Solute carrier organic anion transporter family member 1B1 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Cyclosporin A	IC50	700.0 [1], 1200.0 [2]
	Cyclosporin A	Ki	200.0 [1], 238.0 [2], 1300.0 [3]
	Rifampicin	IC50	300.0 [1], 1200.0 [2], 2200.0 [3], 2300.0 [4]
	Rifampicin	Ki	17000.0 [1]
	Sodium	IC50	50.0 [1], 1949.84 [2]
	Sodium	Ki	44.0 [1], 1070.0 [2]
	Verapamil	IC50	32000.0 [1], 64000.0 [2], 600000.0 [3]
	Verapamil	Ki	52000.0 [1]
	Simvastatin	IC50	4400.0 [1], 6000.0 [2], 9700.0 [3], 11000.0 [4]
	Ritonavir	IC50	700.0 [1], 1000.0 [2], 1300.0 [3], 5000.0 [4]
	Gemfibrozil	IC50	4073.8 [1], 11000.0 [2], 38000.0 [3], 130000.0 [4]
	Atorvastatin	IC50	600.0 [1], 800.0 [2], 1600.0 [3]
	Glyburide	IC50	1400.0 [1], 2200.0 [2], 21000.0 [3]
	Silymarin	IC50	6165.95 [1], 9700.0 [2]
	Silymarin	Ki	3370.0 [1]
	Calcium	IC50	812.83 [1]
	Calcium	Ki	450.0 [1]
	Bilirubin	IC50	1318.26 [1]
	Bilirubin	Ki	720.0 [1]
	Arachidonic acid	IC50	602.56 [1]
	Arachidonic acid	Ki	330.0 [1]
	Genistein	IC50	9120.11 [1]
	Genistein	Ki	5000.0 [1]
	Losartan	IC50	288.4 [1]
	Losartan	Ki	160.0 [1]
	beta-Carotene	IC50	616.6 [1]
	beta-Carotene	Ki	340.0 [1]
	Tannic acid	IC50	2630.27 [1]
	Tannic acid	Ki	1460.0 [1]
	Telmisartan	IC50	1862.09 [1]
	Telmisartan	Ki	1030.0 [1]
	Enoxolone	IC50	524.81 [1]
	Enoxolone	Ki	290.0 [1]
	Gossypol	IC50	3235.94 [1]
	Gossypol	Ki	1780.0 [1]
	Hydroxyzine pamoate	IC50	812.83 [1]
	Hydroxyzine pamoate	Ki	450.0 [1]
	Olmesartan medoxomil	IC50	977.24 [1]
	Olmesartan medoxomil	Ki	540.0 [1]
	Mometasone furoate	IC50	2951.21 [1]
	Mometasone furoate	Ki	1620.0 [1]
	Nonoxynol-9	IC50	3467.37 [1]
	Nonoxynol-9	Ki	1920.0 [1]
	Lasalocid sodium	IC50	478.63 [1]
	Lasalocid sodium	Ki	260.0 [1]
	Candesartan cilexetil	IC50	724.44 [1]
	Candesartan cilexetil	Ki	400.0 [1]
	Dicloxacillin sodium monohydrate	IC50	676.08 [1]
	Dicloxacillin sodium monohydrate	Ki	370.0 [1]
	Erythromycin ethylsuccinate	IC50	3019.95 [1]
	Erythromycin ethylsuccinate	Ki	1670.0 [1]
	Retinyl acetate	IC50	2238.72 [1]
	Retinyl acetate	Ki	1220.0 [1]
	(-)-Epicatechin gallate	IC50	3801.89 [1]
	(-)-Epicatechin gallate	Ki	2070.0 [1]
	Rifamycin	IC50	230.0 [1]
	Rifamycin	Ki	2000.0 [1]
	Abietic acid	IC50	2691.53 [1]
	Abietic acid	Ki	1470.0 [1]
	Erythromycin estolate	IC50	4365.16 [1]
	Erythromycin estolate	Ki	2410.0 [1]
	Sarsasapogenin	IC50	245.47 [1]
	Sarsasapogenin	Ki	130.0 [1]
	Hederagenin	IC50	3801.89 [1]
	Hederagenin	Ki	2110.0 [1]
	Alisporivir	IC50	180.0 [1], 800.0 [2]
	Aurin	IC50	2630.27 [1]
	Aurin	Ki	1430.0 [1]
	Lobaric acid	IC50	724.44 [1]
	Lobaric acid	Ki	400.0 [1]
	Methyl cholate	IC50	8317.64 [1]
	Methyl cholate	Ki	4580.0 [1]
	Norstictic acid	IC50	1148.15 [1]
	Norstictic acid	Ki	630.0 [1]
	Theasinensin B	IC50	3715.35 [1]
	Theasinensin B	Ki	2050.0 [1]
	Scandenin	IC50	1071.52 [1]
	Scandenin	Ki	590.0 [1]
	Anthothecol	IC50	3019.95 [1]
	Anthothecol	Ki	1650.0 [1]
	(2S,3S,4S,5R,6R)-6-[[(3S,4S,6Ar,6bR,8R,8aR,9R,10R,14aR,14bS)-9-acetyloxy-8-hydroxy-4,8a-bis(hydroxymethyl)-6a,6b,11,11,14b-pentamethyl-10-[(E)-2-methylbut-2-enoyl]oxy-2,3,4,4a,5,6,7,8,9,10,12,12a,14,14a-tetradecahydro-1H-picen-3-yl]oxy]-4-hydroxy-3,5-bis[[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy]oxane-2-carboxylic acid	IC50	1412.54 [1]
	(2S,3S,4S,5R,6R)-6-[[(3S,4S,6Ar,6bR,8R,8aR,9R,10R,14aR,14bS)-9-acetyloxy-8-hydroxy-4,8a-bis(hydroxymethyl)-6a,6b,11,11,14b-pentamethyl-10-[(E)-2-methylbut-2-enoyl]oxy-2,3,4,4a,5,6,7,8,9,10,12,12a,14,14a-tetradecahydro-1H-picen-3-yl]oxy]-4-hydroxy-3,5-bis[[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy]oxane-2-carboxylic acid	Ki	780.0 [1]
	Acetyl isogambogic acid	IC50	4073.8 [1]
	Acetyl isogambogic acid	Ki	2240.0 [1]
	Methyl (2S,3R,4R,5S)-4-[(1S,3aS,5R,6R,7R,7aR)-6-formyloxy-1-(furan-3-yl)-3a-hydroxy-7-[(2R,3R)-2-hydroxy-3-methylpentanoyl]oxy-7a-methyl-4-methylidene-3-oxo-2,5,6,7-tetrahydro-1H-inden-5-yl]-5-acetyloxy-2-(acetyloxymethyl)-2,4-dimethyl-7-oxooxepane-3-carboxylate	IC50	2344.23 [1]
	Methyl (2S,3R,4R,5S)-4-[(1S,3aS,5R,6R,7R,7aR)-6-formyloxy-1-(furan-3-yl)-3a-hydroxy-7-[(2R,3R)-2-hydroxy-3-methylpentanoyl]oxy-7a-methyl-4-methylidene-3-oxo-2,5,6,7-tetrahydro-1H-inden-5-yl]-5-acetyloxy-2-(acetyloxymethyl)-2,4-dimethyl-7-oxooxepane-3-carboxylate	Ki	1280.0 [1]
	Methyl 6-acetoxyangolensate	IC50	1445.44 [1]
	Methyl 6-acetoxyangolensate	Ki	800.0 [1]
	Leoidin	IC50	144.54 [1]
	Leoidin	Ki	80.0 [1]
	Gangaleoidin	IC50	102.33 [1]
	Gangaleoidin	Ki	60.0 [1]
	Bussein	IC50	691.83 [1]
	Bussein	Ki	380.0 [1]
	Utilin	IC50	676.08 [1]
	Utilin	Ki	380.0 [1]
	Chukrasin methyl ether	IC50	758.58 [1]
	Chukrasin methyl ether	Ki	420.0 [1]
	Dimethyl gambogate	IC50	2290.87 [1]
	Dimethyl gambogate	Ki	1260.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

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References

This online tool may be cited as follows

MLA	"Quest Database™ Solute carrier organic anion transporter family member 1B1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Feb. 2025, https://www.aatbio.com/data-sets/solute-carrier-organic-anion-transporter-family-member-1b1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, February 21). Quest Database™ Solute carrier organic anion transporter family member 1B1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/solute-carrier-organic-anion-transporter-family-member-1b1-inhibitors-ic50-ki.
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