![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_e9ddbfd3b6f07208dc97db4e7ef39cb0.svg) | 4-(3-Pyridin-2-YL-1H-pyrazol-4-YL)quinoline | IC50 | 51.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_3d7fd13de900a9c7fee5495394736fdb.svg) | Benzamide, 3-((4-(6-methyl-2-pyridinyl)-5-(6-quinoxalinyl)-1H-imidazol-2-yl)methyl)- | IC50 | 17.2 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_d2360a97a2e83af674174c745c41140d.svg) | 4-(4-(Benzo[d][1,3]dioxol-5-yl)-5-(pyridin-2-yl)-1H-imidazol-2-yl)benzamide | IC50 | 94.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_d2360a97a2e83af674174c745c41140d.svg) | 4-(4-(Benzo[d][1,3]dioxol-5-yl)-5-(pyridin-2-yl)-1H-imidazol-2-yl)benzamide | Ki | 17.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_d8c9f64db0b5aad78138a2dd34a08b59.svg) | 2-(4-(Benzo[d][1,3]dioxol-5-yl)-2-tert-butyl-1H-imidazol-5-yl)-6-methylpyridine | IC50 | 54.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_e783c2adc532ed706f74adae49c2b479.svg) | RepSox | IC50 | 4.0 [1], 10.0 [2], 20.0 [3], 181.0 [4] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_bca7f3db243d5647ee899b9d088c6b6c.svg) | Vactosertib | IC50 | 7.0 [1], 9.67 [2], 16.5 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_bca7f3db243d5647ee899b9d088c6b6c.svg) | Vactosertib | Ki | 6.3 [1], 20.59 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_836af37d10c5d6dfb4a7491f582cf02e.svg) | 4-(3-Chlorophenyl)-5-(1,5-naphthyridin-2-yl)-1,3-thiazol-2-amine | IC50 | 10.0 [1], 13.0 [2], 20.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_3e6bd5f7b4a571b8f74aa37a6047fdee.svg) | Galunisertib | IC50 | 4.1 [1], 51.0 [2], 69.4 [3], 100.0 [4] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_f8f162e67a22db8d9b92500349990590.svg) | 4-(4-Fluorophenyl)-5-(1,5-naphthyridin-2-yl)thiazol-2-amine | IC50 | 10.0 [1], 11.0 [2], 30.0 [3], 40.0 [4] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_0b615c20b63ab538af14dd2362acbf2a.svg) | 5-[1,5]Naphthyridin-2-yl-4-pyridin-2-yl-thiazol-2-ylamine | IC50 | 20.0 [1], 40.0 [2], 120.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_b2c170fb55bc6e210aab26936c9f40de.svg) | 4-(3-(6-Methylpyridin-2-yl)-1H-pyrazol-4-yl)phenol | IC50 | 31.0 [1], 32.0 [2], 44.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_14a4fe5bb7fa98e23f44757ee31fed45.svg) | 4-(1-Benzyl-3-pyridin-2-yl-1H-pyrazol-4-yl)-quinoline | IC50 | 369.0 [1], 399.0 [2], 1340.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_67793dfeb7160c43b3983e6839021dbd.svg) | 4-(5-Cyclopropyl-3-pyridin-2-yl-1H-pyrazol-4-yl)-quinoline | IC50 | 94.0 [1], 203.0 [2], 538.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_9afd77d92c6fd0885d0145a5873e55f9.svg) | 2-(4-Phenyl-1H-pyrazol-3-yl)pyridine | IC50 | 3990.0 [1], 9000.0 [2], 9540.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_b7fb3ea14da658be3130019616feb476.svg) | 4-(3-(5-Fluoropyridin-2-yl)-1H-pyrazol-4-yl)quinoline | IC50 | 76.0 [1], 91.0 [2], 94.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_ddf4a0b262be3eb3c59bb530b071eff4.svg) | 4-(3-(Thiophen-2-yl)-1H-pyrazol-4-yl)quinoline | IC50 | 353.0 [1], 1660.0 [2], 2810.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_bb5f8e8288e9acc7dc877c5f5b747291.svg) | 4-(3-(5-Chloropyridin-2-yl)-1H-pyrazol-4-yl)quinoline | IC50 | 1760.0 [1], 4670.0 [2], 10000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_fd1f855133ea171ec83514fb4ef73a9e.svg) | 4-(4-Pyridin-2-yl-1H-pyrazol-3-yl)-quinoline | IC50 | 150.0 [1], 683.0 [2], 1680.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_f6239344e62db5889619de7028020509.svg) | 4-(3-Phenyl-1H-pyrazol-4-yl)quinoline | IC50 | 382.0 [1], 1200.0 [2], 2920.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_2ff79cb4feef2522c25dcb5edf6abf64.svg) | 4-(3-(3-(Trifluoromethyl)phenyl)-1H-pyrazol-4-yl)quinoline | IC50 | 217.0 [1], 355.0 [2], 524.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_157fad50be5e555e06cb4fbb0e45353a.svg) | 2-(3-Pyridin-2-yl-1H-pyrazol-4-yl)-[1,5]naphthyridine | IC50 | 10.0 [1], 19.0 [2], 30.0 [3], 50.0 [4] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_396c1809408622de3bb9a7557734ad35.svg) | N-[4-[3-[5-(Trideuteriomethoxy)pyridin-2-yl]-1H-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl]acetamide | IC50 | 2.0 [1], 17.0 [2], 110.0 [3], 450.0 [4] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_f384cf90a821872663a388f61dc6bc3a.svg) | N-[4-[3-[6-(Difluoromethyl)pyridin-2-yl]-1H-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl]acetamide | IC50 | 1.0 [1], 50.0 [2], 68.0 [3], 94.0 [4] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_d2aaae557a3df420b61b69998679cc44.svg) | Dorsomorphin | IC50 | 10000.0 [1], 10760.0 [2], 17090.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_4744f719e061d188f64f7298e92769bc.svg) | 4-(6-(4-(Piperazin-1-yl)phenyl)pyrazolo[1,5-a]pyrimidin-3-yl)quinoline | IC50 | 27.15 [1], 500.0 [2], 565.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_5ccd1ebeb7ee5003bbac158cd721cb49.svg) | 4-[2-[4-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)quinolin-7-yl]oxyethyl]morpholine | IC50 | 3.7 [1], 69.0 [2], 370.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_3aeedd1127f0020f9820de743bbea753.svg) | 4-(4-(3-(Pyridin-2-yl)-1H-pyrazol-4-yl)pyridin-2-yl)-N-(tetrahydro-2H-pyran-4-yl)benzamide | IC50 | 18.0 [1], 446.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_2ac762e24d3564bc0ada32a6ed72aec7.svg) | 4-(3-(6-Methylpyridin-2-yl)-1H-pyrazol-4-yl)quinoline | IC50 | 2.9 [1], 7.1 [2], 34.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_02c8af48926a785574973f3f64b4c02c.svg) | 4-((5-(6-Ethylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H-imidazol-2-yl)methylamino)benzamide | IC50 | 92.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_ac87a7701686c7c63d5a704e344afca2.svg) | 4-[4-(4-Fluorophenyl)-5-(2-pyridyl)-1H-imidazole-2-yl]benzoic acid | IC50 | 1500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_6bad3df0a8f4743f2718943d69c2c4f6.svg) | 4-[3-[6-[2-(6-Methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]benzimidazol-1-yl]propyl]morpholine | IC50 | 69.0 [1], 186.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_170881ac8d622079d40ac3bd5ef19194.svg) | 5-(6-Methyl-1,5-naphthyridin-4-yl)-4-(pyridin-2-yl)thiazol-2-amine | IC50 | 260.0 [1], 380.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_04b474e997b3aa2e10ba21466fd85b78.svg) | 5-Quinolin-4-yl-4-(1,3-thiazol-2-yl)-1,3-thiazol-2-amine | IC50 | 1170.0 [1], 1175.0 [2], 6580.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_7d8f087881be7ac4c11dad0b68e02ca8.svg) | 4-Pyridin-3-yl-5-quinolin-4-yl-thiazol-2-ylamine | IC50 | 3980.0 [1], 3981.0 [2], 10000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_cc16da50e72bc7166acb2961cffaded6.svg) | 4-(2-Fluorophenyl)-5-(quinolin-4-yl)thiazol-2-amine | IC50 | 1250.0 [1], 1259.0 [2], 6670.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_93cfaaff9f9dce622781f97bd19446eb.svg) | 4-(4-Chloropyridin-2-yl)-5-(quinolin-4-yl)thiazol-2-amine | IC50 | 1020.0 [1], 1023.0 [2], 10000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_efb8f90261ceaa3e93d6615d3a613550.svg) | 5-Naphthalen-1-yl-4-pyridin-2-yl-thiazol-2-ylamine | IC50 | 10000.0 [1], 10960.0 [2], 10965.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_08529250ec2ce2c613602b3955d91e73.svg) | 3-[6-[2-(6-Methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]benzimidazol-1-yl]propan-1-ol | IC50 | 41.0 [1], 78.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_04ec58793b8aaed2736ba79437754f96.svg) | SB-505124 hydrochloride | IC50 | 54.0 [1], 54.4 [2], 594.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_679cfd0590ae1f0d16e0c64b14500fbe.svg) | N,N-Diethyl-3-[6-[2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]benzimidazol-1-yl]propan-1-amine | IC50 | 100.0 [1], 122.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_32260304c881c7e9a838fa55a76af1ee.svg) | 6-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1-(3-pyrrolidin-1-ylpropyl)benzimidazole | IC50 | 226.0 [1], 246.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_74db2a8634f6c3131b5d37658561544e.svg) | 4-Pyridin-2-yl-5-quinolin-4-yl-thiazol-2-ylamine | IC50 | 274.0 [1], 420.0 [2], 720.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_885c36d84f7c8650c8d42d67f1ce1914.svg) | 4-[5-Methyl-3-(6-methyl-pyridin-2-yl)-1H-pyrazol-4-yl]-quinoline | IC50 | 24.0 [1], 82.0 [2], 148.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_f237176dd561ac07a67709432afd9aa3.svg) | 2-(4-(4-Fluorophenyl)-1H-pyrazol-3-yl)-6-methylpyridine | IC50 | 41.0 [1], 70.0 [2], 139.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_8d91b2a1b387aa9bd72a18a18a3160bb.svg) | 4-[3-(6-Bromo-pyridin-2-yl)-1H-pyrazol-4-yl]-quinoline | IC50 | 1.2 [1], 2.9 [2], 31.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_4f10dae7830ba8c10b94659e68dabf95.svg) | 3-(2-Pyridinyl)-4-(4-fluorophenyl)-1H-pyrazole | IC50 | 275.0 [1], 2590.0 [2], 3530.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_afecd5c497c14ea95fa9048dd67f3ce1.svg) | 2-[4-(4-Chloro-phenyl)-1H-pyrazol-3-yl]-6-methyl-pyridine | IC50 | 57.0 [1], 421.0 [2], 551.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_a992f4652f6be277e8956a2f42f818cc.svg) | 2-Methyl-6-(4-phenyl-1H-pyrazol-3-yl)-pyridine | IC50 | 543.0 [1], 2160.0 [2], 3370.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_ef0e4b3846a70fee77c86e17ed8ea761.svg) | 2-[4-(3,4-Difluoro-phenyl)-1H-pyrazol-3-yl]-6-methyl-pyridine | IC50 | 151.0 [1], 683.0 [2], 788.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_edcf1c8ccd068a90139a554edee26dea.svg) | 2-[4-(4-Methoxyphenyl)-1-methylpyrazol-3-yl]-6-methylpyridine | IC50 | 44.0 [1], 47.0 [2], 61.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_85f600dfa279e3171ebfcf535bc63cf2.svg) | 4-(6-Methyl-pyridin-2-yl)-5-[1,5]naphthyridin-2-yl-thiazol-2-ylamine | IC50 | 6.0 [1], 10.0 [2], 20.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_87a908686fba16f8b7b77efdff44c154.svg) | 2-[4-Methyl-2-(6-methyl-pyridin-2-yl)-2H-pyrazol-3-yl]thieno[3,2-c]pyridine | IC50 | 6.65 [1], 35.9 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_d734a0668dc15dc0288598331ada425a.svg) | 2-[2-(6-Methylpyridin-2-yl)pyrazol-3-yl]thieno[3,2-c]pyridine | IC50 | 23.4 [1], 149.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_3d7e78277d65064399703bb35464d261.svg) | 2-[5-Methyl-2-(6-methylpyridin-2-yl)pyrazol-3-yl]thieno[3,2-c]pyridine | IC50 | 94.1 [1], 440.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_7a17249c76ea1a65cd90fcd0fbe0406d.svg) | 2-[5-Ethyl-2-(6-methylpyridin-2-yl)pyrazol-3-yl]thieno[3,2-c]pyridine | IC50 | 108.0 [1], 403.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_2cd5a1652530eb846695d3776ba622d9.svg) | 2-[4-Ethyl-2-(6-methylpyridin-2-yl)pyrazol-3-yl]thieno[3,2-c]pyridine | IC50 | 4.33 [1], 21.5 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_de7a6b75e077f41fd2b2daf306190322.svg) | 2-[2-(6-Methylpyridin-2-yl)-5,6-dihydro-4H-cyclopenta[c]pyrazol-3-yl]thieno[3,2-c]pyridine | IC50 | 12.9 [1], 30.8 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_3b6035957cd7c804e4c0d5b86d5b72c1.svg) | 2-[4,5-Dimethyl-2-(6-methylpyridin-2-yl)pyrazol-3-yl]thieno[3,2-c]pyridine | IC50 | 35.2 [1], 244.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_afc05c499561fd28d432b45933a35860.svg) | 2-[4-Methyl-2-(6-methylpyridin-2-yl)pyrazol-3-yl]thieno[2,3-c]pyridine | IC50 | 7.94 [1], 42.5 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_51cd4d95feba74ec2a326dfe57d3f7b4.svg) | 2-[2-(6-Methylpyridin-2-yl)-5,6-dihydro-4H-cyclopenta[c]pyrazol-3-yl]thieno[2,3-c]pyridine | IC50 | 18.9 [1], 57.5 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 6870.0 [1], 18500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_b96c95589239aa5fc9b995c3e9055da0.svg) | 4-(4-Fluorophenyl)-2-(4-methylsulfinylphenyl)-5-(4-pyridyl)-1H-imidazole | IC50 | 6000.0 [1], 30000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_ff0d43edb17f983137c243b2b294bebc.svg) | 3-[6-Amino-5-(3,4,5-Trimethoxyphenyl)pyridin-3-Yl]phenol | IC50 | 280.0 [1], 3400.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_77133570e896153ed2bcf3545f22a0e5.svg) | 1-(4-(6-Methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl)phenyl)piperazine | IC50 | 3000.0 [1], 16000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_a3eb1c0196423a11d157d89a65d61d29.svg) | 2-Phenyl-4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridine | IC50 | 107.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_4d9372d552e995d0cae5a543bff064c8.svg) | 4-[4-(1,3-Benzodioxole-5-yl)-5-(2-pyridyl)-1H-imidazole-2-yl]benzyl alcohol | IC50 | 260.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_367c8c616e3bc9ceadb1375485a54f31.svg) | 2-(4-(2-(1H-Imidazol-1-yl)ethoxy)phenyl)-4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridine | IC50 | 30.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_ec48d6555446a000627b90bb84146829.svg) | 3-Benzo[1,3]dioxol-5-yl-2-pyridin-2-yl-6,7-dihydro-5H-pyrrolo[1,2-a]imidazole | IC50 | 460.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_7c0dc9192eeac8359b048be64ae65627.svg) | 2-(4-Fluorophenyl)-4-(5-pyridin-2-yl-1H-pyrazol-4-yl)pyridine | IC50 | 48.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_38e42a57fc1c3093bdc8a1547a18c603.svg) | 2-[3-Methoxyphenyl]-4-(3-pyridin-2-yl-1H-pyrazol-4-yl)pyridine | IC50 | 115.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_e64996fea835b8cfe100ac9f6c1a845a.svg) | N-[[4-(1,3-Benzothiazol-6-yl)-5-(4-methyl-1,3-thiazol-2-yl)-1H-imidazol-2-yl]methyl]butanamide | IC50 | 8.2 [1], 32.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_26d82b9748acbf3308fb8957664e459f.svg) | 4-[[4-(1,3-Benzodioxol-5-yl)-5-(6-methylpyridin-2-yl)-1H-imidazol-2-yl]methylamino]benzonitrile | IC50 | 46.0 [1], 174.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_ae61be283e2497c869eba322d5cf92f9.svg) | 4-[[4-(1,3-Benzodioxol-5-yl)-5-(6-ethylpyridin-2-yl)-1H-imidazol-2-yl]methylamino]benzonitrile | IC50 | 360.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_870389911b97886dbdffae994d2d5aee.svg) | 3-((5-(6-Methylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H-imidazol-2-yl)methylamino)benzamide | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_d47bc9e22c0c2a0b52d3b8f84b88474c.svg) | 4-[[[4-(1,3-Benzodioxol-5-yl)-5-(6-methylpyridin-2-yl)-1H-imidazol-2-yl]amino]methyl]benzonitrile | IC50 | 24.0 [1], 153.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_26304f1eeda6ee0aefdb220dc709f37c.svg) | 3-[[4-(1,3-Benzodioxol-5-yl)-5-(6-ethylpyridin-2-yl)-1H-imidazol-2-yl]methylamino]benzonitrile | IC50 | 73.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_6335abb3a09e6922b9a07d6000f47c27.svg) | 4-((5-(6-Ethylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H-imidazol-2-yl)methylamino)benzonitrile | IC50 | 47.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_5dde7406865fc01fa73ec8fe69869e5d.svg) | 4-[[4-(1,3-Benzodioxol-5-yl)-5-(6-methylpyridin-2-yl)-1H-imidazol-2-yl]methylamino]benzamide | IC50 | 21.0 [1], 262.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_8484589f036e6ff32aa1745dc3a76e0b.svg) | 4-[[4-(1,3-Benzodioxol-5-yl)-5-(6-ethylpyridin-2-yl)-1H-imidazol-2-yl]methylamino]benzamide | IC50 | 46.0 [1], 385.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_8887e50869a64ff6a30bdc92e8476d88.svg) | 4-((5-(6-Methylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H-imidazol-2-yl)methylamino)benzamide | IC50 | 75.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_61d4778f101390b6dbc64262f4e45155.svg) | 4-(4-(Benzo[d][1,3]dioxol-5-yl)-5-(pyridin-2-yl)-1H-imidazol-2-yl)benzoic acid | IC50 | 170.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_0841d37f2eca69619cfd675ea4d0a3d8.svg) | N-[2-(Methoxy)ethyl]-4-{4-[3-(pyridin-2-yl)-1H-pyrazol-4-yl]-pyridin-2-yl}benzamide | IC50 | 91.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_5f66b01171ce3f3ad49418853898f25d.svg) | 4-(3-(Pyridin-2-yl)-1H-pyrazol-4-yl)-2-(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)pyridine | IC50 | 40.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_135745c63ed912627deefccdab2cf518.svg) | 3-[6-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)benzimidazol-1-yl]propan-1-ol | IC50 | 79.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_a7084205209e18e63b9c23d025e38ba6.svg) | 3-(4-Methoxyphenyl)-2-(2-pyridyl)-6,7-dihydro-5H-pyrrolo[1,2-a]imidazole | IC50 | 5100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_686f494d1981008dd525659972ae99a6.svg) | 2-(4-(2-Cyclohexylethoxy)phenyl)-4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridine | IC50 | 81.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_0f4b0887be9dc6749114be639b288164.svg) | 2-[4-Cyanophenyl]-4-(3-pyridin-2-yl-1H-pyrazol-4-yl)pyridine | IC50 | 35.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_6ec229f837654047ef5e159a17cebec1.svg) | 2-[3-(Trifluoromethyl)phenyl]-4-(3-pyridin-2-yl-1H-pyrazol-4-yl)pyridine | IC50 | 240.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_3429e430f22ef510031ac69935c1c0ce.svg) | N-(4-{4-[3-(Pyridin-2-yl)-1H-pyrazol-4-yl]-pyridin-2-yl}phenyl)-tetrahydro-2H-pyran-4-carboxamide | IC50 | 112.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_308392e1e97a8a801f267080126818a6.svg) | N-Methyl-4-{4-[3-(pyridin-2-yl)-1H-pyrazol-4-yl]-pyridin-2-yl}-N-(tetrahydro-2H-pyran-4-yl)benzamide | IC50 | 214.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_e5d04ca1b9990ebe3e9adb2d2b0742fc.svg) | 2-[2-Fluorophenyl]-4-(3-pyridin-2-yl-1H-pyrazol-4-yl)pyridine | IC50 | 59.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_0989c247dd4f4e30adcca1325db55edc.svg) | 1-(4-(4-(3-(Pyridin-2-yl)-1H-pyrazol-4-yl)pyridin-2-yl)phenoxy)propan-2-one | IC50 | 25.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_b49f7d577fb47cefba8247892cb8b29b.svg) | Dimethyl-{2-[(4-{4-[3-(pyridin-2-yl)-1H-pyrazol-4-yl]-2-pyridinyl}phenyl)oxy]ethyl}amine | IC50 | 15.0 [1], 19.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_54abc3db88e6fe927dda07174acf81a1.svg) | 6-[4-(4-Methyl-2-thiazolyl)-1H-imidazole-5-yl]benzothiazole | IC50 | 2.7 [1], 8.7 [2] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_769ce4aa7c0619a5f9feca1796231fc8.svg) | 5-(4-Fluorophenyl)-6-(2-pyridyl)-2,3-dihydroimidazo[2,1-b]thiazole | IC50 | 1600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_6099a4fdf497b4b0144e6375146edb81.svg) | 5-(5-Fluoro-6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H-imidazol-2-amine | IC50 | 33.5 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_6099a4fdf497b4b0144e6375146edb81.svg) | 5-(5-Fluoro-6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H-imidazol-2-amine | Ki | 0.7 [1] |
![](https://images.aatbio.com/dataset/ic50/tgf-beta-receptor-type-i_886cc511bac3440bd0acee965fdf5ac1.svg) | N-(4-Methoxyphenyl)-3-(6-methylpyridin-2-yl)-4-([1,2,4]triazolo[1,5-a]pyridin-6-yl)pyrazole-1-carbothioamide | IC50 | 0.57 [1], 6360.0 [2] |