Solute carrier family 22 member 1 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Clonidine	IC50	18980.0 [1], 22600.0 [2]
	Clonidine	Ki	550.0 [1]
	Imipramine	IC50	7950.0 [1], 17100.0 [2], 37000.0 [3]
	Cimetidine	IC50	100000.0 [1], 149000.0 [2]
	Cimetidine	Ki	166000.0 [1]
	Quinidine	IC50	23400.0 [1], 113800.0 [2]
	Quinidine	Ki	17500.0 [1]
	Tetraethylammonium	Ki	158000.0 [1], 161000.0 [2], 163000.0 [3]
	Desipramine	IC50	9180.0 [1], 56800.0 [2]
	Desipramine	Ki	5360.0 [1]
	Ondansetron	IC50	20400.0 [1], 100000.0 [2], 300000.0 [3]
	Pseudoisocyanine	IC50	980.0 [1]
	Pseudoisocyanine	Ki	2730.0 [1], 4400.0 [2]
	Corticosterone	IC50	21700.0 [1]
	Corticosterone	Ki	7020.0 [1]
	Verapamil	IC50	6800.0 [1]
	Verapamil	Ki	2900.0 [1]
	Metformin	IC50	1230000.0 [1], 2010000.0 [2]
	Chlorpromazine	IC50	4300.0 [1], 27000.0 [2]
	Prazosin	IC50	1840.0 [1], 9900.0 [2]
	Quinine	IC50	51600.0 [1]
	Quinine	Ki	22900.0 [1]
	Trimethoprim	IC50	50680.0 [1], 56800.0 [2]
	Phenoxybenzamine	IC50	2720.0 [1], 15100.0 [2]
	Vecuronium	Ki	120000.0 [1], 232000.0 [2]
	Tacrine	IC50	21720.0 [1], 83000.0 [2]
	Disopyramide	IC50	81700.0 [1], 100000.0 [2]
	Propafenone	IC50	11100.0 [1], 15540.0 [2]
	Tetrabutylammonium	IC50	52000.0 [1]
	Tetrabutylammonium	Ki	29600.0 [1]
	Orphenadrine	IC50	12600.0 [1], 100000.0 [2]
	Bithionol	IC50	2230.0 [1], 3900.0 [2]
	Tetrapropylammonium	IC50	90000.0 [1]
	Tetrapropylammonium	Ki	102000.0 [1]
	Estradiol	IC50	5730.0 [1]
	Progesterone	IC50	3050.0 [1]
	Morphine	IC50	28000.0 [1]
	Propranolol	IC50	63200.0 [1]
	Atropine	IC50	12200.0 [1]
	Imatinib	IC50	107000.0 [1]
	Haloperidol	IC50	141900.0 [1]
	Midazolam	Ki	3700.0 [1]
	Thiamine	IC50	4354000.0 [1]
	Irinotecan	IC50	20800.0 [1]
	Apomorphine	IC50	20800.0 [1]
	Dipyridamole	IC50	81000.0 [1]
	Amiloride	IC50	57000.0 [1]
	Amitriptyline	IC50	16900.0 [1]
	Ketoconazole	IC50	2600.0 [1]
	Citalopram	IC50	18800.0 [1]
	Diltiazem	IC50	12400.0 [1]
	Chlorhexidine	IC50	210.0 [1]
	Ritonavir	IC50	33900.0 [1]
	Erlotinib	IC50	16200.0 [1]
	Mitoxantrone	IC50	43900.0 [1]
	Metoclopramide	IC50	94800.0 [1]
	Dobutamine	IC50	4170.0 [1]
	Pyrimethamine	IC50	13570.0 [1]
	Carvedilol	IC50	3400.0 [1]
	Procainamide	Ki	73900.0 [1]
	Clomipramine	IC50	19300.0 [1]
	Promethazine	IC50	35100.0 [1]
	Sunitinib	IC50	6100.0 [1]
	Indinavir	IC50	208000.0 [1]
	Nandrolone	IC50	35100.0 [1]
	Griseofulvin	IC50	7300.0 [1]
	Ultram	IC50	52500.0 [1]
	Clotrimazole	IC50	11970.0 [1]
	Cyperquat	Ki	12300.0 [1]
	Fluphenazine	IC50	110000.0 [1]
	Pantoprazole	IC50	500000.0 [1]
	Pentamidine	IC50	22100.0 [1]
	Memantine	IC50	27200.0 [1]
	Dextromethorphan	IC50	10450.0 [1]
	Loperamide	IC50	23700.0 [1]
	Pepcid	IC50	300000.0 [1]
	Phenformin	IC50	10000.0 [1]
	Agmatine	Ki	24000000.0 [1]
	Amsacrine	IC50	5000.0 [1]
	Prochlorperazine	IC50	49600.0 [1]
	Promazine	IC50	17200.0 [1]
	Doxepin	IC50	11190.0 [1]
	Tetramethylammonium	Ki	12400000.0 [1]
	Repaglinide	IC50	9200.0 [1]
	Oxprenolol	IC50	28600.0 [1]
	Terazosin	IC50	23700.0 [1]
	Acebutolol	Ki	95800.0 [1]
	Flupentixol	IC50	89500.0 [1]
	Alfuzosin	IC50	14870.0 [1]
	Eltrombopag	Ki	103000.0 [1]
	Chlorprothixene	IC50	77800.0 [1]
	Trimipramine	IC50	27700.0 [1]
	Clemastine	IC50	4900.0 [1]
	N-(2,6-Dichlorobenzylidene)-N'-amidinohydrazine	IC50	4850.0 [1]
	N-Methylnicotinamide	Ki	7700000.0 [1]
	Closantel	IC50	3000.0 [1]
	Nifekalant	IC50	300000.0 [1]
	Dichlorophen	IC50	8410.0 [1]
	Bucindolol	IC50	27200.0 [1]
	Denopamine	IC50	46900.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 100 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Solute carrier family 22 member 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 31 Mar. 2025, https://www.aatbio.com/data-sets/solute-carrier-family-22-member-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, March 31). Quest Database™ Solute carrier family 22 member 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/solute-carrier-family-22-member-1-inhibitors-ic50-ki.
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