![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_0a83b01cf93719a90ccaeda771089c43.svg) | Doramapimod | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_99d590530c99b53efc4907213bcd8b23.svg) | 7-Chloro-3-oxo-8-(1,3-thiazol-5-ylmethylamino)-11,16-dioxa-2,4,19,21-tetrazatricyclo[15.3.1.05,10]henicosa-1(20),5,7,9,17(21),18-hexaene-18-carbonitrile | Ki | 1526.0 [1] |
![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_21aa752395444707db3d7c65ae53dc35.svg) | 1-({4-[(3,4-Dichlorophenyl)methoxy]phenyl}methyl)azetidine-3-carboxylic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_d019ff4da979aeb51ea88bb93c1f1472.svg) | 5-(4-Chlorophenyl)-N-(4-piperazin-1-ylphenyl)furan-2-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_262c5527ba96216e81ae5e081ba9279f.svg) | 3-Methyl-N-[6-methylsulfanyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]-1,2-thiazol-5-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_77eb8e9cdf9ebb4dafaaacd9407e9c0b.svg) | 3-[(1R)-1-[(2S,6R)-2,6-Dimethylmorpholin-4-yl]ethyl]-N-[6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]-1,2-thiazol-5-amine | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_400786f64062ecb5f10a9d3b11455207.svg) | 1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_3e5e956fd3311d2f1725fa72559e89d1.svg) | CID 59627005 | IC50 | 30.6 [1] |
![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_5b5057f07ba36d969b42e83280bc9205.svg) | 2-[3-(3-Piperidin-4-ylpropoxy)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_61551f1612b1d03b33f689e3fdae85ae.svg) | 2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_be3215402906f80de76893d9c9f28399.svg) | 2-[Ethyl-[[5-[[6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino]-1,2-thiazol-3-yl]methyl]amino]ethanol | IC50 | 500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_09c777664a74d957394c48618430a40f.svg) | 2-(5-Methoxy-3-oxo-1H-isoindol-2-yl)-N-(4-piperazin-1-ylpyridin-3-yl)-1,3-thiazole-4-carboxamide | IC50 | 8900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_2db2a2d148038bcb7681f06d72b80a8e.svg) | N-[6-Methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]-3-(pyridin-2-ylmethyl)-1,2-thiazol-5-amine | IC50 | 500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_b846b3952b86b7c4b437a16a51fb1e05.svg) | 8-[(4-Aminocyclohexyl)amino]-2-(4-chlorophenyl)imidazo[1,2-a]pyrazine-5-carboxamide | IC50 | 12000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_079d46552bd9bfffd84d80bdda6c59b9.svg) | 3-[Dideuterio-(3,3-difluoropyrrolidin-1-yl)methyl]-N-[6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]-1,2-thiazol-5-amine;hydrochloride | IC50 | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_9296ce5228829a70797f4a55b8cdc874.svg) | 2-(4-Chlorophenyl)-8-piperazin-1-yl-5-[(2-pyridin-3-ylphenyl)methyl]-10H-furo[2,3-c][1]benzazepin-4-one | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_a24e3192a9ff50577fd7c3e72a2d7066.svg) | 3-[(3,3-Difluoropyrrolidin-1-yl)methyl]-N-[6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]-1,2-thiazol-5-amine;hydrochloride | IC50 | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_5efd76d03838ecc45636f311fa9c0a92.svg) | SCH-1473759 (hydrochloride) | IC50 | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_2f905efdbe6d8f0fedfc64e5dcd53382.svg) | (3R)-1-[2-[4-(4-Acetylphenyl)piperazin-1-yl]-2-oxoethyl]-N-(3-chloro-4-hydroxyphenyl)pyrrolidine-3-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_700247dab7b9fdcc2d81fe4984afa76c.svg) | 2-[3-(3-Piperazin-1-ylpropoxy)phenyl]-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/testis-specific-serine-threonine-protein-kinase-2_f28e47e67ea642604198866d9f11a2d4.svg) | 1-[4-[2-[5-(4-Chlorophenyl)furan-2-yl]imidazol-1-yl]phenyl]piperazine | IC50 | 30000.0 [1] |