![](https://images.aatbio.com/dataset/ic50/tankyrase-2_7de353ee3e6da7d439f1ec3aa8996b73.svg) | 3,5,7,8-Tetrahydro-2-[4-(trifluoromethyl)phenyl]-4H-thiopyrano[4,3-d]pyrimidin-4-one | IC50 | 5.25 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_bba0e8ca6afb314c59542be5b90d2370.svg) | Olaparib | IC50 | 5.2 [1], 1200.0 [2], 1700.0 [3], 2344.23 [4] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_f2b198c2d504e236c39c9f094ca41530.svg) | IWR-1-endo | IC50 | 38.0 [1], 39.0 [2], 56.0 [3], 134.9 [4] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_fbc186dc6ed96f500ea5b572e86e159c.svg) | 1-[3-[4-(2-Chlorophenyl)-5-pyrimidin-4-yl-1,2,4-triazol-3-yl]cyclobutyl]-2-oxo-3H-benzimidazole-5-carbonitrile | IC50 | 6.3 [1], 19.0 [2], 70.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_4f9590108cda1b4f92b634af74a38a7e.svg) | 3-[4-[4-(2-Chlorophenyl)-5-pyrimidin-4-yl-1,2,4-triazol-3-yl]cyclohexyl]-1H-benzimidazol-2-one | IC50 | 430.0 [1], 1060.0 [2], 1800.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_9f096f0e8d0df4552419673fb8b4f954.svg) | 1-[4-[4-(2-Chlorophenyl)-5-pyrimidin-4-yl-1,2,4-triazol-3-yl]cyclohexyl]-2-oxo-3H-benzimidazole-5-carbonitrile | IC50 | 120.0 [1], 330.0 [2], 1490.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_bd0528e8a6fb9307aba0b8786efa083e.svg) | 3-[3-[4-(2-Chlorophenyl)-5-pyrimidin-4-yl-1,2,4-triazol-3-yl]cyclobutyl]-1H-benzimidazol-2-one | IC50 | 9.8 [1], 200.0 [2], 410.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_9d37a00818f71911ddc7ae7fb3af75a7.svg) | N~2~,N~2~-Dimethyl-N~1~-(6-oxo-5,6-dihydrophenanthridin-2-YL)glycinamide | IC50 | 219.0 [1], 2951.21 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_4ce1e392071f9a35d153ee0e21369703.svg) | Rucaparib | IC50 | 14.0 [1], 891.25 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_0736bd1a9c6d0fc2d5d01fcfa8a8fe5a.svg) | 2-(4-Chlorophenyl)quinazolin-4-ol | IC50 | 54.0 [1], 200.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_9702119f8d8353419fd0adaa755f86bb.svg) | Nvp-tnks656 | IC50 | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_028a11317906182ba0740511a9b10018.svg) | 4,4'-Oxydibenzamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_0d917f12b4f21e18825c944259cad2ab.svg) | 2-(4-Methylphenyl)-4H-chromen-4-one | IC50 | 190.0 [1], 1100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_f0ddb6875e45fa0e6cdffc2a25da2c26.svg) | 5-[[4-(4-Methoxyphenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]sulfanylmethyl]-3-(4-methylphenyl)-1,2,4-oxadiazole | IC50 | 460.0 [1], 650.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_dd293d72769226a0e0dafb5851d2a4b7.svg) | 4-[(3Ar,4r,7s,7as)-1,3-Dioxooctahydro-2h-4,7-Methanoisoindol-2-Yl]-N-(Quinolin-8-Yl)benzamide | IC50 | 31.0 [1], 56.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_5644794b80cfe89001355cea696d6311.svg) | 2-[4-(Trifluoromethyl)phenyl]-3h-Quinazolin-4-One | IC50 | 21.5 [1], 133.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_42cb637297ccd2eab77731f4608ef765.svg) | 2-[4-(Trifluoromethyl)phenyl]-3,5,6,8-tetrahydrothiopyrano[3,4-d]pyrimidin-4-one | IC50 | 2.0 [1], 4.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_b4add25d1d6e7553e07e230307eda588.svg) | 1-[4-[4-(2-Chlorophenyl)-5-pyrimidin-4-yl-1,2,4-triazol-3-yl]phenyl]-2-oxo-3H-benzimidazole-5-carbonitrile | IC50 | 340.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_5990b92b8b207aaa055fb0a86512c4bc.svg) | 2-[4-(4-Fluorobenzoyl)piperidin-1-yl]-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]-N-(thiophen-2-ylmethyl)acetamide | IC50 | 7.5 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_841732ebe8b3ab4c3c60886e582b565f.svg) | 4-[3-(8-Methyl-4-oxo-3H-quinazolin-2-yl)propanoylamino]-N-quinolin-8-ylbenzamide | IC50 | 0.1 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_59fb4f7f48babb39c7b1fc9f7648ba3f.svg) | 2-[4-(4-Fluorobenzoyl)piperidin-1-yl]-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]-N-propylacetamide | IC50 | 11.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_9640d72ce10399f21864841df59636d7.svg) | N-[(4-Oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]-3-phenyl-N-(thiophen-2-ylmethyl)propanamide | IC50 | 216.0 [1], 222.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_f17fe138053a8c5198acb5f732046b14.svg) | 3-(4-Fluorophenyl)-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]-N-(thiophen-2-ylmethyl)propanamide | IC50 | 78.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_ffb1ae5afe444c60a2edc3d344878ebf.svg) | 3-(2-Fluorophenyl)-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]-N-(thiophen-2-ylmethyl)propanamide | IC50 | 64.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_74a5a8cedc2a6fd5521beb4cf63a56eb.svg) | 3-(3-Fluorophenyl)-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]-N-(thiophen-2-ylmethyl)propanamide | IC50 | 284.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_81d20e37d642d79ebf46fecba2591204.svg) | 3-(2-Hydroxyphenyl)-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]-N-(thiophen-2-ylmethyl)propanamide | IC50 | 766.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_e51f5257e4b0add6e02102390d50f025.svg) | 3-(3-Hydroxyphenyl)-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]-N-(thiophen-2-ylmethyl)propanamide | IC50 | 178.0 [1], 180.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_fcad33cfa2f84ff6b0591f27a51b0774.svg) | 3-(4-Hydroxyphenyl)-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]-N-(thiophen-2-ylmethyl)propanamide | IC50 | 341.0 [1], 345.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_bd03a894b9a40276de9464345a2d5160.svg) | N-[(4-Oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]-3-pyridin-4-yl-N-(thiophen-2-ylmethyl)propanamide | IC50 | 958.0 [1], 962.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_25562a38eb9729404835d85db16a6a8c.svg) | N-Ethyl-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]-3-phenylpropanamide | IC50 | 4780.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_4667a5d9a8b83caa371123bbce4c495e.svg) | N-[(4-Oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]-3-phenyl-N-(thiophen-3-ylmethyl)propanamide | IC50 | 1030.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_d6e687c802ab565b500c07fcbfa3d912.svg) | 2-[4-(4-Fluorobenzoyl)piperidin-1-yl]-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]acetamide | IC50 | 23.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_046f3de6eb4d2d97f4263a9f01986ecc.svg) | 2-[4-(4-Fluorobenzoyl)piperidin-1-yl]-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]-N-(pyridin-2-ylmethyl)acetamide | IC50 | 31.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_98b2062b6bf4308499c3cdd361da78ca.svg) | N-(Cyclopropylmethyl)-2-[4-(4-fluorobenzoyl)piperidin-1-yl]-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]acetamide | IC50 | 10.7 [1], 11.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_e4d6a30808f19ef02288b0b5233ffa46.svg) | 2-[4-(4-Fluorobenzoyl)piperidin-1-yl]-N-(2-methylpropyl)-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]acetamide | IC50 | 18.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_deb7bcaf1390912e2f5b7aaac1bf1ef1.svg) | 2-[4-(4-Fluorobenzoyl)piperidin-1-yl]-N-methyl-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]acetamide | IC50 | 57.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_1dfd9162a8d3412bf049216cb53b22fb.svg) | N-Benzyl-2-[4-(4-fluorobenzoyl)piperidin-1-yl]-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]acetamide | IC50 | 16.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_0e07bfbff2c180fabed4d01060dfe29f.svg) | N-[(4-Oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]-3-pyridin-3-yl-N-(thiophen-2-ylmethyl)propanamide | IC50 | 7960.0 [1], 10100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_72c7cc5ac6d5063ed4c906a9aa4f57bc.svg) | (4s)-3-{4-[6-Amino-5-(Pyrimidin-2-Yl)pyridin-3-Yl]phenyl}-5,5-Dimethyl-4-Phenyl-1,3-Oxazolidin-2-One | IC50 | 25.9 [1], 26.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_b27ee95b8ae62e1e37aae710aa7107a5.svg) | 4-[[1-[[2-Cyano-3-(trifluoromethyl)phenyl]methyl]-2,4-dioxoquinazolin-3-yl]methyl]cyclohexane-1-carboxylic acid | IC50 | 19.95 [1], 79.43 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_eb81af17281212e35497b075b4976117.svg) | 4-[[1-[[2-Cyano-3-(trifluoromethyl)phenyl]methyl]-6-fluoro-5-methyl-2,4-dioxoquinazolin-3-yl]methyl]cyclohexane-1-carboxylic acid | IC50 | 19.95 [1], 79.43 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_fae0683caff6602ef4aa10d3914d0529.svg) | 2-[4-(Aminomethyl)phenyl]-8-methyl-3H-quinazolin-4-one | IC50 | 43.0 [1], 100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_a2cf57bd6f8c46fcf64697efa5bb4d5b.svg) | Apigenin | IC50 | 2900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_ae75139455e150d724bbd6242680ee8e.svg) | Luteolin | IC50 | 1100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_862307a24e133d7a8e87a44ad1554b52.svg) | Flavone | IC50 | 140.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_587dbc3ae22354d383980900bdf85d4d.svg) | 2-Hydroxyquinoline | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_5bde39defdeb9b3639f2a3e58f77f3b5.svg) | Veliparib | IC50 | 23988.33 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_67f6ced2b72cac0cc2b4d65f0d199019.svg) | Niraparib | IC50 | 5128.61 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_60c3f20b0f42dbc4974f096cbfd3e3d0.svg) | 6(5H)-Phenanthridinone | IC50 | 14.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_979b4880256c881f24510e2d72655f5e.svg) | Bmn-673 8R,9S | IC50 | 107.15 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_ed5423d1fea4d2aa003b77f5700b59a3.svg) | 3',4'-Dihydroxyflavone | IC50 | 170.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_e22fbcee4d1b44d65842d118f749f8f1.svg) | 7,3',4'-Trihydroxyflavone | IC50 | 870.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_d766d480fe5526460281bc46a7f9336b.svg) | 4H-Thieno[2,3-c]isoquinolin-5-one | IC50 | 24.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_b2b5a3d0592918a9be8fe77088de2d91.svg) | 2-Phenylquinazolin-4-ol | IC50 | 2200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_fcd7153670da8d30810bab38d0db23c5.svg) | 2-(4-Methoxyphenyl)-1H-quinazolin-4-one | IC50 | 611.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_a9d5afe1eb72fca8cbb3e3ef44a1cf3c.svg) | CID 67960134 | IC50 | 25.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_fefd68655cfe1bcbb8b6fcd49ef27f88.svg) | 4-Methylquinolin-2-ol | IC50 | 12000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_8f0cb53e167ee65c11f6c35cf45d912b.svg) | Pratol | IC50 | 450.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_35aec792bbfc6c95d4c64c30a66ec983.svg) | 4-Methoxybenzamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_20a8fd36c01b010ea5d95a8099282287.svg) | 4'-Fluoroflavone | IC50 | 1100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_dea69defff582730421352373662e055.svg) | 2-(4-Nitrophenyl)quinazolin-4-ol | IC50 | 259.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_a1e76a8488fc5ccbc552c80b14d4ce30.svg) | 7,3'-Dihydroxyflavone | IC50 | 620.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_7bfac7be1a991d1d508432f91e80551f.svg) | 8-(3-Chloro-5-(4-(1-methyl-1H-pyrazol-4-yl)phenyl)pyridin-4-yl)-2,8-diazaspiro[4.5]decan-1-one | IC50 | 15000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_aff7e02f0bec3cdbd5af3b2187f127b2.svg) | 2-(4-Methoxyphenyl)-2,3-dihydroquinazolin-4(1H)-one | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_b7c1de4a3b880cd0247e145bc7a0dcfe.svg) | 2-(4-Bromophenyl)-3,4-Dihydroquinazolin-4-One | IC50 | 101.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_aa0974474c3754d928b4d05f08aff109.svg) | 3-(4-Oxo-3,4-dihydroquinazolin-2-yl)propanoic acid | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_dd2e30a1d532fd0f0282933ea64e7e88.svg) | 2-Phenyl-2,3-dihydroquinazolin-4(1h)-one | IC50 | 5495.41 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_b96387d19fb60c745fd82c5b553f23f0.svg) | 2-(4-Fluorophenyl)quinazolin-4-ol | IC50 | 1102.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_e5b2ba75b17264c8f95259d87396926e.svg) | 3'-Hydroxyflavone | IC50 | 310.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_2fbb4add00da292625e0fdc82d875028.svg) | 2-(4-Chlorophenyl)-2,3-dihydroquinazolin-4(1H)-one | IC50 | 416.87 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_65e4c9abcd55739e5a0236b7516bb1de.svg) | 5H-Pyrano[4,3-b]pyridine-3-carbonitrile, 2-hydroxy-7-isopropyl-7,8-dihydro- | IC50 | 1700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_8a8178990d3fbb389a88c088c3ee5e97.svg) | 2-(2-Chlorophenyl)-2,3-dihydro-1H-quinazolin-4-one | IC50 | 31200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_88ccee9ebb6dbe831416b672fdc0f7fd.svg) | 2-(4-Hydroxyphenyl)-3h-Quinazolin-4-One | IC50 | 189.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_bfd34a07f7bd6135041a404c06ee84be.svg) | 5-Ethyl-2-[4-(2-fluoro-phenyl)-piperazin-1-yl]-6-methyl-3H-pyrimidin-4-one | IC50 | 724.44 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_54a1b21a36e0bc6ef2d5bfe03211adb3.svg) | 2-[4-(2-Fluorophenyl)piperazin-1-yl]-6-methyl-5-propylpyrimidin-4(3H)-one | IC50 | 63095.73 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_36aad2118efb42fc02387e783b2d2457.svg) | N-[4-[[[4-(4-Methoxyphenyl)-4-oxanyl]methylamino]-oxomethyl]phenyl]-2-furancarboxamide | IC50 | 1995.26 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_da759c45c4a5813431ec3296123568ca.svg) | 4-[[3-[(6S)-3-(1,1-Difluoroethyl)-6-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl]phenyl]-difluoromethyl]-2H-phthalazin-1-one | IC50 | 3000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_b38e7300dfef6363df76af9b0a060601.svg) | 2-(4-Methoxy-phenyl)-8-methyl-3H-quinazolin-4-one | IC50 | 12.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_43aa27e94eda0f82cbe31b9263fcbe44.svg) | 8-Methyl-2-(4-nitro-phenyl)-3H-quinazolin-4-one | IC50 | 30.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_001d916e82575e7e5d056f4c536db2f6.svg) | 2-(4-Amino-phenyl)-8-methyl-3H-quinazolin-4-one | IC50 | 3.3 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_fd0ecae9850589ebb00411badca6e227.svg) | 2-(4-Hydroxy-phenyl)-8-methyl-3H-quinazolin-4-one | IC50 | 3.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_9782dae799147b0a38eb9c4587333f0b.svg) | 8-Methyl-2-phenylquinazolin-4(3H)-one | IC50 | 41.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_8e4dd4f310216d806e4334f529f789e9.svg) | 2-(3-Benzyloxyphenyl)-1,2-dihydro-4(3H)-quinazolinone | IC50 | 7244.36 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_58e01c0bb8eff75743ac57fac59fc826.svg) | 2-(4-Nitrophenyl)-4H-chromen-4-one | IC50 | 140.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_22bfa2cad69571110b65106c86895b47.svg) | 2-(4-Aminophenyl)-3,4-Dihydroquinazolin-4-One | IC50 | 690.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_41feab3c9fd34f20ec15f681338460cd.svg) | 4-Quinazolinol, 5,6,7,8-tetrahydro-2-(4-methyl-1-piperazinyl)- | IC50 | 302.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_a4fa529c8182febcafe88e97cde76e05.svg) | 2-(4-Methoxyphenyl)-8-methoxyquinazoline-4(3H)-one | IC50 | 128.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_7362302d52d88fc7bdf6b3491a4eb693.svg) | 8-Methoxy-2-(4-nitro-phenyl)-3H-quinazolin-4-one | IC50 | 863.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_5750baca8423e7c362467cf03d973560.svg) | 8-Methoxy-2-phenyl-quinazolin-4-ol | IC50 | 1029.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_7856958589f29d2161f0841f53db7345.svg) | 2-(4-Methylphenyl)quinazolin-4(3H)-one | IC50 | 540.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_8d5a3e82a8dab0474b51e286a372e735.svg) | 8-Methyl-2-[4-(Trifluoromethyl)phenyl]-3h-Quinazolin-4-One | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_fda4bed4c721d7533cd665b904b64110.svg) | 2-(4-Amino-phenyl)-8-hydroxy-3H-quinazolin-4-one | IC50 | 219.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_77dbeb52853d0bbc3a516b376532e57f.svg) | 8-Hydroxy-2-(4-nitro-phenyl)-3H-quinazolin-4-one | IC50 | 191.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_1026fa9ebfa5585657242db3acf2d0f9.svg) | 2-(4-Hydroxyphenyl)-8-hydroxyquinazoline-4(3H)-one | IC50 | 86.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_90e980d4e7b3fc3c5f4944bc4e1ac8f4.svg) | 8-Methoxy-2-[4-(Trifluoromethyl)phenyl]-3,4-Dihydroquinazolin-4-One | IC50 | 87.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_9456dcb072ef0622cc11785509ac0978.svg) | 8-Hydroxy-2-phenyl-3H-quinazolin-4-one | IC50 | 180.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_3278563b2825e1a509bf053e94a95b99.svg) | 5-({[5-(2-Furyl)-4-phenyl-4H-1,2,4-triazol-3-yl]thio}methyl)-3-phenyl-1,2,4-oxadiazole | IC50 | 19000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_3740a0a21ff3ca353bc2d4cc0ce3c9e8.svg) | 4'-Isopropylflavone | IC50 | 72.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_d0cbe3ae5e2077efb72eb6824b10f4c6.svg) | CID 41783892 | IC50 | 2760.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-2_9f55c70eef839ae3878767dd7b8cd018.svg) | 2-(4-Tert-Butylphenyl)-2,3-dihydroquinazoline-4(1H)-one | IC50 | 154.88 [1] |