 | Benzenesulfonamide, 4-methyl-N-8-quinolinyl- | IC50 | 49900.0 [1] |
 | 8-(4-Benzenesulfonylamino)quinoline | IC50 | 4590.0 [1] |
 | 5H-Quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide | IC50 | 2900.0 [1] |
 | 2-Nitro-N-quinolin-8-ylbenzenesulfonamide | IC50 | 2900.0 [1] |
 | 2-Amino-N-quinolin-8-yl-benzenesulfonamide | IC50 | 20800.0 [1] |
 | 2-Amino-N-(2-methylquinolin-8-yl)benzenesulfonamide | IC50 | 100000.0 [1] |
 | 9-Trifluoromethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 130.0 [1] |
 | 2-Amino-N-(6-methoxyquinolin-8-yl)-4-methylbenzenesulfonamide | IC50 | 585.0 [1] |
 | 2-Nitro-N-quinolin-8-yl-4-(trifluoromethyl)benzenesulfonamide | IC50 | 100000.0 [1] |
 | 9-Fluoro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 1560.0 [1] |
 | 9-Methyl-5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide | IC50 | 3200.0 [1] |
 | 9-Chloro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 770.0 [1] |
 | 9-Methoxy-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 1580.0 [1] |
 | 5-Bromo-N-quinolin-8-ylthiophene-2-sulfonamide | IC50 | 6800.0 [1] |
 | N-(2-Methylquinolin-8-yl)benzenesulfonamide | IC50 | 100000.0 [1] |
 | 2,4-Dichloro-N-quinolin-8-yl-benzenesulfonamide | IC50 | 989.0 [1] |
 | 4-Methoxy-N-quinolin-8-ylbenzenesulfonamide | IC50 | 100000.0 [1] |
 | N-(6-Methoxyquinolin-8-yl)benzenesulfonamide | IC50 | 6400.0 [1] |
 | 4-Chloro-N-(8-quinolinyl)benzenesulfonamide | IC50 | 3200.0 [1] |
 | N-(5,7-Dichloroquinolin-8-yl)-4-methylbenzenesulfonamide | IC50 | 79000.0 [1] |
 | N-(6-Fluoroquinolin-8-yl)-4-(trifluoromethyl)benzenesulfonamide | IC50 | 25000.0 [1] |
 | 1-[2-Fluoro-5-(3-methyl-2,2-dioxo-1,4-dihydropyrido[3,2-h][2,1,3]benzothiadiazin-4-yl)phenyl]ethanone | IC50 | 5430.0 [1] |
 | N-(7-Hydroxyquinolin-8-yl)benzenesulfonamide | IC50 | 100000.0 [1] |
 | N-(5,7-Dichloroquinolin-8-yl)-2,4,6-trimethylbenzenesulfonamide | IC50 | 100000.0 [1] |
 | 2-Amino-4-methoxy-N-quinolin-8-ylbenzenesulfonamide | IC50 | 100000.0 [1] |
 | 3-Methyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 100000.0 [1] |
 | 4-Methoxy-2-nitro-N-(quinolin-8-yl)benzene-1-sulfonamide | IC50 | 1810.0 [1] |
 | 2-Amino-N-quinolin-8-yl-4-(trifluoromethyl)benzenesulfonamide | IC50 | 760.0 [1] |
 | 2-Amino-4-methyl-N-quinolin-8-ylbenzenesulfonamide | IC50 | 300.0 [1] |
 | 4-Fluoro-2-nitro-N-quinolin-8-ylbenzenesulfonamide | IC50 | 920.0 [1] |
 | 2-Amino-4-fluoro-N-quinolin-8-ylbenzenesulfonamide | IC50 | 3940.0 [1] |
 | 12-Chloro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 320.0 [1] |
 | 12-Bromo-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 12600.0 [1] |
 | 2-Amino-4-methoxy-N-(2-methylquinolin-8-yl)benzenesulfonamide | IC50 | 100000.0 [1] |
 | N-(Quinolin-8-yl)-2-(trifluoromethoxy)benzene-1-sulfonamide | IC50 | 2500.0 [1] |
 | N-Quinolin-8-ylpyridine-2-sulfonamide | IC50 | 1890.0 [1] |
 | 8-Methoxy-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 2110.0 [1] |
 | 8-Trifluoromethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 2340.0 [1] |
 | 8-Methyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 360.0 [1] |
 | 8-Fluoro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 1620.0 [1] |
 | N-Quinolin-8-ylpyridine-3-sulfonamide | IC50 | 3640.0 [1] |
 | 2,6-Dichloro-N-quinolin-8-ylbenzenesulfonamide | IC50 | 100000.0 [1] |
 | 2-Cyano-N-quinolin-8-ylbenzenesulfonamide | IC50 | 815.0 [1] |
 | Methyl 3-[(quinolin-8-yl)sulfamoyl]benzoate | IC50 | 1420.0 [1] |
 | N-Quinolin-8-yl-3-(trifluoromethoxy)benzenesulfonamide | IC50 | 1200.0 [1] |
 | N-(5-Chloroquinolin-8-yl)benzenesulfonamide | IC50 | 1670.0 [1] |
 | 2-Chloro-N-(quinolin-8-yl)benzene-1-sulfonamide | IC50 | 8000.0 [1] |
 | 2,6-Difluoro-N-quinolin-8-ylbenzenesulfonamide | IC50 | 1140.0 [1] |
 | N-(8-Quinolinyl)-3-(trifluoromethyl)benzenesulfonamide | IC50 | 720.0 [1] |
 | 2-Methyl-N-(8-quinolinyl)benzenesulfonamide | IC50 | 100000.0 [1] |
 | N-(5-Bromoquinolin-8-yl)benzenesulfonamide | IC50 | 100000.0 [1] |
 | 3-Methyl-N-(8-quinolinyl)benzenesulfonamide | IC50 | 2090.0 [1] |
 | 2-Methoxy-N-quinolin-8-ylbenzenesulfonamide | IC50 | 100000.0 [1] |
 | 1-[4-(4-Fluorophenyl)-3-methyl-2,2-dioxo-1,4-dihydropyrido[3,2-h][2,1,3]benzothiadiazin-6-yl]ethanone | IC50 | 250.0 [1] |
 | 1-(3,4-Difluoro-phenyl)-2-methyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene 3,3-dioxide | IC50 | 250.0 [1] |
 | N-(7-Methylquinolin-8-yl)benzenesulfonamide | IC50 | 100000.0 [1] |
 | N-(6-Chloroquinolin-8-yl)benzenesulfonamide | IC50 | 100000.0 [1] |
 | N-(3-Methylquinolin-8-yl)benzenesulfonamide | IC50 | 610.0 [1] |
 | 2,4,6-Trichloro-N-quinolin-8-ylbenzenesulfonamide | IC50 | 857.0 [1] |
 | 2-Methyl-N-[2-(quinolin-8-ylsulfamoyl)phenyl]propanamide | IC50 | 24600.0 [1] |
 | 2,2,2-Trifluoro-N-[2-(quinolin-8-ylsulfamoyl)phenyl]acetamide | IC50 | 307.0 [1] |
 | 4-Chloro-N-(5-chloroquinolin-8-yl)-2-fluorobenzenesulfonamide | IC50 | 1380.0 [1] |
 | CID 60163923 | IC50 | 1750.0 [1] |
 | N-(6-Methoxyquinolin-8-yl)pyridine-3-sulfonamide | IC50 | 2800.0 [1] |
 | N-(5-Chloroquinolin-8-yl)pyridine-3-sulfonamide | IC50 | 1780.0 [1] |
 | 2-Amino-N-(6-methoxyquinolin-8-yl)-4-(trifluoromethyl)benzenesulfonamide | IC50 | 1000.0 [1] |
 | 2,4-Dichloro-N-(3-methylquinolin-8-yl)benzenesulfonamide | IC50 | 100000.0 [1] |
 | N-(3-Methylquinolin-8-yl)pyridine-3-sulfonamide | IC50 | 1390.0 [1] |
 | N-(5-Chloro-6-methylquinolin-8-yl)benzenesulfonamide | IC50 | 100000.0 [1] |
 | N-(7-Chloroquinolin-8-yl)benzenesulfonamide | IC50 | 100000.0 [1] |
 | N-(7-Methoxyquinolin-8-yl)benzenesulfonamide | IC50 | 100000.0 [1] |
 | 8,9-Dimethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 4020.0 [1] |
 | 12-Methyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 599.0 [1] |
 | 11-Methoxy-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 100000.0 [1] |
 | 1-Methoxy-9-trifluoromethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 979.0 [1] |
 | 2-Phenyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene 3,3-dioxide | IC50 | 460.0 [1] |
 | 1,4-Dihydro-2H-3-thia-2,4,5-triaza-phenanthrene 3,3-dioxide | IC50 | 39500.0 [1] |
 | 2-Methyl-1-phenyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene 3,3-dioxide | IC50 | 870.0 [1] |
 | N-Quinolin-8-yl-1,3-thiazole-2-sulfonamide | IC50 | 4580.0 [1] |
 | N-Quinolin-8-ylpyrazine-2-sulfonamide | IC50 | 1910.0 [1] |
 | N-[6-(Trifluoromethoxy)quinolin-8-yl]-6-(trifluoromethyl)pyridine-3-sulfonamide | IC50 | 12500.0 [1] |
 | 6-(Trifluoromethyl)-N-[5-(trifluoromethyl)quinolin-8-yl]pyridine-3-sulfonamide | IC50 | 25000.0 [1] |
 | N-[5-(Trifluoromethyl)quinolin-8-yl]pyridine-2-sulfonamide | IC50 | 460.0 [1] |
 | N-[6-(Trifluoromethoxy)quinolin-8-yl]pyridine-2-sulfonamide | IC50 | 1090.0 [1] |
 | N-(6-Fluoroquinolin-8-yl)pyridine-2-sulfonamide | IC50 | 2370.0 [1] |
 | 6-Cyano-N-[6-(trifluoromethoxy)quinolin-8-yl]pyridine-3-sulfonamide | IC50 | 2110.0 [1] |
 | 6-Cyano-N-(6-fluoroquinolin-8-yl)pyridine-3-sulfonamide | IC50 | 3750.0 [1] |
 | Methyl 6,6-dioxo-5H-quinolino[8,7-c][1,2]benzothiazine-9-carboxylate | IC50 | 4180.0 [1] |
 | 6,6-Dioxo-5H-quinolino[8,7-c][1,2]benzothiazine-9-carbonitrile | IC50 | 2830.0 [1] |
 | 1-Trifluoromethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 25000.0 [1] |
 | 9-Chloro-1-trifluoromethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 25000.0 [1] |
 | 12-Trifluoromethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 14100.0 [1] |
 | 9-Chloro-12-trifluoromethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 8510.0 [1] |
 | 3-Chloro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 25000.0 [1] |
 | 8,12-Dichloro-9-fluoro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 25000.0 [1] |
 | 12-Chloro-8,9-difluoro-5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide | IC50 | 25000.0 [1] |
 | 9-Chloro-6,6-dioxo-5H-quinolino[8,7-c][1,2]benzothiazine-12-carbonitrile | IC50 | 25000.0 [1] |
 | 3,9-Dichloro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 25000.0 [1] |
 | 12-Chloro-9-methanesulfonyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide | IC50 | 25000.0 [1] |
 | Methyl 6,6-dioxo-5H-quinolino[8,7-c][1,2]benzothiazine-1-carboxylate | IC50 | 2940.0 [1] |