 | 3-(1-((3,5-Dimethylisoxazol-4-yl)methyl)-1H-pyrazol-4-yl)-1-(3-hydroxybenzyl)imidazolidine-2,4-dione | IC50 | 30.0 [1], 35.0 [2] |
 | 4-[Benzyl-[(4-methoxyphenyl)methyl]sulfamoyl]benzoic acid | IC50 | 200.0 [1] |
 | N-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]imidazol-4-yl]-2,3-dihydro-1H-indene-5-carboxamide | IC50 | 12100.0 [1] |
 | N-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-2-phenylpropanamide | IC50 | 300.0 [1] |
 | N-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-3-methoxybenzamide | IC50 | 400.0 [1] |
 | Methyl 3-[[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]sulfamoyl]thiophene-2-carboxylate | IC50 | 1252.0 [1] |
 | 1-(2,5-Dimethoxyphenyl)-3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]thiourea | IC50 | 5240.0 [1] |
 | [2-[[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]amino]-2-oxo-1-phenylethyl] acetate | IC50 | 830.0 [1] |
 | 3-Chloro-N-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-4-methylsulfonylthiophene-2-carboxamide | IC50 | 2090.0 [1] |
 | (5S)-1-Benzyl-3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5-methylimidazolidine-2,4-dione | IC50 | 10.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(3-hydroxy-5-methoxyphenyl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 20.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(4-fluoro-3-hydroxyphenyl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 10.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[2-(4-methoxyphenyl)ethyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 120.0 [1] |
 | 6-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-4-[(3-hydroxyphenyl)methyl]-4,6-diazaspiro[2.4]heptane-5,7-dione | IC50 | 20.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethyl-1-(1-phenylethyl)imidazolidine-2,4-dione | IC50 | 150.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(1,5-dimethylpyrazol-3-yl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 160.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-(2-methoxyethyl)-5,5-dimethylimidazolidine-2,4-dione | IC50 | 590.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(2-methoxyphenyl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 80.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(4-methoxyphenyl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 110.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[[3-(methoxymethyl)phenyl]methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 130.0 [1] |
 | (5R)-1-Benzyl-3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5-methylimidazolidine-2,4-dione | IC50 | 10.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(4-hydroxyphenyl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 70.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(6-methoxypyridin-2-yl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 80.0 [1] |
 | 1-[(2,3-Dihydroxyphenyl)methyl]-3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 100.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(3-fluorophenyl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 120.0 [1] |
 | 1-[2-(3,4-Dimethoxyphenyl)ethyl]-3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 130.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(2,5-dimethylpyrazol-3-yl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 230.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(4-fluorophenyl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 80.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(3-methoxyphenyl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 80.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[[3-(hydroxymethyl)phenyl]methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 110.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethyl-1-(pyridin-3-ylmethyl)imidazolidine-2,4-dione | IC50 | 220.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(2-hydroxyphenyl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 70.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[2-(3-fluorophenyl)ethyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 150.0 [1] |
 | 1-[(2,6-Difluorophenyl)methyl]-3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 100.0 [1] |
 | 1-[(3,4-Dihydroxyphenyl)methyl]-3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 120.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethyl-1-(2-phenoxyethyl)imidazolidine-2,4-dione | IC50 | 350.0 [1] |
 | 1-[(3,4-Dimethoxyphenyl)methyl]-3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 80.0 [1] |
 | 3-[[3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethyl-2,4-dioxoimidazolidin-1-yl]methyl]benzonitrile | IC50 | 90.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(2-fluorophenyl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 110.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethyl-1-[(3-methylphenyl)methyl]imidazolidine-2,4-dione | IC50 | 120.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(5-methoxypyridin-2-yl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 190.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[2-(2-fluorophenyl)ethyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 200.0 [1] |
 | Methyl 3-[[3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethyl-2,4-dioxoimidazolidin-1-yl]methyl]benzoate | IC50 | 220.0 [1] |
 | Methyl 4-[[3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethyl-2,4-dioxoimidazolidin-1-yl]methyl]benzoate | IC50 | 230.0 [1] |
 | 1-[(2,5-Difluorophenyl)methyl]-3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 240.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethyl-1-(pyridin-2-ylmethyl)imidazolidine-2,4-dione | IC50 | 260.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[[3-(2-hydroxyethoxy)phenyl]methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 280.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(2-fluoro-6-methoxyphenyl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 310.0 [1] |
 | 1-Benzyl-3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 320.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[2-(4-fluorophenyl)ethyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 330.0 [1] |
 | 1-[(2,5-Dimethoxyphenyl)methyl]-3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 200.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethyl-1-(2-phenylethyl)imidazolidine-2,4-dione | IC50 | 230.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[2-(2-methoxyphenyl)ethyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 240.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[2-(3-methoxyphenyl)ethyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 250.0 [1] |
 | 1-(2,3-Dihydro-1,4-benzodioxin-6-ylmethyl)-3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 270.0 [1] |
 | 1-[(2,3-Dimethoxyphenyl)methyl]-3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 300.0 [1] |
 | 1-[(2,3-Difluorophenyl)methyl]-3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 310.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(3-fluoro-4-methoxyphenyl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 330.0 [1] |
 | 1-[2-(3,5-Difluorophenyl)ethyl]-3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 400.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethyl-1-[(1-methylpyrazol-3-yl)methyl]imidazolidine-2,4-dione | IC50 | 420.0 [1] |
 | 3-[[3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethyl-2,4-dioxoimidazolidin-1-yl]methyl]benzoic acid | IC50 | 460.0 [1] |
 | Methyl 2-[3-[[3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethyl-2,4-dioxoimidazolidin-1-yl]methyl]phenoxy]acetate | IC50 | 530.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-(2-hydroxyethyl)-5,5-dimethylimidazolidine-2,4-dione | IC50 | 560.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethyl-1-[(4-methylphenyl)methyl]imidazolidine-2,4-dione | IC50 | 740.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(3,4-dimethylphenyl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 1220.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(2,6-dimethylphenyl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 1580.0 [1] |
 | 1-[[3-[2-(Dimethylamino)ethoxy]phenyl]methyl]-3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 2080.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethyl-1-[(6-oxo-1H-pyridin-2-yl)methyl]imidazolidine-2,4-dione | IC50 | 440.0 [1] |
 | 1-[(2,4-Difluorophenyl)methyl]-3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 530.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(4-methoxy-3-methylphenyl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 540.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethyl-1-(3-phenylpropyl)imidazolidine-2,4-dione | IC50 | 580.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[[3-(2-methoxyethoxy)phenyl]methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 710.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(2-fluoro-3-methylphenyl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 810.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethyl-1-[[3-(trifluoromethyl)phenyl]methyl]imidazolidine-2,4-dione | IC50 | 1540.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(2,4-dimethylphenyl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 1890.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[[4-(hydroxymethyl)phenyl]methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 360.0 [1] |
 | 4-[[3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethyl-2,4-dioxoimidazolidin-1-yl]methyl]benzoic acid | IC50 | 2310.0 [1] |
 | 2-[3-[[3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethyl-2,4-dioxoimidazolidin-1-yl]methyl]phenoxy]acetic acid | IC50 | 2850.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[[4-(methoxymethyl)phenyl]methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 280.0 [1] |
 | (10As)-2-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-7-hydroxy-10,10a-dihydro-5H-imidazo[1,5-b]isoquinoline-1,3-dione | IC50 | 30.0 [1] |
 | 2-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-8-hydroxy-10,10a-dihydro-5H-imidazo[1,5-b]isoquinoline-1,3-dione | IC50 | 30.0 [1] |
 | (10Ar)-2-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-7-hydroxy-10,10a-dihydro-5H-imidazo[1,5-b]isoquinoline-1,3-dione | IC50 | 30.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethyl-1-(pyridin-4-ylmethyl)imidazolidine-2,4-dione | IC50 | 190.0 [1] |
 | Unii-7S06P17S1V | IC50 | 50.0 [1] |
 | 1-[(3,5-Dihydroxyphenyl)methyl]-3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 10.0 [1] |
 | 7-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5-[(3-hydroxyphenyl)methyl]-5,7-diazaspiro[3.4]octane-6,8-dione | IC50 | 30.0 [1] |
 | (5S)-3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(3-hydroxyphenyl)methyl]-5-methylimidazolidine-2,4-dione | IC50 | 20.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(3-hydroxy-4-methoxyphenyl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 60.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(3-hydroxyphenyl)methyl]-1,3-diazaspiro[4.4]nonane-2,4-dione | IC50 | 70.0 [1] |
 | (5R)-3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(3-hydroxyphenyl)methyl]-5-methylimidazolidine-2,4-dione | IC50 | 20.0 [1] |
 | (5S)-3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5-(hydroxymethyl)-1-[(3-hydroxyphenyl)methyl]imidazolidine-2,4-dione | IC50 | 40.0 [1] |
 | 6-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-4-[(3-hydroxy-4-methoxyphenyl)methyl]-4,6-diazaspiro[2.4]heptane-5,7-dione | IC50 | 20.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5-(hydroxymethyl)-1-[(3-hydroxyphenyl)methyl]-5-methylimidazolidine-2,4-dione | IC50 | 130.0 [1] |
 | 4-[(3,4-Dimethoxyphenyl)methyl]-6-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-4,6-diazaspiro[2.4]heptane-5,7-dione | IC50 | 20.0 [1] |
 | 1-[(3,5-Dimethoxyphenyl)methyl]-3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 300.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(4-fluoro-3-methoxyphenyl)methyl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 180.0 [1] |
 | 1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]-3-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethylimidazolidine-2,4-dione | IC50 | 80.0 [1] |
 | 3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethyl-1-[(2-methylphenyl)methyl]imidazolidine-2,4-dione | IC50 | 100.0 [1] |
 | 4-[[3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-5,5-dimethyl-2,4-dioxoimidazolidin-1-yl]methyl]benzonitrile | IC50 | 50.0 [1] |
 | (5S)-3-[1-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]pyrazol-4-yl]-1-[(3-hydroxyphenyl)methyl]-5-propan-2-ylimidazolidine-2,4-dione | IC50 | 650.0 [1] |