![](https://images.aatbio.com/dataset/ic50/tankyrase-1_7de353ee3e6da7d439f1ec3aa8996b73.svg) | 3,5,7,8-Tetrahydro-2-[4-(trifluoromethyl)phenyl]-4H-thiopyrano[4,3-d]pyrimidin-4-one | IC50 | 11.1 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_bba0e8ca6afb314c59542be5b90d2370.svg) | Olaparib | IC50 | 1230.27 [1], 1500.0 [2], 1800.0 [3], 1900.0 [4], 3534.0 [5] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_465f984f663a4d46ba38e496f97de95c.svg) | (4S)-3-[4-(6-Amino-5-pyrimidin-2-ylpyridin-3-yl)cyclohexyl]-5,5-dimethyl-4-phenyl-1,3-oxazolidin-2-one | IC50 | 1.47 [1], 2.0 [2], 370.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_9d37a00818f71911ddc7ae7fb3af75a7.svg) | N~2~,N~2~-Dimethyl-N~1~-(6-oxo-5,6-dihydrophenanthridin-2-YL)glycinamide | IC50 | 570.0 [1], 1300.0 [2], 1698.24 [3] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_f2b198c2d504e236c39c9f094ca41530.svg) | IWR-1-endo | IC50 | 131.0 [1], 150.0 [2], 151.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_f8ac584aeb8831a7376c015c49b7ae16.svg) | 4-[(4S)-5,5-Dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]-N-quinolin-8-ylcyclohexane-1-carboxamide | IC50 | 16.0 [1], 16.8 [2], 5200.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_e3d255343eb86bef4ede7696f4cffee1.svg) | [4-(1-Methylimidazole-4-carbonyl)piperazin-1-yl]-[4-(tetrazolo[1,5-a]quinoxalin-4-ylamino)phenyl]methanone | IC50 | 2.51 [1], 31.62 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_ca230c02c816061886a0a8b9ffdd2715.svg) | (4-Pyrimidin-2-ylpiperazin-1-yl)-[4-(tetrazolo[1,5-a]quinoxalin-4-ylamino)phenyl]methanone | IC50 | 7.94 [1], 15.85 [2], 19.95 [3] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_da0178ee87eb5587a87e83d9ebd8baac.svg) | 3-(4-(Dimethylaminomethyl)phenyl)isoquinoline-1(2H)-one | IC50 | 18.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_fc92ca04458c0e96d45b62813cfa179f.svg) | 3-(4-(Dimethylaminomethyl)phenyl)-5-methylisoquinoline-1(2H)-one | IC50 | 12.0 [1], 72.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_862307a24e133d7a8e87a44ad1554b52.svg) | Flavone | IC50 | 320.0 [1], 330.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_5bde39defdeb9b3639f2a3e58f77f3b5.svg) | Veliparib | IC50 | 10000.0 [1], 10715.19 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_4ce1e392071f9a35d153ee0e21369703.svg) | Rucaparib | IC50 | 25.0 [1], 144.54 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_67f6ced2b72cac0cc2b4d65f0d199019.svg) | Niraparib | IC50 | 570.0 [1], 2344.23 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_d766d480fe5526460281bc46a7f9336b.svg) | 4H-Thieno[2,3-c]isoquinolin-5-one | IC50 | 200.0 [1], 100000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_b2b5a3d0592918a9be8fe77088de2d91.svg) | 2-Phenylquinazolin-4-ol | IC50 | 59.0 [1], 1406.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_20a8fd36c01b010ea5d95a8099282287.svg) | 4'-Fluoroflavone | IC50 | 280.0 [1], 700.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_0736bd1a9c6d0fc2d5d01fcfa8a8fe5a.svg) | 2-(4-Chlorophenyl)quinazolin-4-ol | IC50 | 140.0 [1], 485.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_251879f72243b062e422fd4644dceb33.svg) | N-Phenyltetrazolo[1,5-a]quinoxalin-4-amine | IC50 | 251.19 [1], 1995.26 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_028a11317906182ba0740511a9b10018.svg) | 4,4'-Oxydibenzamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_0d917f12b4f21e18825c944259cad2ab.svg) | 2-(4-Methylphenyl)-4H-chromen-4-one | IC50 | 47.0 [1], 52.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_66d28150a01ef0379ed488fd6fe1c582.svg) | N-(3-Methylphenyl)-4-tetrazolo[1,5-a]quinoxalinamine | IC50 | 10000.0 [1], 15848.93 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_5fa8e76aa24b2b81f34c6348d2952249.svg) | N-(4-Chlorophenyl)tetrazolo[1,5-a]quinoxalin-4-amine | IC50 | 398.11 [1], 1258.93 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_566629e35339f632bfa3667c313ae140.svg) | N-(4-Methylphenyl)-4-tetrazolo[1,5-a]quinoxalinamine | IC50 | 125.89 [1], 1258.93 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_472c3cf9d774b2094ec1f932ca6c063b.svg) | Morpholin-4-Yl[4-(Tetrazolo[1,5-A]quinoxalin-4-Ylamino)phenyl]methanone | IC50 | 50.12 [1], 158.49 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_8736d006c0d7f06954fe2bbdc4f53745.svg) | 4-[(1R,2S,6R,7S)-3,5-Dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]-N-(4-methylquinolin-8-yl)benzamide | IC50 | 160.0 [1], 192.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_bde678acc27e2df12f907857c17377a9.svg) | 5H-Benzothiopheno[2,3-c]quinolin-6-one | IC50 | 90.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_1429faacc2c24ca8da9bfe6f7406325a.svg) | N-(2-Methoxyphenyl)-4-{[3-(4-Oxo-3,4-Dihydroquinazolin-2-Yl)propanoyl]amino}benzamide | IC50 | 8.0 [1], 10.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_5644794b80cfe89001355cea696d6311.svg) | 2-[4-(Trifluoromethyl)phenyl]-3h-Quinazolin-4-One | IC50 | 50.0 [1], 425.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_42cb637297ccd2eab77731f4608ef765.svg) | 2-[4-(Trifluoromethyl)phenyl]-3,5,6,8-tetrahydrothiopyrano[3,4-d]pyrimidin-4-one | IC50 | 11.0 [1], 5000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_08ec09e888945152ff9e57296979530d.svg) | 4-N,4-N-Dimethyl-1-N-(tetrazolo[1,5-a]quinoxalin-4-yl)benzene-1,4-diamine | IC50 | 63.1 [1], 1258.93 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_43b819bf557a989bdd7ed1f5240914b3.svg) | N-(2-Methoxyphenyl)-4-[3-(4-oxo-3H-quinazolin-2-yl)propanoylamino]cyclohexane-1-carboxamide | IC50 | 31.0 [1], 7460.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_63c311979c541c9492a33c3e0b88d02c.svg) | [4-(Oxan-4-yl)piperazin-1-yl]-[4-(tetrazolo[1,5-a]quinoxalin-4-ylamino)phenyl]methanone | IC50 | 31.62 [1], 251.19 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_1563704fb488ffb7b73b82a95920d7ab.svg) | Morpholin-4-yl-[3-(tetrazolo[1,5-a]quinoxalin-4-ylamino)phenyl]methanone | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_17b74b29df437c2229876ee0fe28ce8b.svg) | N-(3-Propan-2-ylphenyl)tetrazolo[1,5-a]quinoxalin-4-amine | IC50 | 10000.0 [1], 199526.23 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_7d12a5a52ffcb7f8f0c60ccb5e67fe5c.svg) | [3-Fluoro-4-(tetrazolo[1,5-a]quinoxalin-4-ylamino)phenyl]-morpholin-4-ylmethanone | IC50 | 7943.28 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_a232277d06b5fd2ce56de5d083f76a21.svg) | N-(2-Methylphenyl)tetrazolo[1,5-a]quinoxalin-4-amine | IC50 | 10000.0 [1], 63095.73 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_cb41bb76f2957c3de9b8220a5befa801.svg) | (4-Pyrimidin-4-ylpiperazin-1-yl)-[4-(tetrazolo[1,5-a]quinoxalin-4-ylamino)phenyl]methanone | IC50 | 2.0 [1], 6.31 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_8340d97b066188e10434a26defce91f8.svg) | N-(4-Propan-2-ylphenyl)tetrazolo[1,5-a]quinoxalin-4-amine | IC50 | 125.89 [1], 199.53 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_6dd67df46403ca92911e559bba057d24.svg) | (4-Pyridin-2-ylpiperazin-1-yl)-[4-(tetrazolo[1,5-a]quinoxalin-4-ylamino)phenyl]methanone | IC50 | 31.62 [1], 100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_3bb58b78666709abaa6f98a7c7ffa1e9.svg) | N-(4-Fluorophenyl)tetrazolo[1,5-a]quinoxalin-4-amine | IC50 | 630.96 [1], 3981.07 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_2ba5f314ffdf95299e65431a1041bfb6.svg) | N-[4-(Tetrazolo[1,5-a]quinoxalin-4-ylamino)phenyl]acetamide | IC50 | 19.95 [1], 251.19 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_64a36171129b71301828f12d468cff2f.svg) | 4-[(4s)-5,5-Dimethyl-2-Oxo-4-Phenyl-1,3-Oxazolidin-3-Yl]-N-(Quinolin-8-Yl)benzamide | IC50 | 198.0 [1], 200.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_c3334db838615edd5224dcc9654f75b7.svg) | 4-[(4S)-5,5-Dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]-N-(1,5-naphthyridin-4-yl)benzamide | IC50 | 18.0 [1], 18.3 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_edbceffaaf4f63b81e3f63b78f71848a.svg) | N-[4-[(4S)-5,5-Dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]cyclohexyl]quinoline-8-carboxamide | IC50 | 10.0 [1], 22.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_dace1aaf30dea92033527981f05f4a3c.svg) | N-[4-[(4S)-5,5-Dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]cyclohexyl]-1,5-naphthyridine-4-carboxamide | IC50 | 4.0 [1], 4.56 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_8db9571a4ef89d9dc27ebe53c025a1ee.svg) | N-[4-[(4S)-5,5-Dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]cyclohexyl]-7-fluoro-1,5-naphthyridine-4-carboxamide | IC50 | 3.86 [1], 4.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_f3d64f974e8eaa4b642b305d21c36a9a.svg) | (4S)-5,5-Dimethyl-3-[4-(2-oxo-3H-imidazo[4,5-c]pyridin-1-yl)cyclohexyl]-4-phenyl-1,3-oxazolidin-2-one | IC50 | 3.0 [1], 3.04 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_fde2fbcaa8725caf9957d855e94a3862.svg) | (4S)-5,5-Dimethyl-3-[4-(2-oxo-3H-imidazo[4,5-b]pyridin-1-yl)cyclohexyl]-4-phenyl-1,3-oxazolidin-2-one | IC50 | 10.7 [1], 11.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_95bcda1f0470c82fa4f3d799e2e36689.svg) | 1-[4-[(4S)-5,5-Dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]cyclohexyl]-2-oxo-3H-benzimidazole-5-carbonitrile | IC50 | 1.0 [1], 1.12 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_82fdbea39d7da663faff98415c23fa8f.svg) | 1-[4-[(4S)-5,5-Dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]cyclohexyl]-2-oxo-3H-benzimidazole-4-carbonitrile | IC50 | 3.56 [1], 4.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_ffb006c7e2bf7638f2944032b6c722fb.svg) | 1-[4-[(4S)-5,5-Dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]cyclohexyl]-6-fluoro-2-oxo-3H-benzimidazole-5-carbonitrile | IC50 | 3.0 [1], 3.48 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_33f88d4dccba9c52445ae6d27ddc06b3.svg) | 1-[4-[(4S)-5,5-Dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]cyclohexyl]-4-fluoro-2-oxo-3H-benzimidazole-5-carbonitrile | IC50 | 1.0 [1], 1.09 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_eec74de64a5cb4e4d80f3875765f6fe3.svg) | 3-[4-[(4S)-5,5-Dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]cyclohexyl]-2-oxo-1H-imidazo[4,5-b]pyridine-6-carbonitrile | IC50 | 143.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_a653a6c1dd8d94f537ca50e4419d58f7.svg) | (4S)-5,5-Dimethyl-3-[4-(2-oxo-1H-imidazo[4,5-b]pyridin-3-yl)cyclohexyl]-4-phenyl-1,3-oxazolidin-2-one | IC50 | 4.0 [1], 11.8 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_88e9d6f8c834fdbf4fdeb3f0c449e483.svg) | (4S)-5,5-Dimethyl-3-[4-(2-oxo-1H-imidazo[4,5-c]pyridin-3-yl)cyclohexyl]-4-phenyl-1,3-oxazolidin-2-one | IC50 | 4.0 [1], 4.07 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_de3ca4e3eb74c24111a9ead2b5ebe77e.svg) | (4S)-5,5-Dimethyl-3-[4-(8-oxo-7H-purin-9-yl)cyclohexyl]-4-phenyl-1,3-oxazolidin-2-one | IC50 | 5.0 [1], 5.11 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_72c7cc5ac6d5063ed4c906a9aa4f57bc.svg) | (4s)-3-{4-[6-Amino-5-(Pyrimidin-2-Yl)pyridin-3-Yl]phenyl}-5,5-Dimethyl-4-Phenyl-1,3-Oxazolidin-2-One | IC50 | 49.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_b27ee95b8ae62e1e37aae710aa7107a5.svg) | 4-[[1-[[2-Cyano-3-(trifluoromethyl)phenyl]methyl]-2,4-dioxoquinazolin-3-yl]methyl]cyclohexane-1-carboxylic acid | IC50 | 7.94 [1], 31.62 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_eb81af17281212e35497b075b4976117.svg) | 4-[[1-[[2-Cyano-3-(trifluoromethyl)phenyl]methyl]-6-fluoro-5-methyl-2,4-dioxoquinazolin-3-yl]methyl]cyclohexane-1-carboxylic acid | IC50 | 6.31 [1], 50.12 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_6f53d2fb4772516b8348dddcbd436861.svg) | 2-Amino-5-[4-[(4S)-5,5-dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]cyclohexyl]pyridine-3-carbonitrile | IC50 | 6.98 [1], 9.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_ec6bae798a152ab8fd165681eefce1a1.svg) | Cyclopropyl-[4-[4-(tetrazolo[1,5-a]quinoxalin-4-ylamino)benzoyl]piperazin-1-yl]methanone | IC50 | 19.95 [1], 5011.87 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_2d0ff5966e9b29d87a0d805b76e9700c.svg) | [4-(1H-Pyrazole-5-carbonyl)piperazin-1-yl]-[4-(tetrazolo[1,5-a]quinoxalin-4-ylamino)phenyl]methanone | IC50 | 10.0 [1], 125.89 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_b6f81f19b2e9176a08ea223379a73724.svg) | [4-(3-Methylimidazole-4-carbonyl)piperazin-1-yl]-[4-(tetrazolo[1,5-a]quinoxalin-4-ylamino)phenyl]methanone | IC50 | 25.12 [1], 398.11 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_48d159677654cd605fe9cd0a437363ed.svg) | [4-(1H-Imidazole-5-carbonyl)piperazin-1-yl]-[4-(tetrazolo[1,5-a]quinoxalin-4-ylamino)phenyl]methanone | IC50 | 3.98 [1], 251.19 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_0ed8884e04b241bf500d4726c6c9f548.svg) | 1-[4-[4-(Tetrazolo[1,5-a]quinoxalin-4-ylamino)benzoyl]piperazin-1-yl]ethanone | IC50 | 15.85 [1], 125.89 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_bbc60ce120ce85388dc37ae6aac2cd0e.svg) | (4-Pyridin-3-ylpiperazin-1-yl)-[4-(tetrazolo[1,5-a]quinoxalin-4-ylamino)phenyl]methanone | IC50 | 25.12 [1], 63.1 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_00cd697ea879d801abe1a1a0dc0d0b94.svg) | Tnks-IN-41 | IC50 | 7.94 [1], 100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_36879f959a07907538ace106d1cb8acc.svg) | [4-(Pyrimidine-2-carbonyl)piperazin-1-yl]-[4-(tetrazolo[1,5-a]quinoxalin-4-ylamino)phenyl]methanone | IC50 | 15.85 [1], 398.11 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_4fc881f484bf9838d22c2835f4820409.svg) | N-(2-Methoxyethyl)-4-(tetrazolo[1,5-a]quinoxalin-4-ylamino)benzamide | IC50 | 199.53 [1], 630.96 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_294dd74efd8a1d459ada5a0fc7ca0de1.svg) | (4-Pyridin-4-ylpiperazin-1-yl)-[4-(tetrazolo[1,5-a]quinoxalin-4-ylamino)phenyl]methanone | IC50 | 6.31 [1], 125.89 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_324da6fffc64a704311160613d7e09b8.svg) | 4-(Tetrazolo[1,5-a]quinoxalin-4-ylamino)benzoic acid | IC50 | 398.11 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_79f84ab499a67ed8244bdd519d8a130c.svg) | Piperazin-1-yl-[4-(tetrazolo[1,5-a]quinoxalin-4-ylamino)phenyl]methanone | IC50 | 50.12 [1], 794.33 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_e235f9d982029bccdcf3a2c611dc8c34.svg) | N-(2-Methoxyethyl)-N-methyl-4-(tetrazolo[1,5-a]quinoxalin-4-ylamino)benzamide | IC50 | 19.95 [1], 79.43 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_d46161df8f74ee167c1da985bbdddd4a.svg) | 1-[4-(Tetrazolo[1,5-a]quinoxalin-4-ylamino)phenyl]pyrrolidin-2-one | IC50 | 7.94 [1], 100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_abfb521bf80ccd1d7b5328def376b913.svg) | 4-[4-(Tetrazolo[1,5-a]quinoxalin-4-ylamino)phenyl]morpholin-3-one | IC50 | 7.94 [1], 100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_017c542465229113f7cce53d526854d9.svg) | N-Methyl-N-[4-(tetrazolo[1,5-a]quinoxalin-4-ylamino)phenyl]acetamide | IC50 | 10.0 [1], 79.43 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_21f9d027f23d7a7bcb186a2faaccc285.svg) | Piperidin-1-yl-[4-(tetrazolo[1,5-a]quinoxalin-4-ylamino)phenyl]methanone | IC50 | 63.1 [1], 501.19 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_79d50247cf3a822ce48528cc66cadd25.svg) | Oxan-4-yl-[4-[4-(tetrazolo[1,5-a]quinoxalin-4-ylamino)benzoyl]piperazin-1-yl]methanone | IC50 | 25.12 [1], 199.53 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_85be8858585233ccc0f5cb4a26752fe0.svg) | 3-(4-(3-(Dimethylamino)azetidine-1-ylmethyl)phenyl)-5-methylisoquinoline-1(2H)-one | IC50 | 21.0 [1], 35.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_a6b98e4d1e4ef8e95adc92b8acfafd02.svg) | 3-(4-(Trifluoromethyl)phenyl)-5-chloroisoquinoline-1(2H)-one | IC50 | 128.0 [1], 483.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_222a2d112356f1644cd5dc69f72aa814.svg) | 3-(4-Fluorophenyl)-5-methoxyisoquinoline-1(2H)-one | IC50 | 104.0 [1], 120.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_99a530bed3b6fe90b5ca346f10e7b10d.svg) | 3-(4-(Dimethylaminomethyl)phenyl)-5-chloroisoquinoline-1(2H)-one | IC50 | 151.0 [1], 364.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_abe66d813aaed915ffa48b5dcef71677.svg) | 3-(4-(Dimethylaminomethyl)phenyl)-5-fluoroisoquinoline-1(2H)-one | IC50 | 16.0 [1], 1730.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_dca9ee09367c7bfd219da6026bd4b1d5.svg) | 3-(4-(Morpholinomethyl)phenyl)-5-methylisoquinoline-1(2H)-one | IC50 | 12.0 [1], 25.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_554dd22d3cb3df606116c11961600f62.svg) | 3-(4-(4-Methylpiperazinomethyl)phenyl)-5-methylisoquinoline-1(2H)-one | IC50 | 17.0 [1], 43.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_064da9d3000666a146ba4cc38eed0b20.svg) | 3-(4-{[4-(Dimethylamino)piperidin-1-Yl]methyl}phenyl)-5-Methylisoquinolin-1(2h)-One | IC50 | 13.0 [1], 61.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_0216bc00307d0cf3260bdc9a49385135.svg) | 5-Methyl-3-[4-(Piperazin-1-Ylmethyl)phenyl]isoquinolin-1(2h)-One | IC50 | 17.0 [1], 117.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_4177c8607b44adf067b56d4b143170a0.svg) | 3-(4-Methylphenyl)-5-methoxyisoquinoline-1(2H)-one | IC50 | 34.0 [1], 59.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_5f07d15e94908c30abd29038ca22ae35.svg) | (4S)-5,5-Dimethyl-3-[4-(6-oxo-5-pyrimidin-2-yl-1H-pyridin-3-yl)cyclohexyl]-4-phenyl-1,3-oxazolidin-2-one | IC50 | 267.0 [1], 511.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_238d59984811add487cfd7662ab557e0.svg) | (4S)-3-[4-[6-Amino-5-(1,4,5,6-tetrahydropyrimidin-2-yl)pyridin-3-yl]cyclohexyl]-5,5-dimethyl-4-phenyl-1,3-oxazolidin-2-one | IC50 | 1650.0 [1], 9840.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_e8cf37eca9c2feef810007a6df8f4c05.svg) | (4S)-5,5-Dimethyl-4-phenyl-3-[4-(1H-pyrrolo[3,2-b]pyridin-6-yl)cyclohexyl]-1,3-oxazolidin-2-one | IC50 | 19.0 [1], 1250.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_017b51e6bfb53c6134262c8763ae4c45.svg) | 3-{4-[(Dimethylamino)methyl]phenyl}-5-Methoxyisoquinolin-1(2h)-One | IC50 | 19.0 [1], 136.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_a2cf57bd6f8c46fcf64697efa5bb4d5b.svg) | Apigenin | IC50 | 3100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_ae75139455e150d724bbd6242680ee8e.svg) | Luteolin | IC50 | 2400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_60c3f20b0f42dbc4974f096cbfd3e3d0.svg) | 6(5H)-Phenanthridinone | IC50 | 110.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_979b4880256c881f24510e2d72655f5e.svg) | Bmn-673 8R,9S | IC50 | 323.59 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_ed5423d1fea4d2aa003b77f5700b59a3.svg) | 3',4'-Dihydroxyflavone | IC50 | 230.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_d09edca9883e8148a7e2e779f76697ab.svg) | 4'-Methoxyflavone | IC50 | 71.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1_e22fbcee4d1b44d65842d118f749f8f1.svg) | 7,3',4'-Trihydroxyflavone | IC50 | 630.0 [1] |