenyl-2,3,4a,8a-tetrahydroquinolin-6-yl]carbamate	IC50	100.0 [1]
	N-[(4R)-1-Acetyl-4-methyl-4-phenyl-2,3-dihydroquinolin-6-yl]-2-(3-chloro-4-fluorophenyl)acetamide	IC50	100.0 [1]
	3-Methylbutyl N-(1-acetyl-4-methyl-4-phenyl-2,3-dihydroquinolin-6-yl)carbamate	IC50	100.0 [1]
	(1-Methylcyclopropyl)methyl N-(1-acetyl-4-methyl-4-phenyl-2,3-dihydroquinolin-6-yl)carbamate	IC50	100.0 [1]
	Cyclobutylmethyl N-(1-acetyl-4-methyl-4-phenyl-2,3-dihydroquinolin-6-yl)carbamate	IC50	100.0 [1]
	N-(1-Acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)hexanamide	IC50	100.0 [1]
	N-(1-Acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)pyridine-2-carboxamide	IC50	100.0 [1]
	2-Phenoxyethyl N-(1-acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)carbamate	IC50	100.0 [1]
	Butyl N-(1-acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)carbamate	IC50	100.0 [1]
	(3-Chloro-4-fluorophenyl)methyl N-(1-acetyl-4-methyl-4-phenyl-2,3-dihydroquinolin-6-yl)carbamate	IC50	47.0 [1]
	Cyclopentyl N-(1-acetyl-4-methyl-4-phenyl-2,3,4a,8a-tetrahydroquinolin-6-yl)carbamate	IC50	12.0 [1]
	N-(1-Acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)-3-(3-chlorophenyl)propanamide	IC50	100.0 [1]
	N-(1-Acetyl-4-methyl-4-phenyl-2,3-dihydroquinolin-6-yl)-5-bromothiophene-2-carboxamide	IC50	100.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 24 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Thyroid stimulating hormone receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Feb. 2025, https://www.aatbio.com/data-sets/thyroid-stimulating-hormone-receptor-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, February 21). Quest Database™ Thyroid stimulating hormone receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/thyroid-stimulating-hormone-receptor-inhibitors-ic50-ki.
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