Terminal deoxynucleotidyltransferase Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Ethyl (E)-6-[4-(4-cyanobenzoyl)-1H-pyrrol-2-yl]-2,4-dioxohex-5-enoate	Ki	1500.0 [1], 1700.0 [2]
	(E)-6-[4-(2-Fluorobenzoyl)-1H-pyrrol-2-yl]-2,4-dioxohex-5-enoic acid	Ki	400.0 [1], 500.0 [2]
	(E)-6-[1-[(4-Hydroxyphenyl)methyl]indol-3-yl]-2,4-dioxohex-5-enoic acid	Ki	450.0 [1], 500.0 [2]
	Untenone A	IC50	16000.0 [1]
	(1S,2S)-2-Hexadecyl-2-methoxymethoxy-5-oxo-cyclopent-3-enecarboxylic acid methyl ester	IC50	18000.0 [1]
	(3As,4S,7R,7aR)-1,6-dihexadecyl-2,7-bis(methoxycarbonyl)-3-oxo-3a,4,7,7a-tetrahydroindene-4-carboxylic acid	IC50	2500.0 [1]
	(3As,4S,7R,7aR)-1,6-diethyl-2,7-bis(methoxycarbonyl)-3-oxo-3a,4,7,7a-tetrahydroindene-4-carboxylic acid	IC50	50000.0 [1]
	2-Hexadecyl-5-oxo-cyclopent-1-enecarboxylic acid methyl ester	IC50	129000.0 [1]
	Trimethyl (1aR,1bR,2R,5S,5aS,6aS)-1a,3-dihexadecyl-6-oxo-1b,2,5,5a-tetrahydro-1H-cyclopropa[a]indene-2,5,6a-tricarboxylate	IC50	12500.0 [1]
	(R)-4-Hexadecyl-4-hydroxy-cyclopent-2-enone	IC50	200000.0 [1]
	(1R,2S)-2-Hexadecyl-5-oxo-cyclopent-3-enecarboxylic acid methyl ester	IC50	84000.0 [1]
	(3As,4R,7R,7aR)-1,6-dihexadecyl-7-methoxycarbonyl-3a,4,7,7a-tetrahydro-3H-indene-2,4-dicarboxylic acid	IC50	2500.0 [1]
	(3As,4S,7R,7aR)-1,6-didodecyl-2,7-bis(methoxycarbonyl)-3-oxo-3a,4,7,7a-tetrahydroindene-4-carboxylic acid	IC50	8600.0 [1]
	(3As,4S,7R,7aR)-1,6-dihexadecyl-3-oxo-2,7-bis(propan-2-yloxycarbonyl)-3a,4,7,7a-tetrahydroindene-4-carboxylic acid	IC50	20000.0 [1]
	Methyl (2S,3S,4R,5E)-2-ethyl-4-hydroxy-5-(2-oxononadecylidene)-1-(2-phenylethyl)pyrrolidine-3-carboxylate	IC50	25000.0 [1]
	Methyl (2R,3S,4R,5E)-4-hydroxy-5-(2-oxononadecylidene)-2-phenyl-1-(2-phenylethyl)pyrrolidine-3-carboxylate	IC50	50000.0 [1]
	7-O-Ethyl 2-O,4-O-dimethyl (3aR,4R,7S,7aS)-3,5-dihexadecyl-1-oxo-3a,4,7,7a-tetrahydroindene-2,4,7-tricarboxylate	IC50	39700.0 [1]
	7-O-Ethyl 2-O,4-O-dimethyl (3aR,4S,7S,7aS)-3,5-dihexadecyl-1-oxo-3a,4,7,7a-tetrahydroindene-2,4,7-tricarboxylate	IC50	48400.0 [1]
	Methyl (2S,3S,4R,5E)-2-ethyl-4-hydroxy-5-(2-oxotetradecylidene)-1-(2-phenylethyl)pyrrolidine-3-carboxylate	IC50	50000.0 [1]
	Methyl (2S,3S,4R,5E)-1-benzyl-2-ethyl-4-hydroxy-5-(2-oxotetradecylidene)pyrrolidine-3-carboxylate	IC50	50000.0 [1]
	Methyl (2S,3S,4S,5E)-1-benzyl-2-ethyl-4-hydroxy-5-(2-oxotetradecylidene)pyrrolidine-3-carboxylate	IC50	50000.0 [1]
	Dimethyl (3aR,4R,7S,7aS)-3,5-dihexadecyl-1-oxo-7-(2-phenylethylcarbamoyl)-3a,4,7,7a-tetrahydroindene-2,4-dicarboxylate	IC50	12500.0 [1]
	Methyl (2R,3S,4R,5E)-4-hydroxy-1-[2-(1H-indol-3-yl)ethyl]-5-(2-oxotetradecylidene)-2-phenylpyrrolidine-3-carboxylate	IC50	50000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 23 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Terminal deoxynucleotidyltransferase Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/terminal-deoxynucleotidyltransferase-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, November 21). Quest Database™ Terminal deoxynucleotidyltransferase Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/terminal-deoxynucleotidyltransferase-inhibitors-ic50-ki.
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