![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_ebac36f7213da3162d29205ab4152aca.svg) | Prazosin | IC50 | 13600.0 [1], 100000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_35003ced678586a25de172e3d06d122a.svg) | Cimetidine | IC50 | 23000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_35003ced678586a25de172e3d06d122a.svg) | Cimetidine | Ki | 57000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_04cbfb18d4637aa7607c73b2f21de570.svg) | Ondansetron | IC50 | 890.0 [1], 1700.0 [2] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_a93f87e7386d15f182665420dd81b9e5.svg) | Pepcid | IC50 | 36100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_a93f87e7386d15f182665420dd81b9e5.svg) | Pepcid | Ki | 1800000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_2cb3539cbcab54cd61d20691715b1d3e.svg) | Tetramethylammonium | IC50 | 150000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_2cb3539cbcab54cd61d20691715b1d3e.svg) | Tetramethylammonium | Ki | 180000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_8cafaa409fb2dcc84d3240fee93c8314.svg) | Pseudoisocyanine | IC50 | 1130.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_8cafaa409fb2dcc84d3240fee93c8314.svg) | Pseudoisocyanine | Ki | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_3f6592008acb912de238d3aaaf8e5ad5.svg) | Metiprenaline | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_3f6592008acb912de238d3aaaf8e5ad5.svg) | Metiprenaline | Ki | 570000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_28dba8f145b0b6293925c8c01ab57119.svg) | Estradiol | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_84be4cdb308fb643cf288980a1c24c41.svg) | Progesterone | IC50 | 26700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_30efcd8594e5a6ac05921ba868878567.svg) | Corticosterone | IC50 | 34200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_393a6636008719cf0eb93219e05af350.svg) | Metformin | IC50 | 1700000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_b2d54f313fd6fae3559ad99a1d264705.svg) | Imatinib | IC50 | 4200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_0f6f978fc95318968a1d88f8481932fe.svg) | Irinotecan | IC50 | 2700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_be4565ca8c20c1d9804fa640fd1584d5.svg) | Risperidone | IC50 | 11000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_8871e5bc150daca600c47dd7893b11be.svg) | Ethinyl estradiol | IC50 | 2200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_6c3911c895bcf58e15c1ea316421d8fe.svg) | Imipramine | IC50 | 600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_2019d6686c0079c33ef9d229dcb67e59.svg) | Dipyridamole | IC50 | 2600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_3fb59b292039fb68c21d347565286601.svg) | Quinine | Ki | 3400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_49a577a7a8bf4807ce110cac0f81baf9.svg) | Chlorhexidine | IC50 | 400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_9eea3482ccbd85339d3c08d99095be33.svg) | Ritonavir | IC50 | 24800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_926035c06d9d341c1f456b3b189f3e17.svg) | Mitoxantrone | IC50 | 73300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_0f4d8b43fb0367336924afd47b02995d.svg) | Tetraethylammonium | IC50 | 156000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_b2f3218cdbd5f04949eaaf044a21d56f.svg) | Desipramine | Ki | 16000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_c3fec52b171093040a67f2fb6c9d8f8e.svg) | Phenoxybenzamine | IC50 | 4900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_201d087333f42d154ec5c63fa41ae425.svg) | Tubocurarine | IC50 | 78800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_22ca1744345a750f98669f67193f6275.svg) | Carvedilol | IC50 | 7500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_abaf387535b47aae3a9dfa84743be0c3.svg) | Aripiprazole | IC50 | 239000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_0a51bf7eacaa481a84c82d93eeacce50.svg) | Topotecan | IC50 | 61000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_b517d83684d06e6ce0554cacfb470fe9.svg) | Procainamide | Ki | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_0cb63da9824d08dd47365ca9791b812b.svg) | Amantadine | IC50 | 23000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_07d34a94b97fbbe747832a79cffe07a8.svg) | Dabigatran | IC50 | 4700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_c9960c7f038fe75af1672de453506a31.svg) | Indinavir | IC50 | 142000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_0eb0b8c599a479d8d1ad1fc42fa97400.svg) | Vecuronium | IC50 | 3500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_47eddd337dafa05fe9d237d27dca82c1.svg) | Buspirone | IC50 | 12000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_8b6095c409ba14f4a2a342d36e7e5bfb.svg) | Cyperquat | Ki | 2400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_4ecf014c739d4d7f4bb8c1e87b900db7.svg) | Domperidone | IC50 | 7900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_168624a25c3c9d480db32878243c3257.svg) | Pantoprazole | IC50 | 1500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_32a1a4e75a5409dde1a18f2173a90394.svg) | Pentamidine | IC50 | 1200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_170f5263dd119f2c9f5904c3d6347c33.svg) | Pimozide | IC50 | 34200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_922e591df45814020ba0e2ba5eca1f5b.svg) | Tacrine | IC50 | 680.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_284bf47e1ecb17282f21d485720c2e90.svg) | Dihydroergotamine | IC50 | 49900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_db5d2aaeb82f333bc390f7a61d20cd50.svg) | Disopyramide | IC50 | 2900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_dc63e4f696179991c762c163b5bf9476.svg) | Tetrabutylammonium | IC50 | 120000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_f1389cd1d8b6ba9f0bf28775189ca42b.svg) | Phenformin | IC50 | 65000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_f1e44219327ec5d3833ac42aff528e73.svg) | Maraviroc | IC50 | 255000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_9c3656ff341e5e268acece6a306b8bb8.svg) | Granisetron | IC50 | 4300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_10e671aa0c2e8af205d779ba113db7f0.svg) | Zafirlukast | IC50 | 9700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_2dee02d8b672dc9ec123450abcbff8e6.svg) | Gabexate | IC50 | 900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_39f28c7db5b571077dbf34394d5beb87.svg) | Dolutegravir | IC50 | 1900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_307582b656256d08794edf3f5613a5a3.svg) | Orphenadrine | IC50 | 2500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_633e6dfffcf9d327a06f2856f979b0cb.svg) | Rimantadine | IC50 | 4400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_2f012b29ba88fd87f54d5e4eef19a971.svg) | Noscapine | IC50 | 2600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_7a511f64478fb8b75838455bd83206be.svg) | Camostat | IC50 | 16500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_7530b8355d72841ecace9c03543eb9af.svg) | Epinastine | IC50 | 4300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_89f632ef3482ab6e2214fd7116ba7ca0.svg) | N-Methylnicotinamide | Ki | 266000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_5a5b2db7898174efe1b0850be1ba01e3.svg) | Bithionol | IC50 | 1900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_c3b9e7bcc43f821330e3f557e266aed4.svg) | Nifekalant | IC50 | 10300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_f06ab1a946a0ffbca194ab5d5dd3b18c.svg) | Tetrapropylammonium | IC50 | 128000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_1e8fe7dc68e113ec523db30fe281f377.svg) | Tetrapentylammonium | Ki | 1500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_a546464b88610fa579feb5df8dfacc85.svg) | 1-Phenylguanidine | IC50 | 89000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_e16a5f1aa99ef1b9070f88ea04250c01.svg) | 1-(3-Chlorophenyl)guanidine | IC50 | 60500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_6cd16eb86c6b73a79066c78df73d9382.svg) | Mepiperphenidol | Ki | 4800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_87a95a663c107992e86d429c9d49a6c2.svg) | 1-(4-Chlorophenyl)guanidine | IC50 | 18900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_22c21e0636d3044d8d727d3d92ca2400.svg) | N-p-Tolyl-guanidine | IC50 | 9300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_3292fb283895da0b7e94f7f360c67d47.svg) | 1-(4-Fluorophenyl)guanidine | IC50 | 48300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_b29fe561edfaf81ae3a689ddfaf285ac.svg) | N-(2-Chloroethyl)-N-methyl-9H-fluoren-9-amine | IC50 | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_fdb652ef248d83e5f37e08b9fd843da4.svg) | 1-(4-Bromophenyl)guanidine | IC50 | 11300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_ef2fdb95f641edcf8dba5fdf2fe93b36.svg) | N-(4-Benzylphenyl)guanidine | IC50 | 96200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_c70d15dfd1d0a23ae55c35ce8bb8579d.svg) | N-(4-Iodo-phenyl)-guanidine | IC50 | 4400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_9f6debcc42c46c2923c07b4798bc815a.svg) | 1-(4-Tert-Butylphenyl)guanidine | IC50 | 8300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-2_9162db67eec8773ed7eebc9e4b11ee52.svg) | 2-[(3,6-Dimethyl-2-phenyl-4H-pyrimidin-4-yl)methyl]-1-ethylquinolin-1-ium | Ki | 210.0 [1] |