| N-[[3-[2-(4-Fluorophenyl)ethoxy]phenyl]methyl]-2-(4-methoxyphenyl)-N-(pyridin-4-ylmethyl)acetamide | IC50 | 18200.0 [1] |
| 4-Methoxy-N-[[3-[(3-methoxyphenyl)methoxy]phenyl]methyl]-N-(pyridin-4-ylmethyl)benzamide | IC50 | 11000.0 [1] |
| Chembl4164091 | IC50 | 20000.0 [1] |
| Chembl4171968 | IC50 | 1700.0 [1] |
| 4-[[2-(4-Chlorophenyl)-6-(2-fluorophenyl)imidazo[1,2-a]pyridin-3-yl]methyl]morpholine | IC50 | 6.0 [1] |
| (2S)-3-(4-Fluorophenyl)-2-[[2-(3-hydroxyphenyl)acetyl]amino]-N-[(1S)-1-phenylethyl]propanamide | IC50 | 195.0 [1] |
| (2S)-3-(2-Bromophenyl)-2-[[2-(4-methoxyphenyl)acetyl]amino]-N-[(1S)-1-phenylethyl]propanamide | IC50 | 90.0 [1] |
| 4-[[2-(4-Chlorophenyl)-6-(4-fluorophenyl)imidazo[1,2-a]pyridin-3-yl]methyl]morpholine | IC50 | 10000.0 [1] |
| 4-[[6-(2-Chlorophenyl)-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-3-yl]methyl]morpholine | IC50 | 6.0 [1] |
| 4-[[2-(4-Chlorophenyl)-6-(2,6-difluorophenyl)imidazo[1,2-a]pyridin-3-yl]methyl]morpholine | IC50 | 6.0 [1] |
| 4-[[2-(2,4-Dichlorophenyl)-6-phenylimidazo[1,2-a]pyridin-3-yl]methyl]morpholine | IC50 | 6.0 [1] |
| 4-[[2-(4-Chlorophenyl)-5-methyl-6-phenylimidazo[1,2-a]pyridin-3-yl]methyl]morpholine | IC50 | 6.0 [1] |
| 4-[[2-(4-Chlorophenyl)-6-cyclopropylimidazo[1,2-a]pyrazin-3-yl]methyl]morpholine | IC50 | 6.0 [1] |
| 1-[4-[[2-(4-Chlorophenyl)-6-cyclopropylimidazo[1,2-a]pyrazin-3-yl]methyl]piperazin-1-yl]ethanone | IC50 | 6.0 [1] |
| 2-[3-[(4-Acetylpiperazin-1-yl)methyl]-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-6-yl]benzonitrile | IC50 | 6.0 [1] |
| 4-[[2-(4-Chlorophenyl)-6-(2,6-difluorophenyl)imidazo[1,2-a]pyrazin-3-yl]methyl]morpholine | IC50 | 6.0 [1] |
| N-[2-(4-Chlorophenyl)-3-(morpholin-4-ylmethyl)imidazo[1,2-a]pyridin-6-yl]-N-methylmethanesulfonamide | IC50 | 6.0 [1] |
| [4-[[2-(4-Chlorophenyl)-6-cyclopropylimidazo[1,2-a]pyrazin-3-yl]methyl]piperazin-1-yl]-pyridin-4-ylmethanone | IC50 | 6.0 [1] |
| 1-[4-[[6-Cyclopropyl-2-(2,4-dichlorophenyl)imidazo[1,2-a]pyrazin-3-yl]methyl]piperazin-1-yl]ethanone | IC50 | 6.0 [1] |
| [4-[[6-Cyclopropyl-2-(2,4-dichlorophenyl)imidazo[1,2-a]pyrazin-3-yl]methyl]piperazin-1-yl]-pyrazin-2-ylmethanone | IC50 | 6.0 [1] |
| [4-[[6-Cyclopropyl-2-(2,4-dichlorophenyl)imidazo[1,2-a]pyrazin-3-yl]methyl]piperazin-1-yl]-pyridazin-4-ylmethanone | IC50 | 6.0 [1] |
| [4-[[6-Cyclopropyl-2-(2,4-dichlorophenyl)imidazo[1,2-a]pyrazin-3-yl]methyl]piperazin-1-yl]-(oxan-4-yl)methanone | IC50 | 6.0 [1] |
| [4-[[6-Cyclopropyl-2-(2,4-dichlorophenyl)imidazo[1,2-a]pyrazin-3-yl]methyl]piperazin-1-yl]-(1,3-thiazol-4-yl)methanone | IC50 | 6.0 [1] |
| N-[2-(4-Chlorophenyl)-3-[[4-(2-methoxyacetyl)piperazin-1-yl]methyl]imidazo[1,2-a]pyridin-6-yl]-N-methylmethanesulfonamide | IC50 | 6.0 [1] |
| N-[2-(4-Chlorophenyl)-3-[[4-(oxetane-3-carbonyl)piperazin-1-yl]methyl]imidazo[1,2-a]pyridin-6-yl]-N-methylmethanesulfonamide | IC50 | 6.0 [1] |
| N-[2-(4-Chlorophenyl)-3-[[4-(pyridazine-4-carbonyl)piperazin-1-yl]methyl]imidazo[1,2-a]pyridin-6-yl]-N-methylmethanesulfonamide | IC50 | 6.0 [1] |
| 1-[4-[[6-Cyclopropyl-2-(2,4-dichlorophenyl)imidazo[1,2-a]pyrazin-3-yl]methyl]piperazin-1-yl]-2-methoxyethanone | IC50 | 6.0 [1] |
| N-[3-[(4-Acetylpiperazin-1-yl)methyl]-2-(2,4-dichlorophenyl)imidazo[1,2-a]pyridin-6-yl]methanesulfonamide | IC50 | 6.0 [1] |
| N-[3-[(4-Acetylpiperazin-1-yl)methyl]-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-6-yl]ethanesulfonamide | IC50 | 6.0 [1] |
| N-[3-[(4-Acetylpiperazin-1-yl)methyl]-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-6-yl]-N-methylethanesulfonamide | IC50 | 6.0 [1] |
| 1-[4-[[6-Cyclopropyl-2-(2,4-dichlorophenyl)imidazo[1,2-a]pyrazin-3-yl]methyl]piperazin-1-yl]-2-hydroxy-2-methylpropan-1-one | IC50 | 6.0 [1] |
| 1-[4-[[6-Cyclopropyl-2-(2,4-dichlorophenyl)imidazo[1,2-a]pyrazin-3-yl]methyl]piperazin-1-yl]-2-hydroxyethanone | IC50 | 6.0 [1] |
| 1-[4-[[2-(4-Chlorophenyl)-6-(1,1-dioxothiazinan-2-yl)imidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]ethanone | IC50 | 6.0 [1] |
| N-[3-[(4-Acetylpiperazin-1-yl)methyl]-2-(2,4-dichlorophenyl)imidazo[1,2-a]pyridin-6-yl]-N-methylmethanesulfonamide | IC50 | 6.0 [1] |
| N-[2-(2,4-Dichlorophenyl)-3-[[4-(oxetane-3-carbonyl)piperazin-1-yl]methyl]imidazo[1,2-a]pyridin-6-yl]methanesulfonamide | IC50 | 6.0 [1] |
| N-[2-(2,4-Dichlorophenyl)-3-[[4-(2-methoxyacetyl)piperazin-1-yl]methyl]imidazo[1,2-a]pyridin-6-yl]-N-methylmethanesulfonamide | IC50 | 6.0 [1] |
| N-[2-(2,4-Dichlorophenyl)-3-[[4-(oxetane-3-carbonyl)piperazin-1-yl]methyl]imidazo[1,2-a]pyridin-6-yl]-N-methylmethanesulfonamide | IC50 | 6.0 [1] |
| N-[2-(2,4-Dichlorophenyl)-3-[[4-(2-methoxyacetyl)piperazin-1-yl]methyl]imidazo[1,2-a]pyridin-6-yl]methanesulfonamide | IC50 | 6.0 [1] |
| 1-[4-[[2-(2,4-Dichlorophenyl)-6-(1,1-dioxo-1,2-thiazolidin-2-yl)imidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]ethanone | IC50 | 6.0 [1] |
| N-[3-[(4-Acetylpiperazin-1-yl)methyl]-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-6-yl]-N-methylpropane-2-sulfonamide | IC50 | 6.0 [1] |
| N-[3-[(4-Acetylpiperazin-1-yl)methyl]-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-6-yl]-N-methylpropane-1-sulfonamide | IC50 | 6.0 [1] |
| N-[2-(2,4-Dichlorophenyl)-3-(6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazin-7-ylmethyl)imidazo[1,2-a]pyridin-6-yl]-N-methylmethanesulfonamide | IC50 | 6.0 [1] |
| 3-[(4-Acetylpiperazin-1-yl)methyl]-2-(4-chlorophenyl)-N,N-dimethylimidazo[1,2-a]pyridine-6-sulfonamide | IC50 | 6.0 [1] |
| N-[3-[(4-Acetylpiperazin-1-yl)methyl]-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-6-yl]-N-ethylmethanesulfonamide | IC50 | 6.0 [1] |
| N-[2-(2,4-Dichlorophenyl)-3-[[4-(pyridazine-4-carbonyl)piperazin-1-yl]methyl]imidazo[1,2-a]pyridin-6-yl]methanesulfonamide | IC50 | 6.0 [1] |
| N-[2-(2,4-Dichlorophenyl)-3-[(3-oxopiperazin-1-yl)methyl]imidazo[1,2-a]pyridin-6-yl]-N-methylmethanesulfonamide | IC50 | 6.0 [1] |
| N-[2-(2,4-Dichlorophenyl)-3-[[4-(4-fluorobenzoyl)piperazin-1-yl]methyl]imidazo[1,2-a]pyridin-6-yl]methanesulfonamide | IC50 | 6.0 [1] |
| N-[2-(2,4-Dichlorophenyl)-3-[[4-(2-hydroxy-2-methylpropanoyl)piperazin-1-yl]methyl]imidazo[1,2-a]pyridin-6-yl]methanesulfonamide | IC50 | 6.0 [1] |
| N-[2-(2,4-Dichlorophenyl)-3-[[4-(4-fluorobenzoyl)piperazin-1-yl]methyl]imidazo[1,2-a]pyridin-6-yl]-N-methylmethanesulfonamide | IC50 | 6.0 [1] |
| N-[2-(2,4-Dichlorophenyl)-3-[[4-(1-methylpyrazole-4-carbonyl)piperazin-1-yl]methyl]imidazo[1,2-a]pyridin-6-yl]methanesulfonamide | IC50 | 6.0 [1] |
| N-[2-(2,4-Dichlorophenyl)-3-[(4-hydroxypiperazin-1-yl)methyl]imidazo[1,2-a]pyridin-6-yl]methanesulfonamide | IC50 | 6.0 [1] |
| 4-[[2-(2,4-Dichlorophenyl)-6-propan-2-ylimidazo[1,2-a]pyrazin-3-yl]methyl]morpholine | IC50 | 6.0 [1] |
| N-[3-[(4-Acetylpiperazin-1-yl)methyl]-2-(2,4-dichlorophenyl)imidazo[1,2-a]pyridin-6-yl]-N-(difluoromethyl)methanesulfonamide | IC50 | 6.0 [1] |
| N-[3-[(4-Acetylpiperazin-1-yl)methyl]-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-6-yl]-N-(difluoromethyl)methanesulfonamide | IC50 | 6.0 [1] |
| N-[2-(2,4-Dichlorophenyl)-3-[[4-(oxane-4-carbonyl)piperazin-1-yl]methyl]imidazo[1,2-a]pyridin-6-yl]-N-methylmethanesulfonamide | IC50 | 6.0 [1] |
| N-[2-(2,4-Dichlorophenyl)-3-[(6-oxo-1,3,4,7,8,8a-hexahydropyrrolo[1,2-a]pyrazin-2-yl)methyl]imidazo[1,2-a]pyridin-6-yl]methanesulfonamide | IC50 | 6.0 [1] |
| N-[2-(2,4-Dichlorophenyl)-3-[[4-(2-hydroxyacetyl)piperazin-1-yl]methyl]imidazo[1,2-a]pyridin-6-yl]-N-methylmethanesulfonamide | IC50 | 6.0 [1] |
| 1-[4-[[2-(4-Chlorophenyl)-6-methylsulfanylimidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]ethanone | IC50 | 6.0 [1] |
| 1-[4-[[2-(4-Chlorophenyl)-6-propan-2-ylsulfonylimidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]ethanone | IC50 | 6.0 [1] |
| N-[2-(2,4-Dichlorophenyl)-3-[(6-oxo-1,3,4,7,8,8a-hexahydropyrrolo[1,2-a]pyrazin-2-yl)methyl]imidazo[1,2-a]pyridin-6-yl]-N-methylmethanesulfonamide | IC50 | 6.0 [1] |
| N-[2-(2,4-Dichlorophenyl)-3-[[4-(2-hydroxy-2-methylpropanoyl)piperazin-1-yl]methyl]imidazo[1,2-a]pyridin-6-yl]-N-methylmethanesulfonamide | IC50 | 6.0 [1] |
| 1-[4-[[2-(4-Chlorophenyl)-6-ethylsulfonylimidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]ethanone | IC50 | 6.0 [1] |
| N-[3-[(4-Acetylpiperazin-1-yl)methyl]-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-6-yl]-N-propan-2-ylmethanesulfonamide | IC50 | 6.0 [1] |
| N-[2-(2,4-Dichlorophenyl)-3-[[4-(pyridazine-4-carbonyl)piperazin-1-yl]methyl]imidazo[1,2-a]pyridin-6-yl]-N-methylmethanesulfonamide | IC50 | 6.0 [1] |
| 1-[4-[[2-(4-Chlorophenyl)-6-methylsulfonylimidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]ethanone | IC50 | 6.0 [1] |
| 2-[[2-(4-Chlorophenyl)-6-cyclopropylimidazo[1,2-a]pyrazin-3-yl]methyl]-1,3,4,7,8,8a-hexahydropyrrolo[1,2-a]pyrazin-6-one | IC50 | 6.0 [1] |
| N-[2-(2,4-Dichlorophenyl)-3-[[4-(oxane-4-carbonyl)piperazin-1-yl]methyl]imidazo[1,2-a]pyridin-6-yl]methanesulfonamide | IC50 | 6.0 [1] |
| 3-[(4-Acetylpiperazin-1-yl)methyl]-2-(4-chlorophenyl)-N-methylimidazo[1,2-a]pyridine-6-sulfonamide | IC50 | 6.0 [1] |
| [4-[[2-(4-Chlorophenyl)-6-phenylimidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-(3-fluorophenyl)methanone | IC50 | 6.0 [1] |