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Somatostatin receptor 2 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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SomatostatinIC500.4 [1], 0.67 [2], 0.7 [3]
SomatostatinKi0.04 [1], 0.05 [2], 0.08 [3]
(4R,7S,10R,13S,16R,19S,22R,25S,28R,31S,34R,37S)-37-[[2-[[(2S)-2-[[(2S)-6-Amino-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-4-amino-2-[[(2S)-2-[[(2S)-4-amino-2-[[(2S)-2-[[(2S)-2-amino-3-hydroxypropanoyl]amino]propanoyl]amino]-4-oxobutanoyl]amino]-3-hydroxypropanoyl]amino]-4-oxobutanoyl]pyrrolidine-2-carbonyl]amino]propanoyl]amino]-4-methylsulfanylbutanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-4-carboxybutanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]hexanoyl]amino]propanoyl]amino]acetyl]amino]-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-13,25,28-tribenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxylic acidIC502.3 [1]
(4R,7S,10R,13S,16R,19S,22R,25S,28R,31S,34R,37S)-37-[[2-[[(2S)-2-[[(2S)-6-Amino-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-4-amino-2-[[(2S)-2-[[(2S)-4-amino-2-[[(2S)-2-[[(2S)-2-amino-3-hydroxypropanoyl]amino]propanoyl]amino]-4-oxobutanoyl]amino]-3-hydroxypropanoyl]amino]-4-oxobutanoyl]pyrrolidine-2-carbonyl]amino]propanoyl]amino]-4-methylsulfanylbutanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-4-carboxybutanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]hexanoyl]amino]propanoyl]amino]acetyl]amino]-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-13,25,28-tribenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxylic acidKi0.31 [1]
(4R,7S,10S,13R,16S,19R)-10-(4-Aminobutyl)-19-[[(2R)-2-amino-3-phenylpropanoyl]amino]-16-benzyl-N-[(2S,3R)-1,3-dihydroxybutan-2-yl]-7-[(1R)-1-hydroxyethyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamideIC500.02 [1], 1.0 [2]
(4R,7S,10S,13S,16R,19S,22S,25R)-25-Amino-13-(4-aminobutyl)-7,19,22-tribenzyl-10-[(1R)-1-hydroxyethyl]-16-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23-heptazacyclohexacosane-4-carboxylic acidIC5041.0 [1]
(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37-[[2-[[(2S)-2-[[(2S)-6-Amino-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-4-amino-2-[[(2S)-2-[[(2S)-4-amino-2-[[(2S)-2-[[(2S)-2-amino-3-hydroxypropanoyl]amino]propanoyl]amino]-4-oxobutanoyl]amino]-3-hydroxypropanoyl]amino]-4-oxobutanoyl]pyrrolidine-2-carbonyl]amino]propanoyl]amino]-4-methylsulfanylbutanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-4-carboxybutanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]hexanoyl]amino]propanoyl]amino]acetyl]amino]-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-13,25,28-tribenzyl-10,16-bis[(1S)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-2-ylmethyl)-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxylic acidIC502.1 [1], 2.3 [2], 2.7 [3], 3.3 [4]
SeglitideIC501.6 [1]
SeglitideKi0.08 [1], 0.3 [2]
CID 5311374IC501000.0 [1], 10000.0 [2]
(4R,7S,10S,13S,16S,19S,22S,25R)-25-Amino-13-(4-aminobutyl)-7,19,22-tribenzyl-10-[(1R)-1-hydroxyethyl]-16-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23-heptazacyclohexacosane-4-carboxylic acidIC50130.0 [1]
H-DPhe-c[Cys-Phe-DTrp-Lys-Thr-Cys]-Thr-NH2IC501.9 [1], 2.2 [2]
Cyclo(Pro-Phe-D-Trp-Lys-Thr-Phe)Ki0.63 [1], 5.1 [2]
8-D-Tryptophan-somatostatinIC501.1 [1]
8-D-Tryptophan-somatostatinKi0.0 [1]
CID 15965425Ki0.01 [1]
5-{3,4,5-Tris-benzyloxy-6-[2-(1H-indol-3-yl)-ethoxy]-tetrahydro-pyran-2-ylmethoxy}-pentylamineKi1800.0 [1], 4520.0 [2]
2-(1-(4-Amino-3,5-diethoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-5-sulfonamideKi10000.0 [1]
CID 52936725IC504.8 [1]
CID 52936725Ki0.03 [1]
(4R,7S,10S,13R,16S,19S)-10-(4-Aminobutyl)-19-[[(2S)-2-amino-3-(4-chlorophenyl)propanoyl]amino]-N-[(2S)-1-amino-3-naphthalen-2-yl-1-oxopropan-2-yl]-7-[(1R)-1-hydroxyethyl]-16-[(4-hydroxyphenyl)methyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamideKi5.51 [1], 26.0 [2]
(4R,7S,10S,13S,16S,19S,22S,25R)-25-Amino-13-(4-aminobutyl)-7,22-dibenzyl-10-[(1R)-1-hydroxyethyl]-19-[(4-hydroxyphenyl)methyl]-16-[(1S)-1-naphthalen-2-ylethyl]-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23-heptazacyclohexacosane-4-carboxylic acidIC50110.0 [1], 194.0 [2]
(4R,7S,10S,13S,16R,19S,22S,25R)-25-Amino-13-(4-aminobutyl)-7,22-dibenzyl-10-[(1R)-1-hydroxyethyl]-16-(1H-indol-3-ylmethyl)-19-methyl-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23-heptazacyclohexacosane-4-carboxylic acidIC50183.0 [1]
(4R,7S,10S,13S,16R,19S,22S,25R)-25-Amino-13-(4-aminobutyl)-7,22-dibenzyl-10-[(1R)-1-hydroxyethyl]-19-[(4-hydroxyphenyl)methyl]-16-[(1S)-1-naphthalen-2-ylethyl]-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23-heptazacyclohexacosane-4-carboxylic acidIC5030.0 [1], 339.0 [2]
Des-AA1,2,5-[IAmp9,Tyr11]-SRIFIC501000.0 [1], 10000.0 [2]
(4R,7S,10R,13S,16R,19S,22S,25S,28R,31R,34S)-31-(4-Aminobutyl)-34-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-13,25,28-tribenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33-decaoxo-19-[[4-[(propan-2-ylamino)methyl]phenyl]methyl]-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacontane-4-carboxylic acidIC501000.0 [1]
(4R,7S,10S,13S,16S,19S,22S,25R)-25-Amino-13-(4-aminobutyl)-7,22-dibenzyl-10-[(1R)-1-hydroxyethyl]-16-(1H-indol-3-ylmethyl)-19-methyl-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23-heptazacyclohexacosane-4-carboxylic acidIC50807.0 [1]
(2R,3S)-N-[(5-Amino-1,3-dioxan-2-yl)methyl]-3-(1H-indol-3-yl)-N-methyl-2-[2-oxo-3-(1-phenylpiperidin-3-yl)imidazolidin-1-yl]butanamideKi2.1 [1], 14.0 [2]
7-Chloro-3-(3,5-dimethylphenyl)-6-(1-methylpyrazol-4-yl)-4-[2-[(2S)-piperidin-2-yl]ethoxy]quinolineIC50145.0 [1]
7-Chloro-3-(3,5-dimethylphenyl)-6-(1-methylpyrazol-4-yl)-4-[2-[(2S)-piperidin-2-yl]ethoxy]quinolineKi1.5 [1]
3-{7-Chloro-3-(3,5-dimethylphenyl)-4-[2-(piperidin-2-yl)ethoxy]quinolin-6-yl}benzamideIC500.39 [1]
3-{7-Chloro-3-(3,5-dimethylphenyl)-4-[2-(piperidin-2-yl)ethoxy]quinolin-6-yl}benzamideKi0.04 [1]
3-[7-Chloro-3-(3,5-dimethylphenyl)-4-{2-[(2R)-piperidin-2-yl]ethoxy}quinolin-6-yl]phenolIC501.1 [1]
3-[7-Chloro-3-(3,5-dimethylphenyl)-4-{2-[(2R)-piperidin-2-yl]ethoxy}quinolin-6-yl]phenolKi0.04 [1]
4-[7-Chloro-3-(3,5-dimethylphenyl)-4-{2-[(2R)-piperidin-2-yl]ethoxy}quinolin-6-yl]phenolIC500.38 [1]
4-[7-Chloro-3-(3,5-dimethylphenyl)-4-{2-[(2R)-piperidin-2-yl]ethoxy}quinolin-6-yl]phenolKi0.08 [1]
[4-[7-Chloro-3-(3,5-dimethylphenyl)-4-[2-[(2R)-piperidin-2-yl]ethoxy]quinolin-6-yl]phenyl]methanolIC5013.0 [1]
[4-[7-Chloro-3-(3,5-dimethylphenyl)-4-[2-[(2R)-piperidin-2-yl]ethoxy]quinolin-6-yl]phenyl]methanolKi0.1 [1]
7-Chloro-3-(3,5-dimethylphenyl)-4-[2-[(2R)-piperidin-2-yl]ethoxy]-6-pyridin-4-ylquinolineIC5020.0 [1]
7-Chloro-3-(3,5-dimethylphenyl)-4-[2-[(2R)-piperidin-2-yl]ethoxy]-6-pyridin-4-ylquinolineKi0.11 [1]
7-Chloro-3-(3,5-dimethylphenyl)-6-(6-fluoropyridin-3-yl)-4-[2-[(2R)-piperidin-2-yl]ethoxy]quinolineIC504.7 [1]
7-Chloro-3-(3,5-dimethylphenyl)-6-(6-fluoropyridin-3-yl)-4-[2-[(2R)-piperidin-2-yl]ethoxy]quinolineKi0.12 [1]
3-[4-(3-Aminopropoxy)-7-chloro-3-(3,5-dimethylphenyl)quinolin-6-yl]benzamideIC500.38 [1]
3-[4-(3-Aminopropoxy)-7-chloro-3-(3,5-dimethylphenyl)quinolin-6-yl]benzamideKi0.08 [1]
Tert-butyl (2S)-6-amino-2-[[(2R)-3-(1H-indol-3-yl)-2-[[4-(4-methylphenyl)sulfonylpiperazine-1-carbonyl]amino]propanoyl]amino]hexanoateIC509.2 [1], 7700.0 [2]
Tert-butyl (2S)-6-amino-2-[[(2R)-2-[(4-benzoylpiperazine-1-carbonyl)amino]-3-(1H-indol-3-yl)propanoyl]amino]hexanoateIC506.9 [1], 1600.0 [2]
Tert-butyl (2S)-6-amino-2-[[(2R)-3-(1H-indol-3-yl)-2-[[4-(4-methylbenzoyl)piperazine-1-carbonyl]amino]propanoyl]amino]hexanoateIC504.4 [1], 67.0 [2]
Tert-butyl (2S)-6-amino-2-[[(2R)-2-[[1-(benzenesulfonyl)piperidine-4-carbonyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]hexanoateIC503.2 [1], 120.0 [2]
Tert-butyl (2S)-6-amino-2-[[(2S)-3-(1H-indol-3-yl)-2-[(4-phenylbenzoyl)amino]propanoyl]amino]hexanoateIC5085.0 [1], 1200.0 [2]
(4R,8S,11S,17S)-8-(4-Aminobutyl)-17-[[2-amino-3-(3-fluorophenyl)propanoyl]amino]-N-(1-amino-3-naphthalen-1-yl-1-oxopropan-2-yl)-6-tert-butyl-11-(1H-indol-3-ylmethyl)-7,10,13,16-tetraoxo-14-(pyridin-3-ylmethyl)-1,2-dithia-5,9,12,15-tetrazacyclooctadecane-4-carboxamideIC504.1 [1], 270.0 [2]
Methyl (2S)-5-(diaminomethylideneamino)-2-[[(2S)-3-(3-fluorophenyl)-2-[(4-methylphenyl)sulfonylamino]propanoyl]amino]pentanoateIC502000.0 [1], 6500.0 [2]
Tert-butyl (2S)-6-amino-2-[[(2R)-3-(1H-indol-3-yl)-2-[[4-(2-oxo-3H-benzimidazol-1-yl)piperidine-1-carbonyl]amino]propanoyl]amino]hexanoateIC500.26 [1], 6.5 [2]
Tert-butyl (2S)-6-amino-2-[[(2R)-2-[[4-(benzenesulfonyl)piperazine-1-carbonyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]hexanoateIC502.9 [1], 29.0 [2]
Tert-butyl (2R)-6-amino-2-[[(2R,3S)-3-(1H-indol-3-yl)-2-[2-oxo-3-(4-phenylcyclohexyl)imidazolidin-1-yl]butanoyl]amino]hexanoateKi6.3 [1], 40.0 [2]
(4R,7S,10S,13R,16S,19S)-10-(4-Aminobutyl)-19-[[(2R)-2-amino-3-(4-chlorophenyl)propanoyl]amino]-N-[(2S)-1-amino-3-naphthalen-2-yl-1-oxopropan-2-yl]-7-[(1R)-1-hydroxyethyl]-16-[(4-hydroxyphenyl)methyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamideIC505.7 [1]
(4R,7S,10S,13R,16S,19S)-10-(4-Aminobutyl)-19-[[(2R)-2-amino-3-(4-chlorophenyl)propanoyl]amino]-N-[(2S)-1-amino-3-naphthalen-2-yl-1-oxopropan-2-yl]-7-[(1R)-1-hydroxyethyl]-16-[(4-hydroxyphenyl)methyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamideKi26.0 [1]
(4R,7S,10S,13R,16S,19S)-19-[[(2R)-2-Amino-3-(4-chlorophenyl)propanoyl]amino]-N-[(2S)-1-amino-3-naphthalen-2-yl-1-oxopropan-2-yl]-7-[(1R)-1-hydroxyethyl]-16-[(4-hydroxyphenyl)methyl]-13-(1H-indol-3-ylmethyl)-10-[4-(methylamino)butyl]-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamideIC5010.0 [1]
(4R,7S,10S,13R,16S,19S)-19-[[(2R)-2-Amino-3-(4-chlorophenyl)propanoyl]amino]-N-[(2S)-1-amino-3-naphthalen-2-yl-1-oxopropan-2-yl]-7-[(1R)-1-hydroxyethyl]-16-[(4-hydroxyphenyl)methyl]-13-(1H-indol-3-ylmethyl)-10-[4-(methylamino)butyl]-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamideKi5.51 [1]
7-Chloro-3-(3,5-dimethylphenyl)-4-[2-[(2R)-piperidin-2-yl]ethoxy]-6-pyridin-3-ylquinolineIC508.3 [1]
7-Chloro-3-(3,5-dimethylphenyl)-4-[2-[(2R)-piperidin-2-yl]ethoxy]-6-pyridin-3-ylquinolineKi0.13 [1]
5-[7-Chloro-3-(3,5-dimethylphenyl)-4-[2-[(2R)-piperidin-2-yl]ethoxy]quinolin-6-yl]-1H-pyridin-2-oneIC500.29 [1]
5-[7-Chloro-3-(3,5-dimethylphenyl)-4-[2-[(2R)-piperidin-2-yl]ethoxy]quinolin-6-yl]-1H-pyridin-2-oneKi0.27 [1]
5-[7-Chloro-3-(3,5-dimethylphenyl)-4-[2-[(2R)-piperidin-2-yl]ethoxy]quinolin-6-yl]pyridin-2-amineIC5034.0 [1]
5-[7-Chloro-3-(3,5-dimethylphenyl)-4-[2-[(2R)-piperidin-2-yl]ethoxy]quinolin-6-yl]pyridin-2-amineKi0.6 [1]
7-Chloro-3-(3,5-dimethylphenyl)-6-(6-methoxypyridin-3-yl)-4-[2-[(2R)-piperidin-2-yl]ethoxy]quinolineIC5050.0 [1]
7-Chloro-3-(3,5-dimethylphenyl)-6-(6-methoxypyridin-3-yl)-4-[2-[(2R)-piperidin-2-yl]ethoxy]quinolineKi0.65 [1]
7-Chloro-6-(6-chloropyridin-3-yl)-3-(3,5-dimethylphenyl)-4-[2-[(2R)-piperidin-2-yl]ethoxy]quinolineIC5011.0 [1]
7-Chloro-6-(6-chloropyridin-3-yl)-3-(3,5-dimethylphenyl)-4-[2-[(2R)-piperidin-2-yl]ethoxy]quinolineKi0.13 [1]
[3-[7-Chloro-6-(1-methylpyrazol-4-yl)-4-[2-[(2R)-piperidin-2-yl]ethoxy]quinolin-3-yl]phenyl]methanolIC508.3 [1]
[3-[7-Chloro-6-(1-methylpyrazol-4-yl)-4-[2-[(2R)-piperidin-2-yl]ethoxy]quinolin-3-yl]phenyl]methanolKi0.13 [1]
[3-[3-[3-(Hydroxymethyl)phenyl]-4-[2-[(2R)-piperidin-2-yl]ethoxy]quinolin-6-yl]phenyl]methanolIC5011.0 [1]
[3-[3-[3-(Hydroxymethyl)phenyl]-4-[2-[(2R)-piperidin-2-yl]ethoxy]quinolin-6-yl]phenyl]methanolKi0.13 [1]
7-Chloro-3-(3,5-dimethylphenyl)-6-(1-methylpyrazol-4-yl)-4-[2-[(2R)-piperidin-2-yl]ethoxy]quinolineIC504.8 [1]
7-Chloro-3-(3,5-dimethylphenyl)-6-(1-methylpyrazol-4-yl)-4-[2-[(2R)-piperidin-2-yl]ethoxy]quinolineKi0.03 [1]
7-Chloro-3-(3,5-dimethylphenyl)-6-phenyl-4-(2-piperidin-2-ylethoxy)-1,2-dihydroquinolineIC507.6 [1]
7-Chloro-3-(3,5-dimethylphenyl)-6-phenyl-4-(2-piperidin-2-ylethoxy)-1,2-dihydroquinolineKi0.18 [1]
(4R,7S,10R,13S,16R,19R,22S,25R,28S,31R,34S,37R)-19,34-Bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25-dibenzyl-10,16-bis[(1S)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-28-(pyrazin-2-ylmethyl)-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxylic acidKi1.0 [1], 7.0 [2]
AstemizoleKi10000.0 [1]
LanreotideKi0.5 [1]
PasireotideKi1.0 [1]
EdotreotideIC5014.0 [1]
VapreotideKi0.08 [1]
(4R,7S,10S,13S,16S,19S,22R,25S,28S,31S,34R)-34-Amino-31-(4-aminobutyl)-13,25,28-tribenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33-decaoxo-19-[[4-[(propan-2-ylamino)methyl]phenyl]methyl]-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacontane-4-carboxylic acidIC501000.0 [1]
1-[3-[(5-Bromopyridin-2-yl)-[(3,4-dichlorophenyl)methyl]amino]propyl]-3-[3-(1H-imidazol-5-yl)propyl]thioureaKi621.0 [1]
CID 56927659IC504025.0 [1]
(1R,3R)-1-(Oxan-4-yl)-3-(5-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indoleIC501000.0 [1]
(3R)-1,1-Dibutyl-3-(5-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indoleKi10000.0 [1]
3-[3-(1H-Imidazole-4-yl)propyl]-1-[2-[(5-bromo-2-pyridinyl)(3,4-dichlorobenzyl)amino]ethyl]thioureaKi310.0 [1]
(2R,5R)-5-(4-Aminobutyl)-2-(1H-indol-3-ylmethyl)-7-(naphthalen-1-ylmethyl)-1,4,7-thiadiazonane-3,6-dioneIC501585.0 [1]
H-c[Cys-Phe-DTrp-Lys-Thr-Cys]-OHIC50378.0 [1]
(3S)-1,1-Dibutyl-3-(5-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indoleKi10000.0 [1]
5-[[(2R,3R,4S,5R,6R)-5-(1H-Imidazol-5-ylmethoxy)-6-[2-(1H-indol-3-yl)ethoxy]-4-phenylmethoxy-3-(pyridin-3-ylmethoxy)oxan-2-yl]methoxy]pentan-1-amineIC502250.0 [1]
N-(1-(3-Ethoxy-4-methoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amineKi10000.0 [1]
2-(1-(3-Ethoxy-4-methoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-5-sulfonamideKi10000.0 [1]
N-(1-(4-Chloro-3-ethoxybenzyl)piperidin-4-yl)-5-methylnicotinamideKi10000.0 [1]
3-[(1R,3R)-3-[5-(5-Fluoropyridin-2-yl)-1H-imidazol-2-yl]-1-(1-methylpyrazol-4-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-5-methyl-1,2,4-oxadiazoleIC5010000.0 [1]
4-((4-(Benzo[d]oxazol-2-ylamino)piperidin-1-yl)methyl)-2-ethoxyphenolKi10000.0 [1]
N-(1-(3-(Cyclopentyloxy)-4-methoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amineKi10000.0 [1]
Benzooxazol-2-yl-[1-(3-isobutoxy-4-methoxy-benzyl)-piperidin-4-yl]-amineKi10000.0 [1]
Items per page: 1 - 10 of 99
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References

This online tool may be cited as follows

MLA

"Quest Database™ Somatostatin receptor 2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/somatostatin-receptor-2-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ Somatostatin receptor 2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/somatostatin-receptor-2-inhibitors-ic50-ki.
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