| Probenecid | IC50 | 6300.0 [1], 7400.0 [2], 12300.0 [3], 12500.0 [4] |
| Probenecid | Ki | 4300.0 [1], 4410.0 [2], 12100.0 [3] |
| Aminohippuric acid | IC50 | 8800.0 [1], 127000.0 [2] |
| Aminohippuric acid | Ki | 6020.0 [1] |
| Betamipron | IC50 | 6000.0 [1], 39000.0 [2] |
| Betamipron | Ki | 23600.0 [1] |
| Indoxyl sulfate | IC50 | 83000.0 [1] |
| Indoxyl sulfate | Ki | 22700.0 [1], 23000.0 [2] |
| Ketoprofen | IC50 | 1300.0 [1], 1400.0 [2] |
| Piroxicam | IC50 | 20500.0 [1] |
| Piroxicam | Ki | 19800.0 [1] |
| Hippuric acid | IC50 | 20000.0 [1] |
| Hippuric acid | Ki | 66000.0 [1] |
| Cilastatin | IC50 | 2550000.0 [1] |
| Cilastatin | Ki | 1470000.0 [1] |
| Citrinin | Ki | 3080000.0 [1] |
| (6R,7R)-8-Oxo-3-(pyridin-1-ium-1-ylmethyl)-7-[(2-thiophen-2-ylacetyl)amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid | IC50 | 1250000.0 [1] |
| (6R,7R)-8-Oxo-3-(pyridin-1-ium-1-ylmethyl)-7-[(2-thiophen-2-ylacetyl)amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid | Ki | 740.0 [1] |
| Indomethacin | IC50 | 3000.0 [1] |
| Ibuprofen | IC50 | 8000.0 [1] |
| Diclofenac | IC50 | 4000.0 [1] |
| Salicylic acid | IC50 | 280000.0 [1] |
| Cimetidine | IC50 | 492000.0 [1] |
| Naproxen | IC50 | 5800.0 [1] |
| Pravastatin | IC50 | 408000.0 [1] |
| Ceftriaxone | Ki | 230.0 [1] |
| Cefotaxime | Ki | 3130.0 [1] |
| Cefazolin | Ki | 180.0 [1] |
| Flurbiprofen | IC50 | 1500.0 [1] |
| Cephalothin | Ki | 220.0 [1] |
| Phenacetin | IC50 | 200000.0 [1] |
| Cidofovir | IC50 | 60000.0 [1] |
| Octanoic acid | Ki | 5410.0 [1] |
| Ellagic acid | IC50 | 270.0 [1] |
| Cefoperazone | Ki | 210.0 [1] |
| Adefovir | IC50 | 28000.0 [1] |
| Cefamandole | Ki | 30.0 [1] |
| Glutaric acid | IC50 | 4900.0 [1] |
| Diflunisal | IC50 | 850.0 [1] |
| Cephradine | IC50 | 1600000.0 [1] |
| Cefadroxil | Ki | 6140.0 [1] |
| 2,3-Dimercapto-1-propanesulfonic acid | Ki | 22400.0 [1] |
| Benzbromarone | IC50 | 4600.0 [1] |
| Etodolac | IC50 | 50000.0 [1] |
| 3-Acetoxyindole | IC50 | 83000.0 [1] |
| Salicyluric acid | IC50 | 27000.0 [1] |
| 3-Hydroxyglutaric acid | Ki | 98000.0 [1] |
| Rolofylline | Ki | 7820.0 [1] |
| Oseltamivir acid | Ki | 45100000.0 [1] |
| Zonampanel | IC50 | 3000.0 [1] |
| Cyclic-hpmpc | IC50 | 1100000.0 [1] |
| 4-Hydroxyhippuric acid | IC50 | 25000.0 [1] |
| S-(2-Benzothiazolyl)cysteine | IC50 | 9900.0 [1] |
| (2S)-2-Amino-3-[(Z)-1,2-dichloroethenyl]sulfanylpropanoic acid | IC50 | 208000.0 [1] |
| Benzothiazolylcysteine | IC50 | 9900.0 [1] |
| 1-Methylpyrenyl Mercapturic Acid | Ki | 14500.0 [1] |
| 2-Sulfanyl-3-[(2-sulfanyl-2-sulfoethyl)disulfanyl]propane-1-sulfonic acid | Ki | 66000.0 [1] |
| (2S)-2-Amino-3-(2-chloro-1,1,2-trifluoroethyl)sulfanylpropanoic acid | IC50 | 177000.0 [1] |
| 2-(Trifluoromethyl)-N-[6-(trifluoromethyl)pyridin-3-yl]benzenesulfonamide | IC50 | 12300.0 [1] |
| 2-(Trifluoromethyl)-N-[5-(trifluoromethyl)pyridin-3-yl]benzenesulfonamide | IC50 | 9300.0 [1] |
| CID 86271138 | IC50 | 14300.0 [1] |
| CID 86294663 | IC50 | 14000.0 [1] |