![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_1a2ef0969fddb77e7c383253c8b871b7.svg) | Clonidine | IC50 | 18980.0 [1], 22600.0 [2] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_1a2ef0969fddb77e7c383253c8b871b7.svg) | Clonidine | Ki | 550.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_6c3911c895bcf58e15c1ea316421d8fe.svg) | Imipramine | IC50 | 7950.0 [1], 17100.0 [2], 37000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_35003ced678586a25de172e3d06d122a.svg) | Cimetidine | IC50 | 100000.0 [1], 149000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_35003ced678586a25de172e3d06d122a.svg) | Cimetidine | Ki | 166000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_d9d88c2a7bdabc45b702c06047b28bae.svg) | Quinidine | IC50 | 23400.0 [1], 113800.0 [2] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_d9d88c2a7bdabc45b702c06047b28bae.svg) | Quinidine | Ki | 17500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_0f4d8b43fb0367336924afd47b02995d.svg) | Tetraethylammonium | Ki | 158000.0 [1], 161000.0 [2], 163000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_b2f3218cdbd5f04949eaaf044a21d56f.svg) | Desipramine | IC50 | 9180.0 [1], 56800.0 [2] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_b2f3218cdbd5f04949eaaf044a21d56f.svg) | Desipramine | Ki | 5360.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_04cbfb18d4637aa7607c73b2f21de570.svg) | Ondansetron | IC50 | 20400.0 [1], 100000.0 [2], 300000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_8cafaa409fb2dcc84d3240fee93c8314.svg) | Pseudoisocyanine | IC50 | 980.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_8cafaa409fb2dcc84d3240fee93c8314.svg) | Pseudoisocyanine | Ki | 2730.0 [1], 4400.0 [2] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_30efcd8594e5a6ac05921ba868878567.svg) | Corticosterone | IC50 | 21700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_30efcd8594e5a6ac05921ba868878567.svg) | Corticosterone | Ki | 7020.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_01814a6086009d7440d5f435a324c600.svg) | Verapamil | IC50 | 6800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_01814a6086009d7440d5f435a324c600.svg) | Verapamil | Ki | 2900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_393a6636008719cf0eb93219e05af350.svg) | Metformin | IC50 | 1230000.0 [1], 2010000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_a7e11d7bcee94c9af8c42c557a082c25.svg) | Chlorpromazine | IC50 | 4300.0 [1], 27000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_ebac36f7213da3162d29205ab4152aca.svg) | Prazosin | IC50 | 1840.0 [1], 9900.0 [2] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_3fb59b292039fb68c21d347565286601.svg) | Quinine | IC50 | 51600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_3fb59b292039fb68c21d347565286601.svg) | Quinine | Ki | 22900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_3f59bab9b954f7e2737294dc8b7f1b51.svg) | Trimethoprim | IC50 | 50680.0 [1], 56800.0 [2] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_c3fec52b171093040a67f2fb6c9d8f8e.svg) | Phenoxybenzamine | IC50 | 2720.0 [1], 15100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_0eb0b8c599a479d8d1ad1fc42fa97400.svg) | Vecuronium | Ki | 120000.0 [1], 232000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_922e591df45814020ba0e2ba5eca1f5b.svg) | Tacrine | IC50 | 21720.0 [1], 83000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_db5d2aaeb82f333bc390f7a61d20cd50.svg) | Disopyramide | IC50 | 81700.0 [1], 100000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_89fd1058473b46f547fd6ef0c68156d1.svg) | Propafenone | IC50 | 11100.0 [1], 15540.0 [2] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_dc63e4f696179991c762c163b5bf9476.svg) | Tetrabutylammonium | IC50 | 52000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_dc63e4f696179991c762c163b5bf9476.svg) | Tetrabutylammonium | Ki | 29600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_307582b656256d08794edf3f5613a5a3.svg) | Orphenadrine | IC50 | 12600.0 [1], 100000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_5a5b2db7898174efe1b0850be1ba01e3.svg) | Bithionol | IC50 | 2230.0 [1], 3900.0 [2] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_f06ab1a946a0ffbca194ab5d5dd3b18c.svg) | Tetrapropylammonium | IC50 | 90000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_f06ab1a946a0ffbca194ab5d5dd3b18c.svg) | Tetrapropylammonium | Ki | 102000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_28dba8f145b0b6293925c8c01ab57119.svg) | Estradiol | IC50 | 5730.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_84be4cdb308fb643cf288980a1c24c41.svg) | Progesterone | IC50 | 3050.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_629c398a4b53125db843b1930cacf26a.svg) | Morphine | IC50 | 28000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_c70f5b79af37726016ec15cea0b55e94.svg) | Propranolol | IC50 | 63200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_42b65f9d06589482f6ee80cb71d05669.svg) | Atropine | IC50 | 12200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_b2d54f313fd6fae3559ad99a1d264705.svg) | Imatinib | IC50 | 107000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_7ce5c90b273b41810bee3170ac9401d3.svg) | Haloperidol | IC50 | 141900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_94fca8d3b15a98bf35a0a3961e7494ec.svg) | Midazolam | Ki | 3700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_58cd7b84d6fa6df8bbd156b30a5cc7f2.svg) | Thiamine | IC50 | 4354000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_0f6f978fc95318968a1d88f8481932fe.svg) | Irinotecan | IC50 | 20800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_3e94330ba1527a829fecddbee5acde55.svg) | Apomorphine | IC50 | 20800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_2019d6686c0079c33ef9d229dcb67e59.svg) | Dipyridamole | IC50 | 81000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_3a9de7e3ee99440d6e854c271aa6a7d6.svg) | Amiloride | IC50 | 57000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_946b0b501eb57b26c13e79111c2b1587.svg) | Amitriptyline | IC50 | 16900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_a69f1db31ed30d6a63db389cb16202f2.svg) | Ketoconazole | IC50 | 2600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_a8f1d2cb44ef2c1d22b45cacb1b70229.svg) | Citalopram | IC50 | 18800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_1651d7921a8facf41c6a5623ae7707ce.svg) | Diltiazem | IC50 | 12400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_49a577a7a8bf4807ce110cac0f81baf9.svg) | Chlorhexidine | IC50 | 210.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_9eea3482ccbd85339d3c08d99095be33.svg) | Ritonavir | IC50 | 33900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_e2f99194617c96946324b426e112d809.svg) | Erlotinib | IC50 | 16200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_926035c06d9d341c1f456b3b189f3e17.svg) | Mitoxantrone | IC50 | 43900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_38c87cbf7f5f12f867d108fcf8a921dc.svg) | Metoclopramide | IC50 | 94800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_69f1e2f0b60a6951de28604d3a1311ba.svg) | Dobutamine | IC50 | 4170.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_8055fdb52a0be4690c7a5f93e8cd44e9.svg) | Pyrimethamine | IC50 | 13570.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_22ca1744345a750f98669f67193f6275.svg) | Carvedilol | IC50 | 3400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_b517d83684d06e6ce0554cacfb470fe9.svg) | Procainamide | Ki | 73900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_3b2da37f0b0ee76d72c81525a0edc58c.svg) | Clomipramine | IC50 | 19300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_75b4a3ad6d84cdf5a40e35cf9ff23287.svg) | Promethazine | IC50 | 35100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_7de5848be93196a6906eba944a298431.svg) | Sunitinib | IC50 | 6100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_c9960c7f038fe75af1672de453506a31.svg) | Indinavir | IC50 | 208000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_afa07ba3e0b5b4b9daf2ed5946367072.svg) | Nandrolone | IC50 | 35100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_5c2b082f47ad336563283b75e1db518a.svg) | Griseofulvin | IC50 | 7300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_c45117ad154c21e4110d8ec236a71e57.svg) | Ultram | IC50 | 52500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_6c5a78e8ca55529a3f6c3b506ecb26d6.svg) | Clotrimazole | IC50 | 11970.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_8b6095c409ba14f4a2a342d36e7e5bfb.svg) | Cyperquat | Ki | 12300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_53e0258413dfe8503285a6d017480c2b.svg) | Fluphenazine | IC50 | 110000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_168624a25c3c9d480db32878243c3257.svg) | Pantoprazole | IC50 | 500000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_32a1a4e75a5409dde1a18f2173a90394.svg) | Pentamidine | IC50 | 22100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_5a2477912e4297575ff778ccf17d2ed0.svg) | Memantine | IC50 | 27200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_c59762588b8a03ebb9fb4e148eed366e.svg) | Dextromethorphan | IC50 | 10450.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_84d4469c2b25f634938bff679377ae62.svg) | Loperamide | IC50 | 23700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_a93f87e7386d15f182665420dd81b9e5.svg) | Pepcid | IC50 | 300000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_f1389cd1d8b6ba9f0bf28775189ca42b.svg) | Phenformin | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_8a9232a5ccb991c66d47d0b1f1ca286c.svg) | Agmatine | Ki | 24000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_07992946abda58514c65c68057ac00b7.svg) | Amsacrine | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_9a5260e763e5868fc0aa2cf7ef33f02a.svg) | Prochlorperazine | IC50 | 49600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_f4df25a7afebf1dbe9c187a14c4ccbb0.svg) | Promazine | IC50 | 17200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_651e93ab94925b96a9fd90c4ef0d6a82.svg) | Doxepin | IC50 | 11190.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_2cb3539cbcab54cd61d20691715b1d3e.svg) | Tetramethylammonium | Ki | 12400000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_45749eb7b9e4c6bf2c1fd1cfc4a3eb27.svg) | Repaglinide | IC50 | 9200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_8841e892211cc25a2f4450fae2129018.svg) | Oxprenolol | IC50 | 28600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_1726a98f5c906c983c15d93ec617b7f6.svg) | Terazosin | IC50 | 23700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_e2827ec41e052d65c1bbfd99d08fc9a9.svg) | Acebutolol | Ki | 95800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_ae6519a1ba4a52a978e2c8af2e3ff158.svg) | Flupentixol | IC50 | 89500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_be653f89bf9757f77ea6b06dba105b92.svg) | Alfuzosin | IC50 | 14870.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_99974635fe8d76f26549fd768a4d73f4.svg) | Eltrombopag | Ki | 103000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_602cd641a77ba903b85b3fdb24fee22c.svg) | Chlorprothixene | IC50 | 77800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_9199bb281567131db622f149ca71e2fc.svg) | Trimipramine | IC50 | 27700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_99243ad70f3782906d99e25d725ca7ff.svg) | Clemastine | IC50 | 4900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_83f1e5770f1d25a6183bdc3153445774.svg) | N-(2,6-Dichlorobenzylidene)-N'-amidinohydrazine | IC50 | 4850.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_89f632ef3482ab6e2214fd7116ba7ca0.svg) | N-Methylnicotinamide | Ki | 7700000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_f1f3f8e79e46812022d51644a92a50df.svg) | Closantel | IC50 | 3000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_c3b9e7bcc43f821330e3f557e266aed4.svg) | Nifekalant | IC50 | 300000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_966c0c9f833b76ce684ab637ec5135ff.svg) | Dichlorophen | IC50 | 8410.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_4dcc515bda8dfad73cc0eb95dd9c2a87.svg) | Bucindolol | IC50 | 27200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/solute-carrier-family-22-member-1_cda5dec816d821139ec91e51d81c961b.svg) | Denopamine | IC50 | 46900.0 [1] |