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Sphingosine 1-phosphate receptor Edg-5 Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
[3-(4-Nonyl-benzylamino)-propyl]-phosphonic acidIC500.7 [1], 5.5 [2], 320.0 [3], 750.0 [4], 10000.0 [5]
3-(Tetradecylamino)propylphosphonic acidIC5013.0 [1], 580.0 [2]
4-[3-(4-Fluorophenoxy)-5-[[4-(4-fluorophenyl)-4-hydroxypiperidine-1-carbonyl]amino]phenoxy]benzoic acidIC506.2 [1], 430.0 [2]
N-[3-(4-Carbamoylphenoxy)-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamideIC503.7 [1], 39.0 [2]
Sphingosine 1-phosphateIC500.23 [1], 0.35 [2], 3.6 [3]
CID 10223146IC5010.0 [1], 20.0 [2], 58.4 [3]
[(1R,3R)-3-Amino-1-hydroxy-5-(4-octylphenyl)pentyl]phosphonic acidIC504.5 [1], 33.0 [2], 10000.0 [3]
3-(3-Bromo-5-methoxy-4-(octyloxy)benzylamino)propylphosphonic acidIC5010.0 [1], 10000.0 [2]
Phosphonic acid, [3-amino-5-(4-octylphenyl)pentyl]-IC50100.0 [1], 10000.0 [2]
4-(2-Ethylbutyl)-N-[3-(4-fluorophenoxy)phenyl]-4-hydroxypiperidine-1-carboxamideIC501200.0 [1]
FTY720 phosphateIC500.77 [1], 1100.0 [2]
\n\n - Open Babel Depiction\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\n\nN\nO\nS\nF\nF\nF\nO\nHO\n\n\n\n\n1-(4-((4-Phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)azetidine-3-carboxylic acidIC5010000.0 [1]
Merck SIP AgonistIC5010000.0 [1]
CID 90309142IC508.2 [1], 500.0 [2]
[3-(4-Octyl-benzylamino)-propyl]-phosphonic acidIC505.5 [1], 10000.0 [2]
1-(4-Nonylbenzyl)pyrrolidin-3-ylphosphonic acidIC501000.0 [1], 10000.0 [2]
(3-Amino-heptadecyl)-phosphonic acidIC50830.0 [1], 1200.0 [2]
2-Hydroxy-4-(4-nonyl-benzylamino)-butyric acidIC5099.0 [1], 10000.0 [2]
3-Fluoro-4-(4-nonyl-benzylamino)-butyric acidIC5057.0 [1], 1000.0 [2]
[3-(3-Chloro-4-octyloxy-benzylamino)-propyl]-phosphonic acidIC501.7 [1], 10000.0 [2]
[3-(3-Ethoxy-4-octyloxy-benzylamino)-propyl]-phosphonic acidIC5012.0 [1], 10000.0 [2]
[3-(3-Methyl-4-octyloxy-benzylamino)-propyl]-phosphonic acidIC501.8 [1], 10000.0 [2]
[3-(3,5-Dichloro-4-octyloxy-benzylamino)-propyl]-phosphonic acidIC501.0 [1], 10000.0 [2]
[3-(4-Octyloxy-benzylamino)-propyl]-phosphonic acidIC506.3 [1], 4600.0 [2]
[3-(4-Nonanoyl-benzylamino)-propyl]-phosphonic acidIC504.0 [1], 8600.0 [2]
[3-(4-Nonyloxy-benzylamino)-propyl]-phosphonic acidIC501.7 [1], 840.0 [2]
[3-(3-Methoxy-5-methyl-4-octyloxy-benzylamino)-propyl]-phosphonic acidIC5019.0 [1], 10000.0 [2]
[3-(3-Chloro-5-methoxy-4-octyloxy-benzylamino)-propyl]-phosphonic acidIC508.0 [1], 10000.0 [2]
[3-(3-Bromo-5-methoxy-4-nonyloxy-benzylamino)-propyl]-phosphonic acidIC503.9 [1], 10000.0 [2]
[3-(3-Bromo-5-methoxy-4-undecyloxy-benzylamino)-propyl]-phosphonic acidIC501.9 [1], 10000.0 [2]
2,2-Difluoro-4-(4-nonyl-benzylamino)-butyric acidIC50200.0 [1], 10000.0 [2]
[3-(3-Fluoro-4-octyloxy-benzylamino)-propyl]-phosphonic acidIC502.0 [1], 4700.0 [2]
(3-Amino-hexadecyl)-phosphonic acidIC5086.0 [1], 10000.0 [2]
4-[(3-Phosphono-propylamino)-methyl]-benzoic acid heptyl esterIC50680.0 [1], 10000.0 [2]
(3-Amino-henicosyl)-phosphonic acidIC501500.0 [1], 10000.0 [2]
4-(4-Nonyl-benzylamino)-butyric acidIC50200.0 [1], 10000.0 [2]
Methyl-[3-(4-nonyl-benzylamino)-propyl]-phosphinic acidIC5060.0 [1], 10000.0 [2]
{3-[4-(1-Hydroxy-nonyl)-benzylamino]-propyl}-phosphonic acidIC50110.0 [1], 5400.0 [2]
[3-(3-Methoxy-4-octyloxy-benzylamino)-propyl]-phosphonic acidIC5024.0 [1], 10000.0 [2]
3-[[4-(4-Hexylphenyl)phenyl]methylamino]propylphosphonic acidIC502.6 [1], 3400.0 [2]
[3-(3-Bromo-4-heptyloxy-5-methoxy-benzylamino)-propyl]-phosphonic acidIC506.1 [1], 10000.0 [2]
[3-(3,5-Dibromo-4-octyloxy-benzylamino)-propyl]-phosphonic acidIC503.0 [1], 10000.0 [2]
3-Hydroxy-4-(4-nonyl-benzylamino)-butyric acidIC5066.0 [1], 10000.0 [2]
[3-(3-Hydroxy-4-octyloxy-benzylamino)-propyl]-phosphonic acidIC5041.0 [1], 10000.0 [2]
[3-(3,5-Dimethyl-4-octyloxy-benzylamino)-propyl]-phosphonic acidIC500.8 [1], 10000.0 [2]
[3-(3-Bromo-4-octyloxy-benzylamino)-propyl]-phosphonic acidIC502.9 [1], 10000.0 [2]
[3-(3-Bromo-4-decyloxy-5-methoxy-benzylamino)-propyl]-phosphonic acidIC501.5 [1], 10000.0 [2]
4-(2-Ethylbutyl)-N-[3-(4-fluorophenoxy)-5-methylphenyl]-4-hydroxypiperidine-1-carboxamideIC50500.0 [1]
N-[3-Chloro-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamideIC50860.0 [1]
N-[3-Ethoxy-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamideIC501400.0 [1]
N-[3,5-Bis(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamideIC50980.0 [1]
N-[3-(3-Carbamoylphenoxy)-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamideIC5013.0 [1], 150.0 [2]
N-[3-[4-(Dimethylcarbamoyl)phenoxy]-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamideIC508.8 [1], 43.0 [2]
4-(2-Ethylbutyl)-N-[3-(4-fluorophenoxy)-5-pyridin-4-yloxyphenyl]-4-hydroxypiperidine-1-carboxamideIC5045.0 [1], 93.0 [2]
4-(2-Ethylbutyl)-N-[3-(4-fluorophenoxy)-5-pyridin-3-yloxyphenyl]-4-hydroxypiperidine-1-carboxamideIC50210.0 [1], 940.0 [2]
4-(2-Ethylbutyl)-N-[3-(4-fluorophenoxy)-5-pyridin-2-yloxyphenyl]-4-hydroxypiperidine-1-carboxamideIC50260.0 [1], 390.0 [2]
(3-Hexadecylamino-propyl)-phosphonic acidIC5012.0 [1], 740.0 [2]
[2-Amino-1-hydroxy-4-(4-octylphenyl)butan-2-yl] dihydrogen phosphateIC500.8 [1], 1100.0 [2]
(3-Tridecylamino-propyl)-phosphonic acidIC5038.0 [1], 150.0 [2]
(3-Dodecylamino-propyl)-phosphonic acidIC5019.0 [1], 10000.0 [2]
3-[[4-(5-Heptyl-1,2,4-oxadiazol-3-yl)phenyl]methylamino]propylphosphonic acidIC501.8 [1], 1500.0 [2]
{3-[4-(2-Heptyl-2H-tetrazol-5-yl)-benzylamino]-propyl}-phosphonic acidIC501.4 [1], 2300.0 [2]
{3-[4-(4-Heptyl-phenyl)-butylamino]-propyl}-phosphonic acidIC50590.0 [1], 2000.0 [2]
3-[(4-Nonylphenyl)methylamino]propylphosphonous acidIC50140.0 [1], 10000.0 [2]
[3-(10-Phenyl-decylamino)-propyl]-phosphonic acidIC5059.0 [1], 530.0 [2]
(3-Pentadecylamino-propyl)-phosphonic acidIC5011.0 [1], 740.0 [2]
{3-[3-(4-Heptyl-phenyl)-propylamino]-propyl}-phosphonic acidIC5042.0 [1], 2200.0 [2]
{3-[2-(4-Octyl-phenyl)-ethylamino]-propyl}-phosphonic acidIC5045.0 [1], 10000.0 [2]
(3-Amino-octadecyl)-phosphonic acidIC50450.0 [1], 10000.0 [2]
(3-Amino-13-phenyl-tridecyl)-phosphonic acidIC50110.0 [1], 2100.0 [2]
2-[4-[3-(4-Fluorophenoxy)-5-[[4-hydroxy-4-(2-methylpropyl)piperidine-1-carbonyl]amino]phenoxy]phenyl]-2-methylpropanoic acidIC502.3 [1]
2-[4-[3-(4-Fluorophenoxy)-5-[[3-hydroxy-3-(2-methylpropyl)azetidine-1-carbonyl]amino]phenoxy]phenyl]-2-methylpropanoic acidIC505.2 [1], 9.4 [2]
4-(2-Ethylbutyl)-N-[3-(4-fluorophenoxy)-5-(4-sulfamoylphenoxy)phenyl]-4-hydroxypiperidine-1-carboxamideIC504.1 [1], 21.0 [2]
4-(2-Ethylbutyl)-N-[3-(4-fluorophenoxy)-5-[4-(methylcarbamoyl)phenoxy]phenyl]-4-hydroxypiperidine-1-carboxamideIC503.0 [1], 27.0 [2]
N-[3-(2-Carbamoylphenoxy)-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamideIC5049.0 [1], 88.0 [2]
4-(2-Ethylbutyl)-N-[3-(4-fluorophenoxy)-5-(4-methylsulfonylphenoxy)phenyl]-4-hydroxypiperidine-1-carboxamideIC5045.0 [1], 58.0 [2]
(3-Amino-pentadecyl)-phosphonic acidIC5086.0 [1], 10000.0 [2]
[3-(3-Bromo-4-hexyloxy-5-methoxy-benzylamino)-propyl]-phosphonic acidIC506.2 [1], 6500.0 [2]
FingolimodIC5010000.0 [1]
5-[4-Phenyl-5-(trifluoromethyl)-2-thienyl]-3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazoleIC5010000.0 [1]
Fingolimod phosphate ester, S-IC505.9 [1]
CeralifimodKi5450.0 [1]
N-(4-(Aminomethyl)-2,6-dimethylphenyl)-5-(2,5-dichlorophenyl)furan-2-carboxamideIC503900.0 [1]
CID 59393720IC5010000.0 [1]
(2R)-2-Amino-2-[(phosphonooxy)methyl]-4-(4-octylphenyl)-1-butanolIC5022000.0 [1]
1-[[4-[5-[4-Phenyl-5-(trifluoromethyl)thiophen-2-yl]-1,2,4-oxadiazol-3-yl]phenyl]methyl]azetidine-3-carboxylic acidIC5010000.0 [1]
3-(4-(5-(3-Cyano-4-isopropyloxyphenyl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acidIC5010000.0 [1]
4-Amino-6-(4-octylphenyl)hexanoic AcidIC501000.0 [1]
3-Amino-5-(4-octylphenyl)pentanoic AcidIC503300.0 [1]
[2-Amino-4-(4-octylphenyl)butyl] dihydrogen phosphateIC501.8 [1]
[3-Amino-3-hydroxymethyl-5-(4-octyl-phenyl)-pentyl]-phosphonic acidIC50230.0 [1]
1-{4-[5-(4-Tert-butylphenyl)-1,3,4-oxadiazol-2-yl]benzyl}azetidine-3-carboxylic acidIC5010000.0 [1]
1-{4-[3-(4-Tert-butylphenyl)-1,2,4-oxadiazol-5-yl]benzyl}azetidine-3-carboxylic acidIC5010000.0 [1]
3-[3-Methyl-4-[5-[4-propan-2-yloxy-3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-3-yl]phenyl]propanoic acidIC5010000.0 [1]
1-({4-[5-(4-Butylphenyl)-1,2,4-oxadiazol-3-yl]phenyl}methyl)azetidine-3-carboxylic acidIC5010000.0 [1]
1-(4-Nonylbenzyl)azetidine-3-carboxylic acidIC5010000.0 [1]
[3-Amino-2-hydroxy-5-(4-octylphenyl)pentyl]phosphonic acidIC50240.0 [1]
1-(4-((4-Phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)pyrrolidine-3-carboxylic acidIC5010000.0 [1]
1-(4-Nonylbenzyl)pyrrolidine-3-carboxylic acidIC5010000.0 [1]
1-(3-Chloro-4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)azetidine-3-carboxylic acidIC5010000.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Sphingosine 1-phosphate receptor Edg-5 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/sphingosine-1-phosphate-receptor-edg-5-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ Sphingosine 1-phosphate receptor Edg-5 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/sphingosine-1-phosphate-receptor-edg-5-inhibitors-ic50-ki.
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