![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_d2360a97a2e83af674174c745c41140d.svg) | 4-(4-(Benzo[d][1,3]dioxol-5-yl)-5-(pyridin-2-yl)-1H-imidazol-2-yl)benzamide | IC50 | 66.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_d2aaae557a3df420b61b69998679cc44.svg) | Dorsomorphin | IC50 | 102.9 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_4744f719e061d188f64f7298e92769bc.svg) | 4-(6-(4-(Piperazin-1-yl)phenyl)pyrazolo[1,5-a]pyrimidin-3-yl)quinoline | IC50 | 140.4 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_3e6bd5f7b4a571b8f74aa37a6047fdee.svg) | Galunisertib | IC50 | 1300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_5ccd1ebeb7ee5003bbac158cd721cb49.svg) | 4-[2-[4-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)quinolin-7-yl]oxyethyl]morpholine | IC50 | 190.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_e9ddbfd3b6f07208dc97db4e7ef39cb0.svg) | 4-(3-Pyridin-2-YL-1H-pyrazol-4-YL)quinoline | IC50 | 400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_c212e894513b08a44a48498579ea742a.svg) | LY-2090314 | IC50 | 1200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_f0a154106aee26d2cb409ff4c746c070.svg) | 3-Imidazo[1,2-a]pyridin-3-yl-4-[10-(morpholine-4-carbonyl)-1,10-diazatricyclo[6.4.1.04,13]trideca-2,4,6,8(13)-tetraen-3-yl]pyrrole-2,5-dione | IC50 | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_7c61426636de742e3bc9e56260715465.svg) | 5-[6-[4-(1-Piperazinyl)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | IC50 | 327.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_eb821ad270fe42b5a86634d12bb3a821.svg) | Ethyl 2,7,7-trimethyl-5-oxo-4-(4-phenylphenyl)-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 850.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_5bfa3a49106f8bec3217517a478b526a.svg) | Methyl 2,7,7-trimethyl-5-oxo-4-phenyl-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_498d85cce39dd7384f7a0bb29cf8216c.svg) | 3-(4-Imidazo[1,2-a]pyridin-3-yl-2,5-dioxopyrrol-3-yl)-N,N-dimethyl-1,10-diazatricyclo[6.4.1.04,13]trideca-2,4,6,8(13)-tetraene-10-carboxamide | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_135745c63ed912627deefccdab2cf518.svg) | 3-[6-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)benzimidazol-1-yl]propan-1-ol | IC50 | 352.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_6bad3df0a8f4743f2718943d69c2c4f6.svg) | 4-[3-[6-[2-(6-Methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]benzimidazol-1-yl]propyl]morpholine | IC50 | 19750.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_ed98d3f7c09ac11edc8356dc5b0faed9.svg) | 3-Imidazo[1,2-a]pyridin-3-yl-4-[10-(piperidine-1-carbonyl)-1,10-diazatricyclo[6.4.1.04,13]trideca-2,4,6,8(13)-tetraen-3-yl]pyrrole-2,5-dione | IC50 | 3100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_08529250ec2ce2c613602b3955d91e73.svg) | 3-[6-[2-(6-Methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]benzimidazol-1-yl]propan-1-ol | IC50 | 690.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_c7c3df679c3f2be78c0d5228a1850316.svg) | N-Ethyl-2-hydroxy-N-methyl-3-[C-phenyl-N-[4-(piperidin-1-ylmethyl)phenyl]carbonimidoyl]-1H-indole-6-carboxamide | IC50 | 19000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_62e5e5463f68a262f3a04054e212b325.svg) | Methyl 4-(biphenyl-4-yl)-2,7,7-trimethyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate | IC50 | 1490.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_6c7d29ccfb8f2b82860a3a3ff1e1bf60.svg) | 4-Methoxybenzyl 4-(biphenyl-4-yl)-2,7,7-trimethyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate | IC50 | 830.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_6ea384a833fe7c94fd437af047856629.svg) | Methyl 4-(4-tert-butylphenyl)-2,7,7-trimethyl-5-oxo-1,4,5,6,7,8-hexahydro-3-quinolinecarboxylate | IC50 | 560.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_0b3bef4951982c7469a1048c590b1d9c.svg) | Methyl 4-(4-fluorophenyl)-2,7,7-trimethyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_3690b6820a353232ff0cbe080abaf2b0.svg) | 4-(6-(4-Methoxyphenyl)pyrazolo[1,5-a]pyrimidin-3-yl)quinoline | IC50 | 236.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_679cfd0590ae1f0d16e0c64b14500fbe.svg) | N,N-Diethyl-3-[6-[2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]benzimidazol-1-yl]propan-1-amine | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_32260304c881c7e9a838fa55a76af1ee.svg) | 6-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1-(3-pyrrolidin-1-ylpropyl)benzimidazole | IC50 | 10840.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_f3d5c8a5dc74fd33094ffd0debe977a6.svg) | Ethyl 2-ethyl-7,7-dimethyl-5-oxo-4-(4-pyridin-2-ylphenyl)-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 3570.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_79211104fa9e8935353baf3730f88af5.svg) | [(4-{2-[(3-Hydroxyphenyl)amino]-1h-Benzimidazol-1-Yl}-1,3,5-Triazin-2-Yl)amino]acetonitrile | IC50 | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_f72122e87910200fe1ed05192270f4db.svg) | Methyl 4-[3-(3-chlorophenyl)phenyl]-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_e287ed5dd991a46defbc256f0e26d2fa.svg) | Methyl 7-ethyl-2-methyl-5-oxo-4-(4-phenylphenyl)-4,6,7,8-tetrahydro-1H-quinoline-3-carboxylate | IC50 | 790.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_a0d66fac974572abb0a34798a5b34dc1.svg) | Methyl 4-[4-(3-chlorophenyl)phenyl]-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 1520.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_e9f8419afde2394ffca30fe93aae6891.svg) | Ethyl 7,7-dimethyl-5-oxo-4-(4-phenylphenyl)-2-propyl-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 830.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_1d4a5c87634293dd705b9faf16621270.svg) | Methyl 2,7,7-trimethyl-5-oxo-4-(4-pyrazol-1-ylphenyl)-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 8800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_70b5cca739072559b6006713ee053286.svg) | Methyl 2-methyl-5-oxo-7-phenyl-4-(4-phenylphenyl)-4,6,7,8-tetrahydro-1H-quinoline-3-carboxylate | IC50 | 1920.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_12ca6da21f5fd32ed946d0ce3dcbb3ef.svg) | CID 60182364 | IC50 | 15.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_9ff18c07942722398a15ef844b620ff9.svg) | CID 60182389 | IC50 | 26.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_412de614e4031e722d3d92aad63f1520.svg) | 4-(4-(3-(1H-Pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-6-yl)phenyl)morpholine | IC50 | 1.37 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_e0e006ee9feaaec7d074b14392d6e557.svg) | Methyl 4-[3-(1H-indol-5-yl)phenyl]-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 4450.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_73c11cd52b9bf8be9152dabff6255236.svg) | Methyl 2-methyl-5-oxo-4-(4-phenylphenyl)-7-propyl-4,6,7,8-tetrahydro-1H-quinoline-3-carboxylate | IC50 | 530.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_ba54ea9e69adaa96041cceb25e7dd261.svg) | Methyl 7-[4-(dimethylamino)phenyl]-2-methyl-5-oxo-4-(4-phenylphenyl)-4,6,7,8-tetrahydro-1H-quinoline-3-carboxylate | IC50 | 3970.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_09f374893c3e804876339c51c52852a2.svg) | Methyl 2-methyl-7-(2-methylpropyl)-5-oxo-4-(4-phenylphenyl)-4,6,7,8-tetrahydro-1H-quinoline-3-carboxylate | IC50 | 590.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_cf9fb5bec15bed3ed098f2e7d95819a9.svg) | Methyl 2,7,7-trimethyl-5-oxo-4-(3-pyridin-3-ylphenyl)-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_38971a90f8e0f83ffe778df37a65f179.svg) | Methyl 2,7-dimethyl-5-oxo-4-(4-phenylphenyl)-4,6,7,8-tetrahydro-1H-quinoline-3-carboxylate | IC50 | 2730.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_9bdbfe38e3b4ef16a3edbe97bfa905eb.svg) | Methyl 4-(3-fluoro-4-phenylphenyl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 1840.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_88b147d238d5892c0fe0bd3e8bbb6ead.svg) | 2-Methylpropyl 4-(4-tert-butylphenyl)-2-methyl-5-oxo-7-propyl-4,6,7,8-tetrahydro-1H-quinoline-3-carboxylate | IC50 | 170.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_6201f6030a5ce9e9b9ccca1cf68fff7f.svg) | 2-Methylpropyl 2,7,7-trimethyl-5-oxo-4-(4-phenylphenyl)-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 530.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_c573eca3d5477e5828e35a19aa255c36.svg) | 3-Methylbutyl 2,7,7-trimethyl-5-oxo-4-(4-phenylphenyl)-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 1460.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_f3490cf2ec13191c7482203cc800b36b.svg) | Methyl 4-[4-(2-fluorophenyl)phenyl]-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 2060.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_3cd9888427d6dd37085dd5e611fb6638.svg) | Methyl 2-methyl-5-oxo-4-(4-phenylphenyl)-7-propan-2-yl-4,6,7,8-tetrahydro-1H-quinoline-3-carboxylate | IC50 | 940.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_29932908502cd1fbb0ded3485b8733bc.svg) | Methyl 4-(4-cyclohexylphenyl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 590.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_e106e8072675f3c80af614bafd6c5ea1.svg) | Methyl 4-[4-(1H-indol-5-yl)phenyl]-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 4050.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_0a434d2d2c97d9e0ad778ecb3ab11fc3.svg) | Methyl 4-[3-(4-methoxyphenyl)phenyl]-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_b4d680649874c966c46241d2f6093c9a.svg) | N-[(4-Methoxyphenyl)methyl]-2,7,7-trimethyl-5-oxo-4-(4-phenylphenyl)-1,4,6,8-tetrahydroquinoline-3-carboxamide | IC50 | 4060.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_e0505fc2cbee4d58c79680770e50df89.svg) | Methyl 4-[4-(4-methoxycarbonylphenyl)phenyl]-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 1350.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_764ef83ab707c6cb723ddae93831890b.svg) | Ethyl 4-(4-tert-butylphenyl)-2-methyl-5-oxo-7-propyl-4,6,7,8-tetrahydro-1H-quinoline-3-carboxylate | IC50 | 170.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_1f9d63e151317d67d7271a1eddad14e7.svg) | Methyl 2,7,7-trimethyl-5-oxo-4-(3-phenylphenyl)-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_40574e344d22bac4bb53932015862df6.svg) | 2,2,2-Trifluoroethyl 2,7,7-trimethyl-5-oxo-4-(4-phenylphenyl)-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 760.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_b2f2d3bad3be053f4442e5e3e36a5fee.svg) | Methyl 2,7,7-trimethyl-4-[4-(2-methylphenyl)phenyl]-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 890.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_59c6aab724852b8d67b99c2de32605b3.svg) | 6-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzimidazole | IC50 | 8730.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_c04fbddbc0ab9108e3eb71dae12a8a8d.svg) | 6-[2-(6-Methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1-(3-pyrrolidin-1-ylpropyl)benzimidazole | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_c1026b7908f4e5db836f77ab3d7edfde.svg) | 5-[2-(6-Methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1-[3-(oxan-2-yloxy)propyl]benzimidazole | IC50 | 14540.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_6f471ec8d26cc3f90ae463ae0799ae2d.svg) | 1-Methyl-6-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)benzimidazole | IC50 | 395.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_fcfcb9f09c76afcf95bfeac6aed6c031.svg) | 1-[3-(Oxan-2-yloxy)propyl]-5-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)benzimidazole | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_5552e6487f0ab3659321a0f425845e04.svg) | 6-[2-(6-Methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1-(3-piperidin-1-ylpropyl)benzimidazole | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_ae92bb23f717566f8e8e99089aa41b22.svg) | 1-Methyl-6-[2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]benzimidazole | IC50 | 668.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_5715f628b864353ae465bb7190af2e4e.svg) | Propan-2-yl 3-(4-imidazo[1,2-a]pyridin-3-yl-2,5-dioxopyrrol-3-yl)-1,10-diazatricyclo[6.4.1.04,13]trideca-2,4,6,8(13)-tetraene-10-carboxylate | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_7b77b20b9648173942886c5c04d36a35.svg) | 5-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-indole | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_a9be5c77c459be6a3988366cde650110.svg) | 6-[2-(6-Methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-benzimidazole | IC50 | 1300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_009f3e443fe19236d7793cb540927bcc.svg) | N-{4-[3-(5-Methoxypyridin-2-yl)-1H-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamide | IC50 | 15000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_396c1809408622de3bb9a7557734ad35.svg) | N-[4-[3-[5-(Trideuteriomethoxy)pyridin-2-yl]-1H-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl]acetamide | IC50 | 7600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_183f91508fae7ae9276cc4180c51e6ca.svg) | N-[4-[3-(6-Methylpyridin-2-yl)-1H-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl]acetamide | IC50 | 730.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_fc9a6c3f353922a1bc56bb7d7d59b927.svg) | N-{4-[3-(6-Methoxypyridin-3-yl)-1H-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamide | IC50 | 40.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_64d20c8c70fcc4994db4bb7188a54097.svg) | N-[4-[3-[6-(Trifluoromethyl)pyridin-2-yl]-1H-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl]acetamide | IC50 | 15000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_392e3b3d0093e13d08fc0e4b00560358.svg) | N-[4-[3-(6-Fluoropyridin-3-yl)-1H-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl]acetamide | IC50 | 7.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_bec1b48f17d66973c6c9fd52dd9ee440.svg) | N-[4-[3-[5-(Difluoromethoxy)pyridin-2-yl]-1H-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl]acetamide | IC50 | 14000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_703c26940dc4b65e5c1fb21a27a7c753.svg) | N-[4-[3-(5-Chloropyridin-2-yl)-1H-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl]acetamide | IC50 | 14000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_c7094de4b1a176533513649ff9750dc0.svg) | N-[4-[3-(5-Methylpyridin-2-yl)-1H-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl]acetamide | IC50 | 15000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_f384cf90a821872663a388f61dc6bc3a.svg) | N-[4-[3-[6-(Difluoromethyl)pyridin-2-yl]-1H-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl]acetamide | IC50 | 4300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_8c6b99acfadfd4e1d1e6fa09084e67e8.svg) | N-[4-[3-(5-Fluoropyridin-2-yl)-1H-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl]acetamide | IC50 | 390.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_2cfb3131248fc17811e1753392afae07.svg) | (3S,4S)-4-Amino-1-[[4-[(3-fluoropyridin-4-yl)amino]-2-pyridin-2-ylpyrrolo[2,1-f][1,2,4]triazin-5-yl]methyl]piperidin-3-ol | IC50 | 810.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_eec136fd5125342528fdc24f7b43017e.svg) | N-[5-Fluoro-4-[[2-[6-(trifluoromethyl)pyridin-2-yl]pyrrolo[2,1-f][1,2,4]triazin-4-yl]amino]pyridin-2-yl]acetamide | IC50 | 15000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_76ed7331d898c4bf22a67a4840d283ea.svg) | 2-(6-Methylpyridin-2-yl)-N-pyridin-4-ylpyrrolo[2,1-f][1,2,4]triazin-4-amine | IC50 | 550.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_91c9a0dc38e40ab68a80a46b8cdb38bc.svg) | N-Pyridin-4-yl-2-[6-(trifluoromethyl)pyridin-2-yl]pyrrolo[2,1-f][1,2,4]triazin-4-amine | IC50 | 8500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_4657324bd95c19d189be9c38f76a5fb0.svg) | N-(3-Fluoropyridin-4-yl)-2-pyridin-2-ylpyrrolo[2,1-f][1,2,4]triazin-4-amine | IC50 | 110.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_c931b636c65246a6af6a198669373352.svg) | 2-(6-Methoxypyridin-2-yl)-N-pyridin-4-ylpyrrolo[2,1-f][1,2,4]triazin-4-amine | IC50 | 15000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_e34f79f3d933cbf9babdf574419eb2e4.svg) | 4-[[2-(6-Methylpyridin-2-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]amino]-N-propan-2-ylpyridine-3-carboxamide | IC50 | 15000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_a7d318871c3dc2b68b2e9da62707ab37.svg) | N-(3-Fluoropyridin-4-yl)-2-[6-(trifluoromethyl)pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine | IC50 | 15000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_0c5abe85ec685a3cff4930cd04e250d9.svg) | N-[4-[[2-[6-(Trifluoromethyl)pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino]pyridin-2-yl]acetamide | IC50 | 940.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_b6c8e0b0c669d91870517864398c41d5.svg) | N-(3-Fluoropyridin-4-YL)-2-(6-methylpyridin-2-YL)-7H-pyrrolo[2,3-D]pyrimidin-4-amine | IC50 | 310.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_924674928efae6a950123e1d6cbff298.svg) | N-(3-Fluoropyridin-4-yl)-2-(6-methylpyridin-2-yl)-7H-purin-6-amine | IC50 | 1100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_7ed2fde712ec3dfe21da65fae29aefd2.svg) | CID 126677289 | IC50 | 1100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_70a8a2efd98d17b78514773e1d5308ac.svg) | N-(3,5-Difluoropyridin-4-yl)-2-(6-methylpyridin-2-yl)pyrrolo[2,1-f][1,2,4]triazin-4-amine | IC50 | 15000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_74b31a67ac193daebfb2bb4c5836b26d.svg) | 2-Pyridin-2-yl-N-pyridin-4-ylpyrrolo[2,1-f][1,2,4]triazin-4-amine | IC50 | 77.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_67073b31d107ba98447ac74d037b8660.svg) | 4-N-[[4-[(3-Fluoropyridin-4-yl)amino]-2-pyridin-2-ylpyrrolo[2,1-f][1,2,4]triazin-5-yl]methyl]cyclohexane-1,4-diamine | IC50 | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_d21590cc5ed96c469ec4286e6f73af8b.svg) | (3R,4R)-4-Amino-1-[[4-[(3-fluoropyridin-4-yl)amino]-2-pyridin-2-ylpyrrolo[2,1-f][1,2,4]triazin-5-yl]methyl]piperidin-3-ol | IC50 | 3000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_b5737ec8a578fb63e6da72d7dad4b428.svg) | N-(3-Fluoropyridin-4-yl)-2-(6-methylpyridin-2-yl)pyrrolo[2,1-f][1,2,4]triazin-4-amine | IC50 | 570.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_7465485b49f08e4cd9a2cea57d31727d.svg) | Alk2-IN-2 | IC50 | 698.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_4554dea7c0c950ec7103c94eb0c5aa1b.svg) | 3-Imidazo[1,2-a]pyridin-3-yl-4-[6-methyl-10-(piperidine-1-carbonyl)-1,10-diazatricyclo[6.4.1.04,13]trideca-2,4,6,8(13)-tetraen-3-yl]pyrrole-2,5-dione | IC50 | 9500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_da569f46166fb5a4efb41e6800f2a157.svg) | N,N-Dimethyl-3-[6-[2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]benzimidazol-1-yl]propan-1-amine | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_f29c45ad374a44e3cd2130f61df14c63.svg) | N,N-Dimethyl-3-[6-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)benzimidazol-1-yl]propan-1-amine | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-ii_7042a2bfb0bfc3bafa0ee59fb6233e6a.svg) | Indolocarbazole deriv. 14m | IC50 | 20000.0 [1] |