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Synaptic vesicular amine transporter Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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Standard Type
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Standard Values (in nM)
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▼
SerotoninIC501430.0 [1]
SerotoninKi2290.0 [1], 7690.0 [2], 640000.0 [3]
ReserpineIC5013.2 [1]
ReserpineKi5.26 [1], 410.0 [2], 630.0 [3]
DL-MethamphetamineIC503620.0 [1]
DL-MethamphetamineKi6400.0 [1], 24500.0 [2], 346000.0 [3]
KetanserinIC50180.0 [1]
KetanserinKi77.0 [1], 353.0 [2], 1190.0 [3]
LobelineIC504200.0 [1]
LobelineKi1840.0 [1], 1950.0 [2], 10000.0 [3]
DihydrotetrabenazineIC5028.1 [1]
DihydrotetrabenazineKi70.0 [1], 152.0 [2], 10000.0 [3]
2H-Benzo(a)quinolizin-2-ol, 2-ethyl-1,3,4,6,7,11b-hexahydro-9,10-dimethoxy-3-(2-methylpropyl)-IC50154.0 [1]
2H-Benzo(a)quinolizin-2-ol, 2-ethyl-1,3,4,6,7,11b-hexahydro-9,10-dimethoxy-3-(2-methylpropyl)-Ki64.0 [1], 83.0 [2], 1932.0 [3]
Ethyl (3S,4R)-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]-4-(4-fluorophenyl)piperidine-3-carboxylateIC5085.5 [1]
Ethyl (3S,4R)-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]-4-(4-fluorophenyl)piperidine-3-carboxylateKi176.0 [1], 750.0 [2], 1150.0 [3]
Ethyl (3S,4S)-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]-4-thiophen-2-ylpiperidine-3-carboxylateIC50101.0 [1]
Ethyl (3S,4S)-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]-4-thiophen-2-ylpiperidine-3-carboxylateKi450.0 [1], 900.0 [2], 6160.0 [3]
Ethyl (3S,4S)-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]-4-(4-fluorophenyl)piperidine-3-carboxylateIC5039.4 [1]
Ethyl (3S,4S)-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]-4-(4-fluorophenyl)piperidine-3-carboxylateKi74.0 [1], 161.0 [2], 7400.0 [3]
Ethyl (3S,4S)-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]-4-phenylpiperidine-3-carboxylateIC5019.7 [1]
Ethyl (3S,4S)-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]-4-phenylpiperidine-3-carboxylateKi70.0 [1], 287.0 [2], 7700.0 [3]
Ethyl (3S,4S)-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]-4-(4-methylphenyl)piperidine-3-carboxylateIC502700.0 [1]
Ethyl (3S,4S)-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]-4-(4-methylphenyl)piperidine-3-carboxylateKi452.0 [1], 9100.0 [2], 10000.0 [3]
Ethyl (3S,4S)-4-(2,3-dihydro-1,4-benzodioxin-5-yl)-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]piperidine-3-carboxylateIC50142.0 [1]
Ethyl (3S,4S)-4-(2,3-dihydro-1,4-benzodioxin-5-yl)-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]piperidine-3-carboxylateKi652.0 [1], 700.0 [2], 7900.0 [3]
Ethyl (3S,4S)-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]-4-[4-(trifluoromethyl)phenyl]piperidine-3-carboxylateIC502900.0 [1]
Ethyl (3S,4S)-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]-4-[4-(trifluoromethyl)phenyl]piperidine-3-carboxylateKi720.0 [1], 10000.0 [2]
Ethyl (3S,4S)-4-[4-(dimethylamino)phenyl]-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]piperidine-3-carboxylateIC505800.0 [1]
Ethyl (3S,4S)-4-[4-(dimethylamino)phenyl]-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]piperidine-3-carboxylateKi1960.0 [1], 10000.0 [2]
Ethyl (3S,4S)-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]-4-[3-(trifluoromethyl)phenyl]piperidine-3-carboxylateIC50125.0 [1]
Ethyl (3S,4S)-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]-4-[3-(trifluoromethyl)phenyl]piperidine-3-carboxylateKi350.0 [1], 990.0 [2], 10000.0 [3]
Ethyl (3S,4S)-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]-4-(4-phenylphenyl)piperidine-3-carboxylateIC5010000.0 [1]
Ethyl (3S,4S)-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]-4-(4-phenylphenyl)piperidine-3-carboxylateKi3770.0 [1], 10000.0 [2]
Ethyl (3S,4S)-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]-4-(4-ethoxycarbonylphenyl)piperidine-3-carboxylateIC5010000.0 [1]
Ethyl (3S,4S)-1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]-4-(4-ethoxycarbonylphenyl)piperidine-3-carboxylateKi1660.0 [1], 10000.0 [2]
Ethyl 1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]-4-(4-fluorophenyl)piperidine-3-carboxylateIC5051.1 [1]
Ethyl 1-[2-(2,4-dioxo-1H-quinazolin-3-yl)ethyl]-4-(4-fluorophenyl)piperidine-3-carboxylateKi179.0 [1], 290.0 [2], 10000.0 [3]
LobelinKi2760.0 [1]
FlorbenazineKi0.1 [1]
LobelaneKi970.0 [1]
10S-Hydroxylobel-7-eneKi6060.0 [1]
(2R,6S)-1-Methyl-2,6-bis-(2-naphthalen-1-yl-ethyl)-piperidineKi630.0 [1]
2-[4-[4-(7-(111C)Methoxynaphthalen-1-yl)piperazin-1-yl]butyl]-4-methyl-1,2,4-triazine-3,5-dioneKi10000.0 [1]
8R-Hydroxylobel-9-eneKi5160.0 [1]
Items per page: 1 - 10 of 45
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References

This online tool may be cited as follows

MLA

"Quest Database™ Synaptic vesicular amine transporter Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/synaptic-vesicular-amine-transporter-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ Synaptic vesicular amine transporter Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/synaptic-vesicular-amine-transporter-inhibitors-ic50-ki.
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