Solute carrier organic anion transporter family member 1B3 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Dioscin	Ki	1030.0 [1], 1430.0 [2], 4550.0 [3], 8290.0 [4]
	Silymarin	IC50	2700.0 [1], 4265.8 [2]
	Silymarin	Ki	3270.0 [1]
	Calcium	IC50	3388.44 [1]
	Calcium	Ki	2580.0 [1]
	Sodium	IC50	1905.46 [1]
	Sodium	Ki	1480.0 [1]
	Bilirubin	IC50	3388.44 [1]
	Bilirubin	Ki	2630.0 [1]
	Vincristine	IC50	11000.0 [1], 36780.0 [2]
	Rifampicin	IC50	1500.0 [1]
	Rifampicin	Ki	5000.0 [1]
	Arachidonic acid	IC50	1071.52 [1]
	Arachidonic acid	Ki	820.0 [1]
	Genistein	IC50	3890.45 [1]
	Genistein	Ki	2960.0 [1]
	Losartan	IC50	1148.15 [1]
	Losartan	Ki	890.0 [1]
	beta-Carotene	IC50	2951.21 [1]
	beta-Carotene	Ki	2260.0 [1]
	Tannic acid	IC50	4168.69 [1]
	Tannic acid	Ki	3230.0 [1]
	Telmisartan	IC50	1258.93 [1]
	Telmisartan	Ki	960.0 [1]
	Enoxolone	IC50	549.54 [1]
	Enoxolone	Ki	420.0 [1]
	Gossypol	IC50	4570.88 [1]
	Gossypol	Ki	3470.0 [1]
	Hydroxyzine pamoate	IC50	1230.27 [1]
	Hydroxyzine pamoate	Ki	940.0 [1]
	Olmesartan medoxomil	IC50	977.24 [1]
	Olmesartan medoxomil	Ki	750.0 [1]
	Mometasone furoate	IC50	1148.15 [1]
	Mometasone furoate	Ki	870.0 [1]
	Nonoxynol-9	IC50	3715.35 [1]
	Nonoxynol-9	Ki	2870.0 [1]
	Lasalocid sodium	IC50	776.25 [1]
	Lasalocid sodium	Ki	590.0 [1]
	Candesartan cilexetil	IC50	2454.71 [1]
	Candesartan cilexetil	Ki	1900.0 [1]
	Dicloxacillin sodium monohydrate	IC50	1995.26 [1]
	Dicloxacillin sodium monohydrate	Ki	1550.0 [1]
	Erythromycin ethylsuccinate	IC50	2089.3 [1]
	Erythromycin ethylsuccinate	Ki	1610.0 [1]
	Retinyl acetate	IC50	5011.87 [1]
	Retinyl acetate	Ki	3890.0 [1]
	(-)-Epicatechin gallate	IC50	4466.84 [1]
	(-)-Epicatechin gallate	Ki	3460.0 [1]
	Abietic acid	IC50	5248.07 [1]
	Abietic acid	Ki	4080.0 [1]
	Erythromycin estolate	IC50	3090.3 [1]
	Erythromycin estolate	Ki	2350.0 [1]
	Sarsasapogenin	IC50	104.71 [1]
	Sarsasapogenin	Ki	80.0 [1]
	Hederagenin	IC50	891.25 [1]
	Hederagenin	Ki	680.0 [1]
	Aurin	IC50	4073.8 [1]
	Aurin	Ki	3150.0 [1]
	Lobaric acid	IC50	1621.81 [1]
	Lobaric acid	Ki	1250.0 [1]
	Methyl cholate	IC50	3715.35 [1]
	Methyl cholate	Ki	2890.0 [1]
	Norstictic acid	IC50	549.54 [1]
	Norstictic acid	Ki	420.0 [1]
	Theasinensin B	IC50	8511.38 [1]
	Theasinensin B	Ki	6500.0 [1]
	Scandenin	IC50	741.31 [1]
	Scandenin	Ki	560.0 [1]
	Anthothecol	IC50	3467.37 [1]
	Anthothecol	Ki	2640.0 [1]
	(2S,3S,4S,5R,6R)-6-[[(3S,4S,6Ar,6bR,8R,8aR,9R,10R,14aR,14bS)-9-acetyloxy-8-hydroxy-4,8a-bis(hydroxymethyl)-6a,6b,11,11,14b-pentamethyl-10-[(E)-2-methylbut-2-enoyl]oxy-2,3,4,4a,5,6,7,8,9,10,12,12a,14,14a-tetradecahydro-1H-picen-3-yl]oxy]-4-hydroxy-3,5-bis[[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy]oxane-2-carboxylic acid	IC50	3388.44 [1]
	(2S,3S,4S,5R,6R)-6-[[(3S,4S,6Ar,6bR,8R,8aR,9R,10R,14aR,14bS)-9-acetyloxy-8-hydroxy-4,8a-bis(hydroxymethyl)-6a,6b,11,11,14b-pentamethyl-10-[(E)-2-methylbut-2-enoyl]oxy-2,3,4,4a,5,6,7,8,9,10,12,12a,14,14a-tetradecahydro-1H-picen-3-yl]oxy]-4-hydroxy-3,5-bis[[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy]oxane-2-carboxylic acid	Ki	2610.0 [1]
	Acetyl isogambogic acid	IC50	5370.32 [1]
	Acetyl isogambogic acid	Ki	4170.0 [1]
	Methyl (2S,3R,4R,5S)-4-[(1S,3aS,5R,6R,7R,7aR)-6-formyloxy-1-(furan-3-yl)-3a-hydroxy-7-[(2R,3R)-2-hydroxy-3-methylpentanoyl]oxy-7a-methyl-4-methylidene-3-oxo-2,5,6,7-tetrahydro-1H-inden-5-yl]-5-acetyloxy-2-(acetyloxymethyl)-2,4-dimethyl-7-oxooxepane-3-carboxylate	IC50	3388.44 [1]
	Methyl (2S,3R,4R,5S)-4-[(1S,3aS,5R,6R,7R,7aR)-6-formyloxy-1-(furan-3-yl)-3a-hydroxy-7-[(2R,3R)-2-hydroxy-3-methylpentanoyl]oxy-7a-methyl-4-methylidene-3-oxo-2,5,6,7-tetrahydro-1H-inden-5-yl]-5-acetyloxy-2-(acetyloxymethyl)-2,4-dimethyl-7-oxooxepane-3-carboxylate	Ki	2630.0 [1]
	Methyl 6-acetoxyangolensate	IC50	3801.89 [1]
	Methyl 6-acetoxyangolensate	Ki	2920.0 [1]
	Leoidin	IC50	2398.83 [1]
	Leoidin	Ki	1840.0 [1]
	Gangaleoidin	IC50	2630.27 [1]
	Gangaleoidin	Ki	2020.0 [1]
	Bussein	IC50	691.83 [1]
	Bussein	Ki	530.0 [1]
	Utilin	IC50	776.25 [1]
	Utilin	Ki	600.0 [1]
	Chukrasin methyl ether	IC50	724.44 [1]
	Chukrasin methyl ether	Ki	560.0 [1]
	Dimethyl gambogate	IC50	5128.61 [1]
	Dimethyl gambogate	Ki	3940.0 [1]
	Dihydrogambogic acid	IC50	2884.03 [1]
	Dihydrogambogic acid	Ki	2240.0 [1]
	Garcinolic acid	IC50	2238.72 [1]
	Garcinolic acid	Ki	1730.0 [1]
	[(2R,3R,4S,5R)-3-[(2R,3R,4S,5R,6S)-5-[(2S,3R,4S,5R)-3,5-Dihydroxy-4-[(2R,3R,4R,5R,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxyoxan-2-yl]oxy-3,4-dihydroxy-6-methyloxan-2-yl]oxy-4,5-dihydroxyoxan-2-yl] (4aR,5R,6aR,6aS,6bR,8aR,10S,12aR,14bR)-5-hydroxy-2,2,6a,6b,9,9,12a-heptamethyl-10-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydropicene-4a-carboxylate	IC50	5248.07 [1]
	[(2R,3R,4S,5R)-3-[(2R,3R,4S,5R,6S)-5-[(2S,3R,4S,5R)-3,5-Dihydroxy-4-[(2R,3R,4R,5R,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxyoxan-2-yl]oxy-3,4-dihydroxy-6-methyloxan-2-yl]oxy-4,5-dihydroxyoxan-2-yl] (4aR,5R,6aR,6aS,6bR,8aR,10S,12aR,14bR)-5-hydroxy-2,2,6a,6b,9,9,12a-heptamethyl-10-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydropicene-4a-carboxylate	Ki	4020.0 [1]
	Decahydrogambogic acid	IC50	2290.87 [1]
	Decahydrogambogic acid	Ki	1770.0 [1]
	[(1R,2R,4S,7R,8R,11R,12S,13S,15R,17S,19R)-13-Acetyloxy-7-(furan-3-yl)-19-hydroxy-1,8,12,16,16-pentamethyl-5-oxo-3,6-dioxapentacyclo[9.8.0.02,4.02,8.012,17]nonadecan-15-yl] acetate	IC50	2951.21 [1]
	[(1R,2R,4S,7R,8R,11R,12S,13S,15R,17S,19R)-13-Acetyloxy-7-(furan-3-yl)-19-hydroxy-1,8,12,16,16-pentamethyl-5-oxo-3,6-dioxapentacyclo[9.8.0.02,4.02,8.012,17]nonadecan-15-yl] acetate	Ki	2270.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 100 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Solute carrier organic anion transporter family member 1B3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 22 Feb. 2025, https://www.aatbio.com/data-sets/solute-carrier-organic-anion-transporter-family-member-1b3-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, February 22). Quest Database™ Solute carrier organic anion transporter family member 1B3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/solute-carrier-organic-anion-transporter-family-member-1b3-inhibitors-ic50-ki.
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