Solute carrier family 22 member 2 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Prazosin	IC50	13600.0 [1], 100000.0 [2]
	Cimetidine	IC50	23000.0 [1]
	Cimetidine	Ki	57000.0 [1]
	Ondansetron	IC50	890.0 [1], 1700.0 [2]
	Pepcid	IC50	36100.0 [1]
	Pepcid	Ki	1800000.0 [1]
	Tetramethylammonium	IC50	150000.0 [1]
	Tetramethylammonium	Ki	180000.0 [1]
	Pseudoisocyanine	IC50	1130.0 [1]
	Pseudoisocyanine	Ki	100.0 [1]
	Metiprenaline	IC50	100000.0 [1]
	Metiprenaline	Ki	570000.0 [1]
	Estradiol	IC50	30000.0 [1]
	Progesterone	IC50	26700.0 [1]
	Corticosterone	IC50	34200.0 [1]
	Metformin	IC50	1700000.0 [1]
	Imatinib	IC50	4200.0 [1]
	Irinotecan	IC50	2700.0 [1]
	Risperidone	IC50	11000.0 [1]
	Ethinyl estradiol	IC50	2200.0 [1]
	Imipramine	IC50	600.0 [1]
	Dipyridamole	IC50	2600.0 [1]
	Quinine	Ki	3400.0 [1]
	Chlorhexidine	IC50	400.0 [1]
	Ritonavir	IC50	24800.0 [1]
	Mitoxantrone	IC50	73300.0 [1]
	Tetraethylammonium	IC50	156000.0 [1]
	Desipramine	Ki	16000.0 [1]
	Phenoxybenzamine	IC50	4900.0 [1]
	Tubocurarine	IC50	78800.0 [1]
	Carvedilol	IC50	7500.0 [1]
	Aripiprazole	IC50	239000.0 [1]
	Topotecan	IC50	61000.0 [1]
	Procainamide	Ki	50000.0 [1]
	Amantadine	IC50	23000.0 [1]
	Dabigatran	IC50	4700.0 [1]
	Indinavir	IC50	142000.0 [1]
	Vecuronium	IC50	3500.0 [1]
	Buspirone	IC50	12000.0 [1]
	Cyperquat	Ki	2400.0 [1]
	Domperidone	IC50	7900.0 [1]
	Pantoprazole	IC50	1500.0 [1]
	Pentamidine	IC50	1200.0 [1]
	Pimozide	IC50	34200.0 [1]
	Tacrine	IC50	680.0 [1]
	Dihydroergotamine	IC50	49900.0 [1]
	Disopyramide	IC50	2900.0 [1]
	Tetrabutylammonium	IC50	120000.0 [1]
	Phenformin	IC50	65000.0 [1]
	Maraviroc	IC50	255000.0 [1]
	Granisetron	IC50	4300.0 [1]
	Zafirlukast	IC50	9700.0 [1]
	Gabexate	IC50	900.0 [1]
	Dolutegravir	IC50	1900.0 [1]
	Orphenadrine	IC50	2500.0 [1]
	Rimantadine	IC50	4400.0 [1]
	Noscapine	IC50	2600.0 [1]
	Camostat	IC50	16500.0 [1]
	Epinastine	IC50	4300.0 [1]
	N-Methylnicotinamide	Ki	266000.0 [1]
	Bithionol	IC50	1900.0 [1]
	Nifekalant	IC50	10300.0 [1]
	Tetrapropylammonium	IC50	128000.0 [1]
	Tetrapentylammonium	Ki	1500.0 [1]
	1-Phenylguanidine	IC50	89000.0 [1]
	1-(3-Chlorophenyl)guanidine	IC50	60500.0 [1]
	Mepiperphenidol	Ki	4800.0 [1]
	1-(4-Chlorophenyl)guanidine	IC50	18900.0 [1]
	N-p-Tolyl-guanidine	IC50	9300.0 [1]
	1-(4-Fluorophenyl)guanidine	IC50	48300.0 [1]
	N-(2-Chloroethyl)-N-methyl-9H-fluoren-9-amine	IC50	100.0 [1]
	1-(4-Bromophenyl)guanidine	IC50	11300.0 [1]
	N-(4-Benzylphenyl)guanidine	IC50	96200.0 [1]
	N-(4-Iodo-phenyl)-guanidine	IC50	4400.0 [1]
	1-(4-Tert-Butylphenyl)guanidine	IC50	8300.0 [1]
	2-[(3,6-Dimethyl-2-phenyl-4H-pyrimidin-4-yl)methyl]-1-ethylquinolin-1-ium	Ki	210.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 76 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Solute carrier family 22 member 2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 30 Mar. 2025, https://www.aatbio.com/data-sets/solute-carrier-family-22-member-2-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, March 30). Quest Database™ Solute carrier family 22 member 2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/solute-carrier-family-22-member-2-inhibitors-ic50-ki.
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