![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_7de353ee3e6da7d439f1ec3aa8996b73.svg) | 3,5,7,8-Tetrahydro-2-[4-(trifluoromethyl)phenyl]-4H-thiopyrano[4,3-d]pyrimidin-4-one | IC50 | 11.0 [1], 707.0 [2], 272000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_465f984f663a4d46ba38e496f97de95c.svg) | (4S)-3-[4-(6-Amino-5-pyrimidin-2-ylpyridin-3-yl)cyclohexyl]-5,5-dimethyl-4-phenyl-1,3-oxazolidin-2-one | IC50 | 12.0 [1], 91.0 [2], 6550.0 [3] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_f2b198c2d504e236c39c9f094ca41530.svg) | IWR-1-endo | IC50 | 250.0 [1], 136000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_72c7cc5ac6d5063ed4c906a9aa4f57bc.svg) | (4s)-3-{4-[6-Amino-5-(Pyrimidin-2-Yl)pyridin-3-Yl]phenyl}-5,5-Dimethyl-4-Phenyl-1,3-Oxazolidin-2-One | IC50 | 96.0 [1], 233.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_6f53d2fb4772516b8348dddcbd436861.svg) | 2-Amino-5-[4-[(4S)-5,5-dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]cyclohexyl]pyridine-3-carbonitrile | IC50 | 43.0 [1], 392.0 [2] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_825d74a1a3b92831caf077e800d861cb.svg) | Cinnamic acid | IC50 | 685.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_bba0e8ca6afb314c59542be5b90d2370.svg) | Olaparib | IC50 | 3000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_a9d5afe1eb72fca8cbb3e3ef44a1cf3c.svg) | CID 67960134 | IC50 | 50.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_f0ddb6875e45fa0e6cdffc2a25da2c26.svg) | 5-[[4-(4-Methoxyphenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]sulfanylmethyl]-3-(4-methylphenyl)-1,2,4-oxadiazole | IC50 | 1010.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_36aad2118efb42fc02387e783b2d2457.svg) | N-[4-[[[4-(4-Methoxyphenyl)-4-oxanyl]methylamino]-oxomethyl]phenyl]-2-furancarboxamide | IC50 | 1230.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_da759c45c4a5813431ec3296123568ca.svg) | 4-[[3-[(6S)-3-(1,1-Difluoroethyl)-6-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl]phenyl]-difluoromethyl]-2H-phthalazin-1-one | IC50 | 3000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_8736d006c0d7f06954fe2bbdc4f53745.svg) | 4-[(1R,2S,6R,7S)-3,5-Dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]-N-(4-methylquinolin-8-yl)benzamide | IC50 | 163000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_1429faacc2c24ca8da9bfe6f7406325a.svg) | N-(2-Methoxyphenyl)-4-{[3-(4-Oxo-3,4-Dihydroquinazolin-2-Yl)propanoyl]amino}benzamide | IC50 | 36000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_42cb637297ccd2eab77731f4608ef765.svg) | 2-[4-(Trifluoromethyl)phenyl]-3,5,6,8-tetrahydrothiopyrano[3,4-d]pyrimidin-4-one | IC50 | 11.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_c18e776e19bcb8483ae899b1f9dd2f26.svg) | 2-[4-[3-[(4-Oxo-3H-phthalazin-1-yl)methyl]benzoyl]piperazin-1-yl]pyridine-3-carbonitrile | IC50 | 222.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_cc06a47ef1cd90f88c44822007ee39ab.svg) | N-{4-[(2-Chlorophenyl)(Pyrimidin-4-Yl)carbamoyl]phenyl}-4-Methoxybenzamide | IC50 | 1910.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_580c5e3910f3ecc604f8441e360d3d6d.svg) | 2-Chloro-4-[(4-methoxybenzoyl)amino]-N-[[4-(4-methoxyphenyl)oxan-4-yl]methyl]benzamide | IC50 | 790.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_b396bc4c4b9a29e8d5561fdc4f3ced55.svg) | 2-(4-Tert-butylphenyl)-3H-[1]benzothiolo[3,2-d]pyrimidin-4-one | IC50 | 832.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_02906230b65507ef6e47b05a3bafdf17.svg) | 4-[5-[[4-(2-Chlorophenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3,4-oxadiazol-2-yl]benzonitrile | IC50 | 140.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_5a8f9a0269f68dd7837c78be8affbf8a.svg) | 2-[2-[4-(2-Chlorophenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]ethyl]-5-(4-methylphenyl)-1,3,4-oxadiazole | IC50 | 420.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_34fd9db7745db0271cd6a8632220654a.svg) | 5-[[4-(4-Methoxyphenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]oxymethyl]-3-(4-methylphenyl)-1,2,4-oxadiazole | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_af8b5b30f667fc5317b62b48c5a73ab9.svg) | 4-[5-[(E)-2-[4-(2-Chlorophenyl)-5-(4-fluorophenyl)-1,2,4-triazol-3-yl]ethenyl]-1,3,4-oxadiazol-2-yl]-1H-pyridin-2-one | IC50 | 6300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_7db1bfeb8c2092db3bfd2e993ea64edd.svg) | 2-[(E)-2-[4-(2-Chlorophenyl)-5-(5-methylsulfonylpyridin-2-yl)-1,2,4-triazol-3-yl]ethenyl]-5-(2-methoxypyridin-4-yl)-1,3,4-oxadiazole | IC50 | 70.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_f716737a37b56a10ae1ed27956688f4f.svg) | 5-(2-Aminoquinazolin-6-Yl)-N-(4,4-Dimethyl-2-Oxo-1,2,3,4-Tetrahydroquinolin-7-Yl)-2-Fluorobenzamide | IC50 | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_c2db1dc87c3fe8452f4872dcd3437fd0.svg) | 4-(4-Methoxyphenyl)-N-[[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-5-pyridin-4-yl-1,2,4-triazol-3-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_16f0e3ebbb8079e08cccd4eff620a7ef.svg) | 3-(4-Methylphenyl)-5-[[1-(2-methylphenyl)-5-pyridin-4-ylimidazol-2-yl]sulfanylmethyl]-1,2,4-oxadiazole | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_90d9e36c87d4154ffe280aa8c6842884.svg) | 3-[3-[3-[5-[[4-(2-Chlorophenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,2,4-oxadiazol-3-yl]phenoxy]propoxy]propan-1-amine | IC50 | 3920.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_45e771b6b7d60dfb7adaade32b949429.svg) | 2-[[4-(2-Chlorophenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]sulfanylmethyl]-7,8-dimethylpyrido[1,2-a]pyrimidin-4-one | IC50 | 4530.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_be74b7ee227d499d318a3b6aa867c587.svg) | 2-(4-Chlorophenyl)-5-[[4-(2-chlorophenyl)-5-(5-methylsulfonylpyridin-2-yl)-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3,4-oxadiazole | IC50 | 50.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_64a36171129b71301828f12d468cff2f.svg) | 4-[(4s)-5,5-Dimethyl-2-Oxo-4-Phenyl-1,3-Oxazolidin-3-Yl]-N-(Quinolin-8-Yl)benzamide | IC50 | 2100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_e013ed40f7442ae631d9e5f09bf509e9.svg) | N-(4-(((4-(4-Methoxyphenyl)oxan-4-Yl)methyl)carbamoyl)phenyl)-5-Methylfuran-2-Carboxamide | IC50 | 380.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_8a657c793a6c6dbbececeec220524a4a.svg) | 4-(2,2-Dimethyl-5-oxopyrrolidin-1-yl)-N-quinolin-8-ylbenzamide | IC50 | 7300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_6cfc9389a46ace5eb9467d641b9daa4e.svg) | 4-[2-(4-Fluorophenyl)-5-oxopyrrolidin-1-yl]-N-quinolin-8-ylbenzamide | IC50 | 1100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_2233bcd1f6532a8c3916f51ebfa1dd2a.svg) | 4-[(4S)-2-Oxo-4-phenyl-1,3-oxazolidin-3-yl]-N-quinolin-8-ylbenzamide | IC50 | 4000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_c3334db838615edd5224dcc9654f75b7.svg) | 4-[(4S)-5,5-Dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]-N-(1,5-naphthyridin-4-yl)benzamide | IC50 | 189.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_f8ac584aeb8831a7376c015c49b7ae16.svg) | 4-[(4S)-5,5-Dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]-N-quinolin-8-ylcyclohexane-1-carboxamide | IC50 | 390.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_edbceffaaf4f63b81e3f63b78f71848a.svg) | N-[4-[(4S)-5,5-Dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]cyclohexyl]quinoline-8-carboxamide | IC50 | 200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_dace1aaf30dea92033527981f05f4a3c.svg) | N-[4-[(4S)-5,5-Dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]cyclohexyl]-1,5-naphthyridine-4-carboxamide | IC50 | 73.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_8db9571a4ef89d9dc27ebe53c025a1ee.svg) | N-[4-[(4S)-5,5-Dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]cyclohexyl]-7-fluoro-1,5-naphthyridine-4-carboxamide | IC50 | 270.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_f3d64f974e8eaa4b642b305d21c36a9a.svg) | (4S)-5,5-Dimethyl-3-[4-(2-oxo-3H-imidazo[4,5-c]pyridin-1-yl)cyclohexyl]-4-phenyl-1,3-oxazolidin-2-one | IC50 | 140.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_fde2fbcaa8725caf9957d855e94a3862.svg) | (4S)-5,5-Dimethyl-3-[4-(2-oxo-3H-imidazo[4,5-b]pyridin-1-yl)cyclohexyl]-4-phenyl-1,3-oxazolidin-2-one | IC50 | 1100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_95bcda1f0470c82fa4f3d799e2e36689.svg) | 1-[4-[(4S)-5,5-Dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]cyclohexyl]-2-oxo-3H-benzimidazole-5-carbonitrile | IC50 | 54.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_82fdbea39d7da663faff98415c23fa8f.svg) | 1-[4-[(4S)-5,5-Dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]cyclohexyl]-2-oxo-3H-benzimidazole-4-carbonitrile | IC50 | 270.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_ffb006c7e2bf7638f2944032b6c722fb.svg) | 1-[4-[(4S)-5,5-Dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]cyclohexyl]-6-fluoro-2-oxo-3H-benzimidazole-5-carbonitrile | IC50 | 67.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_33f88d4dccba9c52445ae6d27ddc06b3.svg) | 1-[4-[(4S)-5,5-Dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]cyclohexyl]-4-fluoro-2-oxo-3H-benzimidazole-5-carbonitrile | IC50 | 150.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_eec74de64a5cb4e4d80f3875765f6fe3.svg) | 3-[4-[(4S)-5,5-Dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]cyclohexyl]-2-oxo-1H-imidazo[4,5-b]pyridine-6-carbonitrile | IC50 | 170.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_a653a6c1dd8d94f537ca50e4419d58f7.svg) | (4S)-5,5-Dimethyl-3-[4-(2-oxo-1H-imidazo[4,5-b]pyridin-3-yl)cyclohexyl]-4-phenyl-1,3-oxazolidin-2-one | IC50 | 520.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_88e9d6f8c834fdbf4fdeb3f0c449e483.svg) | (4S)-5,5-Dimethyl-3-[4-(2-oxo-1H-imidazo[4,5-c]pyridin-3-yl)cyclohexyl]-4-phenyl-1,3-oxazolidin-2-one | IC50 | 1710.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_de3ca4e3eb74c24111a9ead2b5ebe77e.svg) | (4S)-5,5-Dimethyl-3-[4-(8-oxo-7H-purin-9-yl)cyclohexyl]-4-phenyl-1,3-oxazolidin-2-one | IC50 | 290.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_dbc6428aeaa6a1ab3935c16d0a8095af.svg) | 4-[(5R)-2-Oxo-5-phenylpyrrolidin-1-yl]-N-quinolin-8-ylbenzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_addf6acc0b6b6de0df1b5237774f0605.svg) | 2-(4-Chlorophenyl)-5-[[4-(2-chlorophenyl)-5-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3,4-oxadiazole | IC50 | 4500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_6dc4e95105142949e67c23ebee87d33e.svg) | 4-[(1S,2R,6S,7R)-4-Azatricyclo[5.2.1.02,6]dec-8-en-4-yl]-N-quinolin-8-ylbenzamide | IC50 | 131.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_4e7c0feae5d022b6821abafe5f8403dc.svg) | 2-[N-(Benzenesulfonyl)-5-chloro-2-methoxyanilino]-N-[4-(2-oxo-3H-benzimidazol-1-yl)cyclohexyl]acetamide | IC50 | 150.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_329e6f978feb6d6e3d8d0bd501cd3c9d.svg) | N-[3-Chloranyl-4-[[4-(4-Methoxyphenyl)oxan-4-Yl]methylcarbamoyl]phenyl]furan-2-Carboxamide | IC50 | 360.0 [1] |
![](https://images.aatbio.com/dataset/ic50/tankyrase-1-2_495cae331f81feb60ce76443fbdecf13.svg) | N-[3-Chloro-4-[[4-(4-methoxyphenyl)oxan-4-yl]methylcarbamoyl]phenyl]-2-methyl-1,3-oxazole-5-carboxamide | IC50 | 690.0 [1] |