| Tifenazoxide | IC50 | 286.0 [1], 320.0 [2], 165000.0 [3], 685000.0 [4], 696000.0 [5] |
| Diazoxide | IC50 | 194000.0 [1], 198000.0 [2], 740000.0 [3], 750000.0 [4] |
| 6-Chloro-3-isopropylamino-4H-thieno(3,2-E)-1,2,4-thiadiazine 1,1-dioxide | IC50 | 340.0 [1], 187000.0 [2], 554000.0 [3] |
| 6-Chloro-N-(1-methylcyclobutyl)-1,1-dioxo-4H-thieno[3,2-e][1,2,4]thiadiazin-3-imine | IC50 | 3.0 [1], 10800.0 [2], 859000.0 [3] |
| (2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithia-4,6-diaza-inden-5-yl)-propyl-amine | IC50 | 2270.0 [1], 584000.0 [2], 924000.0 [3] |
| N-[(2R)-Butan-2-yl]-6-chloro-1,1-dioxo-4H-thieno[3,2-e][1,2,4]thiadiazin-3-imine | IC50 | 640.0 [1], 224000.0 [2], 487000.0 [3] |
| 6-Chloro-N-(2-methylbutan-2-yl)-1,1-dioxo-4H-thieno[3,2-e][1,2,4]thiadiazin-3-imine | IC50 | 180.0 [1], 375000.0 [2], 899000.0 [3] |
| Tert-Butyl-(2-chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithia-4,6-diaza-inden-5-yl)-amine | IC50 | 230.0 [1], 393000.0 [2], 1350000.0 [3] |
| (2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithia-4,6-diaza-inden-5-yl)-cyclobutyl-amine | IC50 | 120.0 [1], 146000.0 [2], 943000.0 [3] |
| N-[(2S)-Butan-2-yl]-6-chloro-1,1-dioxo-4H-thieno[3,2-e][1,2,4]thiadiazin-3-imine | IC50 | 460.0 [1], 309000.0 [2], 420000.0 [3] |
| 6-Chloro-1,1-dioxo-N-(2-phenylpropan-2-yl)-4H-thieno[3,2-e][1,2,4]thiadiazin-3-imine | IC50 | 81.0 [1], 360000.0 [2] |
| Glyburide | IC50 | 4.3 [1] |
| Clamikalant | IC50 | 8200.0 [1] |
| 4-Methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide | IC50 | 19952.62 [1] |